| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | SRPK1 | SRPK1_HUMAN | 6FADA | Q96SB4 | 55 | 655 | 655.0 | No_ligand | No_ligand | Inactive | DFGin | 6.2199 | 15.1362 | BLAminus | -122.93, 179.12 | 57.38, 61.42 | -78.03, 19.0 | 277.69, 78.02 | -68.08, -18.77 | in-out | in | 9.9288 | Saltbr-out | 5.6991 | HRD-in | -65.55, -50.38 | 76.6, 9.52 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.0457 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -121.2, 171.46 | APE9-dihe-na | 71.78, 143.02 | APE8-dihe-in | -86.05, 154.67 | APE8-rot-out | 81.2 | APE67-dihe-in | -62.54, -19.42 | -41.68, -58.38 | APE12-dist-in | 12.82 | APE11-dist-in | 10.9878 | APE10-dist-in | 7.6723 | APE9-dist-in | 3.1383 | None | None | None | XRAY | 2.801 | 0.201 | 0.257 | A | 618.0 | 356.0 | 245 | 25 | 25 | 0 | [[80, 653]] | 1.0 | 6fad | CMGC_SRPK1_HUMAN | CMGC | 1.7e-138 | 466.8 | 1.0 | 301.0 | 301.0 | 496 | 497 | 498 | 500 | 502 | 109 | 124 | 128 | 210 | 212 | 211 | 213.0 | 533 | 521 | 516 | 515 | 514 | 513 | 512 | 511 | 510 | 166 | SRSF protein kinase 1 |
| CMGC | SRPK1 | SRPK1_HUMAN | 6FADB | Q96SB4 | 55 | 655 | 655.0 | No_ligand | No_ligand | Inactive | DFGin | 6.2322 | 14.9856 | BLAminus | -113.6, 174.2 | 60.21, 87.3 | -102.47, 28.18 | 286.78, 61.47 | -69.13, -15.83 | in-out | in | 9.7481 | Saltbr-out | 4.624 | HRD-in | -75.61, -45.96 | 73.19, 8.23 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8797 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -125.25, 164.85 | APE9-dihe-na | 73.22, 157.16 | APE8-dihe-in | -99.01, 141.77 | APE8-rot-out | 60.06 | APE67-dihe-in | -66.35, -13.73 | -20.25, -68.69 | APE12-dist-in | 12.6174 | APE11-dist-in | 10.9073 | APE10-dist-in | 7.7495 | APE9-dist-in | 3.1803 | None | None | None | XRAY | 2.801 | 0.201 | 0.257 | B | 618.0 | 356.0 | 245 | 25 | 25 | 0 | [[80, 653]] | 1.0 | 6fad | CMGC_SRPK1_HUMAN | CMGC | 1.7e-138 | 466.8 | 1.0 | 301.0 | 301.0 | 496 | 497 | 498 | 500 | 502 | 109 | 124 | 128 | 210 | 212 | 211 | 213.0 | 533 | 521 | 516 | 515 | 514 | 513 | 512 | 511 | 510 | 166 | SRSF protein kinase 1 |
| CMGC | SRPK1 | SRPK1_HUMAN | 6FADC | Q96SB4 | 55 | 655 | 655.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5172 | 15.2946 | BLAminus | -123.52, -178.15 | 55.08, 85.74 | -104.19, 20.56 | 276.3, 81.28 | -67.88, -18.36 | in-out | in | 9.9668 | Saltbr-out | 5.5582 | HRD-in | -74.58, -44.68 | 71.07, 8.29 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7854 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.77, 164.16 | APE9-dihe-na | 77.72, 151.02 | APE8-dihe-in | -86.55, 133.38 | APE8-rot-in | 273.9 | APE67-dihe-in | -62.07, -14.6 | -22.9, -73.33 | APE12-dist-in | 12.6911 | APE11-dist-in | 10.7186 | APE10-dist-in | 7.6395 | APE9-dist-in | 3.2358 | None | None | None | XRAY | 2.801 | 0.201 | 0.257 | C | 618.0 | 359.0 | 242 | 25 | 25 | 0 | [[80, 653]] | 1.0 | 6fad | CMGC_SRPK1_HUMAN | CMGC | 1.7e-138 | 466.8 | 1.0 | 301.0 | 301.0 | 496 | 497 | 498 | 500 | 502 | 109 | 124 | 128 | 210 | 212 | 211 | 213.0 | 533 | 521 | 516 | 515 | 514 | 513 | 512 | 511 | 510 | 166 | SRSF protein kinase 1 |
| CMGC | SRPK1 | SRPK1_HUMAN | 6FADD | Q96SB4 | 55 | 655 | 655.0 | No_ligand | No_ligand | Inactive | DFGin | 6.3771 | 15.3304 | BLAminus | -119.7, -178.47 | 48.47, 81.81 | -91.0, 13.61 | 274.63, 34.06 | -64.49, -20.18 | out-out | out | 10.1938 | Saltbr-out | 5.1793 | HRD-in | -73.88, -47.0 | 76.16, 9.55 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.856 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.69, 159.48 | APE9-dihe-na | 80.31, 146.18 | APE8-dihe-in | -75.32, 143.12 | APE8-rot-in | 297.81 | APE67-dihe-in | -63.2, -18.62 | -40.87, -60.1 | APE12-dist-in | 12.7857 | APE11-dist-in | 10.6244 | APE10-dist-in | 7.7559 | APE9-dist-in | 3.1639 | None | None | None | XRAY | 2.801 | 0.201 | 0.257 | D | 618.0 | 356.0 | 245 | 25 | 25 | 0 | [[80, 653]] | 1.0 | 6fad | CMGC_SRPK1_HUMAN | CMGC | 1.7e-138 | 466.8 | 1.0 | 301.0 | 301.0 | 496 | 497 | 498 | 500 | 502 | 109 | 124 | 128 | 210 | 212 | 211 | 213.0 | 533 | 521 | 516 | 515 | 514 | 513 | 512 | 511 | 510 | 166 | SRSF protein kinase 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | SRPK1 | SRPK1_HUMAN | 6FADA | Q96SB4 | 55 | 655 | 655.0 | No_ligand | No_ligand | Inactive | DFGin | 6.2199 | 15.1362 | BLAminus | -122.93, 179.12 | 57.38, 61.42 | -78.03, 19.0 | 277.69, 78.02 | -68.08, -18.77 | in-out | in | 9.9288 | Saltbr-out | 5.6991 | HRD-in | -65.55, -50.38 | 76.6, 9.52 | out-in-out | SNCoio | in-out | ActLoopNT-in | 3.0457 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -121.2, 171.46 | APE9-dihe-na | 71.78, 143.02 | APE8-dihe-in | -86.05, 154.67 | APE8-rot-out | 81.2 | APE67-dihe-in | -62.54, -19.42 | -41.68, -58.38 | APE12-dist-in | 12.82 | APE11-dist-in | 10.9878 | APE10-dist-in | 7.6723 | APE9-dist-in | 3.1383 | None | None | None | XRAY | 2.801 | 0.201 | 0.257 | A | 618.0 | 356.0 | 245 | 25 | 25 | 0 | [[80, 653]] | 1.0 | 6fad | Homo sapiens | CMGC_SRPK1_HUMAN | CMGC | 1.7e-138 | 466.8 | 1.0 | 301.0 | 301.0 | 496 | 497 | 498 | 500 | 502 | 109 | 124 | 128 | 210 | 212 | 211 | 213.0 | 533 | 521 | 516 | 515 | 514 | 513 | 512 | 511 | 510 | 166 | SRSF protein kinase 1 |
| CMGC | SRPK1 | SRPK1_HUMAN | 6FADB | Q96SB4 | 55 | 655 | 655.0 | No_ligand | No_ligand | Inactive | DFGin | 6.2322 | 14.9856 | BLAminus | -113.6, 174.2 | 60.21, 87.3 | -102.47, 28.18 | 286.78, 61.47 | -69.13, -15.83 | in-out | in | 9.7481 | Saltbr-out | 4.624 | HRD-in | -75.61, -45.96 | 73.19, 8.23 | out-in-out | SNCoio | in-out | ActLoopNT-in | 2.8797 | ActLoopCT-out | nonTYR | APEdihe_aaioi | APEdist_iiii | APE10-dihe-na | -125.25, 164.85 | APE9-dihe-na | 73.22, 157.16 | APE8-dihe-in | -99.01, 141.77 | APE8-rot-out | 60.06 | APE67-dihe-in | -66.35, -13.73 | -20.25, -68.69 | APE12-dist-in | 12.6174 | APE11-dist-in | 10.9073 | APE10-dist-in | 7.7495 | APE9-dist-in | 3.1803 | None | None | None | XRAY | 2.801 | 0.201 | 0.257 | B | 618.0 | 356.0 | 245 | 25 | 25 | 0 | [[80, 653]] | 1.0 | 6fad | Homo sapiens | CMGC_SRPK1_HUMAN | CMGC | 1.7e-138 | 466.8 | 1.0 | 301.0 | 301.0 | 496 | 497 | 498 | 500 | 502 | 109 | 124 | 128 | 210 | 212 | 211 | 213.0 | 533 | 521 | 516 | 515 | 514 | 513 | 512 | 511 | 510 | 166 | SRSF protein kinase 1 |
| CMGC | SRPK1 | SRPK1_HUMAN | 6FADC | Q96SB4 | 55 | 655 | 655.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5172 | 15.2946 | BLAminus | -123.52, -178.15 | 55.08, 85.74 | -104.19, 20.56 | 276.3, 81.28 | -67.88, -18.36 | in-out | in | 9.9668 | Saltbr-out | 5.5582 | HRD-in | -74.58, -44.68 | 71.07, 8.29 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.7854 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.77, 164.16 | APE9-dihe-na | 77.72, 151.02 | APE8-dihe-in | -86.55, 133.38 | APE8-rot-in | 273.9 | APE67-dihe-in | -62.07, -14.6 | -22.9, -73.33 | APE12-dist-in | 12.6911 | APE11-dist-in | 10.7186 | APE10-dist-in | 7.6395 | APE9-dist-in | 3.2358 | None | None | None | XRAY | 2.801 | 0.201 | 0.257 | C | 618.0 | 359.0 | 242 | 25 | 25 | 0 | [[80, 653]] | 1.0 | 6fad | Homo sapiens | CMGC_SRPK1_HUMAN | CMGC | 1.7e-138 | 466.8 | 1.0 | 301.0 | 301.0 | 496 | 497 | 498 | 500 | 502 | 109 | 124 | 128 | 210 | 212 | 211 | 213.0 | 533 | 521 | 516 | 515 | 514 | 513 | 512 | 511 | 510 | 166 | SRSF protein kinase 1 |
| CMGC | SRPK1 | SRPK1_HUMAN | 6FADD | Q96SB4 | 55 | 655 | 655.0 | No_ligand | No_ligand | Inactive | DFGin | 6.3771 | 15.3304 | BLAminus | -119.7, -178.47 | 48.47, 81.81 | -91.0, 13.61 | 274.63, 34.06 | -64.49, -20.18 | out-out | out | 10.1938 | Saltbr-out | 5.1793 | HRD-in | -73.88, -47.0 | 76.16, 9.55 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.856 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -123.69, 159.48 | APE9-dihe-na | 80.31, 146.18 | APE8-dihe-in | -75.32, 143.12 | APE8-rot-in | 297.81 | APE67-dihe-in | -63.2, -18.62 | -40.87, -60.1 | APE12-dist-in | 12.7857 | APE11-dist-in | 10.6244 | APE10-dist-in | 7.7559 | APE9-dist-in | 3.1639 | None | None | None | XRAY | 2.801 | 0.201 | 0.257 | D | 618.0 | 356.0 | 245 | 25 | 25 | 0 | [[80, 653]] | 1.0 | 6fad | Homo sapiens | CMGC_SRPK1_HUMAN | CMGC | 1.7e-138 | 466.8 | 1.0 | 301.0 | 301.0 | 496 | 497 | 498 | 500 | 502 | 109 | 124 | 128 | 210 | 212 | 211 | 213.0 | 533 | 521 | 516 | 515 | 514 | 513 | 512 | 511 | 510 | 166 | SRSF protein kinase 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|