| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 4J98B | P21802 | 461 | 764 | 821.0 | ACP:804 | ATPlike | Inactive | DFGin | 6.5497 | 14.0416 | BLAminus | -130.09, -172.54 | 52.51, 78.98 | -94.32, 21.96 | 285.07, 86.18 | -63.61, -22.45 | in-in | in | 7.1129 | Saltbr-in | 3.0165 | HRD-in | -86.21, -48.16 | 74.7, -12.01 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8085 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -116.22, 26.63 | APE9-dihe-in | -99.48, 124.84 | APE8-dihe-in | -50.97, 125.51 | APE8-rot-na | 328.99 | APE67-dihe-in | -68.16, -7.57 | -60.28, -41.11 | APE12-dist-na | 15.0958 | APE11-dist-na | 10.4175 | APE10-dist-na | 7.5796 | APE9-dist-in | 4.8265 | C491A,K659Q | None | None | XRAY | 2.307 | 0.19 | 0.234 | B | 324.0 | 304.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j98 | TYR_FGFR2_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J98A | P21802 | 461 | 764 | 821.0 | No_ligand | No_ligand | Inactive | DFGin | 6.8949 | 14.189 | BLAminus | -127.05, -173.93 | 55.52, 75.94 | -94.55, 21.07 | 285.33, 84.3 | -62.1, -22.56 | in-in | in | 7.2723 | Saltbr-in | 2.7079 | HRD-in | -84.97, -48.15 | 77.1, -13.76 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8915 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.08, 26.13 | APE9-dihe-in | -100.11, 126.32 | APE8-dihe-in | -52.05, 125.82 | APE8-rot-na | 328.58 | APE67-dihe-in | -66.67, -7.8 | -60.08, -40.94 | APE12-dist-na | 15.2032 | APE11-dist-na | 10.4996 | APE10-dist-na | 7.5006 | APE9-dist-in | 5.0053 | C491A,K659Q | None | None | XRAY | 2.307 | 0.19 | 0.234 | A | 324.0 | 304.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j98 | TYR_FGFR2_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 4J98B | P21802 | 461 | 764 | 821.0 | ACP:804 | ATPlike | Inactive | DFGin | 6.5497 | 14.0416 | BLAminus | -130.09, -172.54 | 52.51, 78.98 | -94.32, 21.96 | 285.07, 86.18 | -63.61, -22.45 | in-in | in | 7.1129 | Saltbr-in | 3.0165 | HRD-in | -86.21, -48.16 | 74.7, -12.01 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8085 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -116.22, 26.63 | APE9-dihe-in | -99.48, 124.84 | APE8-dihe-in | -50.97, 125.51 | APE8-rot-na | 328.99 | APE67-dihe-in | -68.16, -7.57 | -60.28, -41.11 | APE12-dist-na | 15.0958 | APE11-dist-na | 10.4175 | APE10-dist-na | 7.5796 | APE9-dist-in | 4.8265 | C491A,K659Q | None | None | XRAY | 2.307 | 0.19 | 0.234 | B | 324.0 | 304.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j98 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 4J98A | P21802 | 461 | 764 | 821.0 | No_ligand | No_ligand | Inactive | DFGin | 6.8949 | 14.189 | BLAminus | -127.05, -173.93 | 55.52, 75.94 | -94.55, 21.07 | 285.33, 84.3 | -62.1, -22.56 | in-in | in | 7.2723 | Saltbr-in | 2.7079 | HRD-in | -84.97, -48.15 | 77.1, -13.76 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8915 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -114.08, 26.13 | APE9-dihe-in | -100.11, 126.32 | APE8-dihe-in | -52.05, 125.82 | APE8-rot-na | 328.58 | APE67-dihe-in | -66.67, -7.8 | -60.08, -40.94 | APE12-dist-na | 15.2032 | APE11-dist-na | 10.4996 | APE10-dist-na | 7.5006 | APE9-dist-in | 5.0053 | C491A,K659Q | None | None | XRAY | 2.307 | 0.19 | 0.234 | A | 324.0 | 304.0 | 0 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 4j98 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.1e-104 | 354.4 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|