| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK1 | GRK1_BOVIN | 4L9IA | P28327 | 30 | 533 | 561.0 | 8PR:601 | Type1 | Inactive | DFGin | 5.7724 | 13.4538 | BLAminus | -149.91, 178.73 | 54.74, 79.81 | -98.99, 23.91 | 282.53, 102.36 | -68.07, -19.68 | in-out | in | 8.693 | Saltbr-out | 3.808 | HRD-in | -75.83, -53.93 | 68.31, 13.36 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8273 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -162.8, 142.88 | APE9-dihe-na | 125.17, -158.26 | APE8-dihe-in | -112.07, 133.06 | APE8-rot-in | 301.6 | APE67-dihe-inflip | 94.99, -2.22 | -45.66, 120.79 | APE12-dist-in | 10.6157 | APE11-dist-in | 11.3826 | APE10-dist-in | 5.8078 | APE9-dist-in | 3.7234 | None | None | None | XRAY | 2.32 | 0.188 | 0.231 | A | 504.0 | 504.0 | 0 | 28 | 28 | 0 | [[187, 452]] | 1.0 | 4l9i | Bos taurus | AGC_GRK1_BOVIN | AGC | 2.5e-80 | 275.4 | 4.0 | 260.0 | 257.0 | 331 | 332 | 333 | 335 | 337 | 216 | 235 | 239 | 311 | 313 | 312 | 314.0 | 371 | 359 | 354 | 353 | 352 | 351 | 350 | 349 | 348 | 265 | Rhodopsin kinase GRK1 |
| AGC | GRK1 | GRK1_BOVIN | 4L9IB | P28327 | 31 | 533 | 561.0 | 8PR:601 | Type1 | Active | DFGin | 5.7147 | 13.0643 | BLAminus | -147.41, -179.95 | 59.09, 74.76 | -90.68, 22.77 | 285.65, 103.28 | -76.71, -12.5 | in-in | in | 8.7578 | Saltbr-in | 3.1172 | HRD-in | -77.55, -56.18 | 71.16, 4.39 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7658 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.45, 143.07 | APE9-dihe-na | 140.89, -160.87 | APE8-dihe-in | -115.15, 127.72 | APE8-rot-in | 297.19 | APE67-dihe-inflip | 102.74, -33.6 | -52.94, 132.06 | APE12-dist-in | 10.2921 | APE11-dist-in | 11.2208 | APE10-dist-in | 5.6416 | APE9-dist-in | 3.766 | None | None | None | XRAY | 2.32 | 0.188 | 0.231 | B | 504.0 | 493.0 | 0 | 28 | 28 | 0 | [[187, 452]] | 1.0 | 4l9i | Bos taurus | AGC_GRK1_BOVIN | AGC | 2.5e-80 | 275.4 | 4.0 | 260.0 | 257.0 | 331 | 332 | 333 | 335 | 337 | 216 | 235 | 239 | 311 | 313 | 312 | 314.0 | 371 | 359 | 354 | 353 | 352 | 351 | 350 | 349 | 348 | 265 | Rhodopsin kinase GRK1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| AGC | GRK1 | GRK1_BOVIN | 4L9IA | P28327 | 30 | 533 | 561.0 | 8PR:601 | Type1 | Inactive | DFGin | 5.7724 | 13.4538 | BLAminus | -149.91, 178.73 | 54.74, 79.81 | -98.99, 23.91 | 282.53, 102.36 | -68.07, -19.68 | in-out | in | 8.693 | Saltbr-out | 3.808 | HRD-in | -75.83, -53.93 | 68.31, 13.36 | out-in-in | SNCoii | in-in | ActLoopNT-in | 2.8273 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -162.8, 142.88 | APE9-dihe-na | 125.17, -158.26 | APE8-dihe-in | -112.07, 133.06 | APE8-rot-in | 301.6 | APE67-dihe-inflip | 94.99, -2.22 | -45.66, 120.79 | APE12-dist-in | 10.6157 | APE11-dist-in | 11.3826 | APE10-dist-in | 5.8078 | APE9-dist-in | 3.7234 | None | None | None | XRAY | 2.32 | 0.188 | 0.231 | A | 504.0 | 504.0 | 0 | 28 | 28 | 0 | [[187, 452]] | 1.0 | 4l9i | Bos taurus | AGC_GRK1_BOVIN | AGC | 2.5e-80 | 275.4 | 4.0 | 260.0 | 257.0 | 331 | 332 | 333 | 335 | 337 | 216 | 235 | 239 | 311 | 313 | 312 | 314.0 | 371 | 359 | 354 | 353 | 352 | 351 | 350 | 349 | 348 | 265 | Rhodopsin kinase GRK1 |
| AGC | GRK1 | GRK1_BOVIN | 4L9IB | P28327 | 31 | 533 | 561.0 | 8PR:601 | Type1 | Active | DFGin | 5.7147 | 13.0643 | BLAminus | -147.41, -179.95 | 59.09, 74.76 | -90.68, 22.77 | 285.65, 103.28 | -76.71, -12.5 | in-in | in | 8.7578 | Saltbr-in | 3.1172 | HRD-in | -77.55, -56.18 | 71.16, 4.39 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.7658 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -160.45, 143.07 | APE9-dihe-na | 140.89, -160.87 | APE8-dihe-in | -115.15, 127.72 | APE8-rot-in | 297.19 | APE67-dihe-inflip | 102.74, -33.6 | -52.94, 132.06 | APE12-dist-in | 10.2921 | APE11-dist-in | 11.2208 | APE10-dist-in | 5.6416 | APE9-dist-in | 3.766 | None | None | None | XRAY | 2.32 | 0.188 | 0.231 | B | 504.0 | 493.0 | 0 | 28 | 28 | 0 | [[187, 452]] | 1.0 | 4l9i | Bos taurus | AGC_GRK1_BOVIN | AGC | 2.5e-80 | 275.4 | 4.0 | 260.0 | 257.0 | 331 | 332 | 333 | 335 | 337 | 216 | 235 | 239 | 311 | 313 | 312 | 314.0 | 371 | 359 | 354 | 353 | 352 | 351 | 350 | 349 | 348 | 265 | Rhodopsin kinase GRK1 |