| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4ZSAA | P11362 | 464 | 765 | 822.0 | 4UT:801 | Type1 | Inactive | DFGin | 5.2357 | 13.3584 | BLAplus | -116.62, 164.17 | 62.61, 38.9 | -97.55, -0.8 | 57.69, 84.31 | -93.9, -12.07 | in-in | in | 7.7271 | Saltbr-in | 3.0735 | HRD-in | -75.4, -51.03 | 78.41, -18.38 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.8014 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -100.19, 166.07 | APE9-dihe-in | -106.61, 111.7 | APE8-dihe-out | -53.66, -24.02 | APE8-rot-na | 328.26 | APE67-dihe-in | -75.2, -3.02 | -58.56, -21.55 | APE12-dist-na | 20.9966 | APE11-dist-na | 22.3196 | APE10-dist-na | 20.7954 | APE9-dist-out | 11.8029 | C488A,C584S | None | None | XRAY | 2.0 | 0.206 | 0.254 | A | 308.0 | 290.0 | 12 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 4zsa | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4ZSAB | P11362 | 462 | 761 | 822.0 | 4UT:801 | Type1 | Inactive | DFGin | 5.3779 | 12.914 | BLAplus | -118.54, 160.55 | 64.46, 37.46 | -95.07, -9.43 | 54.72, 89.6 | -73.6, -19.27 | in-in | in | 7.6413 | Saltbr-in | 3.1631 | HRD-in | -75.52, -45.77 | 74.73, -25.0 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.36, 172.16 | APE9-dihe-in | -104.52, 114.27 | APE8-dihe-out | -53.39, -26.0 | APE8-rot-na | 330.81 | APE67-dihe-in | -73.62, -3.9 | -59.13, -21.5 | APE12-dist-na | 20.7248 | APE11-dist-na | 22.162 | APE10-dist-na | 20.8587 | APE9-dist-out | 11.5249 | C488A,C584S | None | None | XRAY | 2.0 | 0.206 | 0.254 | B | 308.0 | 282.0 | 18 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4zsa | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4ZSAA | P11362 | 464 | 765 | 822.0 | 4UT:801 | Type1 | Inactive | DFGin | 5.2357 | 13.3584 | BLAplus | -116.62, 164.17 | 62.61, 38.9 | -97.55, -0.8 | 57.69, 84.31 | -93.9, -12.07 | in-in | in | 7.7271 | Saltbr-in | 3.0735 | HRD-in | -75.4, -51.03 | 78.41, -18.38 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.8014 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -100.19, 166.07 | APE9-dihe-in | -106.61, 111.7 | APE8-dihe-out | -53.66, -24.02 | APE8-rot-na | 328.26 | APE67-dihe-in | -75.2, -3.02 | -58.56, -21.55 | APE12-dist-na | 20.9966 | APE11-dist-na | 22.3196 | APE10-dist-na | 20.7954 | APE9-dist-out | 11.8029 | C488A,C584S | None | None | XRAY | 2.0 | 0.206 | 0.254 | A | 308.0 | 290.0 | 12 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 4zsa | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4ZSAB | P11362 | 462 | 761 | 822.0 | 4UT:801 | Type1 | Inactive | DFGin | 5.3779 | 12.914 | BLAplus | -118.54, 160.55 | 64.46, 37.46 | -95.07, -9.43 | 54.72, 89.6 | -73.6, -19.27 | in-in | in | 7.6413 | Saltbr-in | 3.1631 | HRD-in | -75.52, -45.77 | 74.73, -25.0 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.36, 172.16 | APE9-dihe-in | -104.52, 114.27 | APE8-dihe-out | -53.39, -26.0 | APE8-rot-na | 330.81 | APE67-dihe-in | -73.62, -3.9 | -59.13, -21.5 | APE12-dist-na | 20.7248 | APE11-dist-na | 22.162 | APE10-dist-na | 20.8587 | APE9-dist-out | 11.5249 | C488A,C584S | None | None | XRAY | 2.0 | 0.206 | 0.254 | B | 308.0 | 282.0 | 18 | 30 | 24 | 6 | [[478, 756]] | 1.0 | 4zsa | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|