| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 3RI1B | P21802 | 468 | 766 | 821.0 | 3RH:1 | Type1 | Inactive | DFGin | 6.6686 | 14.1679 | BLAminus | -125.05, -168.18 | 44.8, 79.48 | -91.34, 24.45 | 292.18, 85.49 | -61.68, -38.04 | in-in | in | 7.681 | Saltbr-in | 2.7144 | HRD-in | -78.4, -46.06 | 72.66, -13.3 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9368 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.45, 15.65 | APE9-dihe-in | -96.94, 132.02 | APE8-dihe-in | -54.97, 122.14 | APE8-rot-na | 331.98 | APE67-dihe-in | -73.55, -6.33 | -62.74, -38.58 | APE12-dist-na | 10.0228 | APE11-dist-na | 10.8403 | APE10-dist-na | 7.241 | APE9-dist-in | 5.0053 | None | None | None | XRAY | 2.1 | 0.216 | 0.247 | B | 313.0 | 283.0 | 16 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 3ri1 | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 3RI1A | P21802 | 468 | 765 | 821.0 | 3RH:2 | Type1.5_Back | Inactive | DFGin | 6.8318 | 14.1702 | BLAminus | -123.23, -170.67 | 54.24, 75.33 | -95.71, 30.48 | 294.51, 86.16 | -72.01, -31.85 | in-in | in | 7.7565 | Saltbr-in | 2.712 | HRD-in | -81.62, -48.44 | 74.58, -5.16 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9412 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.86, 17.26 | APE9-dihe-in | -94.17, 130.86 | APE8-dihe-in | -56.98, 120.47 | APE8-rot-na | 333.82 | APE67-dihe-in | -73.48, -11.98 | -59.18, -36.04 | APE12-dist-na | 9.865 | APE11-dist-na | 10.7096 | APE10-dist-na | 7.3823 | APE9-dist-in | 4.8421 | None | None | None | XRAY | 2.1 | 0.216 | 0.247 | A | 313.0 | 285.0 | 13 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 3ri1 | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 3RI1B | P21802 | 468 | 766 | 821.0 | 3RH:1 | Type1 | Inactive | DFGin | 6.6686 | 14.1679 | BLAminus | -125.05, -168.18 | 44.8, 79.48 | -91.34, 24.45 | 292.18, 85.49 | -61.68, -38.04 | in-in | in | 7.681 | Saltbr-in | 2.7144 | HRD-in | -78.4, -46.06 | 72.66, -13.3 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9368 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -103.45, 15.65 | APE9-dihe-in | -96.94, 132.02 | APE8-dihe-in | -54.97, 122.14 | APE8-rot-na | 331.98 | APE67-dihe-in | -73.55, -6.33 | -62.74, -38.58 | APE12-dist-na | 10.0228 | APE11-dist-na | 10.8403 | APE10-dist-na | 7.241 | APE9-dist-in | 5.0053 | None | None | None | XRAY | 2.1 | 0.216 | 0.247 | B | 313.0 | 283.0 | 16 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 3ri1 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 3RI1A | P21802 | 468 | 765 | 821.0 | 3RH:2 | Type1.5_Back | Inactive | DFGin | 6.8318 | 14.1702 | BLAminus | -123.23, -170.67 | 54.24, 75.33 | -95.71, 30.48 | 294.51, 86.16 | -72.01, -31.85 | in-in | in | 7.7565 | Saltbr-in | 2.712 | HRD-in | -81.62, -48.44 | 74.58, -5.16 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9412 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -106.86, 17.26 | APE9-dihe-in | -94.17, 130.86 | APE8-dihe-in | -56.98, 120.47 | APE8-rot-na | 333.82 | APE67-dihe-in | -73.48, -11.98 | -59.18, -36.04 | APE12-dist-na | 9.865 | APE11-dist-na | 10.7096 | APE10-dist-na | 7.3823 | APE9-dist-in | 4.8421 | None | None | None | XRAY | 2.1 | 0.216 | 0.247 | A | 313.0 | 285.0 | 13 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 3ri1 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.5e-104 | 354.1 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|