| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EPHA2 | EPHA2_HUMAN | 6FNHA | P29317 | 602 | 889 | 976.0 | DXK:1001 | Type1 | Inactive | DFGin | 6.0291 | 15.2866 | ABAminus | -132.89, -13.6 | -114.29, 112.91 | -120.16, 34.85 | 297.73, 92.28 | -68.77, 147.18 | in-in | in | 8.5707 | Saltbr-in | 2.5241 | HRD-in | -71.64, -49.56 | 77.94, -13.05 | in-out-in | SNCioi | out-in | ActLoopNT-out | 10.9018 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -86.64, 136.2 | APE9-dihe-in | -91.95, 112.57 | APE8-dihe-in | -77.45, 142.7 | APE8-rot-na | 28.74 | APE67-dihe-in | -60.57, -18.72 | -57.08, -38.55 | APE12-dist-na | 999.0 | APE11-dist-na | 8.3826 | APE10-dist-na | 12.3766 | APE9-dist-in | 5.4468 | None | None | None | XRAY | 1.379 | 0.206 | 0.221 | A | 306.0 | 277.0 | 11 | 31 | 21 | 10 | [[613, 873]] | 1.0 | 6fnh | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 6FNHB | P29317 | 602 | 882 | 976.0 | DXK:1001 | Type1 | Inactive | DFGin | 5.3484 | 15.0683 | ABAminus | -133.93, -15.74 | -121.25, 119.84 | -118.06, 28.52 | 301.16, 87.41 | -78.43, -76.5 | in-in | in | 8.2525 | Saltbr-in | 2.3405 | HRD-in | -74.5, -47.84 | 76.45, -12.42 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.8125 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 153.72 | APE9-dihe-in | -66.55, 140.49 | APE8-dihe-in | -67.49, 153.9 | APE8-rot-na | 28.58 | APE67-dihe-in | -75.86, -2.19 | -123.09, -16.67 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 12.2475 | APE9-dist-out | 8.9534 | None | None | None | XRAY | 1.379 | 0.206 | 0.221 | B | 306.0 | 271.0 | 10 | 31 | 24 | 7 | [[613, 873]] | 1.0 | 6fnh | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 6FNHC | P29317 | 600 | 890 | 976.0 | DXK:1001 | Type1 | None | DFGin | 6.0999 | 15.0776 | BLAminus | -136.98, -166.98 | 54.47, 77.28 | -106.75, 37.52 | 303.15, 87.48 | -109.85, 171.74 | in-in | in | 8.5229 | Saltbr-in | 2.9729 | HRD-in | -71.56, -48.37 | 75.35, -10.7 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 34.12 | APE8-rot-na | 34.55 | APE67-dihe-in | -53.44, -22.38 | -49.0, -43.37 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.379 | 0.206 | 0.221 | C | 306.0 | 270.0 | 21 | 31 | 12 | 19 | [[613, 873]] | 1.0 | 6fnh | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EPHA2 | EPHA2_HUMAN | 6FNHA | P29317 | 602 | 889 | 976.0 | DXK:1001 | Type1 | Inactive | DFGin | 6.0291 | 15.2866 | ABAminus | -132.89, -13.6 | -114.29, 112.91 | -120.16, 34.85 | 297.73, 92.28 | -68.77, 147.18 | in-in | in | 8.5707 | Saltbr-in | 2.5241 | HRD-in | -71.64, -49.56 | 77.94, -13.05 | in-out-in | SNCioi | out-in | ActLoopNT-out | 10.9018 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -86.64, 136.2 | APE9-dihe-in | -91.95, 112.57 | APE8-dihe-in | -77.45, 142.7 | APE8-rot-na | 28.74 | APE67-dihe-in | -60.57, -18.72 | -57.08, -38.55 | APE12-dist-na | 999.0 | APE11-dist-na | 8.3826 | APE10-dist-na | 12.3766 | APE9-dist-in | 5.4468 | None | None | None | XRAY | 1.379 | 0.206 | 0.221 | A | 306.0 | 277.0 | 11 | 31 | 21 | 10 | [[613, 873]] | 1.0 | 6fnh | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 6FNHB | P29317 | 602 | 882 | 976.0 | DXK:1001 | Type1 | Inactive | DFGin | 5.3484 | 15.0683 | ABAminus | -133.93, -15.74 | -121.25, 119.84 | -118.06, 28.52 | 301.16, 87.41 | -78.43, -76.5 | in-in | in | 8.2525 | Saltbr-in | 2.3405 | HRD-in | -74.5, -47.84 | 76.45, -12.42 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.8125 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 153.72 | APE9-dihe-in | -66.55, 140.49 | APE8-dihe-in | -67.49, 153.9 | APE8-rot-na | 28.58 | APE67-dihe-in | -75.86, -2.19 | -123.09, -16.67 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 12.2475 | APE9-dist-out | 8.9534 | None | None | None | XRAY | 1.379 | 0.206 | 0.221 | B | 306.0 | 271.0 | 10 | 31 | 24 | 7 | [[613, 873]] | 1.0 | 6fnh | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 6FNHC | P29317 | 600 | 890 | 976.0 | DXK:1001 | Type1 | None | DFGin | 6.0999 | 15.0776 | BLAminus | -136.98, -166.98 | 54.47, 77.28 | -106.75, 37.52 | 303.15, 87.48 | -109.85, 171.74 | in-in | in | 8.5229 | Saltbr-in | 2.9729 | HRD-in | -71.56, -48.37 | 75.35, -10.7 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, 34.12 | APE8-rot-na | 34.55 | APE67-dihe-in | -53.44, -22.38 | -49.0, -43.37 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.379 | 0.206 | 0.221 | C | 306.0 | 270.0 | 21 | 31 | 12 | 19 | [[613, 873]] | 1.0 | 6fnh | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 5.5e-108 | 366.1 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|