| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 2PY3A | P21802 | 468 | 766 | 821.0 | ACP:805 | ATPlike | Inactive | DFGin | 6.3947 | 14.1248 | BLAminus | -132.09, -167.28 | 46.92, 77.9 | -89.52, 28.18 | 287.97, 74.42 | -64.92, -12.84 | in-in | in | 7.2777 | Saltbr-in | 2.6425 | HRD-in | -69.15, -50.28 | 73.37, -7.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9371 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.57, 22.43 | APE9-dihe-in | -99.04, 131.25 | APE8-dihe-in | -52.37, 122.48 | APE8-rot-na | 325.05 | APE67-dihe-in | -72.14, -6.33 | -51.92, -40.9 | APE12-dist-na | 9.9501 | APE11-dist-na | 10.6713 | APE10-dist-na | 7.3862 | APE9-dist-in | 4.7437 | C491A,E565G | None | None | XRAY | 2.3 | 0.217 | 0.252 | A | 324.0 | 282.0 | 17 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2py3 | TYR_FGFR2_HUMAN | TYR | 2.7e-103 | 350.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PY3B | P21802 | 468 | 766 | 821.0 | ACP:805 | ATPlike | Inactive | DFGin | 6.5146 | 14.301 | BLAminus | -135.62, -170.09 | 51.9, 73.7 | -89.2, 28.31 | 287.78, 75.56 | -66.05, -13.03 | in-in | in | 7.4251 | Saltbr-in | 2.7042 | HRD-in | -75.46, -47.46 | 71.33, -10.27 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8572 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.61, 23.33 | APE9-dihe-in | -100.25, 127.63 | APE8-dihe-in | -52.55, 116.2 | APE8-rot-na | 325.69 | APE67-dihe-in | -68.53, -13.02 | -47.88, -42.42 | APE12-dist-na | 10.0658 | APE11-dist-na | 10.7884 | APE10-dist-na | 7.4188 | APE9-dist-in | 4.9315 | C491A,E565G | None | None | XRAY | 2.3 | 0.217 | 0.252 | B | 324.0 | 284.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2py3 | TYR_FGFR2_HUMAN | TYR | 2.7e-103 | 350.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR2 | FGFR2_HUMAN | 2PY3A | P21802 | 468 | 766 | 821.0 | ACP:805 | ATPlike | Inactive | DFGin | 6.3947 | 14.1248 | BLAminus | -132.09, -167.28 | 46.92, 77.9 | -89.52, 28.18 | 287.97, 74.42 | -64.92, -12.84 | in-in | in | 7.2777 | Saltbr-in | 2.6425 | HRD-in | -69.15, -50.28 | 73.37, -7.92 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9371 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -113.57, 22.43 | APE9-dihe-in | -99.04, 131.25 | APE8-dihe-in | -52.37, 122.48 | APE8-rot-na | 325.05 | APE67-dihe-in | -72.14, -6.33 | -51.92, -40.9 | APE12-dist-na | 9.9501 | APE11-dist-na | 10.6713 | APE10-dist-na | 7.3862 | APE9-dist-in | 4.7437 | C491A,E565G | None | None | XRAY | 2.3 | 0.217 | 0.252 | A | 324.0 | 282.0 | 17 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2py3 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.7e-103 | 350.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| TYR | FGFR2 | FGFR2_HUMAN | 2PY3B | P21802 | 468 | 766 | 821.0 | ACP:805 | ATPlike | Inactive | DFGin | 6.5146 | 14.301 | BLAminus | -135.62, -170.09 | 51.9, 73.7 | -89.2, 28.31 | 287.78, 75.56 | -66.05, -13.03 | in-in | in | 7.4251 | Saltbr-in | 2.7042 | HRD-in | -75.46, -47.46 | 71.33, -10.27 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8572 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | -110.61, 23.33 | APE9-dihe-in | -100.25, 127.63 | APE8-dihe-in | -52.55, 116.2 | APE8-rot-na | 325.69 | APE67-dihe-in | -68.53, -13.02 | -47.88, -42.42 | APE12-dist-na | 10.0658 | APE11-dist-na | 10.7884 | APE10-dist-na | 7.4188 | APE9-dist-in | 4.9315 | C491A,E565G | None | None | XRAY | 2.3 | 0.217 | 0.252 | B | 324.0 | 284.0 | 15 | 30 | 30 | 0 | [[481, 759]] | 1.0 | 2py3 | Homo sapiens | TYR_FGFR2_HUMAN | TYR | 2.7e-103 | 350.7 | 1.0 | 260.0 | 260.0 | 643 | 644 | 645 | 647 | 649 | 517 | 534 | 538 | 623 | 625 | 624 | 626.0 | 685 | 673 | 668 | 667 | 666 | 665 | 664 | 663 | 662 | 565 | Fibroblast growth factor receptor 2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|