| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | PRKACA | KAPCA_HUMAN | 6NO7E | P17612 | 13 | 351 | 351.0 | ATP:60403 | ATPlike | Inactive | DFGin | 6.9335 | 14.1655 | BLAminus | -118.71, 175.9 | 64.55, 75.01 | -86.85, 19.7 | 273.68, 51.02 | -43.49, -41.12 | in-out | in | 9.4189 | Saltbr-out | 5.4559 | HRD-in | -91.66, -53.62 | 73.72, 11.47 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.1639 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.9, 150.23 | APE9-dihe-na | 149.21, -142.3 | APE8-dihe-in | -132.1, 131.95 | APE8-rot-in | 297.19 | APE67-dihe-in | -64.62, -25.64 | -37.25, -53.79 | APE12-dist-in | 8.0557 | APE11-dist-in | 10.9843 | APE10-dist-in | 5.7482 | APE9-dist-in | 3.2156 | None | SEP140,TPO198,SEP339 | SEP140,TPO198,SEP339 | XRAY | 3.55 | 0.259 | 0.269 | E | 350.0 | 339.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6no7 | AGC_PRKACA_HUMAN | AGC | 4.5e-95 | 323.7 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| AGC | PRKACA | KAPCA_HUMAN | 6NO7G | P17612 | 15 | 351 | 351.0 | ATP:60403 | ATPlike | Inactive | DFGin | 6.0359 | 14.0844 | BLAminus | -118.68, 176.55 | 65.34, 76.32 | -85.78, 18.75 | 273.72, 51.07 | -44.34, -41.82 | in-out | in | 9.7125 | Saltbr-out | 5.2149 | HRD-in | -91.95, -53.38 | 74.11, 11.57 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.3017 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.42, 149.81 | APE9-dihe-na | 148.91, -142.4 | APE8-dihe-in | -132.18, 131.68 | APE8-rot-in | 297.12 | APE67-dihe-in | -64.98, -25.0 | -37.42, -54.32 | APE12-dist-in | 7.6679 | APE11-dist-in | 10.658 | APE10-dist-in | 5.5534 | APE9-dist-in | 3.4096 | None | SEP140,TPO198,SEP339 | SEP140,TPO198,SEP339 | XRAY | 3.55 | 0.259 | 0.269 | G | 350.0 | 337.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6no7 | AGC_PRKACA_HUMAN | AGC | 4.5e-95 | 323.7 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| AGC | PRKACA | KAPCA_HUMAN | 6NO7A | P17612 | 16 | 351 | 351.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5833 | 14.5513 | BLAminus | -119.16, 176.65 | 65.47, 76.79 | -85.63, 19.52 | 273.14, 48.34 | -44.12, -41.29 | in-out | in | 9.256 | Saltbr-out | 3.8369 | HRD-in | -93.59, -54.13 | 73.95, 11.29 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.0846 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.66, 149.89 | APE9-dihe-na | 148.72, -142.64 | APE8-dihe-in | -132.35, 131.6 | APE8-rot-in | 297.3 | APE67-dihe-in | -65.08, -25.39 | -37.56, -54.33 | APE12-dist-in | 7.8572 | APE11-dist-in | 10.7351 | APE10-dist-in | 5.368 | APE9-dist-in | 3.3109 | None | SEP140,TPO198,SEP339 | SEP140,TPO198,SEP339 | XRAY | 3.55 | 0.259 | 0.269 | A | 350.0 | 336.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6no7 | AGC_PRKACA_HUMAN | AGC | 4.5e-95 | 323.7 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| AGC | PRKACA | KAPCA_HUMAN | 6NO7C | P17612 | 12 | 351 | 351.0 | No_ligand | No_ligand | Active | DFGin | 5.3091 | 14.0414 | BLAminus | -119.31, 176.37 | 65.24, 77.94 | -84.43, 19.43 | 273.37, 51.07 | -43.97, -41.52 | in-in | in | 8.987 | Saltbr-in | 2.3597 | HRD-in | -94.38, -54.81 | 73.77, 10.87 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9661 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.7, 149.95 | APE9-dihe-na | 149.29, -142.75 | APE8-dihe-in | -132.31, 130.88 | APE8-rot-in | 297.15 | APE67-dihe-in | -65.36, -25.54 | -38.33, -55.04 | APE12-dist-in | 8.372 | APE11-dist-in | 10.8625 | APE10-dist-in | 5.5723 | APE9-dist-in | 3.1598 | None | SEP140,TPO198,SEP339 | SEP140,TPO198,SEP339 | XRAY | 3.55 | 0.259 | 0.269 | C | 350.0 | 340.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6no7 | AGC_PRKACA_HUMAN | AGC | 4.5e-95 | 323.7 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | PRKACA | KAPCA_HUMAN | 6NO7E | P17612 | 13 | 351 | 351.0 | ATP:60403 | ATPlike | Inactive | DFGin | 6.9335 | 14.1655 | BLAminus | -118.71, 175.9 | 64.55, 75.01 | -86.85, 19.7 | 273.68, 51.02 | -43.49, -41.12 | in-out | in | 9.4189 | Saltbr-out | 5.4559 | HRD-in | -91.66, -53.62 | 73.72, 11.47 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.1639 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.9, 150.23 | APE9-dihe-na | 149.21, -142.3 | APE8-dihe-in | -132.1, 131.95 | APE8-rot-in | 297.19 | APE67-dihe-in | -64.62, -25.64 | -37.25, -53.79 | APE12-dist-in | 8.0557 | APE11-dist-in | 10.9843 | APE10-dist-in | 5.7482 | APE9-dist-in | 3.2156 | None | SEP140,TPO198,SEP339 | SEP140,TPO198,SEP339 | XRAY | 3.55 | 0.259 | 0.269 | E | 350.0 | 339.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6no7 | Homo sapiens | AGC_PRKACA_HUMAN | AGC | 4.5e-95 | 323.7 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| AGC | PRKACA | KAPCA_HUMAN | 6NO7G | P17612 | 15 | 351 | 351.0 | ATP:60403 | ATPlike | Inactive | DFGin | 6.0359 | 14.0844 | BLAminus | -118.68, 176.55 | 65.34, 76.32 | -85.78, 18.75 | 273.72, 51.07 | -44.34, -41.82 | in-out | in | 9.7125 | Saltbr-out | 5.2149 | HRD-in | -91.95, -53.38 | 74.11, 11.57 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.3017 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.42, 149.81 | APE9-dihe-na | 148.91, -142.4 | APE8-dihe-in | -132.18, 131.68 | APE8-rot-in | 297.12 | APE67-dihe-in | -64.98, -25.0 | -37.42, -54.32 | APE12-dist-in | 7.6679 | APE11-dist-in | 10.658 | APE10-dist-in | 5.5534 | APE9-dist-in | 3.4096 | None | SEP140,TPO198,SEP339 | SEP140,TPO198,SEP339 | XRAY | 3.55 | 0.259 | 0.269 | G | 350.0 | 337.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6no7 | Homo sapiens | AGC_PRKACA_HUMAN | AGC | 4.5e-95 | 323.7 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| AGC | PRKACA | KAPCA_HUMAN | 6NO7A | P17612 | 16 | 351 | 351.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5833 | 14.5513 | BLAminus | -119.16, 176.65 | 65.47, 76.79 | -85.63, 19.52 | 273.14, 48.34 | -44.12, -41.29 | in-out | in | 9.256 | Saltbr-out | 3.8369 | HRD-in | -93.59, -54.13 | 73.95, 11.29 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.0846 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.66, 149.89 | APE9-dihe-na | 148.72, -142.64 | APE8-dihe-in | -132.35, 131.6 | APE8-rot-in | 297.3 | APE67-dihe-in | -65.08, -25.39 | -37.56, -54.33 | APE12-dist-in | 7.8572 | APE11-dist-in | 10.7351 | APE10-dist-in | 5.368 | APE9-dist-in | 3.3109 | None | SEP140,TPO198,SEP339 | SEP140,TPO198,SEP339 | XRAY | 3.55 | 0.259 | 0.269 | A | 350.0 | 336.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6no7 | Homo sapiens | AGC_PRKACA_HUMAN | AGC | 4.5e-95 | 323.7 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| AGC | PRKACA | KAPCA_HUMAN | 6NO7C | P17612 | 12 | 351 | 351.0 | No_ligand | No_ligand | Active | DFGin | 5.3091 | 14.0414 | BLAminus | -119.31, 176.37 | 65.24, 77.94 | -84.43, 19.43 | 273.37, 51.07 | -43.97, -41.52 | in-in | in | 8.987 | Saltbr-in | 2.3597 | HRD-in | -94.38, -54.81 | 73.77, 10.87 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9661 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -161.7, 149.95 | APE9-dihe-na | 149.29, -142.75 | APE8-dihe-in | -132.31, 130.88 | APE8-rot-in | 297.15 | APE67-dihe-in | -65.36, -25.54 | -38.33, -55.04 | APE12-dist-in | 8.372 | APE11-dist-in | 10.8625 | APE10-dist-in | 5.5723 | APE9-dist-in | 3.1598 | None | SEP140,TPO198,SEP339 | SEP140,TPO198,SEP339 | XRAY | 3.55 | 0.259 | 0.269 | C | 350.0 | 340.0 | 0 | 25 | 25 | 0 | [[44, 298]] | 1.0 | 6no7 | Homo sapiens | AGC_PRKACA_HUMAN | AGC | 4.5e-95 | 323.7 | 1.0 | 260.0 | 260.0 | 184 | 185 | 186 | 188 | 190 | 73 | 92 | 96 | 164 | 166 | 165 | 167.0 | 221 | 209 | 204 | 203 | 202 | 201 | 200 | 199 | 198 | 122 | cAMP-dependent protein kinase catalytic subunit alpha |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|