| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4RWKA | P11362 | 458 | 764 | 822.0 | 66T:60801 | Type1 | Inactive | DFGin | 5.334 | 13.4485 | BLAplus | -119.61, 171.78 | 43.5, 42.06 | -91.27, -13.97 | 55.41, 85.99 | -97.85, 1.35 | in-in | in | 8.3001 | Saltbr-in | 2.8581 | HRD-in | -72.97, -43.98 | 66.64, 7.94 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.6119 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -132.9, 130.16 | APE9-dihe-in | -81.93, 117.68 | APE8-dihe-out | -73.74, -2.4 | APE8-rot-na | 340.19 | APE67-dihe-in | -78.12, -6.2 | -84.98, -15.3 | APE12-dist-na | 17.0094 | APE11-dist-na | 18.9505 | APE10-dist-na | 16.7093 | APE9-dist-out | 11.0044 | C488A,V561M,C584S | None | None | XRAY | 2.982 | 0.244 | 0.299 | A | 317.0 | 307.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 4rwk | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWKB | P11362 | 459 | 763 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.7367 | 13.232 | BLAplus | -119.15, 169.82 | 41.98, 44.21 | -90.47, -9.61 | 54.08, 84.94 | -94.37, 2.45 | in-in | in | 8.4157 | Saltbr-in | 3.448 | HRD-in | -74.45, -44.2 | 66.06, 8.62 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -133.04, 131.77 | APE9-dihe-in | -79.69, 122.84 | APE8-dihe-out | -69.38, -1.04 | APE8-rot-na | 339.66 | APE67-dihe-in | -75.83, -3.81 | -84.39, -12.82 | APE12-dist-na | 999.0 | APE11-dist-na | 21.9267 | APE10-dist-na | 19.8348 | APE9-dist-out | 11.6466 | C488A,V561M,C584S | None | None | XRAY | 2.982 | 0.244 | 0.299 | B | 317.0 | 282.0 | 23 | 30 | 23 | 7 | [[478, 756]] | 1.0 | 4rwk | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4RWKA | P11362 | 458 | 764 | 822.0 | 66T:60801 | Type1 | Inactive | DFGin | 5.334 | 13.4485 | BLAplus | -119.61, 171.78 | 43.5, 42.06 | -91.27, -13.97 | 55.41, 85.99 | -97.85, 1.35 | in-in | in | 8.3001 | Saltbr-in | 2.8581 | HRD-in | -72.97, -43.98 | 66.64, 7.94 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.6119 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -132.9, 130.16 | APE9-dihe-in | -81.93, 117.68 | APE8-dihe-out | -73.74, -2.4 | APE8-rot-na | 340.19 | APE67-dihe-in | -78.12, -6.2 | -84.98, -15.3 | APE12-dist-na | 17.0094 | APE11-dist-na | 18.9505 | APE10-dist-na | 16.7093 | APE9-dist-out | 11.0044 | C488A,V561M,C584S | None | None | XRAY | 2.982 | 0.244 | 0.299 | A | 317.0 | 307.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 4rwk | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWKB | P11362 | 459 | 763 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.7367 | 13.232 | BLAplus | -119.15, 169.82 | 41.98, 44.21 | -90.47, -9.61 | 54.08, 84.94 | -94.37, 2.45 | in-in | in | 8.4157 | Saltbr-in | 3.448 | HRD-in | -74.45, -44.2 | 66.06, 8.62 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -133.04, 131.77 | APE9-dihe-in | -79.69, 122.84 | APE8-dihe-out | -69.38, -1.04 | APE8-rot-na | 339.66 | APE67-dihe-in | -75.83, -3.81 | -84.39, -12.82 | APE12-dist-na | 999.0 | APE11-dist-na | 21.9267 | APE10-dist-na | 19.8348 | APE9-dist-out | 11.6466 | C488A,V561M,C584S | None | None | XRAY | 2.982 | 0.244 | 0.299 | B | 317.0 | 282.0 | 23 | 30 | 23 | 7 | [[478, 756]] | 1.0 | 4rwk | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|