| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 1FGIA | P11362 | 464 | 762 | 822.0 | SU1:1001 | Type1 | Inactive | DFGin | 5.2448 | 13.0507 | BLAplus | -118.43, 166.43 | 66.52, 8.73 | -64.13, -34.61 | 60.57, 85.04 | -94.1, 14.31 | in-out | in | 7.8098 | Saltbr-out | 4.3938 | HRD-in | -65.25, -56.3 | 86.33, -6.46 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.0188 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.01, 168.11 | APE9-dihe-in | -109.23, 108.22 | APE8-dihe-out | -49.03, -28.53 | APE8-rot-na | 326.13 | APE67-dihe-in | -78.81, -8.46 | -60.3, -12.78 | APE12-dist-na | 19.4008 | APE11-dist-na | 20.9219 | APE10-dist-na | 19.2133 | APE9-dist-out | 11.7398 | C488A | None | None | XRAY | 2.5 | 0.19 | 0.27 | A | 310.0 | 283.0 | 16 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 1fgi | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 1FGIB | P11362 | 461 | 761 | 822.0 | SU1:1000 | Type1 | Inactive | DFGin | 5.0855 | 12.8872 | BLAplus | -129.12, 161.76 | 68.96, 4.34 | -61.61, -28.72 | 62.68, 83.75 | -98.14, 18.47 | in-in | in | 7.9774 | Saltbr-in | 3.237 | HRD-in | -67.23, -42.86 | 65.67, 6.81 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -93.03, 163.6 | APE9-dihe-in | -107.58, 116.43 | APE8-dihe-out | -54.66, -25.86 | APE8-rot-na | 323.83 | APE67-dihe-in | -66.67, -9.45 | -56.63, -25.45 | APE12-dist-na | 999.0 | APE11-dist-na | 21.117 | APE10-dist-na | 19.5572 | APE9-dist-out | 11.7854 | C488A | None | None | XRAY | 2.5 | 0.19 | 0.27 | B | 310.0 | 272.0 | 29 | 30 | 21 | 9 | [[478, 756]] | 1.0 | 1fgi | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 1FGIA | P11362 | 464 | 762 | 822.0 | SU1:1001 | Type1 | Inactive | DFGin | 5.2448 | 13.0507 | BLAplus | -118.43, 166.43 | 66.52, 8.73 | -64.13, -34.61 | 60.57, 85.04 | -94.1, 14.31 | in-out | in | 7.8098 | Saltbr-out | 4.3938 | HRD-in | -65.25, -56.3 | 86.33, -6.46 | out-out-out | SNCooo | out-out | ActLoopNT-out | 9.0188 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.01, 168.11 | APE9-dihe-in | -109.23, 108.22 | APE8-dihe-out | -49.03, -28.53 | APE8-rot-na | 326.13 | APE67-dihe-in | -78.81, -8.46 | -60.3, -12.78 | APE12-dist-na | 19.4008 | APE11-dist-na | 20.9219 | APE10-dist-na | 19.2133 | APE9-dist-out | 11.7398 | C488A | None | None | XRAY | 2.5 | 0.19 | 0.27 | A | 310.0 | 283.0 | 16 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 1fgi | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 1FGIB | P11362 | 461 | 761 | 822.0 | SU1:1000 | Type1 | Inactive | DFGin | 5.0855 | 12.8872 | BLAplus | -129.12, 161.76 | 68.96, 4.34 | -61.61, -28.72 | 62.68, 83.75 | -98.14, 18.47 | in-in | in | 7.9774 | Saltbr-in | 3.237 | HRD-in | -67.23, -42.86 | 65.67, 6.81 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -93.03, 163.6 | APE9-dihe-in | -107.58, 116.43 | APE8-dihe-out | -54.66, -25.86 | APE8-rot-na | 323.83 | APE67-dihe-in | -66.67, -9.45 | -56.63, -25.45 | APE12-dist-na | 999.0 | APE11-dist-na | 21.117 | APE10-dist-na | 19.5572 | APE9-dist-out | 11.7854 | C488A | None | None | XRAY | 2.5 | 0.19 | 0.27 | B | 310.0 | 272.0 | 29 | 30 | 21 | 9 | [[478, 756]] | 1.0 | 1fgi | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|