| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | PDPK1 | PDPK1_HUMAN | 5LVPA | O15530 | 75 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.3028 | 14.9979 | BLAminus | -144.92, -168.82 | 66.06, 77.78 | -108.23, 11.17 | 281.99, 93.22 | -63.04, -32.41 | in-in | in | 9.539 | Saltbr-in | 3.1581 | HRD-in | -77.47, -51.83 | 79.92, -12.48 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8481 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.64, 166.02 | APE9-dihe-na | 141.61, 177.5 | APE8-dihe-in | -123.02, 134.29 | APE8-rot-in | 296.02 | APE67-dihe-in | -68.65, -16.53 | -46.89, -50.92 | APE12-dist-in | 7.9068 | APE11-dist-in | 10.6706 | APE10-dist-in | 5.166 | APE9-dist-in | 3.7049 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | A | 311.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| AGC | PDPK1 | PDPK1_HUMAN | 5LVPB | O15530 | 74 | 359 | 556.0 | ATP:401 | ATPlike | Active | DFGin | 6.3283 | 14.5498 | BLAminus | -137.23, -179.71 | 80.14, 74.16 | -105.47, 15.38 | 295.0, 84.83 | -59.91, -31.47 | in-in | in | 9.2741 | Saltbr-in | 3.3024 | HRD-in | -80.68, -44.41 | 73.96, -16.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7443 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.8, 152.43 | APE9-dihe-na | 134.43, -173.75 | APE8-dihe-in | -120.09, 128.28 | APE8-rot-in | 302.93 | APE67-dihe-in | -67.56, -25.72 | -44.99, -47.55 | APE12-dist-in | 7.8719 | APE11-dist-in | 11.0112 | APE10-dist-in | 5.3751 | APE9-dist-in | 3.7868 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | B | 311.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| AGC | PDPK1 | PDPK1_HUMAN | 5LVPC | O15530 | 75 | 359 | 556.0 | ATP:401 | ATPlike | Active | DFGin | 6.3906 | 14.6076 | BLAminus | -132.15, -176.81 | 71.98, 84.02 | -116.53, 7.62 | 291.47, 90.46 | -60.24, -24.5 | in-in | in | 9.3044 | Saltbr-in | 3.0866 | HRD-in | -75.92, -52.06 | 78.45, -5.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8228 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.81, 168.64 | APE9-dihe-na | 131.92, -176.79 | APE8-dihe-in | -126.79, 133.21 | APE8-rot-in | 299.13 | APE67-dihe-in | -67.64, -15.8 | -51.62, -50.49 | APE12-dist-in | 7.6523 | APE11-dist-in | 10.8632 | APE10-dist-in | 5.1235 | APE9-dist-in | 3.6447 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | C | 311.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| AGC | PDPK1 | PDPK1_HUMAN | 5LVPD | O15530 | 74 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.3336 | 14.4328 | BLAminus | -146.99, -174.22 | 74.22, 81.56 | -113.84, 4.02 | 287.97, 93.59 | -56.11, -25.73 | in-in | in | 9.3044 | Saltbr-in | 3.2517 | HRD-in | -82.38, -50.18 | 78.4, -12.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8357 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.65, 165.17 | APE9-dihe-na | 129.1, -166.82 | APE8-dihe-in | -132.84, 129.79 | APE8-rot-in | 300.06 | APE67-dihe-in | -65.46, -17.03 | -48.9, -48.47 | APE12-dist-in | 8.2282 | APE11-dist-in | 10.8909 | APE10-dist-in | 5.3485 | APE9-dist-in | 3.6459 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | D | 311.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | PDPK1 | PDPK1_HUMAN | 5LVPA | O15530 | 75 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.3028 | 14.9979 | BLAminus | -144.92, -168.82 | 66.06, 77.78 | -108.23, 11.17 | 281.99, 93.22 | -63.04, -32.41 | in-in | in | 9.539 | Saltbr-in | 3.1581 | HRD-in | -77.47, -51.83 | 79.92, -12.48 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8481 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -126.64, 166.02 | APE9-dihe-na | 141.61, 177.5 | APE8-dihe-in | -123.02, 134.29 | APE8-rot-in | 296.02 | APE67-dihe-in | -68.65, -16.53 | -46.89, -50.92 | APE12-dist-in | 7.9068 | APE11-dist-in | 10.6706 | APE10-dist-in | 5.166 | APE9-dist-in | 3.7049 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | A | 311.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| AGC | PDPK1 | PDPK1_HUMAN | 5LVPB | O15530 | 74 | 359 | 556.0 | ATP:401 | ATPlike | Active | DFGin | 6.3283 | 14.5498 | BLAminus | -137.23, -179.71 | 80.14, 74.16 | -105.47, 15.38 | 295.0, 84.83 | -59.91, -31.47 | in-in | in | 9.2741 | Saltbr-in | 3.3024 | HRD-in | -80.68, -44.41 | 73.96, -16.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7443 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.8, 152.43 | APE9-dihe-na | 134.43, -173.75 | APE8-dihe-in | -120.09, 128.28 | APE8-rot-in | 302.93 | APE67-dihe-in | -67.56, -25.72 | -44.99, -47.55 | APE12-dist-in | 7.8719 | APE11-dist-in | 11.0112 | APE10-dist-in | 5.3751 | APE9-dist-in | 3.7868 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | B | 311.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| AGC | PDPK1 | PDPK1_HUMAN | 5LVPC | O15530 | 75 | 359 | 556.0 | ATP:401 | ATPlike | Active | DFGin | 6.3906 | 14.6076 | BLAminus | -132.15, -176.81 | 71.98, 84.02 | -116.53, 7.62 | 291.47, 90.46 | -60.24, -24.5 | in-in | in | 9.3044 | Saltbr-in | 3.0866 | HRD-in | -75.92, -52.06 | 78.45, -5.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8228 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -113.81, 168.64 | APE9-dihe-na | 131.92, -176.79 | APE8-dihe-in | -126.79, 133.21 | APE8-rot-in | 299.13 | APE67-dihe-in | -67.64, -15.8 | -51.62, -50.49 | APE12-dist-in | 7.6523 | APE11-dist-in | 10.8632 | APE10-dist-in | 5.1235 | APE9-dist-in | 3.6447 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | C | 311.0 | 276.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| AGC | PDPK1 | PDPK1_HUMAN | 5LVPD | O15530 | 74 | 359 | 556.0 | ATP:500 | ATPlike | Active | DFGin | 6.3336 | 14.4328 | BLAminus | -146.99, -174.22 | 74.22, 81.56 | -113.84, 4.02 | 287.97, 93.59 | -56.11, -25.73 | in-in | in | 9.3044 | Saltbr-in | 3.2517 | HRD-in | -82.38, -50.18 | 78.4, -12.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8357 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.65, 165.17 | APE9-dihe-na | 129.1, -166.82 | APE8-dihe-in | -132.84, 129.79 | APE8-rot-in | 300.06 | APE67-dihe-in | -65.46, -17.03 | -48.9, -48.47 | APE12-dist-in | 8.2282 | APE11-dist-in | 10.8909 | APE10-dist-in | 5.3485 | APE9-dist-in | 3.6459 | Y288G,Q292A | SEP241 | SEP241 | XRAY | 2.5 | 0.176 | 0.226 | D | 311.0 | 277.0 | 9 | 30 | 21 | 9 | [[82, 342]] | 1.0 | 5lvp | Homo sapiens | AGC_PDPK1_HUMAN | AGC | 6.9e-84 | 286.9 | 1.0 | 260.0 | 260.0 | 222 | 223 | 224 | 226 | 228 | 111 | 130 | 134 | 202 | 204 | 203 | 205.0 | 264 | 252 | 247 | 246 | 245 | 244 | 243 | 242 | 241 | 160 | 3-phosphoinositide-dependent protein kinase 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|