| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 5GTYA | P00533 | 700 | 1014 | 1210.0 | 816:1101 | Type1 | Inactive | DFGin | 3.9194 | 14.2537 | BLBplus | -136.6, 160.21 | 83.79, 10.32 | -71.62, 130.12 | 75.47, 69.3 | 84.21, -2.08 | out-out | out | 14.11 | Saltbr-out | 15.1582 | HRD-in | -64.26, -47.89 | 82.5, -11.45 | out-out-none | SNCoon | out-none | ActLoopNT-out | 7.1763 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 130.2 | APE9-dihe-in | -65.39, 157.4 | APE8-dihe-in | -83.63, 78.13 | APE8-rot-na | 34.93 | APE67-dihe-in | -61.71, -42.12 | -62.97, -39.37 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 15.4079 | APE9-dist-in | 7.8159 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | A | 331.0 | 300.0 | 15 | 30 | 19 | 11 | [[712, 970]] | 1.0 | 5gty | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYC | P00533 | 700 | 1013 | 1210.0 | 816:1101 | Type1 | Inactive | DFGin | 4.2836 | 15.8168 | BLBplus | -149.79, 169.46 | 71.39, 12.4 | -62.83, 164.89 | 105.62, 48.04 | 58.84, -127.22 | out-out | out | 13.7801 | Saltbr-out | 14.4025 | HRD-in | -63.98, -44.78 | 76.23, -10.44 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.8431 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -4.61 | APE8-rot-na | 27.64 | APE67-dihe-in | -61.37, -42.92 | -62.91, -38.64 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | C | 331.0 | 295.0 | 19 | 30 | 15 | 15 | [[712, 970]] | 1.0 | 5gty | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYF | P00533 | 700 | 1013 | 1210.0 | 816:1101 | Type1 | Inactive | DFGin | 4.5658 | 15.5911 | BLBplus | -143.69, 172.87 | 60.29, 35.9 | -98.19, 125.74 | 96.55, 67.96 | 83.35, -2.23 | out-none | out | 14.1687 | Saltbr-none | 999.0 | HRD-out | -91.66, 107.92 | -65.69, -38.43 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 6.1022 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -163.83 | APE8-dihe-in | -84.57, 72.91 | APE8-rot-na | 22.97 | APE67-dihe-in | -62.3, -42.82 | -63.85, -40.8 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.491 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | F | 331.0 | 297.0 | 17 | 30 | 17 | 13 | [[712, 970]] | 1.0 | 5gty | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYB | P00533 | 700 | 1014 | 1210.0 | 816:1101 | Type1.5_Back | Inactive | DFGin | 4.2902 | 14.3474 | BLBplus | -138.92, 165.68 | 84.63, 3.85 | -68.43, 135.48 | 78.45, 90.03 | 81.71, -3.27 | out-out | out | 13.4918 | Saltbr-out | 15.5988 | HRD-out | -95.29, 124.61 | -62.89, -41.97 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0604 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, -99.53 | APE9-dihe-in | -66.19, 150.26 | APE8-dihe-in | -83.76, 84.04 | APE8-rot-na | 28.01 | APE67-dihe-in | -63.91, -38.81 | -63.74, -37.31 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 14.1537 | APE9-dist-out | 9.3046 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | B | 331.0 | 299.0 | 16 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 5gty | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYD | P00533 | 701 | 1014 | 1210.0 | 816:1101 | Type1.5_Back | Inactive | DFGin | 3.7439 | 14.9019 | BLBplus | -133.78, 167.12 | 81.14, 4.97 | -64.51, 133.85 | 87.51, 89.95 | 82.67, -5.26 | out-out | out | 14.1252 | Saltbr-out | 12.581 | HRD-in | -64.22, -47.55 | 79.94, -12.61 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.1801 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 35.49 | APE9-dihe-in | -128.38, 151.23 | APE8-dihe-in | -84.12, 67.79 | APE8-rot-na | 27.63 | APE67-dihe-in | -63.81, -37.49 | -62.48, -38.56 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.1549 | APE9-dist-out | 8.3238 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | D | 331.0 | 297.0 | 17 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 5gty | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYE | P00533 | 701 | 1014 | 1210.0 | 816:1101 | Type1.5_Back | Inactive | DFGin | 4.0598 | 15.4006 | BLBplus | -130.28, 163.95 | 73.19, 13.87 | -64.73, 129.08 | 103.21, 59.68 | 78.99, -3.66 | out-none | out | 13.7411 | Saltbr-none | 999.0 | HRD-in | -63.53, -39.57 | 73.37, -57.08 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 5.6794 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, -16.57 | APE9-dihe-in | -63.24, 143.82 | APE8-dihe-in | -84.53, 69.95 | APE8-rot-na | 27.95 | APE67-dihe-in | -63.25, -38.96 | -61.88, -39.39 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 12.9009 | APE9-dist-out | 9.1105 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | E | 331.0 | 297.0 | 17 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 5gty | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYG | P00533 | 699 | 1014 | 1210.0 | 816:1101 | Type1.5_Back | Inactive | DFGin | 5.0674 | 14.6264 | BLBplus | -143.11, 179.85 | 58.12, 44.59 | -112.54, 128.63 | 59.94, 74.31 | 85.4, 3.0 | out-out | out | 14.3004 | Saltbr-out | 16.0055 | HRD-in | -64.4, -40.83 | 72.49, -56.78 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0551 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 152.17 | APE9-dihe-in | -112.88, 128.29 | APE8-dihe-in | -84.62, 80.89 | APE8-rot-na | 19.82 | APE67-dihe-in | -63.68, -40.43 | -63.75, -39.1 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.2616 | APE9-dist-out | 9.0522 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | G | 331.0 | 299.0 | 17 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 5gty | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYH | P00533 | 700 | 1016 | 1210.0 | 816:1101 | Type1.5_Back | Inactive | DFGin | 4.4636 | 14.9962 | BLBplus | -155.19, 174.62 | 58.89, 40.9 | -106.98, 132.32 | 74.94, 82.26 | 87.03, 0.91 | out-out | out | 14.0921 | Saltbr-out | 15.7915 | HRD-in | -64.35, -48.45 | 80.9, -10.31 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8343 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 6.3 | APE9-dihe-in | -114.67, 127.92 | APE8-dihe-in | -87.4, 86.48 | APE8-rot-na | 29.16 | APE67-dihe-in | -62.99, -38.55 | -63.72, -40.61 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 12.5252 | APE9-dist-out | 8.7343 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | H | 331.0 | 300.0 | 16 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 5gty | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 5GTYA | P00533 | 700 | 1014 | 1210.0 | 816:1101 | Type1 | Inactive | DFGin | 3.9194 | 14.2537 | BLBplus | -136.6, 160.21 | 83.79, 10.32 | -71.62, 130.12 | 75.47, 69.3 | 84.21, -2.08 | out-out | out | 14.11 | Saltbr-out | 15.1582 | HRD-in | -64.26, -47.89 | 82.5, -11.45 | out-out-none | SNCoon | out-none | ActLoopNT-out | 7.1763 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 130.2 | APE9-dihe-in | -65.39, 157.4 | APE8-dihe-in | -83.63, 78.13 | APE8-rot-na | 34.93 | APE67-dihe-in | -61.71, -42.12 | -62.97, -39.37 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 15.4079 | APE9-dist-in | 7.8159 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | A | 331.0 | 300.0 | 15 | 30 | 19 | 11 | [[712, 970]] | 1.0 | 5gty | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYC | P00533 | 700 | 1013 | 1210.0 | 816:1101 | Type1 | Inactive | DFGin | 4.2836 | 15.8168 | BLBplus | -149.79, 169.46 | 71.39, 12.4 | -62.83, 164.89 | 105.62, 48.04 | 58.84, -127.22 | out-out | out | 13.7801 | Saltbr-out | 14.4025 | HRD-in | -63.98, -44.78 | 76.23, -10.44 | out-out-none | SNCoon | out-none | ActLoopNT-out | 8.8431 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -4.61 | APE8-rot-na | 27.64 | APE67-dihe-in | -61.37, -42.92 | -62.91, -38.64 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | C | 331.0 | 295.0 | 19 | 30 | 15 | 15 | [[712, 970]] | 1.0 | 5gty | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYF | P00533 | 700 | 1013 | 1210.0 | 816:1101 | Type1 | Inactive | DFGin | 4.5658 | 15.5911 | BLBplus | -143.69, 172.87 | 60.29, 35.9 | -98.19, 125.74 | 96.55, 67.96 | 83.35, -2.23 | out-none | out | 14.1687 | Saltbr-none | 999.0 | HRD-out | -91.66, 107.92 | -65.69, -38.43 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 6.1022 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, -163.83 | APE8-dihe-in | -84.57, 72.91 | APE8-rot-na | 22.97 | APE67-dihe-in | -62.3, -42.82 | -63.85, -40.8 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 9.491 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | F | 331.0 | 297.0 | 17 | 30 | 17 | 13 | [[712, 970]] | 1.0 | 5gty | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYB | P00533 | 700 | 1014 | 1210.0 | 816:1101 | Type1.5_Back | Inactive | DFGin | 4.2902 | 14.3474 | BLBplus | -138.92, 165.68 | 84.63, 3.85 | -68.43, 135.48 | 78.45, 90.03 | 81.71, -3.27 | out-out | out | 13.4918 | Saltbr-out | 15.5988 | HRD-out | -95.29, 124.61 | -62.89, -41.97 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0604 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, -99.53 | APE9-dihe-in | -66.19, 150.26 | APE8-dihe-in | -83.76, 84.04 | APE8-rot-na | 28.01 | APE67-dihe-in | -63.91, -38.81 | -63.74, -37.31 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 14.1537 | APE9-dist-out | 9.3046 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | B | 331.0 | 299.0 | 16 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 5gty | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYD | P00533 | 701 | 1014 | 1210.0 | 816:1101 | Type1.5_Back | Inactive | DFGin | 3.7439 | 14.9019 | BLBplus | -133.78, 167.12 | 81.14, 4.97 | -64.51, 133.85 | 87.51, 89.95 | 82.67, -5.26 | out-out | out | 14.1252 | Saltbr-out | 12.581 | HRD-in | -64.22, -47.55 | 79.94, -12.61 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.1801 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 35.49 | APE9-dihe-in | -128.38, 151.23 | APE8-dihe-in | -84.12, 67.79 | APE8-rot-na | 27.63 | APE67-dihe-in | -63.81, -37.49 | -62.48, -38.56 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.1549 | APE9-dist-out | 8.3238 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | D | 331.0 | 297.0 | 17 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 5gty | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYE | P00533 | 701 | 1014 | 1210.0 | 816:1101 | Type1.5_Back | Inactive | DFGin | 4.0598 | 15.4006 | BLBplus | -130.28, 163.95 | 73.19, 13.87 | -64.73, 129.08 | 103.21, 59.68 | 78.99, -3.66 | out-none | out | 13.7411 | Saltbr-none | 999.0 | HRD-in | -63.53, -39.57 | 73.37, -57.08 | none-out-out | SNCnoo | out-out | ActLoopNT-out | 5.6794 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, -16.57 | APE9-dihe-in | -63.24, 143.82 | APE8-dihe-in | -84.53, 69.95 | APE8-rot-na | 27.95 | APE67-dihe-in | -63.25, -38.96 | -61.88, -39.39 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 12.9009 | APE9-dist-out | 9.1105 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | E | 331.0 | 297.0 | 17 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 5gty | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYG | P00533 | 699 | 1014 | 1210.0 | 816:1101 | Type1.5_Back | Inactive | DFGin | 5.0674 | 14.6264 | BLBplus | -143.11, 179.85 | 58.12, 44.59 | -112.54, 128.63 | 59.94, 74.31 | 85.4, 3.0 | out-out | out | 14.3004 | Saltbr-out | 16.0055 | HRD-in | -64.4, -40.83 | 72.49, -56.78 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.0551 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 152.17 | APE9-dihe-in | -112.88, 128.29 | APE8-dihe-in | -84.62, 80.89 | APE8-rot-na | 19.82 | APE67-dihe-in | -63.68, -40.43 | -63.75, -39.1 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.2616 | APE9-dist-out | 9.0522 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | G | 331.0 | 299.0 | 17 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 5gty | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 5GTYH | P00533 | 700 | 1016 | 1210.0 | 816:1101 | Type1.5_Back | Inactive | DFGin | 4.4636 | 14.9962 | BLBplus | -155.19, 174.62 | 58.89, 40.9 | -106.98, 132.32 | 74.94, 82.26 | 87.03, 0.91 | out-out | out | 14.0921 | Saltbr-out | 15.7915 | HRD-in | -64.35, -48.45 | 80.9, -10.31 | out-out-out | SNCooo | out-out | ActLoopNT-out | 6.8343 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 6.3 | APE9-dihe-in | -114.67, 127.92 | APE8-dihe-in | -87.4, 86.48 | APE8-rot-na | 29.16 | APE67-dihe-in | -62.99, -38.55 | -63.72, -40.61 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 12.5252 | APE9-dist-out | 8.7343 | T790M | None | None | XRAY | 3.14 | 0.258 | 0.28 | H | 331.0 | 300.0 | 16 | 30 | 18 | 12 | [[712, 970]] | 1.0 | 5gty | Homo sapiens | TYR_EGFR_HUMAN | TYR | 8.4e-88 | 300.1 | 3.0 | 259.0 | 257.0 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837.0 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|