| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4F64A | P11362 | 464 | 762 | 822.0 | 0S8:801 | Type1 | Inactive | DFGin | 5.1832 | 13.1182 | BLAplus | -126.63, 159.8 | 67.66, 19.43 | -73.38, -15.37 | 61.14, 82.05 | -112.05, 14.31 | in-in | in | 7.8334 | Saltbr-in | 2.6567 | HRD-in | -75.01, -53.26 | 79.37, -13.8 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8889 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -105.36, 162.32 | APE9-dihe-in | -110.59, 112.62 | APE8-dihe-out | -54.21, -21.82 | APE8-rot-na | 334.94 | APE67-dihe-in | -73.68, -4.51 | -58.01, -22.74 | APE12-dist-na | 19.9252 | APE11-dist-na | 21.6236 | APE10-dist-na | 19.6065 | APE9-dist-out | 11.7397 | C488A,C584S | None | None | XRAY | 2.05 | 0.217 | 0.269 | A | 309.0 | 278.0 | 21 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 4f64 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4F64B | P11362 | 461 | 761 | 822.0 | 0S8:801 | Type1 | Inactive | DFGin | 5.1666 | 12.9047 | BLAplus | -128.73, 164.19 | 64.4, 29.6 | -84.21, -15.05 | 59.33, 82.94 | -106.3, 1.28 | in-in | in | 7.8942 | Saltbr-in | 2.8638 | HRD-in | -73.33, -50.22 | 71.98, 0.27 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -113.2, 170.72 | APE9-dihe-in | -106.18, 108.15 | APE8-dihe-out | -52.36, -27.43 | APE8-rot-na | 328.0 | APE67-dihe-in | -80.92, -6.4 | -55.61, -16.72 | APE12-dist-na | 999.0 | APE11-dist-na | 20.9952 | APE10-dist-na | 19.8534 | APE9-dist-out | 11.5563 | C488A,C584S | None | None | XRAY | 2.05 | 0.217 | 0.269 | B | 309.0 | 272.0 | 29 | 30 | 21 | 9 | [[478, 756]] | 1.0 | 4f64 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4F64A | P11362 | 464 | 762 | 822.0 | 0S8:801 | Type1 | Inactive | DFGin | 5.1832 | 13.1182 | BLAplus | -126.63, 159.8 | 67.66, 19.43 | -73.38, -15.37 | 61.14, 82.05 | -112.05, 14.31 | in-in | in | 7.8334 | Saltbr-in | 2.6567 | HRD-in | -75.01, -53.26 | 79.37, -13.8 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.8889 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -105.36, 162.32 | APE9-dihe-in | -110.59, 112.62 | APE8-dihe-out | -54.21, -21.82 | APE8-rot-na | 334.94 | APE67-dihe-in | -73.68, -4.51 | -58.01, -22.74 | APE12-dist-na | 19.9252 | APE11-dist-na | 21.6236 | APE10-dist-na | 19.6065 | APE9-dist-out | 11.7397 | C488A,C584S | None | None | XRAY | 2.05 | 0.217 | 0.269 | A | 309.0 | 278.0 | 21 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 4f64 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4F64B | P11362 | 461 | 761 | 822.0 | 0S8:801 | Type1 | Inactive | DFGin | 5.1666 | 12.9047 | BLAplus | -128.73, 164.19 | 64.4, 29.6 | -84.21, -15.05 | 59.33, 82.94 | -106.3, 1.28 | in-in | in | 7.8942 | Saltbr-in | 2.8638 | HRD-in | -73.33, -50.22 | 71.98, 0.27 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -113.2, 170.72 | APE9-dihe-in | -106.18, 108.15 | APE8-dihe-out | -52.36, -27.43 | APE8-rot-na | 328.0 | APE67-dihe-in | -80.92, -6.4 | -55.61, -16.72 | APE12-dist-na | 999.0 | APE11-dist-na | 20.9952 | APE10-dist-na | 19.8534 | APE9-dist-out | 11.5563 | C488A,C584S | None | None | XRAY | 2.05 | 0.217 | 0.269 | B | 309.0 | 272.0 | 29 | 30 | 21 | 9 | [[478, 756]] | 1.0 | 4f64 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|