| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | IGF1R | IGF1R_HUMAN | 1JQHA | P08069 | 984 | 1286 | 1367.0 | ANP:301 | ATPlike | Inactive | DFGin | 5.6898 | 16.5691 | None | -66.7, 163.88 | -59.45, 151.32 | -140.18, 178.07 | 43.94, 89.38 | -106.76, 173.06 | in-out | in | 9.9768 | Saltbr-out | 6.0561 | HRD-in | -50.88, -56.96 | 74.77, -3.78 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -84.24, 106.81 | APE9-dihe-in | -58.88, 134.76 | APE8-dihe-in | -78.96, 121.64 | APE8-rot-na | 37.96 | APE67-dihe-in | -60.45, -7.73 | -52.46, -43.95 | APE12-dist-na | 7.1567 | APE11-dist-na | 11.2997 | APE10-dist-na | 15.5969 | APE9-dist-in | 5.8 | E979G,Y980S | None | None | XRAY | 2.1 | 0.195 | 0.219 | A | 308.0 | 291.0 | 12 | 30 | 23 | 7 | [[999, 1268]] | 1.0 | 1jqh | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 1JQHB | P08069 | 984 | 1286 | 1367.0 | ANP:302 | ATPlike | Inactive | DFGin | 5.6866 | 16.5538 | None | -65.78, 164.4 | -59.98, 151.89 | -140.81, 178.2 | 43.68, 89.42 | -109.69, -174.77 | in-out | in | 9.9884 | Saltbr-out | 6.0195 | HRD-in | -51.69, -56.66 | 74.32, -2.97 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -83.6, 107.67 | APE9-dihe-in | -58.75, 135.36 | APE8-dihe-in | -79.54, 122.52 | APE8-rot-na | 37.69 | APE67-dihe-in | -59.25, -7.46 | -52.18, -45.28 | APE12-dist-na | 6.8166 | APE11-dist-na | 10.9316 | APE10-dist-na | 15.2162 | APE9-dist-in | 5.768 | E979G,Y980S | None | None | XRAY | 2.1 | 0.195 | 0.219 | B | 308.0 | 287.0 | 16 | 30 | 23 | 7 | [[999, 1268]] | 1.0 | 1jqh | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 1JQHC | P08069 | 984 | 1286 | 1367.0 | ANP:303 | ATPlike | Inactive | DFGin | 5.6976 | 16.5582 | None | -65.47, 162.73 | -58.75, 151.62 | -140.8, 179.03 | 43.87, 88.98 | -110.24, -177.72 | in-out | in | 9.9987 | Saltbr-out | 6.0347 | HRD-in | -53.2, -57.0 | 74.59, -2.63 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -82.9, 107.89 | APE9-dihe-in | -58.88, 134.76 | APE8-dihe-in | -79.04, 122.75 | APE8-rot-na | 38.27 | APE67-dihe-in | -60.34, -8.42 | -53.61, -43.61 | APE12-dist-na | 6.9265 | APE11-dist-na | 10.9862 | APE10-dist-na | 15.2452 | APE9-dist-in | 5.7735 | E979G,Y980S | None | None | XRAY | 2.1 | 0.195 | 0.219 | C | 308.0 | 291.0 | 12 | 30 | 23 | 7 | [[999, 1268]] | 1.0 | 1jqh | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | IGF1R | IGF1R_HUMAN | 1JQHA | P08069 | 984 | 1286 | 1367.0 | ANP:301 | ATPlike | Inactive | DFGin | 5.6898 | 16.5691 | None | -66.7, 163.88 | -59.45, 151.32 | -140.18, 178.07 | 43.94, 89.38 | -106.76, 173.06 | in-out | in | 9.9768 | Saltbr-out | 6.0561 | HRD-in | -50.88, -56.96 | 74.77, -3.78 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -84.24, 106.81 | APE9-dihe-in | -58.88, 134.76 | APE8-dihe-in | -78.96, 121.64 | APE8-rot-na | 37.96 | APE67-dihe-in | -60.45, -7.73 | -52.46, -43.95 | APE12-dist-na | 7.1567 | APE11-dist-na | 11.2997 | APE10-dist-na | 15.5969 | APE9-dist-in | 5.8 | E979G,Y980S | None | None | XRAY | 2.1 | 0.195 | 0.219 | A | 308.0 | 291.0 | 12 | 30 | 23 | 7 | [[999, 1268]] | 1.0 | 1jqh | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 1JQHB | P08069 | 984 | 1286 | 1367.0 | ANP:302 | ATPlike | Inactive | DFGin | 5.6866 | 16.5538 | None | -65.78, 164.4 | -59.98, 151.89 | -140.81, 178.2 | 43.68, 89.42 | -109.69, -174.77 | in-out | in | 9.9884 | Saltbr-out | 6.0195 | HRD-in | -51.69, -56.66 | 74.32, -2.97 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -83.6, 107.67 | APE9-dihe-in | -58.75, 135.36 | APE8-dihe-in | -79.54, 122.52 | APE8-rot-na | 37.69 | APE67-dihe-in | -59.25, -7.46 | -52.18, -45.28 | APE12-dist-na | 6.8166 | APE11-dist-na | 10.9316 | APE10-dist-na | 15.2162 | APE9-dist-in | 5.768 | E979G,Y980S | None | None | XRAY | 2.1 | 0.195 | 0.219 | B | 308.0 | 287.0 | 16 | 30 | 23 | 7 | [[999, 1268]] | 1.0 | 1jqh | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| TYR | IGF1R | IGF1R_HUMAN | 1JQHC | P08069 | 984 | 1286 | 1367.0 | ANP:303 | ATPlike | Inactive | DFGin | 5.6976 | 16.5582 | None | -65.47, 162.73 | -58.75, 151.62 | -140.8, 179.03 | 43.87, 88.98 | -110.24, -177.72 | in-out | in | 9.9987 | Saltbr-out | 6.0347 | HRD-in | -53.2, -57.0 | 74.59, -2.63 | out-none-in | SNConi | none-in | ActLoopNT-none | 999.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -82.9, 107.89 | APE9-dihe-in | -58.88, 134.76 | APE8-dihe-in | -79.04, 122.75 | APE8-rot-na | 38.27 | APE67-dihe-in | -60.34, -8.42 | -53.61, -43.61 | APE12-dist-na | 6.9265 | APE11-dist-na | 10.9862 | APE10-dist-na | 15.2452 | APE9-dist-in | 5.7735 | E979G,Y980S | None | None | XRAY | 2.1 | 0.195 | 0.219 | C | 308.0 | 291.0 | 12 | 30 | 23 | 7 | [[999, 1268]] | 1.0 | 1jqh | Homo sapiens | TYR_IGF1R_HUMAN | TYR | 1.9e-95 | 325.0 | 1.0 | 260.0 | 260.0 | 1152 | 1153 | 1154 | 1156 | 1158 | 1033 | 1050 | 1054 | 1132 | 1134 | 1133 | 1135.0 | 1194 | 1182 | 1177 | 1176 | 1175 | 1174 | 1173 | 1172 | 1171 | 1080 | Insulin-like growth factor 1 receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|