| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 5UI0B | P21802 | 462 | 765 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.5418 | 14.2132 | BLAminus | -136.98, -171.82 | 50.02, 76.91 | -91.39, 21.0 | 284.06, 84.3 | -70.34, -15.26 | in-in | in | 7.2433 | Saltbr-in | 2.9593 | HRD-in | -80.63, -49.98 | 74.74, -10.37 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9367 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -115.5, 32.27 | APE9-dihe-in | -102.72, 128.27 | APE8-dihe-in | -51.42, 123.86 | APE8-rot-na | 328.96 | APE67-dihe-in | -69.39, -7.95 | -60.08, -38.03 | APE12-dist-na | 14.7842 | APE11-dist-na | 10.1664 | APE10-dist-na | 7.6055 | APE9-dist-in | 4.8551 | C491A,E565A | None | None | XRAY | 2.05 | 0.183 | 0.207 | B | 324.0 | 304.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 5ui0 | TYR_FGFR2_HUMAN | TYR | 2.9e-103 | 350.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 5UI0A | P21802 | 461 | 766 | 821.0 | No_ligand | No_ligand | Inactive | DFGin | 6.7052 | 14.3598 | BLAminus | -135.62, -171.25 | 53.76, 73.69 | -92.94, 20.04 | 285.17, 82.93 | -70.08, -15.73 | in-in | in | 7.2705 | Saltbr-in | 2.8657 | HRD-in | -79.02, -49.38 | 75.99, -10.91 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9351 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -111.85, 29.9 | APE9-dihe-in | -103.97, 128.06 | APE8-dihe-in | -51.81, 123.04 | APE8-rot-na | 328.88 | APE67-dihe-in | -69.55, -8.5 | -59.7, -37.83 | APE12-dist-na | 14.8934 | APE11-dist-na | 10.2909 | APE10-dist-na | 7.5436 | APE9-dist-in | 4.9492 | C491A,E565A | None | None | XRAY | 2.05 | 0.183 | 0.207 | A | 324.0 | 301.0 | 5 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 5ui0 | TYR_FGFR2_HUMAN | TYR | 2.9e-103 | 350.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 5UI0B | P21802 | 462 | 765 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.5418 | 14.2132 | BLAminus | -136.98, -171.82 | 50.02, 76.91 | -91.39, 21.0 | 284.06, 84.3 | -70.34, -15.26 | in-in | in | 7.2433 | Saltbr-in | 2.9593 | HRD-in | -80.63, -49.98 | 74.74, -10.37 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9367 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -115.5, 32.27 | APE9-dihe-in | -102.72, 128.27 | APE8-dihe-in | -51.42, 123.86 | APE8-rot-na | 328.96 | APE67-dihe-in | -69.39, -7.95 | -60.08, -38.03 | APE12-dist-na | 14.7842 | APE11-dist-na | 10.1664 | APE10-dist-na | 7.6055 | APE9-dist-in | 4.8551 | C491A,E565A | None | None | XRAY | 2.05 | 0.183 | 0.207 | B | 324.0 | 304.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 5ui0 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.9e-103 | 350.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 5UI0A | P21802 | 461 | 766 | 821.0 | No_ligand | No_ligand | Inactive | DFGin | 6.7052 | 14.3598 | BLAminus | -135.62, -171.25 | 53.76, 73.69 | -92.94, 20.04 | 285.17, 82.93 | -70.08, -15.73 | in-in | in | 7.2705 | Saltbr-in | 2.8657 | HRD-in | -79.02, -49.38 | 75.99, -10.91 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9351 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -111.85, 29.9 | APE9-dihe-in | -103.97, 128.06 | APE8-dihe-in | -51.81, 123.04 | APE8-rot-na | 328.88 | APE67-dihe-in | -69.55, -8.5 | -59.7, -37.83 | APE12-dist-na | 14.8934 | APE11-dist-na | 10.2909 | APE10-dist-na | 7.5436 | APE9-dist-in | 4.9492 | C491A,E565A | None | None | XRAY | 2.05 | 0.183 | 0.207 | A | 324.0 | 301.0 | 5 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 5ui0 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.9e-103 | 350.6 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|