| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 5UHNA | P21802 | 469 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.5167 | 14.0937 | BLAminus | -136.8, -167.33 | 56.16, 78.56 | -101.45, 21.6 | 294.96, 102.9 | -64.06, -30.14 | in-in | in | 7.8238 | Saltbr-in | 2.5229 | HRD-in | -81.24, -42.19 | 65.24, 0.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9627 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -130.72, 22.85 | APE9-dihe-in | -103.03, 139.99 | APE8-dihe-in | -59.98, 123.73 | APE8-rot-na | 335.04 | APE67-dihe-in | -66.52, -14.98 | -63.65, -42.1 | APE12-dist-na | 14.8547 | APE11-dist-na | 10.9032 | APE10-dist-na | 7.5865 | APE9-dist-in | 4.8843 | N549H,E565A | None | None | XRAY | 2.909 | 0.26 | 0.311 | A | 324.0 | 282.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 5uhn | TYR_FGFR2_HUMAN | TYR | 3.3e-103 | 350.5 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 5UHNB | P21802 | 469 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.5134 | 14.0231 | BLAminus | -136.33, -166.28 | 57.28, 77.94 | -101.83, 20.57 | 295.09, 103.12 | -64.81, -29.84 | in-in | in | 7.6634 | Saltbr-in | 2.4643 | HRD-in | -80.51, -42.21 | 65.56, -0.07 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.1826 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -129.68, 22.67 | APE9-dihe-in | -103.05, 139.67 | APE8-dihe-in | -60.5, 125.01 | APE8-rot-na | 334.93 | APE67-dihe-in | -66.52, -14.36 | -63.18, -41.76 | APE12-dist-na | 999.0 | APE11-dist-na | 10.8143 | APE10-dist-na | 7.5915 | APE9-dist-in | 4.8168 | N549H,E565A | None | None | XRAY | 2.909 | 0.26 | 0.311 | B | 324.0 | 269.0 | 27 | 30 | 19 | 11 | [[481, 759]] | 1.0 | 5uhn | TYR_FGFR2_HUMAN | TYR | 3.3e-103 | 350.5 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 5UHNA | P21802 | 469 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.5167 | 14.0937 | BLAminus | -136.8, -167.33 | 56.16, 78.56 | -101.45, 21.6 | 294.96, 102.9 | -64.06, -30.14 | in-in | in | 7.8238 | Saltbr-in | 2.5229 | HRD-in | -81.24, -42.19 | 65.24, 0.64 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9627 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -130.72, 22.85 | APE9-dihe-in | -103.03, 139.99 | APE8-dihe-in | -59.98, 123.73 | APE8-rot-na | 335.04 | APE67-dihe-in | -66.52, -14.98 | -63.65, -42.1 | APE12-dist-na | 14.8547 | APE11-dist-na | 10.9032 | APE10-dist-na | 7.5865 | APE9-dist-in | 4.8843 | N549H,E565A | None | None | XRAY | 2.909 | 0.26 | 0.311 | A | 324.0 | 282.0 | 14 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 5uhn | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 3.3e-103 | 350.5 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 5UHNB | P21802 | 469 | 764 | 821.0 | ACP:802 | ATPlike | Inactive | DFGin | 6.5134 | 14.0231 | BLAminus | -136.33, -166.28 | 57.28, 77.94 | -101.83, 20.57 | 295.09, 103.12 | -64.81, -29.84 | in-in | in | 7.6634 | Saltbr-in | 2.4643 | HRD-in | -80.51, -42.21 | 65.56, -0.07 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.1826 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -129.68, 22.67 | APE9-dihe-in | -103.05, 139.67 | APE8-dihe-in | -60.5, 125.01 | APE8-rot-na | 334.93 | APE67-dihe-in | -66.52, -14.36 | -63.18, -41.76 | APE12-dist-na | 999.0 | APE11-dist-na | 10.8143 | APE10-dist-na | 7.5915 | APE9-dist-in | 4.8168 | N549H,E565A | None | None | XRAY | 2.909 | 0.26 | 0.311 | B | 324.0 | 269.0 | 27 | 30 | 19 | 11 | [[481, 759]] | 1.0 | 5uhn | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 3.3e-103 | 350.5 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|