| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | IGF1R | IGF1R_HUMAN | 1P4OA | P08069 | 978 | 1285 | 1367.0 | No_ligand | No_ligand | Inactive | DFGinter | 8.9365 | 7.4526 | None | -75.61, 161.81 | -88.19, 167.58 | -62.75, 158.69 | 79.74, 92.2 | 58.69, 28.18 | in-out | in | 9.6686 | Saltbr-out | 8.1614 | HRD-in | -85.36, -54.81 | 81.1, -18.95 | out-out-in | SNCooi | out-in | ActLoopNT-out | 17.8144 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -75.47, 124.06 | APE9-dihe-in | -124.38, 139.88 | APE8-dihe-in | -82.49, 64.57 | APE8-rot-na | 36.92 | APE67-dihe-in | -73.19, -6.91 | -50.14, -35.0 | APE12-dist-na | 22.2752 | APE11-dist-na | 18.248 | APE10-dist-na | 14.5409 | APE9-dist-in | 7.2736 | E1097A,E1099A | None | None | XRAY | 1.5 | 0.209 | 0.236 | A | 322.0 | 308.0 | 0 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 1p4o | TYR_IGF1R_HUMAN | TYR | 2.3e-95 | 324.8 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 1P4OB | P08069 | 977 | 1290 | 1367.0 | No_ligand | No_ligand | Inactive | DFGinter | 8.9729 | 7.3732 | None | -74.95, 163.69 | -90.41, 168.58 | -63.57, 158.6 | 80.11, 88.87 | 59.26, 26.84 | in-out | in | 9.7118 | Saltbr-out | 8.1343 | HRD-in | -85.93, -55.48 | 81.68, -17.46 | out-out-in | SNCooi | out-in | ActLoopNT-out | 17.8706 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -71.53, 126.34 | APE9-dihe-in | -129.41, 143.63 | APE8-dihe-in | -82.98, 67.29 | APE8-rot-na | 36.94 | APE67-dihe-in | -73.89, -4.17 | -52.36, -34.34 | APE12-dist-na | 22.4577 | APE11-dist-na | 18.39 | APE10-dist-na | 14.6946 | APE9-dist-in | 7.1712 | E1097A,E1099A | None | None | XRAY | 1.5 | 0.209 | 0.236 | B | 322.0 | 314.0 | 0 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 1p4o | TYR_IGF1R_HUMAN | TYR | 2.3e-95 | 324.8 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | IGF1R | IGF1R_HUMAN | 1P4OA | P08069 | 978 | 1285 | 1367.0 | No_ligand | No_ligand | Inactive | DFGinter | 8.9365 | 7.4526 | None | -75.61, 161.81 | -88.19, 167.58 | -62.75, 158.69 | 79.74, 92.2 | 58.69, 28.18 | in-out | in | 9.6686 | Saltbr-out | 8.1614 | HRD-in | -85.36, -54.81 | 81.1, -18.95 | out-out-in | SNCooi | out-in | ActLoopNT-out | 17.8144 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -75.47, 124.06 | APE9-dihe-in | -124.38, 139.88 | APE8-dihe-in | -82.49, 64.57 | APE8-rot-na | 36.92 | APE67-dihe-in | -73.19, -6.91 | -50.14, -35.0 | APE12-dist-na | 22.2752 | APE11-dist-na | 18.248 | APE10-dist-na | 14.5409 | APE9-dist-in | 7.2736 | E1097A,E1099A | None | None | XRAY | 1.5 | 0.209 | 0.236 | A | 322.0 | 308.0 | 0 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 1p4o | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 2.3e-95 | 324.8 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 1P4OB | P08069 | 977 | 1290 | 1367.0 | No_ligand | No_ligand | Inactive | DFGinter | 8.9729 | 7.3732 | None | -74.95, 163.69 | -90.41, 168.58 | -63.57, 158.6 | 80.11, 88.87 | 59.26, 26.84 | in-out | in | 9.7118 | Saltbr-out | 8.1343 | HRD-in | -85.93, -55.48 | 81.68, -17.46 | out-out-in | SNCooi | out-in | ActLoopNT-out | 17.8706 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -71.53, 126.34 | APE9-dihe-in | -129.41, 143.63 | APE8-dihe-in | -82.98, 67.29 | APE8-rot-na | 36.94 | APE67-dihe-in | -73.89, -4.17 | -52.36, -34.34 | APE12-dist-na | 22.4577 | APE11-dist-na | 18.39 | APE10-dist-na | 14.6946 | APE9-dist-in | 7.1712 | E1097A,E1099A | None | None | XRAY | 1.5 | 0.209 | 0.236 | B | 322.0 | 314.0 | 0 | 30 | 30 | 0 | [[999, 1268]] | 1.0 | 1p4o | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 2.3e-95 | 324.8 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|