| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4V05A | P11362 | 464 | 765 | 822.0 | 66T:1769 | Type1.5_Back | Inactive | DFGin | 5.4734 | 13.4201 | BLAplus | -110.72, 173.08 | 50.09, 39.57 | -95.62, -19.67 | 60.09, 83.48 | -87.99, 3.34 | in-in | in | 8.0484 | Saltbr-in | 2.7499 | HRD-in | -64.72, -51.32 | 77.65, -23.6 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.3021 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -98.91, 158.86 | APE9-dihe-in | -104.86, 116.5 | APE8-dihe-out | -57.09, -23.19 | APE8-rot-na | 335.63 | APE67-dihe-in | -66.78, -18.31 | -54.95, -24.99 | APE12-dist-na | 20.8412 | APE11-dist-na | 21.8076 | APE10-dist-na | 19.9108 | APE9-dist-out | 11.6016 | None | None | None | XRAY | 2.57 | 0.196 | 0.256 | A | 309.0 | 287.0 | 15 | 30 | 26 | 4 | [[478, 756]] | 1.0 | 4v05 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V05B | P11362 | 459 | 764 | 822.0 | 66T:1767 | Type1.5_Back | Inactive | DFGin | 5.4267 | 13.0724 | BLAplus | -110.08, 173.06 | 48.31, 47.35 | -106.86, -10.85 | 58.74, 86.16 | -77.17, -18.0 | in-in | in | 7.8311 | Saltbr-in | 2.9832 | HRD-in | -65.29, -47.82 | 74.06, -21.09 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.03, 160.1 | APE9-dihe-in | -100.97, 109.95 | APE8-dihe-out | -53.4, -23.19 | APE8-rot-na | 333.98 | APE67-dihe-in | -59.05, -11.55 | -51.93, -35.21 | APE12-dist-na | 21.3913 | APE11-dist-na | 22.0888 | APE10-dist-na | 20.5381 | APE9-dist-out | 11.4653 | None | None | None | XRAY | 2.57 | 0.196 | 0.256 | B | 309.0 | 286.0 | 20 | 30 | 26 | 4 | [[478, 756]] | 1.0 | 4v05 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4V05A | P11362 | 464 | 765 | 822.0 | 66T:1769 | Type1.5_Back | Inactive | DFGin | 5.4734 | 13.4201 | BLAplus | -110.72, 173.08 | 50.09, 39.57 | -95.62, -19.67 | 60.09, 83.48 | -87.99, 3.34 | in-in | in | 8.0484 | Saltbr-in | 2.7499 | HRD-in | -64.72, -51.32 | 77.65, -23.6 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.3021 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -98.91, 158.86 | APE9-dihe-in | -104.86, 116.5 | APE8-dihe-out | -57.09, -23.19 | APE8-rot-na | 335.63 | APE67-dihe-in | -66.78, -18.31 | -54.95, -24.99 | APE12-dist-na | 20.8412 | APE11-dist-na | 21.8076 | APE10-dist-na | 19.9108 | APE9-dist-out | 11.6016 | None | None | None | XRAY | 2.57 | 0.196 | 0.256 | A | 309.0 | 287.0 | 15 | 30 | 26 | 4 | [[478, 756]] | 1.0 | 4v05 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V05B | P11362 | 459 | 764 | 822.0 | 66T:1767 | Type1.5_Back | Inactive | DFGin | 5.4267 | 13.0724 | BLAplus | -110.08, 173.06 | 48.31, 47.35 | -106.86, -10.85 | 58.74, 86.16 | -77.17, -18.0 | in-in | in | 7.8311 | Saltbr-in | 2.9832 | HRD-in | -65.29, -47.82 | 74.06, -21.09 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.03, 160.1 | APE9-dihe-in | -100.97, 109.95 | APE8-dihe-out | -53.4, -23.19 | APE8-rot-na | 333.98 | APE67-dihe-in | -59.05, -11.55 | -51.93, -35.21 | APE12-dist-na | 21.3913 | APE11-dist-na | 22.0888 | APE10-dist-na | 20.5381 | APE9-dist-out | 11.4653 | None | None | None | XRAY | 2.57 | 0.196 | 0.256 | B | 309.0 | 286.0 | 20 | 30 | 26 | 4 | [[478, 756]] | 1.0 | 4v05 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|