| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | IGF1R | IGF1R_HUMAN | 5HZNA | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.5233 | 11.883 | None | -122.71, -134.04 | -48.48, 117.08 | -112.65, 5.39 | 56.52, 89.56 | -80.2, -12.63 | out-out | out | 10.1046 | Saltbr-out | 7.0696 | HRD-in | -68.72, -44.68 | 74.42, -15.27 | out-out-in | SNCooi | out-in | ActLoopNT-out | 9.0816 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.2, 129.26 | APE9-dihe-in | -125.1, 113.12 | APE8-dihe-in | -76.3, 72.6 | APE8-rot-na | 31.29 | APE67-dihe-in | -71.82, -14.27 | -59.77, -33.09 | APE12-dist-na | 12.7798 | APE11-dist-na | 9.3406 | APE10-dist-na | 6.0029 | APE9-dist-in | 7.4125 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | A | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNB | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.6676 | 11.6982 | None | -120.23, -145.7 | -34.99, 114.07 | -109.86, 7.02 | 53.42, 94.67 | -86.81, -17.85 | out-out | out | 10.2303 | Saltbr-out | 7.469 | HRD-in | -74.79, -42.86 | 77.21, -19.92 | out-out-in | SNCooi | out-in | ActLoopNT-out | 8.9724 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -71.8, 127.36 | APE9-dihe-in | -126.61, 120.91 | APE8-dihe-in | -82.51, 72.5 | APE8-rot-na | 31.18 | APE67-dihe-in | -70.34, -12.61 | -56.19, -36.04 | APE12-dist-na | 12.7105 | APE11-dist-na | 9.4364 | APE10-dist-na | 6.0092 | APE9-dist-in | 7.4127 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | B | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNC | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.5039 | 11.8927 | None | -117.5, -144.25 | -35.28, 118.67 | -116.54, 5.75 | 57.58, 87.45 | -83.77, -13.7 | out-out | out | 10.2048 | Saltbr-out | 6.5682 | HRD-in | -68.11, -52.05 | 81.72, -11.87 | out-out-in | SNCooi | out-in | ActLoopNT-out | 8.9794 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -79.64, 128.06 | APE9-dihe-in | -121.48, 117.98 | APE8-dihe-in | -78.81, 67.18 | APE8-rot-na | 28.39 | APE67-dihe-in | -73.45, -14.3 | -52.08, -33.81 | APE12-dist-na | 13.0318 | APE11-dist-na | 9.428 | APE10-dist-na | 6.062 | APE9-dist-in | 7.2753 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | C | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZND | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.5858 | 11.8119 | None | -120.23, -138.34 | -41.88, 115.18 | -111.54, 6.87 | 52.55, 90.98 | -80.5, -21.29 | out-out | out | 10.1558 | Saltbr-out | 7.0568 | HRD-in | -75.17, -45.42 | 77.74, -21.01 | out-out-in | SNCooi | out-in | ActLoopNT-out | 9.0982 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.35, 128.86 | APE9-dihe-in | -120.46, 118.5 | APE8-dihe-in | -79.97, 71.37 | APE8-rot-na | 32.37 | APE67-dihe-in | -73.39, -13.02 | -52.14, -35.35 | APE12-dist-na | 13.1787 | APE11-dist-na | 9.2529 | APE10-dist-na | 6.0206 | APE9-dist-in | 7.4528 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | D | 304.0 | 304.0 | 0 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNE | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.5339 | 11.8843 | None | -122.97, -133.9 | -50.03, 120.11 | -115.89, 7.06 | 56.85, 84.61 | -81.92, -13.97 | out-out | out | 10.0903 | Saltbr-out | 7.0006 | HRD-in | -71.62, -46.82 | 77.23, -15.08 | out-out-in | SNCooi | out-in | ActLoopNT-out | 9.0762 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.35, 128.61 | APE9-dihe-in | -123.88, 113.86 | APE8-dihe-in | -76.92, 69.0 | APE8-rot-na | 31.9 | APE67-dihe-in | -73.44, -14.93 | -54.7, -32.97 | APE12-dist-na | 12.7562 | APE11-dist-na | 9.3201 | APE10-dist-na | 6.0089 | APE9-dist-in | 7.4173 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | E | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNF | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.6688 | 11.6863 | None | -119.91, -143.87 | -36.57, 117.22 | -111.83, 7.84 | 53.92, 93.37 | -86.48, -19.66 | out-out | out | 10.2445 | Saltbr-out | 7.4948 | HRD-in | -71.54, -45.74 | 77.92, -19.28 | out-out-in | SNCooi | out-in | ActLoopNT-out | 8.9724 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.77, 125.58 | APE9-dihe-in | -123.67, 120.15 | APE8-dihe-in | -81.16, 71.31 | APE8-rot-na | 31.34 | APE67-dihe-in | -70.78, -14.02 | -54.99, -34.82 | APE12-dist-na | 12.6961 | APE11-dist-na | 9.4311 | APE10-dist-na | 6.0247 | APE9-dist-in | 7.4146 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | F | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNG | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.4952 | 11.8883 | None | -115.22, -143.92 | -37.17, 121.14 | -119.03, 5.44 | 57.57, 87.05 | -84.31, -13.87 | out-out | out | 10.2119 | Saltbr-out | 6.5677 | HRD-in | -69.56, -54.08 | 84.44, -12.44 | out-out-in | SNCooi | out-in | ActLoopNT-out | 8.9987 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -81.44, 128.11 | APE9-dihe-in | -122.01, 115.9 | APE8-dihe-in | -78.8, 69.19 | APE8-rot-na | 29.58 | APE67-dihe-in | -71.28, -16.87 | -55.78, -34.47 | APE12-dist-na | 13.0183 | APE11-dist-na | 9.4183 | APE10-dist-na | 6.0678 | APE9-dist-in | 7.3121 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | G | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNH | P08069 | 983 | 1285 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.5638 | 11.8399 | None | -117.51, -139.77 | -40.96, 115.52 | -113.35, 4.84 | 52.59, 91.03 | -79.05, -20.18 | out-out | out | 10.169 | Saltbr-out | 7.1318 | HRD-in | -75.23, -47.04 | 79.69, -19.55 | out-out-in | SNCooi | out-in | ActLoopNT-out | 9.1132 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.78, 128.57 | APE9-dihe-in | -119.04, 118.91 | APE8-dihe-in | -80.75, 73.24 | APE8-rot-na | 32.94 | APE67-dihe-in | -74.0, -12.28 | -56.22, -33.69 | APE12-dist-na | 13.1839 | APE11-dist-na | 9.2607 | APE10-dist-na | 6.0308 | APE9-dist-in | 7.4487 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | H | 304.0 | 303.0 | 0 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | IGF1R | IGF1R_HUMAN | 5HZNA | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.5233 | 11.883 | None | -122.71, -134.04 | -48.48, 117.08 | -112.65, 5.39 | 56.52, 89.56 | -80.2, -12.63 | out-out | out | 10.1046 | Saltbr-out | 7.0696 | HRD-in | -68.72, -44.68 | 74.42, -15.27 | out-out-in | SNCooi | out-in | ActLoopNT-out | 9.0816 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.2, 129.26 | APE9-dihe-in | -125.1, 113.12 | APE8-dihe-in | -76.3, 72.6 | APE8-rot-na | 31.29 | APE67-dihe-in | -71.82, -14.27 | -59.77, -33.09 | APE12-dist-na | 12.7798 | APE11-dist-na | 9.3406 | APE10-dist-na | 6.0029 | APE9-dist-in | 7.4125 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | A | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNB | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.6676 | 11.6982 | None | -120.23, -145.7 | -34.99, 114.07 | -109.86, 7.02 | 53.42, 94.67 | -86.81, -17.85 | out-out | out | 10.2303 | Saltbr-out | 7.469 | HRD-in | -74.79, -42.86 | 77.21, -19.92 | out-out-in | SNCooi | out-in | ActLoopNT-out | 8.9724 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -71.8, 127.36 | APE9-dihe-in | -126.61, 120.91 | APE8-dihe-in | -82.51, 72.5 | APE8-rot-na | 31.18 | APE67-dihe-in | -70.34, -12.61 | -56.19, -36.04 | APE12-dist-na | 12.7105 | APE11-dist-na | 9.4364 | APE10-dist-na | 6.0092 | APE9-dist-in | 7.4127 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | B | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNC | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.5039 | 11.8927 | None | -117.5, -144.25 | -35.28, 118.67 | -116.54, 5.75 | 57.58, 87.45 | -83.77, -13.7 | out-out | out | 10.2048 | Saltbr-out | 6.5682 | HRD-in | -68.11, -52.05 | 81.72, -11.87 | out-out-in | SNCooi | out-in | ActLoopNT-out | 8.9794 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -79.64, 128.06 | APE9-dihe-in | -121.48, 117.98 | APE8-dihe-in | -78.81, 67.18 | APE8-rot-na | 28.39 | APE67-dihe-in | -73.45, -14.3 | -52.08, -33.81 | APE12-dist-na | 13.0318 | APE11-dist-na | 9.428 | APE10-dist-na | 6.062 | APE9-dist-in | 7.2753 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | C | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZND | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.5858 | 11.8119 | None | -120.23, -138.34 | -41.88, 115.18 | -111.54, 6.87 | 52.55, 90.98 | -80.5, -21.29 | out-out | out | 10.1558 | Saltbr-out | 7.0568 | HRD-in | -75.17, -45.42 | 77.74, -21.01 | out-out-in | SNCooi | out-in | ActLoopNT-out | 9.0982 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.35, 128.86 | APE9-dihe-in | -120.46, 118.5 | APE8-dihe-in | -79.97, 71.37 | APE8-rot-na | 32.37 | APE67-dihe-in | -73.39, -13.02 | -52.14, -35.35 | APE12-dist-na | 13.1787 | APE11-dist-na | 9.2529 | APE10-dist-na | 6.0206 | APE9-dist-in | 7.4528 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | D | 304.0 | 304.0 | 0 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNE | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.5339 | 11.8843 | None | -122.97, -133.9 | -50.03, 120.11 | -115.89, 7.06 | 56.85, 84.61 | -81.92, -13.97 | out-out | out | 10.0903 | Saltbr-out | 7.0006 | HRD-in | -71.62, -46.82 | 77.23, -15.08 | out-out-in | SNCooi | out-in | ActLoopNT-out | 9.0762 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.35, 128.61 | APE9-dihe-in | -123.88, 113.86 | APE8-dihe-in | -76.92, 69.0 | APE8-rot-na | 31.9 | APE67-dihe-in | -73.44, -14.93 | -54.7, -32.97 | APE12-dist-na | 12.7562 | APE11-dist-na | 9.3201 | APE10-dist-na | 6.0089 | APE9-dist-in | 7.4173 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | E | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNF | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.6688 | 11.6863 | None | -119.91, -143.87 | -36.57, 117.22 | -111.83, 7.84 | 53.92, 93.37 | -86.48, -19.66 | out-out | out | 10.2445 | Saltbr-out | 7.4948 | HRD-in | -71.54, -45.74 | 77.92, -19.28 | out-out-in | SNCooi | out-in | ActLoopNT-out | 8.9724 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.77, 125.58 | APE9-dihe-in | -123.67, 120.15 | APE8-dihe-in | -81.16, 71.31 | APE8-rot-na | 31.34 | APE67-dihe-in | -70.78, -14.02 | -54.99, -34.82 | APE12-dist-na | 12.6961 | APE11-dist-na | 9.4311 | APE10-dist-na | 6.0247 | APE9-dist-in | 7.4146 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | F | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNG | P08069 | 983 | 1286 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.4952 | 11.8883 | None | -115.22, -143.92 | -37.17, 121.14 | -119.03, 5.44 | 57.57, 87.05 | -84.31, -13.87 | out-out | out | 10.2119 | Saltbr-out | 6.5677 | HRD-in | -69.56, -54.08 | 84.44, -12.44 | out-out-in | SNCooi | out-in | ActLoopNT-out | 8.9987 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -81.44, 128.11 | APE9-dihe-in | -122.01, 115.9 | APE8-dihe-in | -78.8, 69.19 | APE8-rot-na | 29.58 | APE67-dihe-in | -71.28, -16.87 | -55.78, -34.47 | APE12-dist-na | 13.0183 | APE11-dist-na | 9.4183 | APE10-dist-na | 6.0678 | APE9-dist-in | 7.3121 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | G | 304.0 | 296.0 | 8 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 5HZNH | P08069 | 983 | 1285 | 1367.0 | 66A:61301 | Type1.5_Front | Inactive | DFGin | 5.5638 | 11.8399 | None | -117.51, -139.77 | -40.96, 115.52 | -113.35, 4.84 | 52.59, 91.03 | -79.05, -20.18 | out-out | out | 10.169 | Saltbr-out | 7.1318 | HRD-in | -75.23, -47.04 | 79.69, -19.55 | out-out-in | SNCooi | out-in | ActLoopNT-out | 9.1132 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.78, 128.57 | APE9-dihe-in | -119.04, 118.91 | APE8-dihe-in | -80.75, 73.24 | APE8-rot-na | 32.94 | APE67-dihe-in | -74.0, -12.28 | -56.22, -33.69 | APE12-dist-na | 13.1839 | APE11-dist-na | 9.2607 | APE10-dist-na | 6.0308 | APE9-dist-in | 7.4487 | E1097A,E1099A | None | None | XRAY | 2.2 | 0.195 | 0.218 | H | 304.0 | 303.0 | 0 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 5hzn | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|