| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | INSR | INSR_HUMAN | 4IBMA | P06213 | 1009 | 1309 | 1382.0 | IR1:61301 | Type1 | Inactive | DFGin | 5.6235 | 15.3135 | None | -76.0, 163.85 | -44.82, 128.63 | -69.67, 135.99 | 297.32, 165.57 | 60.17, 44.87 | out-out | out | 10.6453 | Saltbr-out | 7.271 | HRD-in | -68.74, -46.51 | 75.22, -15.25 | out-out-in | SNCooi | out-in | ActLoopNT-out | 15.6653 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.2, 121.44 | APE9-dihe-in | -109.91, 120.82 | APE8-dihe-in | -81.27, 70.1 | APE8-rot-na | 28.73 | APE67-dihe-in | -71.57, -11.47 | -57.01, -32.73 | APE12-dist-na | 18.7378 | APE11-dist-na | 15.2744 | APE10-dist-na | 11.5056 | APE9-dist-in | 7.3145 | K1278N | None | None | XRAY | 1.8 | 0.184 | 0.218 | A | 306.0 | 301.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 4ibm | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| TYR | INSR | INSR_HUMAN | 4IBMB | P06213 | 1014 | 1310 | 1382.0 | IR1:61301 | Type1 | Inactive | DFGin | 6.943 | 16.4452 | None | -69.6, 155.55 | -45.67, 125.47 | -61.25, 129.45 | 282.72, 8.49 | 78.34, 8.83 | in-out | in | 9.4175 | Saltbr-out | 5.034 | HRD-in | -66.87, -50.14 | 74.82, -11.33 | out-out-in | SNCooi | out-in | ActLoopNT-out | 15.2219 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.04, 122.58 | APE9-dihe-in | -120.44, 134.35 | APE8-dihe-in | -81.79, 69.08 | APE8-rot-na | 32.76 | APE67-dihe-in | -70.68, -10.48 | -58.86, -32.74 | APE12-dist-na | 19.958 | APE11-dist-na | 16.3087 | APE10-dist-na | 12.6646 | APE9-dist-in | 7.3059 | K1278N | None | None | XRAY | 1.8 | 0.184 | 0.218 | B | 306.0 | 294.0 | 3 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 4ibm | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | INSR | INSR_HUMAN | 4IBMA | P06213 | 1009 | 1309 | 1382.0 | IR1:61301 | Type1 | Inactive | DFGin | 5.6235 | 15.3135 | None | -76.0, 163.85 | -44.82, 128.63 | -69.67, 135.99 | 297.32, 165.57 | 60.17, 44.87 | out-out | out | 10.6453 | Saltbr-out | 7.271 | HRD-in | -68.74, -46.51 | 75.22, -15.25 | out-out-in | SNCooi | out-in | ActLoopNT-out | 15.6653 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.2, 121.44 | APE9-dihe-in | -109.91, 120.82 | APE8-dihe-in | -81.27, 70.1 | APE8-rot-na | 28.73 | APE67-dihe-in | -71.57, -11.47 | -57.01, -32.73 | APE12-dist-na | 18.7378 | APE11-dist-na | 15.2744 | APE10-dist-na | 11.5056 | APE9-dist-in | 7.3145 | K1278N | None | None | XRAY | 1.8 | 0.184 | 0.218 | A | 306.0 | 301.0 | 0 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 4ibm | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| TYR | INSR | INSR_HUMAN | 4IBMB | P06213 | 1014 | 1310 | 1382.0 | IR1:61301 | Type1 | Inactive | DFGin | 6.943 | 16.4452 | None | -69.6, 155.55 | -45.67, 125.47 | -61.25, 129.45 | 282.72, 8.49 | 78.34, 8.83 | in-out | in | 9.4175 | Saltbr-out | 5.034 | HRD-in | -66.87, -50.14 | 74.82, -11.33 | out-out-in | SNCooi | out-in | ActLoopNT-out | 15.2219 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -77.04, 122.58 | APE9-dihe-in | -120.44, 134.35 | APE8-dihe-in | -81.79, 69.08 | APE8-rot-na | 32.76 | APE67-dihe-in | -70.68, -10.48 | -58.86, -32.74 | APE12-dist-na | 19.958 | APE11-dist-na | 16.3087 | APE10-dist-na | 12.6646 | APE9-dist-in | 7.3059 | K1278N | None | None | XRAY | 1.8 | 0.184 | 0.218 | B | 306.0 | 294.0 | 3 | 30 | 30 | 0 | [[1023, 1292]] | 1.0 | 4ibm | Homo sapiens | TYR_INSR_HUMAN | TYR | 1.3e-96 | 328.8 | 1.0 | 260.0 | 260.0 | 1176 | 1177 | 1178 | 1180 | 1182 | 1057 | 1074 | 1078 | 1156 | 1158 | 1157 | 1159.0 | 1218 | 1206 | 1201 | 1200 | 1199 | 1198 | 1197 | 1196 | 1195 | 1104 | Insulin receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|