| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 5AM6A | P11362 | 458 | 765 | 822.0 | 38O:61766 | Type1 | Inactive | DFGin | 5.201 | 13.2703 | BLAplus | -112.58, 159.52 | 61.38, 32.49 | -78.96, -18.15 | 54.05, 84.03 | -102.14, 12.3 | in-in | in | 7.7152 | Saltbr-in | 3.2516 | HRD-in | -73.83, -55.77 | 84.43, -16.37 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.7281 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -103.68, 158.35 | APE9-dihe-in | -101.09, 116.06 | APE8-dihe-out | -55.18, -24.78 | APE8-rot-na | 339.12 | APE67-dihe-in | -70.49, -7.18 | -57.16, -24.6 | APE12-dist-na | 19.7602 | APE11-dist-na | 21.181 | APE10-dist-na | 19.8607 | APE9-dist-out | 11.7652 | None | None | None | XRAY | 1.96 | 0.216 | 0.252 | A | 310.0 | 294.0 | 14 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5am6 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5AM6B | P11362 | 458 | 762 | 822.0 | 38O:61763 | Type1 | Inactive | DFGin | 5.2795 | 13.0402 | BLAplus | -109.26, 159.81 | 58.35, 42.16 | -91.18, -11.81 | 51.78, 82.49 | -107.62, 15.27 | in-in | in | 7.6454 | Saltbr-in | 3.4946 | HRD-in | -73.63, -54.03 | 80.88, -21.94 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6147 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -106.73, 157.38 | APE9-dihe-in | -92.88, 109.99 | APE8-dihe-out | -51.36, -29.92 | APE8-rot-na | 334.27 | APE67-dihe-in | -70.82, -6.38 | -56.34, -19.57 | APE12-dist-na | 999.0 | APE11-dist-na | 21.1311 | APE10-dist-na | 19.7444 | APE9-dist-out | 11.6365 | None | None | None | XRAY | 1.96 | 0.216 | 0.252 | B | 310.0 | 280.0 | 25 | 30 | 17 | 13 | [[478, 756]] | 1.0 | 5am6 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 5AM6A | P11362 | 458 | 765 | 822.0 | 38O:61766 | Type1 | Inactive | DFGin | 5.201 | 13.2703 | BLAplus | -112.58, 159.52 | 61.38, 32.49 | -78.96, -18.15 | 54.05, 84.03 | -102.14, 12.3 | in-in | in | 7.7152 | Saltbr-in | 3.2516 | HRD-in | -73.83, -55.77 | 84.43, -16.37 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.7281 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -103.68, 158.35 | APE9-dihe-in | -101.09, 116.06 | APE8-dihe-out | -55.18, -24.78 | APE8-rot-na | 339.12 | APE67-dihe-in | -70.49, -7.18 | -57.16, -24.6 | APE12-dist-na | 19.7602 | APE11-dist-na | 21.181 | APE10-dist-na | 19.8607 | APE9-dist-out | 11.7652 | None | None | None | XRAY | 1.96 | 0.216 | 0.252 | A | 310.0 | 294.0 | 14 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 5am6 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 5AM6B | P11362 | 458 | 762 | 822.0 | 38O:61763 | Type1 | Inactive | DFGin | 5.2795 | 13.0402 | BLAplus | -109.26, 159.81 | 58.35, 42.16 | -91.18, -11.81 | 51.78, 82.49 | -107.62, 15.27 | in-in | in | 7.6454 | Saltbr-in | 3.4946 | HRD-in | -73.63, -54.03 | 80.88, -21.94 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.6147 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -106.73, 157.38 | APE9-dihe-in | -92.88, 109.99 | APE8-dihe-out | -51.36, -29.92 | APE8-rot-na | 334.27 | APE67-dihe-in | -70.82, -6.38 | -56.34, -19.57 | APE12-dist-na | 999.0 | APE11-dist-na | 21.1311 | APE10-dist-na | 19.7444 | APE9-dist-out | 11.6365 | None | None | None | XRAY | 1.96 | 0.216 | 0.252 | B | 310.0 | 280.0 | 25 | 30 | 17 | 13 | [[478, 756]] | 1.0 | 5am6 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|