| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 3C4FA | P11362 | 464 | 765 | 822.0 | C4F:1 | Type1.5_Back | Inactive | DFGin | 5.1138 | 13.3182 | BLAplus | -110.44, 159.78 | 58.59, 34.58 | -81.02, -11.31 | 51.22, 81.2 | -119.48, 23.64 | in-out | in | 7.8662 | Saltbr-out | 4.6321 | HRD-in | -67.82, -57.48 | 84.79, -17.47 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.0691 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.31, 173.6 | APE9-dihe-in | -111.71, 110.92 | APE8-dihe-out | -49.57, -28.9 | APE8-rot-na | 335.93 | APE67-dihe-in | -76.49, -6.67 | -57.78, -16.15 | APE12-dist-na | 19.2924 | APE11-dist-na | 21.1206 | APE10-dist-na | 19.3954 | APE9-dist-out | 11.7567 | C488A | None | None | XRAY | 2.07 | 0.213 | 0.264 | A | 302.0 | 290.0 | 12 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 3c4f | TYR_FGFR1_HUMAN | TYR | 1.3e-104 | 355.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 3C4FB | P11362 | 464 | 765 | 822.0 | C4F:2 | Type1.5_Back | Inactive | DFGin | 5.1863 | 13.0956 | BLAplus | -113.87, 161.2 | 54.21, 44.76 | -88.95, -14.38 | 49.14, 89.01 | -114.94, 24.21 | in-in | in | 7.8308 | Saltbr-in | 3.2478 | HRD-in | -69.91, -54.09 | 86.4, -33.67 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.9335 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -106.54, 164.12 | APE9-dihe-in | -103.97, 111.75 | APE8-dihe-out | -49.46, -30.24 | APE8-rot-na | 330.07 | APE67-dihe-in | -74.8, -7.14 | -56.82, -17.81 | APE12-dist-na | 19.3702 | APE11-dist-na | 21.2959 | APE10-dist-na | 19.6706 | APE9-dist-out | 11.6434 | C488A | None | None | XRAY | 2.07 | 0.213 | 0.264 | B | 302.0 | 290.0 | 12 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 3c4f | TYR_FGFR1_HUMAN | TYR | 1.3e-104 | 355.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 3C4FA | P11362 | 464 | 765 | 822.0 | C4F:1 | Type1.5_Back | Inactive | DFGin | 5.1138 | 13.3182 | BLAplus | -110.44, 159.78 | 58.59, 34.58 | -81.02, -11.31 | 51.22, 81.2 | -119.48, 23.64 | in-out | in | 7.8662 | Saltbr-out | 4.6321 | HRD-in | -67.82, -57.48 | 84.79, -17.47 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.0691 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.31, 173.6 | APE9-dihe-in | -111.71, 110.92 | APE8-dihe-out | -49.57, -28.9 | APE8-rot-na | 335.93 | APE67-dihe-in | -76.49, -6.67 | -57.78, -16.15 | APE12-dist-na | 19.2924 | APE11-dist-na | 21.1206 | APE10-dist-na | 19.3954 | APE9-dist-out | 11.7567 | C488A | None | None | XRAY | 2.07 | 0.213 | 0.264 | A | 302.0 | 290.0 | 12 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 3c4f | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.3e-104 | 355.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 3C4FB | P11362 | 464 | 765 | 822.0 | C4F:2 | Type1.5_Back | Inactive | DFGin | 5.1863 | 13.0956 | BLAplus | -113.87, 161.2 | 54.21, 44.76 | -88.95, -14.38 | 49.14, 89.01 | -114.94, 24.21 | in-in | in | 7.8308 | Saltbr-in | 3.2478 | HRD-in | -69.91, -54.09 | 86.4, -33.67 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.9335 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -106.54, 164.12 | APE9-dihe-in | -103.97, 111.75 | APE8-dihe-out | -49.46, -30.24 | APE8-rot-na | 330.07 | APE67-dihe-in | -74.8, -7.14 | -56.82, -17.81 | APE12-dist-na | 19.3702 | APE11-dist-na | 21.2959 | APE10-dist-na | 19.6706 | APE9-dist-out | 11.6434 | C488A | None | None | XRAY | 2.07 | 0.213 | 0.264 | B | 302.0 | 290.0 | 12 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 3c4f | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.3e-104 | 355.0 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|