| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 5FLFA | P11362 | 460 | 762 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5659 | 13.9215 | BLAminus | -130.07, -173.3 | 57.53, 81.51 | -106.56, 20.58 | 287.47, 88.65 | -65.69, -26.36 | in-in | in | 7.0608 | Saltbr-in | 2.6235 | HRD-in | -77.09, -44.33 | 71.36, -17.68 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8743 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -122.27, 31.65 | APE9-dihe-in | -120.82, 141.16 | APE8-dihe-in | -55.6, 118.0 | APE8-rot-na | 17.74 | APE67-dihe-in | -68.76, -3.74 | -51.76, -42.09 | APE12-dist-na | 14.9694 | APE11-dist-na | 10.4873 | APE10-dist-na | 8.0447 | APE9-dist-in | 5.7595 | R675G | None | None | XRAY | 2.58 | 0.197 | 0.255 | A | 310.0 | 296.0 | 7 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5flf | TYR_FGFR1_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5FLFB | P11362 | 460 | 764 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 6.597 | 14.2709 | BLAminus | -131.38, -174.56 | 57.69, 69.98 | -91.26, 21.65 | 284.1, 89.91 | -69.58, -18.15 | in-in | in | 7.2083 | Saltbr-in | 2.6613 | HRD-in | -77.24, -42.46 | 70.08, -13.13 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9501 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.34, 21.86 | APE9-dihe-in | -108.05, 143.02 | APE8-dihe-in | -54.9, 122.45 | APE8-rot-na | 333.47 | APE67-dihe-in | -66.56, -8.26 | -58.19, -40.45 | APE12-dist-na | 14.7668 | APE11-dist-na | 10.3425 | APE10-dist-na | 7.6761 | APE9-dist-in | 5.5875 | R675G | None | None | XRAY | 2.58 | 0.197 | 0.255 | B | 310.0 | 292.0 | 13 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5flf | TYR_FGFR1_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5FLFC | P11362 | 464 | 763 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 6.8788 | 14.9038 | BLAminus | -128.63, -179.22 | 56.68, 76.02 | -97.55, 23.96 | 288.87, 80.23 | -64.42, -24.4 | in-in | in | 7.8673 | Saltbr-in | 2.5932 | HRD-in | -77.84, -41.46 | 68.92, -13.37 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0119 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.74, 13.42 | APE9-dihe-in | -108.0, 146.11 | APE8-dihe-in | -55.87, 118.95 | APE8-rot-na | 334.41 | APE67-dihe-in | -77.03, -3.15 | -66.33, -25.17 | APE12-dist-na | 14.7227 | APE11-dist-na | 11.0185 | APE10-dist-na | 8.0397 | APE9-dist-in | 5.5345 | R675G | None | None | XRAY | 2.58 | 0.197 | 0.255 | C | 310.0 | 283.0 | 17 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5flf | TYR_FGFR1_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5FLFD | P11362 | 465 | 763 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5626 | 14.0755 | BLAminus | -137.61, -174.47 | 56.6, 77.52 | -99.56, 24.88 | 289.94, 80.48 | -64.3, -28.41 | in-in | in | 7.2769 | Saltbr-in | 2.8242 | HRD-in | -82.09, -46.03 | 69.99, -9.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9337 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -123.36, 26.56 | APE9-dihe-in | -112.27, 140.35 | APE8-dihe-in | -53.21, 117.11 | APE8-rot-na | 330.63 | APE67-dihe-in | -75.55, -3.28 | -53.96, -35.33 | APE12-dist-na | 14.9431 | APE11-dist-na | 10.5064 | APE10-dist-na | 7.9926 | APE9-dist-in | 5.5979 | R675G | None | None | XRAY | 2.58 | 0.197 | 0.255 | D | 310.0 | 290.0 | 9 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5flf | TYR_FGFR1_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5FLFE | P11362 | 466 | 761 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.8568 | 13.3331 | BLAplus | -107.08, 156.12 | 59.3, 89.04 | -145.68, 9.21 | 46.94, 85.34 | -107.07, -8.42 | in-out | in | 7.681 | Saltbr-out | 4.1216 | HRD-in | -76.44, -47.72 | 79.39, -32.07 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iooai | APEdist_aaao | APE10-dihe-in | -134.53, 84.16 | APE9-dihe-out | 70.54, 76.98 | APE8-dihe-out | -73.71, -15.89 | APE8-rot-na | 29.38 | APE67-dihe-in | -66.59, -10.19 | -60.2, -29.73 | APE12-dist-na | 999.0 | APE11-dist-na | 15.329 | APE10-dist-na | 19.6281 | APE9-dist-out | 11.396 | R675G | None | None | XRAY | 2.58 | 0.197 | 0.255 | E | 310.0 | 258.0 | 38 | 30 | 16 | 14 | [[478, 756]] | 1.0 | 5flf | TYR_FGFR1_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 5FLFA | P11362 | 460 | 762 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5659 | 13.9215 | BLAminus | -130.07, -173.3 | 57.53, 81.51 | -106.56, 20.58 | 287.47, 88.65 | -65.69, -26.36 | in-in | in | 7.0608 | Saltbr-in | 2.6235 | HRD-in | -77.09, -44.33 | 71.36, -17.68 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8743 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -122.27, 31.65 | APE9-dihe-in | -120.82, 141.16 | APE8-dihe-in | -55.6, 118.0 | APE8-rot-na | 17.74 | APE67-dihe-in | -68.76, -3.74 | -51.76, -42.09 | APE12-dist-na | 14.9694 | APE11-dist-na | 10.4873 | APE10-dist-na | 8.0447 | APE9-dist-in | 5.7595 | R675G | None | None | XRAY | 2.58 | 0.197 | 0.255 | A | 310.0 | 296.0 | 7 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5flf | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5FLFB | P11362 | 460 | 764 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 6.597 | 14.2709 | BLAminus | -131.38, -174.56 | 57.69, 69.98 | -91.26, 21.65 | 284.1, 89.91 | -69.58, -18.15 | in-in | in | 7.2083 | Saltbr-in | 2.6613 | HRD-in | -77.24, -42.46 | 70.08, -13.13 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9501 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -119.34, 21.86 | APE9-dihe-in | -108.05, 143.02 | APE8-dihe-in | -54.9, 122.45 | APE8-rot-na | 333.47 | APE67-dihe-in | -66.56, -8.26 | -58.19, -40.45 | APE12-dist-na | 14.7668 | APE11-dist-na | 10.3425 | APE10-dist-na | 7.6761 | APE9-dist-in | 5.5875 | R675G | None | None | XRAY | 2.58 | 0.197 | 0.255 | B | 310.0 | 292.0 | 13 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5flf | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5FLFC | P11362 | 464 | 763 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 6.8788 | 14.9038 | BLAminus | -128.63, -179.22 | 56.68, 76.02 | -97.55, 23.96 | 288.87, 80.23 | -64.42, -24.4 | in-in | in | 7.8673 | Saltbr-in | 2.5932 | HRD-in | -77.84, -41.46 | 68.92, -13.37 | in-in-out | SNCiio | in-out | ActLoopNT-in | 3.0119 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.74, 13.42 | APE9-dihe-in | -108.0, 146.11 | APE8-dihe-in | -55.87, 118.95 | APE8-rot-na | 334.41 | APE67-dihe-in | -77.03, -3.15 | -66.33, -25.17 | APE12-dist-na | 14.7227 | APE11-dist-na | 11.0185 | APE10-dist-na | 8.0397 | APE9-dist-in | 5.5345 | R675G | None | None | XRAY | 2.58 | 0.197 | 0.255 | C | 310.0 | 283.0 | 17 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5flf | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5FLFD | P11362 | 465 | 763 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 6.5626 | 14.0755 | BLAminus | -137.61, -174.47 | 56.6, 77.52 | -99.56, 24.88 | 289.94, 80.48 | -64.3, -28.41 | in-in | in | 7.2769 | Saltbr-in | 2.8242 | HRD-in | -82.09, -46.03 | 69.99, -9.21 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9337 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -123.36, 26.56 | APE9-dihe-in | -112.27, 140.35 | APE8-dihe-in | -53.21, 117.11 | APE8-rot-na | 330.63 | APE67-dihe-in | -75.55, -3.28 | -53.96, -35.33 | APE12-dist-na | 14.9431 | APE11-dist-na | 10.5064 | APE10-dist-na | 7.9926 | APE9-dist-in | 5.5979 | R675G | None | None | XRAY | 2.58 | 0.197 | 0.255 | D | 310.0 | 290.0 | 9 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5flf | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5FLFE | P11362 | 466 | 761 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.8568 | 13.3331 | BLAplus | -107.08, 156.12 | 59.3, 89.04 | -145.68, 9.21 | 46.94, 85.34 | -107.07, -8.42 | in-out | in | 7.681 | Saltbr-out | 4.1216 | HRD-in | -76.44, -47.72 | 79.39, -32.07 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iooai | APEdist_aaao | APE10-dihe-in | -134.53, 84.16 | APE9-dihe-out | 70.54, 76.98 | APE8-dihe-out | -73.71, -15.89 | APE8-rot-na | 29.38 | APE67-dihe-in | -66.59, -10.19 | -60.2, -29.73 | APE12-dist-na | 999.0 | APE11-dist-na | 15.329 | APE10-dist-na | 19.6281 | APE9-dist-out | 11.396 | R675G | None | None | XRAY | 2.58 | 0.197 | 0.255 | E | 310.0 | 258.0 | 38 | 30 | 16 | 14 | [[478, 756]] | 1.0 | 5flf | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 2.7e-104 | 354.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|