| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EPHA2 | EPHA2_HUMAN | 4PDOA | P29317 | 590 | 875 | 976.0 | No_ligand | No_ligand | Inactive | DFGin | 5.3167 | 14.8536 | None | -130.75, -10.88 | -121.71, 138.39 | -133.1, 999.0 | 295.74, 93.17 | 999.0, 999.0 | in-out | in | 7.9685 | Saltbr-out | 6.2618 | HRD-in | -77.55, -48.01 | 73.27, -11.62 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.79, 137.86 | APE9-dihe-in | -135.53, 157.5 | APE8-dihe-in | -79.41, 83.0 | APE8-rot-na | 28.9 | APE67-dihe-in | -59.48, -20.71 | -53.52, -46.26 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.4933 | None | None | None | XRAY | 2.104 | 0.162 | 0.184 | A | 299.0 | 261.0 | 25 | 31 | 13 | 18 | [[613, 873]] | 1.0 | 4pdo | TYR_EPHA2_HUMAN | TYR | 5.1e-108 | 366.2 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 4PDOB | P29317 | 590 | 875 | 976.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2883 | 14.8974 | None | -129.53, -11.31 | -121.1, 139.25 | -134.72, 999.0 | 294.46, 94.17 | 999.0, 999.0 | in-out | in | 7.9653 | Saltbr-out | 6.3734 | HRD-in | -76.29, -48.44 | 73.45, -12.19 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -71.42, 139.51 | APE9-dihe-in | -133.49, 157.9 | APE8-dihe-in | -78.68, 83.43 | APE8-rot-na | 28.65 | APE67-dihe-in | -60.39, -20.86 | -55.6, -45.15 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.4952 | None | None | None | XRAY | 2.104 | 0.162 | 0.184 | B | 299.0 | 261.0 | 25 | 31 | 13 | 18 | [[613, 873]] | 1.0 | 4pdo | TYR_EPHA2_HUMAN | TYR | 5.1e-108 | 366.2 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EPHA2 | EPHA2_HUMAN | 4PDOA | P29317 | 590 | 875 | 976.0 | No_ligand | No_ligand | Inactive | DFGin | 5.3167 | 14.8536 | None | -130.75, -10.88 | -121.71, 138.39 | -133.1, 999.0 | 295.74, 93.17 | 999.0, 999.0 | in-out | in | 7.9685 | Saltbr-out | 6.2618 | HRD-in | -77.55, -48.01 | 73.27, -11.62 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.79, 137.86 | APE9-dihe-in | -135.53, 157.5 | APE8-dihe-in | -79.41, 83.0 | APE8-rot-na | 28.9 | APE67-dihe-in | -59.48, -20.71 | -53.52, -46.26 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.4933 | None | None | None | XRAY | 2.104 | 0.162 | 0.184 | A | 299.0 | 261.0 | 25 | 31 | 13 | 18 | [[613, 873]] | 1.0 | 4pdo | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 5.1e-108 | 366.2 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| TYR | EPHA2 | EPHA2_HUMAN | 4PDOB | P29317 | 590 | 875 | 976.0 | No_ligand | No_ligand | Inactive | DFGin | 5.2883 | 14.8974 | None | -129.53, -11.31 | -121.1, 139.25 | -134.72, 999.0 | 294.46, 94.17 | 999.0, 999.0 | in-out | in | 7.9653 | Saltbr-out | 6.3734 | HRD-in | -76.29, -48.44 | 73.45, -12.19 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -71.42, 139.51 | APE9-dihe-in | -133.49, 157.9 | APE8-dihe-in | -78.68, 83.43 | APE8-rot-na | 28.65 | APE67-dihe-in | -60.39, -20.86 | -55.6, -45.15 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-in | 6.4952 | None | None | None | XRAY | 2.104 | 0.162 | 0.184 | B | 299.0 | 261.0 | 25 | 31 | 13 | 18 | [[613, 873]] | 1.0 | 4pdo | Homo sapiens | TYR_EPHA2_HUMAN | TYR | 5.1e-108 | 366.2 | 2.0 | 261.0 | 260.0 | 756 | 757 | 758 | 760 | 762 | 646 | 663 | 667 | 736 | 738 | 737 | 739.0 | 799 | 787 | 782 | 781 | 780 | 779 | 778 | 777 | 776 | 693 | Ephrin type-A receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|