| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WB | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | None | DFGin | 6.749 | 14.2708 | BLAminus | -132.31, -176.87 | 65.1, 94.3 | -111.58, 28.46 | 301.82, 101.23 | -75.68, -15.25 | out-none | out | 12.8234 | Saltbr-none | 999.0 | HRD-in | -62.32, -42.81 | 74.92, -23.29 | none-in-none | SNCnin | in-none | ActLoopNT-in | 3.0593 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -68.9, -14.83 | 999.0, -25.18 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | B | 443.0 | 382.0 | 28 | 27 | 22 | 5 | [[220, 486]] | 1.0 | 3i6w | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WD | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | None | DFGin | 7.1208 | 14.4732 | BLAminus | -130.43, -175.81 | 63.91, 79.02 | -93.96, 27.08 | 301.9, 101.65 | -74.68, -15.75 | out-none | out | 12.8406 | Saltbr-none | 999.0 | HRD-in | -63.78, -41.36 | 74.21, -23.95 | none-in-none | SNCnin | in-none | ActLoopNT-in | 2.8167 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -68.71, -15.0 | 999.0, -25.14 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | D | 443.0 | 382.0 | 28 | 27 | 22 | 5 | [[220, 486]] | 1.0 | 3i6w | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WF | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | None | DFGin | 7.0122 | 14.1916 | BLAminus | -131.41, -176.41 | 64.86, 90.78 | -109.15, 26.06 | 302.9, 101.84 | -74.04, -16.03 | out-none | out | 12.8713 | Saltbr-none | 999.0 | HRD-in | -63.34, -41.92 | 73.76, -23.06 | none-in-none | SNCnin | in-none | ActLoopNT-in | 2.9844 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -68.91, -15.1 | 999.0, -24.96 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | F | 443.0 | 382.0 | 28 | 27 | 22 | 5 | [[220, 486]] | 1.0 | 3i6w | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WH | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | None | DFGin | 6.8741 | 14.2536 | BLAminus | -131.53, -176.78 | 65.02, 88.11 | -104.7, 27.13 | 303.5, 101.73 | -74.81, -16.38 | out-none | out | 12.8827 | Saltbr-none | 999.0 | HRD-in | -62.35, -41.54 | 74.34, -23.8 | none-in-none | SNCnin | in-none | ActLoopNT-in | 3.0871 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -69.26, -15.11 | 999.0, -24.78 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | H | 443.0 | 382.0 | 28 | 27 | 22 | 5 | [[220, 486]] | 1.0 | 3i6w | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WA | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | Inactive | DFGin | 7.3486 | 13.5162 | None | -131.02, -176.1 | 64.38, 89.31 | -97.7, 999.0 | 302.36, 133.8 | 999.0, 999.0 | out-none | out | 13.0764 | Saltbr-none | 999.0 | HRD-in | -64.4, -41.66 | 75.43, -23.93 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -53.49, -47.48 | 999.0, -37.14 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | A | 443.0 | 369.0 | 41 | 27 | 9 | 18 | [[220, 486]] | 1.0 | 3i6w | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WC | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | Inactive | DFGin | 7.5775 | 13.998 | None | -131.8, -178.23 | 63.57, 98.9 | -117.45, 999.0 | 335.54, 98.66 | 999.0, 999.0 | out-none | out | 13.0805 | Saltbr-none | 999.0 | HRD-in | -63.6, -43.12 | 77.0, -24.17 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -53.04, -46.8 | 999.0, -37.07 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | C | 443.0 | 368.0 | 42 | 27 | 9 | 18 | [[220, 486]] | 1.0 | 3i6w | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WE | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | Inactive | DFGin | 7.5459 | 13.6974 | None | -130.93, -177.05 | 65.38, 105.03 | -130.22, 999.0 | 325.6, 106.63 | 999.0, 999.0 | out-none | out | 13.0915 | Saltbr-none | 999.0 | HRD-in | -61.69, -42.13 | 73.77, -23.14 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -53.57, -46.22 | 999.0, -36.71 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | E | 443.0 | 368.0 | 42 | 27 | 9 | 18 | [[220, 486]] | 1.0 | 3i6w | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WG | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | Inactive | DFGin | 7.5136 | 13.8031 | None | -131.95, -176.65 | 65.29, 79.69 | -111.56, 999.0 | 332.1, 109.83 | 999.0, 999.0 | out-none | out | 13.0784 | Saltbr-none | 999.0 | HRD-in | -62.8, -42.52 | 74.63, -23.4 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -53.54, -46.24 | 999.0, -36.98 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | G | 443.0 | 369.0 | 41 | 27 | 9 | 18 | [[220, 486]] | 1.0 | 3i6w | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WB | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | None | DFGin | 6.749 | 14.2708 | BLAminus | -132.31, -176.87 | 65.1, 94.3 | -111.58, 28.46 | 301.82, 101.23 | -75.68, -15.25 | out-none | out | 12.8234 | Saltbr-none | 999.0 | HRD-in | -62.32, -42.81 | 74.92, -23.29 | none-in-none | SNCnin | in-none | ActLoopNT-in | 3.0593 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -68.9, -14.83 | 999.0, -25.18 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | B | 443.0 | 382.0 | 28 | 27 | 22 | 5 | [[220, 486]] | 1.0 | 3i6w | Homo sapiens | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WD | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | None | DFGin | 7.1208 | 14.4732 | BLAminus | -130.43, -175.81 | 63.91, 79.02 | -93.96, 27.08 | 301.9, 101.65 | -74.68, -15.75 | out-none | out | 12.8406 | Saltbr-none | 999.0 | HRD-in | -63.78, -41.36 | 74.21, -23.95 | none-in-none | SNCnin | in-none | ActLoopNT-in | 2.8167 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -68.71, -15.0 | 999.0, -25.14 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | D | 443.0 | 382.0 | 28 | 27 | 22 | 5 | [[220, 486]] | 1.0 | 3i6w | Homo sapiens | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WF | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | None | DFGin | 7.0122 | 14.1916 | BLAminus | -131.41, -176.41 | 64.86, 90.78 | -109.15, 26.06 | 302.9, 101.84 | -74.04, -16.03 | out-none | out | 12.8713 | Saltbr-none | 999.0 | HRD-in | -63.34, -41.92 | 73.76, -23.06 | none-in-none | SNCnin | in-none | ActLoopNT-in | 2.9844 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -68.91, -15.1 | 999.0, -24.96 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | F | 443.0 | 382.0 | 28 | 27 | 22 | 5 | [[220, 486]] | 1.0 | 3i6w | Homo sapiens | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WH | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | None | DFGin | 6.8741 | 14.2536 | BLAminus | -131.53, -176.78 | 65.02, 88.11 | -104.7, 27.13 | 303.5, 101.73 | -74.81, -16.38 | out-none | out | 12.8827 | Saltbr-none | 999.0 | HRD-in | -62.35, -41.54 | 74.34, -23.8 | none-in-none | SNCnin | in-none | ActLoopNT-in | 3.0871 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -69.26, -15.11 | 999.0, -24.78 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | H | 443.0 | 382.0 | 28 | 27 | 22 | 5 | [[220, 486]] | 1.0 | 3i6w | Homo sapiens | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WA | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | Inactive | DFGin | 7.3486 | 13.5162 | None | -131.02, -176.1 | 64.38, 89.31 | -97.7, 999.0 | 302.36, 133.8 | 999.0, 999.0 | out-none | out | 13.0764 | Saltbr-none | 999.0 | HRD-in | -64.4, -41.66 | 75.43, -23.93 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -53.49, -47.48 | 999.0, -37.14 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | A | 443.0 | 369.0 | 41 | 27 | 9 | 18 | [[220, 486]] | 1.0 | 3i6w | Homo sapiens | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WC | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | Inactive | DFGin | 7.5775 | 13.998 | None | -131.8, -178.23 | 63.57, 98.9 | -117.45, 999.0 | 335.54, 98.66 | 999.0, 999.0 | out-none | out | 13.0805 | Saltbr-none | 999.0 | HRD-in | -63.6, -43.12 | 77.0, -24.17 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -53.04, -46.8 | 999.0, -37.07 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | C | 443.0 | 368.0 | 42 | 27 | 9 | 18 | [[220, 486]] | 1.0 | 3i6w | Homo sapiens | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WE | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | Inactive | DFGin | 7.5459 | 13.6974 | None | -130.93, -177.05 | 65.38, 105.03 | -130.22, 999.0 | 325.6, 106.63 | 999.0, 999.0 | out-none | out | 13.0915 | Saltbr-none | 999.0 | HRD-in | -61.69, -42.13 | 73.77, -23.14 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -53.57, -46.22 | 999.0, -36.71 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | E | 443.0 | 368.0 | 42 | 27 | 9 | 18 | [[220, 486]] | 1.0 | 3i6w | Homo sapiens | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| CAMK | CHEK2 | CHK2_HUMAN | 3I6WG | O96017 | 92 | 501 | 543.0 | No_ligand | No_ligand | Inactive | DFGin | 7.5136 | 13.8031 | None | -131.95, -176.65 | 65.29, 79.69 | -111.56, 999.0 | 332.1, 109.83 | 999.0, 999.0 | out-none | out | 13.0784 | Saltbr-none | 999.0 | HRD-in | -62.8, -42.52 | 74.63, -23.4 | none-none-none | SNCnnn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | nonTYR | APEdihe_aannn | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 999.0 | APE8-rot-none | 999.0 | APE67-dihe-none | -53.54, -46.24 | 999.0, -36.98 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | K249R | None | None | XRAY | 3.25 | 0.252 | 0.287 | G | 443.0 | 369.0 | 41 | 27 | 9 | 18 | [[220, 486]] | 1.0 | 3i6w | Homo sapiens | CAMK_CHEK2_HUMAN | CAMK | 7.4e-84 | 287.1 | 1.0 | 256.0 | 256.0 | 367 | 368 | 369 | 371 | 373 | 249 | 273 | 277 | 344 | 346 | 345 | 347.0 | 409 | 394 | 389 | 388 | 387 | 386 | 385 | 384 | 383 | 302 | Serine/threonine-protein kinase Chk2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|