Ligand: VFS

Total number of chains: 9
Active chains: 0
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 9 100.0% 7JOVC

Hover over column headers for tooltip help.

Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
AGC ROCK1 ROCK1_HUMAN 7JOUA Q13464 9 402 1354.0 VFS:4000 Type1 Inactive DFGin 5.9959 13.3389 BLAminus -143.11, 174.9 56.51, 84.53 -111.27, 42.13 313.94, 101.63 -66.46, -29.86 in-in in 8.5845 Saltbr-in 2.6486 HRD-in -50.19, -37.76 57.05, 15.82 in-in-out SNCiio in-out ActLoopNT-in 3.2049 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -96.97, 107.53 APE9-dihe-na 156.7, 175.62 APE8-dihe-in -79.94, 144.48 APE8-rot-out 53.34 APE67-dihe-in -106.84, -34.67 -68.39, -2.9 APE12-dist-in 11.1521 APE11-dist-in 12.0952 APE10-dist-in 6.1966 APE9-dist-in 3.9409 None None None XRAY 3.318 0.218 0.248 A 413.0 388.0 6 29 29 0 [[76, 338]] 1.0 7jou AGC_ROCK1_HUMAN AGC 3.5e-94 320.7 1.0 260.0 260.0 215 216 217 219 221 105 124 128 195 197 196 198.0 260 244 239 238 237 236 235 234 233 154 Rho-associated protein kinase 1
AGC ROCK2 ROCK2_HUMAN 7JOVA O75116 25 417 1388.0 VFS:502 Type1 Inactive DFGin 6.2465 13.2928 BLAminus -141.83, 172.55 62.54, 72.12 -93.6, 17.75 301.11, 105.91 -60.63, -17.81 in-in in 8.505 Saltbr-in 2.6448 HRD-in -61.37, -48.09 70.0, -5.6 in-in-out SNCiio in-out ActLoopNT-in 3.1039 ActLoopCT-out nonTYR APEdihe_aanoi APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 128.41 APE8-rot-out 35.63 APE67-dihe-in -72.9, -30.33 -60.06, -49.57 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.586 0.185 0.217 A 395.0 377.0 12 29 23 6 [[92, 354]] 1.0 7jov AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVB O75116 23 417 1388.0 VFS:501 Type1 None DFGin 6.2716 13.2483 BLAminus -142.1, 173.55 61.9, 71.69 -93.43, 17.34 301.23, 105.57 -59.73, -16.68 in-in in 8.5286 Saltbr-in 2.6299 HRD-in -62.93, -47.02 69.4, -4.67 in-in-none SNCiin in-none ActLoopNT-in 3.0977 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -66.0, -25.51 999.0, -48.59 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.586 0.185 0.217 B 395.0 378.0 11 29 21 8 [[92, 354]] 1.0 7jov AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVC O75116 23 417 1388.0 VFS:501 Type1 Inactive DFGin 6.2684 13.2283 BLAminus -142.15, 173.25 63.2, 71.86 -94.04, 16.61 301.5, 104.97 -62.04, -13.94 in-in in 8.3763 Saltbr-in 2.7548 HRD-in -63.91, -46.28 70.58, -6.77 in-in-out SNCiio in-out ActLoopNT-in 3.102 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_onno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -148.71 APE8-dihe-in -13.99, 103.33 APE8-rot-out 49.66 APE67-dihe-in -50.5, -34.0 -98.95, 10.78 APE12-dist-out 6.1146 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 9.4434 None None None XRAY 2.586 0.185 0.217 C 395.0 389.0 3 29 27 2 [[92, 354]] 1.0 7jov AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVD O75116 25 417 1388.0 VFS:501 Type1 None DFGin 6.2428 13.3572 BLAminus -142.23, 173.1 61.78, 71.13 -91.99, 20.3 301.3, 105.37 -69.47, 5.8 in-in in 8.6714 Saltbr-in 2.7008 HRD-in -54.87, -50.75 69.64, -5.46 in-in-none SNCiin in-none ActLoopNT-in 3.1806 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, -32.28 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.586 0.185 0.217 D 395.0 361.0 26 29 14 15 [[92, 354]] 1.0 7jov AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVE O75116 23 417 1388.0 VFS:501 Type1 None DFGin 6.2985 13.2567 BLAminus -140.47, 172.73 62.89, 72.53 -94.4, 16.26 301.6, 106.26 -62.28, -16.19 in-in in 8.4545 Saltbr-in 2.7399 HRD-in -64.4, -46.2 69.9, -8.61 in-in-none SNCiin in-none ActLoopNT-in 3.1263 ActLoopCT-none nonTYR APEdihe_aanii APEdist_innn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 132.7 APE8-rot-in 314.77 APE67-dihe-in -47.56, -31.02 -61.45, -35.46 APE12-dist-in 8.281 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.586 0.185 0.217 E 395.0 385.0 4 29 26 3 [[92, 354]] 1.0 7jov AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVF O75116 25 417 1388.0 VFS:502 Type1 Inactive DFGin 6.2536 13.3298 BLAminus -142.21, 173.17 67.59, 68.13 -95.04, 16.84 301.9, 107.53 -61.95, -15.75 in-in in 8.5726 Saltbr-in 2.7159 HRD-in -62.26, -47.83 69.9, -5.26 in-in-out SNCiio in-out ActLoopNT-in 3.0981 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -82.91, 164.49 APE9-dihe-na 87.67, 168.25 APE8-dihe-in -79.05, 142.33 APE8-rot-out 46.7 APE67-dihe-in -72.13, -29.81 -50.42, -43.74 APE12-dist-in 8.1458 APE11-dist-in 11.7085 APE10-dist-in 5.7795 APE9-dist-in 4.2858 None None None XRAY 2.586 0.185 0.217 F 395.0 385.0 4 29 29 0 [[92, 354]] 1.0 7jov AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVG O75116 23 417 1388.0 VFS:501 Type1 Inactive DFGin 6.268 13.2068 BLAminus -141.3, 172.73 62.62, 71.55 -93.79, 17.44 301.31, 106.61 -60.9, -17.27 in-in in 8.3572 Saltbr-in 2.6194 HRD-in -63.54, -47.24 68.64, -6.0 in-in-out SNCiio in-out ActLoopNT-in 3.1285 ActLoopCT-out nonTYR APEdihe_aanoi APEdist_innn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 148.83 APE8-rot-out 39.24 APE67-dihe-in -74.92, -26.36 -51.82, -46.1 APE12-dist-in 10.1264 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.586 0.185 0.217 G 395.0 388.0 3 29 26 3 [[92, 354]] 1.0 7jov AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVH O75116 25 417 1388.0 VFS:501 Type1 Inactive DFGin 6.2783 13.2446 BLAminus -141.88, 173.26 61.58, 72.11 -93.64, 17.43 301.68, 105.86 -61.63, -15.37 in-in in 8.4613 Saltbr-in 2.6636 HRD-in -62.24, -47.57 69.31, -6.43 in-in-out SNCiio in-out ActLoopNT-in 3.1108 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -73.76, 175.86 APE9-dihe-na 74.79, 179.62 APE8-dihe-in -84.69, 144.58 APE8-rot-out 45.29 APE67-dihe-in -73.44, -28.15 -53.28, -43.42 APE12-dist-in 8.553 APE11-dist-in 11.9866 APE10-dist-in 5.9693 APE9-dist-in 4.3451 None None None XRAY 2.586 0.185 0.217 H 395.0 386.0 4 29 29 0 [[92, 354]] 1.0 7jov AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2

Ligand: VFS

Total number of chains: 9
Active chains: 0
Total number of genes: 2
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 9 100.0% 7JOVC

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
AGC ROCK1 ROCK1_HUMAN 7JOUA Q13464 9 402 1354.0 VFS:4000 Type1 Inactive DFGin 5.9959 13.3389 BLAminus -143.11, 174.9 56.51, 84.53 -111.27, 42.13 313.94, 101.63 -66.46, -29.86 in-in in 8.5845 Saltbr-in 2.6486 HRD-in -50.19, -37.76 57.05, 15.82 in-in-out SNCiio in-out ActLoopNT-in 3.2049 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -96.97, 107.53 APE9-dihe-na 156.7, 175.62 APE8-dihe-in -79.94, 144.48 APE8-rot-out 53.34 APE67-dihe-in -106.84, -34.67 -68.39, -2.9 APE12-dist-in 11.1521 APE11-dist-in 12.0952 APE10-dist-in 6.1966 APE9-dist-in 3.9409 None None None XRAY 3.318 0.218 0.248 A 413.0 388.0 6 29 29 0 [[76, 338]] 1.0 7jou Homo sapiens AGC_ROCK1_HUMAN AGC 3.5e-94 320.7 1.0 260.0 260.0 215 216 217 219 221 105 124 128 195 197 196 198.0 260 244 239 238 237 236 235 234 233 154 Rho-associated protein kinase 1
AGC ROCK2 ROCK2_HUMAN 7JOVA O75116 25 417 1388.0 VFS:502 Type1 Inactive DFGin 6.2465 13.2928 BLAminus -141.83, 172.55 62.54, 72.12 -93.6, 17.75 301.11, 105.91 -60.63, -17.81 in-in in 8.505 Saltbr-in 2.6448 HRD-in -61.37, -48.09 70.0, -5.6 in-in-out SNCiio in-out ActLoopNT-in 3.1039 ActLoopCT-out nonTYR APEdihe_aanoi APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 128.41 APE8-rot-out 35.63 APE67-dihe-in -72.9, -30.33 -60.06, -49.57 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.586 0.185 0.217 A 395.0 377.0 12 29 23 6 [[92, 354]] 1.0 7jov Homo sapiens AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVB O75116 23 417 1388.0 VFS:501 Type1 None DFGin 6.2716 13.2483 BLAminus -142.1, 173.55 61.9, 71.69 -93.43, 17.34 301.23, 105.57 -59.73, -16.68 in-in in 8.5286 Saltbr-in 2.6299 HRD-in -62.93, -47.02 69.4, -4.67 in-in-none SNCiin in-none ActLoopNT-in 3.0977 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none -66.0, -25.51 999.0, -48.59 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.586 0.185 0.217 B 395.0 378.0 11 29 21 8 [[92, 354]] 1.0 7jov Homo sapiens AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVC O75116 23 417 1388.0 VFS:501 Type1 Inactive DFGin 6.2684 13.2283 BLAminus -142.15, 173.25 63.2, 71.86 -94.04, 16.61 301.5, 104.97 -62.04, -13.94 in-in in 8.3763 Saltbr-in 2.7548 HRD-in -63.91, -46.28 70.58, -6.77 in-in-out SNCiio in-out ActLoopNT-in 3.102 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_onno APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, -148.71 APE8-dihe-in -13.99, 103.33 APE8-rot-out 49.66 APE67-dihe-in -50.5, -34.0 -98.95, 10.78 APE12-dist-out 6.1146 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-out 9.4434 None None None XRAY 2.586 0.185 0.217 C 395.0 389.0 3 29 27 2 [[92, 354]] 1.0 7jov Homo sapiens AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVD O75116 25 417 1388.0 VFS:501 Type1 None DFGin 6.2428 13.3572 BLAminus -142.23, 173.1 61.78, 71.13 -91.99, 20.3 301.3, 105.37 -69.47, 5.8 in-in in 8.6714 Saltbr-in 2.7008 HRD-in -54.87, -50.75 69.64, -5.46 in-in-none SNCiin in-none ActLoopNT-in 3.1806 ActLoopCT-none nonTYR APEdihe_aannn APEdist_nnnn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-none 999.0 APE67-dihe-none 999.0, -32.28 999.0, 999.0 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.586 0.185 0.217 D 395.0 361.0 26 29 14 15 [[92, 354]] 1.0 7jov Homo sapiens AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVE O75116 23 417 1388.0 VFS:501 Type1 None DFGin 6.2985 13.2567 BLAminus -140.47, 172.73 62.89, 72.53 -94.4, 16.26 301.6, 106.26 -62.28, -16.19 in-in in 8.4545 Saltbr-in 2.7399 HRD-in -64.4, -46.2 69.9, -8.61 in-in-none SNCiin in-none ActLoopNT-in 3.1263 ActLoopCT-none nonTYR APEdihe_aanii APEdist_innn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 132.7 APE8-rot-in 314.77 APE67-dihe-in -47.56, -31.02 -61.45, -35.46 APE12-dist-in 8.281 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.586 0.185 0.217 E 395.0 385.0 4 29 26 3 [[92, 354]] 1.0 7jov Homo sapiens AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVF O75116 25 417 1388.0 VFS:502 Type1 Inactive DFGin 6.2536 13.3298 BLAminus -142.21, 173.17 67.59, 68.13 -95.04, 16.84 301.9, 107.53 -61.95, -15.75 in-in in 8.5726 Saltbr-in 2.7159 HRD-in -62.26, -47.83 69.9, -5.26 in-in-out SNCiio in-out ActLoopNT-in 3.0981 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -82.91, 164.49 APE9-dihe-na 87.67, 168.25 APE8-dihe-in -79.05, 142.33 APE8-rot-out 46.7 APE67-dihe-in -72.13, -29.81 -50.42, -43.74 APE12-dist-in 8.1458 APE11-dist-in 11.7085 APE10-dist-in 5.7795 APE9-dist-in 4.2858 None None None XRAY 2.586 0.185 0.217 F 395.0 385.0 4 29 29 0 [[92, 354]] 1.0 7jov Homo sapiens AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVG O75116 23 417 1388.0 VFS:501 Type1 Inactive DFGin 6.268 13.2068 BLAminus -141.3, 172.73 62.62, 71.55 -93.79, 17.44 301.31, 106.61 -60.9, -17.27 in-in in 8.3572 Saltbr-in 2.6194 HRD-in -63.54, -47.24 68.64, -6.0 in-in-out SNCiio in-out ActLoopNT-in 3.1285 ActLoopCT-out nonTYR APEdihe_aanoi APEdist_innn APE10-dihe-na 999.0, 999.0 APE9-dihe-na 999.0, 999.0 APE8-dihe-none 999.0, 148.83 APE8-rot-out 39.24 APE67-dihe-in -74.92, -26.36 -51.82, -46.1 APE12-dist-in 10.1264 APE11-dist-none 999.0 APE10-dist-none 999.0 APE9-dist-none 999.0 None None None XRAY 2.586 0.185 0.217 G 395.0 388.0 3 29 26 3 [[92, 354]] 1.0 7jov Homo sapiens AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2
AGC ROCK2 ROCK2_HUMAN 7JOVH O75116 25 417 1388.0 VFS:501 Type1 Inactive DFGin 6.2783 13.2446 BLAminus -141.88, 173.26 61.58, 72.11 -93.64, 17.43 301.68, 105.86 -61.63, -15.37 in-in in 8.4613 Saltbr-in 2.6636 HRD-in -62.24, -47.57 69.31, -6.43 in-in-out SNCiio in-out ActLoopNT-in 3.1108 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_iiii APE10-dihe-na -73.76, 175.86 APE9-dihe-na 74.79, 179.62 APE8-dihe-in -84.69, 144.58 APE8-rot-out 45.29 APE67-dihe-in -73.44, -28.15 -53.28, -43.42 APE12-dist-in 8.553 APE11-dist-in 11.9866 APE10-dist-in 5.9693 APE9-dist-in 4.3451 None None None XRAY 2.586 0.185 0.217 H 395.0 386.0 4 29 29 0 [[92, 354]] 1.0 7jov Homo sapiens AGC_ROCK2_HUMAN AGC 2.2e-93 318.1 1.0 260.0 260.0 231 232 233 235 237 121 140 144 211 213 212 214.0 276 260 255 254 253 252 251 250 249 170 Rho-associated protein kinase 2

Ligand: VFS

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name