| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4RWJA | P11362 | 458 | 764 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.2638 | 13.5569 | BLAplus | -111.1, 165.72 | 44.3, 59.14 | -104.5, -7.94 | 52.98, 85.2 | -108.93, 18.9 | in-in | in | 8.0637 | Saltbr-in | 3.1247 | HRD-in | -76.03, -43.68 | 72.99, -8.16 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9816 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.41, 138.95 | APE9-dihe-in | -108.01, 100.05 | APE8-dihe-out | -61.04, -14.23 | APE8-rot-na | 22.4 | APE67-dihe-in | -81.18, -2.01 | -65.12, -23.42 | APE12-dist-na | 19.4256 | APE11-dist-na | 20.4566 | APE10-dist-na | 17.046 | APE9-dist-out | 11.3201 | C488A,C584S | None | None | XRAY | 2.489 | 0.204 | 0.25 | A | 317.0 | 306.0 | 1 | 30 | 29 | 1 | [[478, 756]] | 1.0 | 4rwj | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWJB | P11362 | 459 | 763 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.3065 | 13.0754 | BLAplus | -111.81, 166.65 | 44.09, 58.11 | -104.8, -5.62 | 52.57, 84.61 | -105.75, 19.27 | in-in | in | 7.9338 | Saltbr-in | 2.8347 | HRD-in | -75.88, -44.44 | 70.84, -6.0 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.6, 139.99 | APE9-dihe-in | -106.55, 102.92 | APE8-dihe-out | -58.58, -14.6 | APE8-rot-na | 336.03 | APE67-dihe-in | -80.58, -2.45 | -66.06, -21.44 | APE12-dist-na | 999.0 | APE11-dist-na | 21.7066 | APE10-dist-na | 18.4779 | APE9-dist-out | 11.5466 | C488A,C584S | None | None | XRAY | 2.489 | 0.204 | 0.25 | B | 317.0 | 282.0 | 23 | 30 | 20 | 10 | [[478, 756]] | 1.0 | 4rwj | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4RWJA | P11362 | 458 | 764 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.2638 | 13.5569 | BLAplus | -111.1, 165.72 | 44.3, 59.14 | -104.5, -7.94 | 52.98, 85.2 | -108.93, 18.9 | in-in | in | 8.0637 | Saltbr-in | 3.1247 | HRD-in | -76.03, -43.68 | 72.99, -8.16 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9816 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.41, 138.95 | APE9-dihe-in | -108.01, 100.05 | APE8-dihe-out | -61.04, -14.23 | APE8-rot-na | 22.4 | APE67-dihe-in | -81.18, -2.01 | -65.12, -23.42 | APE12-dist-na | 19.4256 | APE11-dist-na | 20.4566 | APE10-dist-na | 17.046 | APE9-dist-out | 11.3201 | C488A,C584S | None | None | XRAY | 2.489 | 0.204 | 0.25 | A | 317.0 | 306.0 | 1 | 30 | 29 | 1 | [[478, 756]] | 1.0 | 4rwj | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWJB | P11362 | 459 | 763 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.3065 | 13.0754 | BLAplus | -111.81, 166.65 | 44.09, 58.11 | -104.8, -5.62 | 52.57, 84.61 | -105.75, 19.27 | in-in | in | 7.9338 | Saltbr-in | 2.8347 | HRD-in | -75.88, -44.44 | 70.84, -6.0 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.6, 139.99 | APE9-dihe-in | -106.55, 102.92 | APE8-dihe-out | -58.58, -14.6 | APE8-rot-na | 336.03 | APE67-dihe-in | -80.58, -2.45 | -66.06, -21.44 | APE12-dist-na | 999.0 | APE11-dist-na | 21.7066 | APE10-dist-na | 18.4779 | APE9-dist-out | 11.5466 | C488A,C584S | None | None | XRAY | 2.489 | 0.204 | 0.25 | B | 317.0 | 282.0 | 23 | 30 | 20 | 10 | [[478, 756]] | 1.0 | 4rwj | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|