| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK10 | MK10_HUMAN | 6EMHC | P53779 | 46 | 400 | 464.0 | BGE:503 | Type1 | Inactive | DFGin | 4.0106 | 14.0393 | ABAminus | -78.44, -28.09 | -141.81, 177.01 | -104.97, 12.36 | 301.49, 97.27 | 78.59, -161.37 | in-in | in | 8.9467 | Saltbr-in | 3.0403 | HRD-in | -74.95, -52.97 | 66.65, 0.5 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.8694 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 130.1 | APE8-dihe-in | -107.4, 124.09 | APE8-rot-in | 288.83 | APE67-dihe-in | -65.02, -21.01 | -106.3, -7.59 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.2912 | None | None | None | XRAY | 1.76 | 999.0 | 999.0 | C | 367.0 | 334.0 | 15 | 27 | 17 | 10 | [[64, 359]] | 1.0 | 6emh | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.0 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 6EMHD | P53779 | 46 | 400 | 464.0 | BGE:503 | Type1 | Inactive | DFGin | 3.9558 | 14.4087 | ABAminus | -86.47, -17.97 | -146.7, 169.61 | -110.56, 12.64 | 296.15, 94.28 | 76.93, -162.97 | in-in | in | 9.2647 | Saltbr-in | 3.3454 | HRD-in | -69.69, -55.56 | 66.61, 3.24 | in-out-none | SNCion | out-none | ActLoopNT-out | 6.3331 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 113.89 | APE8-rot-in | 293.93 | APE67-dihe-in | -67.17, -21.93 | -103.77, -5.89 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.76 | 999.0 | 999.0 | D | 367.0 | 331.0 | 16 | 27 | 16 | 11 | [[64, 359]] | 1.0 | 6emh | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.0 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 6EMHA | P53779 | 46 | 400 | 464.0 | BGE:504,C15:506 | Type1,Allosteric | Inactive | DFGin | 3.9296 | 14.0838 | ABAminus | -88.94, -22.23 | -144.23, 173.35 | -118.59, 4.36 | 304.38, 93.6 | 70.22, -170.04 | in-in | in | 9.2242 | Saltbr-in | 2.9456 | HRD-in | -75.21, -57.6 | 72.31, -9.22 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.35 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -72.6 | APE8-dihe-in | -99.06, 111.23 | APE8-rot-in | 304.28 | APE67-dihe-in | -64.51, -16.6 | -105.92, -9.46 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.8429 | None | None | None | XRAY | 1.76 | 999.0 | 999.0 | A | 367.0 | 344.0 | 11 | 27 | 22 | 5 | [[64, 359]] | 1.0 | 6emh | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.0 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 6EMHB | P53779 | 46 | 400 | 464.0 | BGE:502,C15:504 | Type1,Allosteric | Inactive | DFGin | 3.9838 | 13.9753 | ABAminus | -90.53, -23.08 | -143.55, 174.7 | -119.54, -1.04 | 302.02, 90.55 | 71.56, -172.09 | in-in | in | 9.088 | Saltbr-in | 3.1394 | HRD-in | -71.43, -57.72 | 66.61, -12.51 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.4686 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 150.41 | APE8-dihe-in | -92.15, 115.96 | APE8-rot-in | 304.13 | APE67-dihe-in | -65.86, -16.66 | -109.13, -2.57 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.9796 | None | None | None | XRAY | 1.76 | 999.0 | 999.0 | B | 367.0 | 344.0 | 11 | 27 | 22 | 5 | [[64, 359]] | 1.0 | 6emh | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.0 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | MAPK10 | MK10_HUMAN | 6EMHC | P53779 | 46 | 400 | 464.0 | BGE:503 | Type1 | Inactive | DFGin | 4.0106 | 14.0393 | ABAminus | -78.44, -28.09 | -141.81, 177.01 | -104.97, 12.36 | 301.49, 97.27 | 78.59, -161.37 | in-in | in | 8.9467 | Saltbr-in | 3.0403 | HRD-in | -74.95, -52.97 | 66.65, 0.5 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.8694 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 130.1 | APE8-dihe-in | -107.4, 124.09 | APE8-rot-in | 288.83 | APE67-dihe-in | -65.02, -21.01 | -106.3, -7.59 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.2912 | None | None | None | XRAY | 1.76 | 999.0 | 999.0 | C | 367.0 | 334.0 | 15 | 27 | 17 | 10 | [[64, 359]] | 1.0 | 6emh | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.0 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 6EMHD | P53779 | 46 | 400 | 464.0 | BGE:503 | Type1 | Inactive | DFGin | 3.9558 | 14.4087 | ABAminus | -86.47, -17.97 | -146.7, 169.61 | -110.56, 12.64 | 296.15, 94.28 | 76.93, -162.97 | in-in | in | 9.2647 | Saltbr-in | 3.3454 | HRD-in | -69.69, -55.56 | 66.61, 3.24 | in-out-none | SNCion | out-none | ActLoopNT-out | 6.3331 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 113.89 | APE8-rot-in | 293.93 | APE67-dihe-in | -67.17, -21.93 | -103.77, -5.89 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.76 | 999.0 | 999.0 | D | 367.0 | 331.0 | 16 | 27 | 16 | 11 | [[64, 359]] | 1.0 | 6emh | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.0 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 6EMHA | P53779 | 46 | 400 | 464.0 | BGE:504,C15:506 | Type1,Allosteric | Inactive | DFGin | 3.9296 | 14.0838 | ABAminus | -88.94, -22.23 | -144.23, 173.35 | -118.59, 4.36 | 304.38, 93.6 | 70.22, -170.04 | in-in | in | 9.2242 | Saltbr-in | 2.9456 | HRD-in | -75.21, -57.6 | 72.31, -9.22 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.35 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, -72.6 | APE8-dihe-in | -99.06, 111.23 | APE8-rot-in | 304.28 | APE67-dihe-in | -64.51, -16.6 | -105.92, -9.46 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.8429 | None | None | None | XRAY | 1.76 | 999.0 | 999.0 | A | 367.0 | 344.0 | 11 | 27 | 22 | 5 | [[64, 359]] | 1.0 | 6emh | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.0 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| CMGC | MAPK10 | MK10_HUMAN | 6EMHB | P53779 | 46 | 400 | 464.0 | BGE:502,C15:504 | Type1,Allosteric | Inactive | DFGin | 3.9838 | 13.9753 | ABAminus | -90.53, -23.08 | -143.55, 174.7 | -119.54, -1.04 | 302.02, 90.55 | 71.56, -172.09 | in-in | in | 9.088 | Saltbr-in | 3.1394 | HRD-in | -71.43, -57.72 | 66.61, -12.51 | in-out-out | SNCioo | out-out | ActLoopNT-out | 6.4686 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_nnno | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 150.41 | APE8-dihe-in | -92.15, 115.96 | APE8-rot-in | 304.13 | APE67-dihe-in | -65.86, -16.66 | -109.13, -2.57 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-out | 11.9796 | None | None | None | XRAY | 1.76 | 999.0 | 999.0 | B | 367.0 | 344.0 | 11 | 27 | 22 | 5 | [[64, 359]] | 1.0 | 6emh | Homo sapiens | CMGC_MAPK10_HUMAN | CMGC | 1.4e-85 | 293.0 | 1.0 | 301.0 | 301.0 | 206 | 207 | 208 | 210 | 212 | 93 | 111 | 115 | 186 | 188 | 187 | 189.0 | 245 | 233 | 228 | 227 | 226 | 225 | 224 | 223 | 222 | 147 | Mitogen-activated protein kinase 10 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|