| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4RWIA | P11362 | 460 | 764 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1902 | 13.2874 | BLAplus | -105.16, 163.21 | 56.87, 28.19 | -74.61, -16.94 | 54.32, 87.9 | -104.05, 11.37 | in-in | in | 7.9641 | Saltbr-in | 2.6905 | HRD-in | -73.3, -52.29 | 82.32, -10.23 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.0996 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -101.29, 144.76 | APE9-dihe-in | -100.4, 99.63 | APE8-dihe-out | -55.34, -23.98 | APE8-rot-na | 331.55 | APE67-dihe-in | -74.41, -9.61 | -59.83, -21.73 | APE12-dist-na | 17.4922 | APE11-dist-na | 19.0334 | APE10-dist-na | 16.5776 | APE9-dist-out | 11.2323 | C488A,V561M,C584S | None | None | XRAY | 2.292 | 0.188 | 0.236 | A | 317.0 | 305.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 4rwi | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWIB | P11362 | 461 | 763 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1408 | 13.1536 | BLAplus | -106.54, 164.69 | 57.29, 29.78 | -77.53, -18.65 | 57.49, 89.17 | -101.92, 7.65 | in-in | in | 7.8788 | Saltbr-in | 2.8702 | HRD-in | -73.64, -53.72 | 81.97, -10.53 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -103.37, 146.39 | APE9-dihe-in | -96.99, 106.58 | APE8-dihe-out | -51.08, -23.64 | APE8-rot-na | 329.78 | APE67-dihe-in | -74.22, -7.08 | -61.58, -21.03 | APE12-dist-na | 999.0 | APE11-dist-na | 21.6378 | APE10-dist-na | 19.3161 | APE9-dist-out | 11.6321 | C488A,V561M,C584S | None | None | XRAY | 2.292 | 0.188 | 0.236 | B | 317.0 | 280.0 | 23 | 30 | 25 | 5 | [[478, 756]] | 1.0 | 4rwi | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4RWIA | P11362 | 460 | 764 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1902 | 13.2874 | BLAplus | -105.16, 163.21 | 56.87, 28.19 | -74.61, -16.94 | 54.32, 87.9 | -104.05, 11.37 | in-in | in | 7.9641 | Saltbr-in | 2.6905 | HRD-in | -73.3, -52.29 | 82.32, -10.23 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.0996 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -101.29, 144.76 | APE9-dihe-in | -100.4, 99.63 | APE8-dihe-out | -55.34, -23.98 | APE8-rot-na | 331.55 | APE67-dihe-in | -74.41, -9.61 | -59.83, -21.73 | APE12-dist-na | 17.4922 | APE11-dist-na | 19.0334 | APE10-dist-na | 16.5776 | APE9-dist-out | 11.2323 | C488A,V561M,C584S | None | None | XRAY | 2.292 | 0.188 | 0.236 | A | 317.0 | 305.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 4rwi | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWIB | P11362 | 461 | 763 | 822.0 | No_ligand | No_ligand | Inactive | DFGin | 5.1408 | 13.1536 | BLAplus | -106.54, 164.69 | 57.29, 29.78 | -77.53, -18.65 | 57.49, 89.17 | -101.92, 7.65 | in-in | in | 7.8788 | Saltbr-in | 2.8702 | HRD-in | -73.64, -53.72 | 81.97, -10.53 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -103.37, 146.39 | APE9-dihe-in | -96.99, 106.58 | APE8-dihe-out | -51.08, -23.64 | APE8-rot-na | 329.78 | APE67-dihe-in | -74.22, -7.08 | -61.58, -21.03 | APE12-dist-na | 999.0 | APE11-dist-na | 21.6378 | APE10-dist-na | 19.3161 | APE9-dist-out | 11.6321 | C488A,V561M,C584S | None | None | XRAY | 2.292 | 0.188 | 0.236 | B | 317.0 | 280.0 | 23 | 30 | 25 | 5 | [[478, 756]] | 1.0 | 4rwi | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|