| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 6LVLA | P21802 | 468 | 766 | 821.0 | EVL:802 | Type1 | Inactive | DFGin | 6.6092 | 14.5299 | BLAminus | -146.15, -175.25 | 63.31, 72.06 | -88.46, 19.6 | 283.4, 82.21 | -53.64, -28.47 | in-in | in | 7.721 | Saltbr-in | 2.6325 | HRD-in | -74.18, -46.26 | 67.97, -0.94 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8589 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.16, 11.22 | APE9-dihe-in | -81.14, 133.04 | APE8-dihe-in | -57.2, 120.46 | APE8-rot-na | 339.92 | APE67-dihe-in | -68.23, -11.94 | -62.32, -43.83 | APE12-dist-na | 10.1631 | APE11-dist-na | 10.9531 | APE10-dist-na | 7.5362 | APE9-dist-in | 4.8939 | None | None | None | XRAY | 2.98 | 0.204 | 0.251 | A | 313.0 | 288.0 | 11 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 6lvl | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 6LVLB | P21802 | 468 | 765 | 821.0 | EVL:804 | Type1 | Inactive | DFGin | 6.5042 | 14.3785 | BLAminus | -137.97, -168.86 | 49.59, 89.79 | -98.61, 21.56 | 282.72, 81.93 | -60.4, -25.9 | in-in | in | 7.4759 | Saltbr-in | 2.7729 | HRD-in | -74.99, -51.02 | 79.49, -6.99 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8144 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.2, 10.06 | APE9-dihe-in | -85.19, 131.23 | APE8-dihe-in | -58.17, 126.23 | APE8-rot-na | 336.1 | APE67-dihe-in | -79.35, -7.86 | -72.73, -22.05 | APE12-dist-na | 10.0306 | APE11-dist-na | 10.8423 | APE10-dist-na | 7.4474 | APE9-dist-in | 4.8471 | None | None | None | XRAY | 2.98 | 0.204 | 0.251 | B | 313.0 | 286.0 | 12 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 6lvl | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 6LVLA | P21802 | 468 | 766 | 821.0 | EVL:802 | Type1 | Inactive | DFGin | 6.6092 | 14.5299 | BLAminus | -146.15, -175.25 | 63.31, 72.06 | -88.46, 19.6 | 283.4, 82.21 | -53.64, -28.47 | in-in | in | 7.721 | Saltbr-in | 2.6325 | HRD-in | -74.18, -46.26 | 67.97, -0.94 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8589 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -117.16, 11.22 | APE9-dihe-in | -81.14, 133.04 | APE8-dihe-in | -57.2, 120.46 | APE8-rot-na | 339.92 | APE67-dihe-in | -68.23, -11.94 | -62.32, -43.83 | APE12-dist-na | 10.1631 | APE11-dist-na | 10.9531 | APE10-dist-na | 7.5362 | APE9-dist-in | 4.8939 | None | None | None | XRAY | 2.98 | 0.204 | 0.251 | A | 313.0 | 288.0 | 11 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 6lvl | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 6LVLB | P21802 | 468 | 765 | 821.0 | EVL:804 | Type1 | Inactive | DFGin | 6.5042 | 14.3785 | BLAminus | -137.97, -168.86 | 49.59, 89.79 | -98.61, 21.56 | 282.72, 81.93 | -60.4, -25.9 | in-in | in | 7.4759 | Saltbr-in | 2.7729 | HRD-in | -74.99, -51.02 | 79.49, -6.99 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8144 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.2, 10.06 | APE9-dihe-in | -85.19, 131.23 | APE8-dihe-in | -58.17, 126.23 | APE8-rot-na | 336.1 | APE67-dihe-in | -79.35, -7.86 | -72.73, -22.05 | APE12-dist-na | 10.0306 | APE11-dist-na | 10.8423 | APE10-dist-na | 7.4474 | APE9-dist-in | 4.8471 | None | None | None | XRAY | 2.98 | 0.204 | 0.251 | B | 313.0 | 286.0 | 12 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 6lvl | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|