| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CK1 | VRK2 | VRK2_HUMAN | 2V62A | Q86Y07 | 15 | 330 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.5216 | 14.2783 | BLAminus | -126.42, 177.81 | 61.4, 82.15 | -97.89, 25.94 | 290.77, 86.68 | -60.53, -27.7 | in-in | in | 7.4688 | Saltbr-in | 2.6513 | HRD-in | -85.44, -49.42 | 78.82, -6.43 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -77.49, 164.36 | APE9-dihe-na | 100.65, -175.4 | APE8-dihe-in | -81.64, 115.53 | APE8-rot-in | 300.97 | APE67-dihe-in | -58.37, -37.59 | -55.92, -37.43 | APE12-dist-in | 13.8351 | APE11-dist-in | 13.7728 | APE10-dist-in | 7.9511 | APE9-dist-in | 4.5825 | None | None | None | XRAY | 1.7 | 0.203 | 0.236 | A | 345.0 | 309.0 | 7 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 2v62 | CK1_VRK2_HUMAN | CK1 | 2e-103 | 351.3 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| CK1 | VRK2 | VRK2_HUMAN | 2V62B | Q86Y07 | 15 | 330 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.6633 | 14.235 | BLAminus | -125.07, 178.48 | 58.38, 82.78 | -95.02, 25.08 | 292.21, 85.61 | -65.49, -19.52 | in-in | in | 7.4809 | Saltbr-in | 3.1122 | HRD-in | -84.77, -51.43 | 82.43, -6.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8814 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -78.49, 164.48 | APE9-dihe-na | 105.42, -177.12 | APE8-dihe-in | -82.14, 116.45 | APE8-rot-in | 302.32 | APE67-dihe-in | -58.69, -38.25 | -56.97, -36.01 | APE12-dist-in | 13.7404 | APE11-dist-in | 13.6627 | APE10-dist-in | 7.977 | APE9-dist-in | 4.6212 | None | None | None | XRAY | 1.7 | 0.203 | 0.236 | B | 345.0 | 310.0 | 6 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 2v62 | CK1_VRK2_HUMAN | CK1 | 2e-103 | 351.3 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CK1 | VRK2 | VRK2_HUMAN | 2V62A | Q86Y07 | 15 | 330 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.5216 | 14.2783 | BLAminus | -126.42, 177.81 | 61.4, 82.15 | -97.89, 25.94 | 290.77, 86.68 | -60.53, -27.7 | in-in | in | 7.4688 | Saltbr-in | 2.6513 | HRD-in | -85.44, -49.42 | 78.82, -6.43 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -77.49, 164.36 | APE9-dihe-na | 100.65, -175.4 | APE8-dihe-in | -81.64, 115.53 | APE8-rot-in | 300.97 | APE67-dihe-in | -58.37, -37.59 | -55.92, -37.43 | APE12-dist-in | 13.8351 | APE11-dist-in | 13.7728 | APE10-dist-in | 7.9511 | APE9-dist-in | 4.5825 | None | None | None | XRAY | 1.7 | 0.203 | 0.236 | A | 345.0 | 309.0 | 7 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 2v62 | Homo sapiens | CK1_VRK2_HUMAN | CK1 | 2e-103 | 351.3 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| CK1 | VRK2 | VRK2_HUMAN | 2V62B | Q86Y07 | 15 | 330 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.6633 | 14.235 | BLAminus | -125.07, 178.48 | 58.38, 82.78 | -95.02, 25.08 | 292.21, 85.61 | -65.49, -19.52 | in-in | in | 7.4809 | Saltbr-in | 3.1122 | HRD-in | -84.77, -51.43 | 82.43, -6.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8814 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -78.49, 164.48 | APE9-dihe-na | 105.42, -177.12 | APE8-dihe-in | -82.14, 116.45 | APE8-rot-in | 302.32 | APE67-dihe-in | -58.69, -38.25 | -56.97, -36.01 | APE12-dist-in | 13.7404 | APE11-dist-in | 13.6627 | APE10-dist-in | 7.977 | APE9-dist-in | 4.6212 | None | None | None | XRAY | 1.7 | 0.203 | 0.236 | B | 345.0 | 310.0 | 6 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 2v62 | Homo sapiens | CK1_VRK2_HUMAN | CK1 | 2e-103 | 351.3 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|