| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | CLK2 | CLK2_HUMAN | 6FYKA | P49760 | 137 | 485 | 499.0 | EAZ:501 | Type1 | Active | DFGin | 7.0247 | 13.933 | BLAminus | -128.78, 177.13 | 62.38, 94.51 | -113.34, 21.4 | 294.8, 89.41 | -67.4, -12.68 | in-in | in | 8.6929 | Saltbr-in | 2.6136 | HRD-in | -66.97, -50.97 | 77.07, -17.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7927 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.9, 169.97 | APE9-dihe-na | 71.5, 144.52 | APE8-dihe-in | -67.7, 143.43 | APE8-rot-in | 294.43 | APE67-dihe-in | -55.56, -28.09 | -39.63, -56.25 | APE12-dist-in | 13.2898 | APE11-dist-in | 11.7062 | APE10-dist-in | 7.4097 | APE9-dist-in | 2.9513 | None | None | None | XRAY | 2.39 | 0.196 | 0.228 | A | 363.0 | 349.0 | 0 | 25 | 25 | 0 | [[163, 479]] | 1.0 | 6fyk | CMGC_CLK2_HUMAN | CMGC | 1.7e-92 | 315.7 | 1.0 | 301.0 | 301.0 | 326 | 327 | 328 | 330 | 332 | 193 | 208 | 212 | 287 | 289 | 288 | 290.0 | 363 | 351 | 346 | 345 | 344 | 343 | 342 | 341 | 340 | 244 | Dual specificity protein kinase CLK2 |
| CMGC | CLK2 | CLK2_HUMAN | 6FYKB | P49760 | 137 | 485 | 499.0 | EAZ:501 | Type1 | Active | DFGin | 6.9791 | 13.5453 | BLAminus | -126.36, 176.1 | 65.04, 89.02 | -110.3, 25.2 | 302.84, 96.68 | -72.78, -13.24 | in-in | in | 8.5714 | Saltbr-in | 2.6918 | HRD-in | -74.27, -47.13 | 73.72, -15.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.834 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.26, 173.72 | APE9-dihe-na | 72.32, 147.64 | APE8-dihe-in | -71.42, 138.78 | APE8-rot-in | 296.31 | APE67-dihe-in | -62.52, -26.37 | -31.99, -52.81 | APE12-dist-in | 13.304 | APE11-dist-in | 11.8792 | APE10-dist-in | 7.3646 | APE9-dist-in | 2.8961 | None | None | None | XRAY | 2.39 | 0.196 | 0.228 | B | 363.0 | 349.0 | 0 | 25 | 25 | 0 | [[163, 479]] | 1.0 | 6fyk | CMGC_CLK2_HUMAN | CMGC | 1.7e-92 | 315.7 | 1.0 | 301.0 | 301.0 | 326 | 327 | 328 | 330 | 332 | 193 | 208 | 212 | 287 | 289 | 288 | 290.0 | 363 | 351 | 346 | 345 | 344 | 343 | 342 | 341 | 340 | 244 | Dual specificity protein kinase CLK2 |
| CMGC | CLK2 | CLK2_HUMAN | 6FYKC | P49760 | 137 | 485 | 499.0 | EAZ:501 | Type1 | Active | DFGin | 7.1797 | 13.8088 | BLAminus | -122.42, 175.39 | 66.62, 94.13 | -114.05, 24.08 | 298.67, 87.87 | -71.48, -13.77 | in-in | in | 8.5576 | Saltbr-in | 2.7503 | HRD-in | -70.0, -49.32 | 73.58, -20.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8236 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.75, 171.99 | APE9-dihe-na | 73.44, 147.9 | APE8-dihe-in | -74.12, 135.91 | APE8-rot-in | 297.57 | APE67-dihe-in | -59.91, -18.18 | -29.96, -58.43 | APE12-dist-in | 13.4365 | APE11-dist-in | 12.0418 | APE10-dist-in | 7.4714 | APE9-dist-in | 3.0303 | None | None | None | XRAY | 2.39 | 0.196 | 0.228 | C | 363.0 | 349.0 | 0 | 25 | 25 | 0 | [[163, 479]] | 1.0 | 6fyk | CMGC_CLK2_HUMAN | CMGC | 1.7e-92 | 315.7 | 1.0 | 301.0 | 301.0 | 326 | 327 | 328 | 330 | 332 | 193 | 208 | 212 | 287 | 289 | 288 | 290.0 | 363 | 351 | 346 | 345 | 344 | 343 | 342 | 341 | 340 | 244 | Dual specificity protein kinase CLK2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | CLK2 | CLK2_HUMAN | 6FYKA | P49760 | 137 | 485 | 499.0 | EAZ:501 | Type1 | Active | DFGin | 7.0247 | 13.933 | BLAminus | -128.78, 177.13 | 62.38, 94.51 | -113.34, 21.4 | 294.8, 89.41 | -67.4, -12.68 | in-in | in | 8.6929 | Saltbr-in | 2.6136 | HRD-in | -66.97, -50.97 | 77.07, -17.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7927 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.9, 169.97 | APE9-dihe-na | 71.5, 144.52 | APE8-dihe-in | -67.7, 143.43 | APE8-rot-in | 294.43 | APE67-dihe-in | -55.56, -28.09 | -39.63, -56.25 | APE12-dist-in | 13.2898 | APE11-dist-in | 11.7062 | APE10-dist-in | 7.4097 | APE9-dist-in | 2.9513 | None | None | None | XRAY | 2.39 | 0.196 | 0.228 | A | 363.0 | 349.0 | 0 | 25 | 25 | 0 | [[163, 479]] | 1.0 | 6fyk | Homo sapiens | CMGC_CLK2_HUMAN | CMGC | 1.7e-92 | 315.7 | 1.0 | 301.0 | 301.0 | 326 | 327 | 328 | 330 | 332 | 193 | 208 | 212 | 287 | 289 | 288 | 290.0 | 363 | 351 | 346 | 345 | 344 | 343 | 342 | 341 | 340 | 244 | Dual specificity protein kinase CLK2 |
| CMGC | CLK2 | CLK2_HUMAN | 6FYKB | P49760 | 137 | 485 | 499.0 | EAZ:501 | Type1 | Active | DFGin | 6.9791 | 13.5453 | BLAminus | -126.36, 176.1 | 65.04, 89.02 | -110.3, 25.2 | 302.84, 96.68 | -72.78, -13.24 | in-in | in | 8.5714 | Saltbr-in | 2.6918 | HRD-in | -74.27, -47.13 | 73.72, -15.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.834 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -119.26, 173.72 | APE9-dihe-na | 72.32, 147.64 | APE8-dihe-in | -71.42, 138.78 | APE8-rot-in | 296.31 | APE67-dihe-in | -62.52, -26.37 | -31.99, -52.81 | APE12-dist-in | 13.304 | APE11-dist-in | 11.8792 | APE10-dist-in | 7.3646 | APE9-dist-in | 2.8961 | None | None | None | XRAY | 2.39 | 0.196 | 0.228 | B | 363.0 | 349.0 | 0 | 25 | 25 | 0 | [[163, 479]] | 1.0 | 6fyk | Homo sapiens | CMGC_CLK2_HUMAN | CMGC | 1.7e-92 | 315.7 | 1.0 | 301.0 | 301.0 | 326 | 327 | 328 | 330 | 332 | 193 | 208 | 212 | 287 | 289 | 288 | 290.0 | 363 | 351 | 346 | 345 | 344 | 343 | 342 | 341 | 340 | 244 | Dual specificity protein kinase CLK2 |
| CMGC | CLK2 | CLK2_HUMAN | 6FYKC | P49760 | 137 | 485 | 499.0 | EAZ:501 | Type1 | Active | DFGin | 7.1797 | 13.8088 | BLAminus | -122.42, 175.39 | 66.62, 94.13 | -114.05, 24.08 | 298.67, 87.87 | -71.48, -13.77 | in-in | in | 8.5576 | Saltbr-in | 2.7503 | HRD-in | -70.0, -49.32 | 73.58, -20.32 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8236 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -130.75, 171.99 | APE9-dihe-na | 73.44, 147.9 | APE8-dihe-in | -74.12, 135.91 | APE8-rot-in | 297.57 | APE67-dihe-in | -59.91, -18.18 | -29.96, -58.43 | APE12-dist-in | 13.4365 | APE11-dist-in | 12.0418 | APE10-dist-in | 7.4714 | APE9-dist-in | 3.0303 | None | None | None | XRAY | 2.39 | 0.196 | 0.228 | C | 363.0 | 349.0 | 0 | 25 | 25 | 0 | [[163, 479]] | 1.0 | 6fyk | Homo sapiens | CMGC_CLK2_HUMAN | CMGC | 1.7e-92 | 315.7 | 1.0 | 301.0 | 301.0 | 326 | 327 | 328 | 330 | 332 | 193 | 208 | 212 | 287 | 289 | 288 | 290.0 | 363 | 351 | 346 | 345 | 344 | 343 | 342 | 341 | 340 | 244 | Dual specificity protein kinase CLK2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|