Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 7T4IA | P00533 | 697 | 1017 | 1210.0 | R28:2500 | Type1 | Active | DFGin | 6.176 | 15.419 | BLAminus | -134.59, -174.82 | 67.2, 83.56 | -99.26, 19.99 | 299.76, 93.96 | -46.8, -37.05 | in-in | in | 8.675 | Saltbr-in | 2.804 | HRD-in | -73.31, -54.28 | 79.02, 0.69 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.963 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.0, 142.26 | APE9-dihe-in | -143.46, 152.77 | APE8-dihe-in | -85.15, 103.65 | APE8-rot-na | 32.16 | APE67-dihe-in | -74.65, -13.42 | -69.82, -40.13 | APE12-dist-na | 12.549 | APE11-dist-na | 9.892 | APE10-dist-na | 10.85 | APE9-dist-in | 7.003 | None | None | None | XRAY | 2.61 | 0.184 | 0.238 | A | 328 | 309 | 0 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7t4i | TYR_EGFR_HUMAN | TYR | 1.1e-87 | 299.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8F1XA | P00533 | 696 | 1018 | 1210.0 | R28:1101 | Type1 | Active | DFGin | 5.983 | 15.01 | BLAminus | -136.15, -173.95 | 61.32, 87.85 | -107.98, 33.07 | 295.84, 87.53 | -69.26, -26.04 | in-in | in | 8.386 | Saltbr-in | 2.835 | HRD-in | -75.88, -47.81 | 70.31, 4.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.807 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -56.75, 114.5 | APE9-dihe-in | -126.56, 132.44 | APE8-dihe-in | -61.97, 98.31 | APE8-rot-na | 23.91 | APE67-dihe-in | -74.89, 2.26 | -62.79, -43.67 | APE12-dist-na | 12.267 | APE11-dist-na | 9.833 | APE10-dist-na | 10.674 | APE9-dist-in | 6.627 | None | None | None | XRAY | 2.3 | 0.205 | 0.226 | A | 331 | 317 | 3 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8f1x | TYR_EGFR_HUMAN | TYR | 1.1e-87 | 299.7 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7B85A | P00533 | 697 | 1020 | 1210.0 | R28:1101 | Type1 | None | DFGin | 5.854 | 14.557 | BLAminus | -137.84, -174.1 | 60.63, 85.07 | -103.17, 26.09 | 294.86, 88.23 | -63.8, -24.92 | in-in | in | 7.92 | Saltbr-in | 2.748 | HRD-in | -73.34, -48.14 | 69.22, 2.13 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.018 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 121.75 | APE9-dihe-in | -146.0, 163.38 | APE8-dihe-in | -89.43, 103.15 | APE8-rot-na | 22.0 | APE67-dihe-in | -71.22, -17.13 | -66.77, -37.78 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 10.554 | APE9-dist-in | 6.798 | None | None | None | XRAY | 2.5 | 0.216 | 0.244 | A | 333 | 312 | 6 | 0 | 0 | 2 | [[712, 970]] | 1.0 | 7b85 | TYR_EGFR_HUMAN | TYR | 1.1e-87 | 299.7 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7T4JA | P00533 | 701 | 984 | 1210.0 | R28:61101 | Type1 | Inactive | DFGin | 6.008 | 14.415 | BLAminus | -144.5, 169.5 | 68.77, 85.47 | -96.42, 20.57 | 291.54, 77.61 | -59.75, -25.89 | in-in | in | 8.017 | Saltbr-in | 2.568 | HRD-in | -76.71, -52.5 | 81.16, 2.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.877 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 45.96, 61.38 | APE9-dihe-in | -145.01, 131.44 | APE8-dihe-in | -84.06, 121.96 | APE8-rot-na | 31.03 | APE67-dihe-in | -61.46, 1.98 | -82.97, -44.13 | APE12-dist-na | 11.773 | APE11-dist-na | 11.055 | APE10-dist-na | 8.533 | APE9-dist-in | 6.334 | V948R | None | None | XRAY | 2.2 | 0.227 | 0.278 | A | 331 | 276 | 8 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7t4j | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7T4JB | P00533 | 701 | 984 | 1210.0 | R28:61101 | Type1 | Active | DFGin | 6.154 | 14.095 | BLAminus | -144.13, 179.52 | 58.61, 83.85 | -92.13, 21.8 | 294.24, 75.73 | -54.65, -26.76 | in-in | in | 7.881 | Saltbr-in | 2.775 | HRD-in | -69.57, -54.49 | 84.7, -3.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.806 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.5, 142.26 | APE9-dihe-in | -155.99, 150.11 | APE8-dihe-in | -82.77, 101.36 | APE8-rot-na | 36.83 | APE67-dihe-in | -75.7, -4.6 | -67.21, -37.02 | APE12-dist-na | 11.913 | APE11-dist-na | 10.71 | APE10-dist-na | 10.255 | APE9-dist-in | 6.477 | V948R | None | None | XRAY | 2.2 | 0.227 | 0.278 | B | 331 | 275 | 9 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7t4j | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7A6KA | P00533 | 700 | 984 | 1210.0 | R28:1101 | Type1 | Inactive | DFGin | 5.672 | 16.532 | BLBtrans | -113.38, -178.74 | 66.45, 17.22 | -70.85, 135.38 | 162.57, 71.95 | 93.0, -13.33 | out-out | out | 13.46 | Saltbr-out | 13.73 | HRD-in | -79.28, -53.26 | 81.06, -6.15 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.541 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 9.43 | APE9-dihe-in | -71.11, 126.54 | APE8-dihe-in | -79.69, 67.98 | APE8-rot-na | 32.03 | APE67-dihe-in | -70.72, -4.33 | -56.41, -46.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.919 | APE9-dist-out | 8.412 | T790M,V948R | None | None | XRAY | 2.0 | 0.193 | 0.22 | A | 333 | 266 | 19 | 0 | 0 | 14 | [[712, 970]] | 1.0 | 7a6k | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7A6KB | P00533 | 700 | 982 | 1210.0 | R28:1101 | Type1 | Inactive | DFGin | 5.343 | 15.868 | BLBtrans | -129.04, -178.67 | 62.57, 21.81 | -71.79, 126.77 | 154.84, 72.08 | 83.61, 999.0 | out-none | out | 13.481 | Saltbr-none | 999.0 | HRD-in | -76.88, -46.01 | 73.74, -7.71 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 133.51 | APE9-dihe-in | -84.9, 130.78 | APE8-dihe-in | -77.41, 66.48 | APE8-rot-na | 31.07 | APE67-dihe-in | -72.33, -5.85 | -61.23, -39.01 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.682 | T790M,V948R | None | None | XRAY | 2.0 | 0.193 | 0.22 | B | 333 | 260 | 23 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7a6k | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7A6KC | P00533 | 700 | 984 | 1210.0 | R28:1101 | Type1 | Inactive | DFGin | 5.484 | 15.789 | BLBtrans | -131.64, -174.72 | 61.99, 29.43 | -91.7, 131.8 | 164.71, 64.61 | 141.03, 999.0 | out-none | out | 13.417 | Saltbr-none | 999.0 | HRD-in | -76.77, -47.52 | 68.03, -0.55 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, -68.19 | APE9-dihe-in | -103.13, 125.01 | APE8-dihe-in | -86.91, 68.74 | APE8-rot-na | 26.28 | APE67-dihe-in | -74.92, -1.32 | -57.04, -40.43 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.556 | T790M,V948R | None | None | XRAY | 2.0 | 0.193 | 0.22 | C | 333 | 262 | 23 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7a6k | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7A6KD | P00533 | 702 | 984 | 1210.0 | R28:1101 | Type1 | Inactive | DFGin | 5.163 | 15.725 | BLBtrans | -125.34, -177.59 | 58.43, 37.54 | -98.25, 128.03 | 151.98, 71.88 | 111.44, 999.0 | out-out | out | 13.356 | Saltbr-out | 9.148 | HRD-in | -91.6, -48.16 | 65.02, 0.98 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 116.46 | APE8-dihe-in | -80.89, 70.4 | APE8-rot-na | 24.1 | APE67-dihe-in | -72.66, -6.51 | -57.4, -40.86 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.69 | T790M,V948R | None | None | XRAY | 2.0 | 0.193 | 0.22 | D | 333 | 255 | 28 | 0 | 0 | 18 | [[712, 970]] | 1.0 | 7a6k | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EGFR | EGFR_HUMAN | 7T4IA | P00533 | 697 | 1017 | 1210.0 | R28:2500 | Type1 | Active | DFGin | 6.176 | 15.419 | BLAminus | -134.59, -174.82 | 67.2, 83.56 | -99.26, 19.99 | 299.76, 93.96 | -46.8, -37.05 | in-in | in | 8.675 | Saltbr-in | 2.804 | HRD-in | -73.31, -54.28 | 79.02, 0.69 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.963 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.0, 142.26 | APE9-dihe-in | -143.46, 152.77 | APE8-dihe-in | -85.15, 103.65 | APE8-rot-na | 32.16 | APE67-dihe-in | -74.65, -13.42 | -69.82, -40.13 | APE12-dist-na | 12.549 | APE11-dist-na | 9.892 | APE10-dist-na | 10.85 | APE9-dist-in | 7.003 | None | None | None | XRAY | 2.61 | 0.184 | 0.238 | A | 328 | 309 | 0 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7t4i | Homo sapiens | TYR_EGFR_HUMAN | TYR | 1.1e-87 | 299.8 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 8F1XA | P00533 | 696 | 1018 | 1210.0 | R28:1101 | Type1 | Active | DFGin | 5.983 | 15.01 | BLAminus | -136.15, -173.95 | 61.32, 87.85 | -107.98, 33.07 | 295.84, 87.53 | -69.26, -26.04 | in-in | in | 8.386 | Saltbr-in | 2.835 | HRD-in | -75.88, -47.81 | 70.31, 4.02 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.807 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -56.75, 114.5 | APE9-dihe-in | -126.56, 132.44 | APE8-dihe-in | -61.97, 98.31 | APE8-rot-na | 23.91 | APE67-dihe-in | -74.89, 2.26 | -62.79, -43.67 | APE12-dist-na | 12.267 | APE11-dist-na | 9.833 | APE10-dist-na | 10.674 | APE9-dist-in | 6.627 | None | None | None | XRAY | 2.3 | 0.205 | 0.226 | A | 331 | 317 | 3 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 8f1x | Homo sapiens | TYR_EGFR_HUMAN | TYR | 1.1e-87 | 299.7 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7B85A | P00533 | 697 | 1020 | 1210.0 | R28:1101 | Type1 | None | DFGin | 5.854 | 14.557 | BLAminus | -137.84, -174.1 | 60.63, 85.07 | -103.17, 26.09 | 294.86, 88.23 | -63.8, -24.92 | in-in | in | 7.92 | Saltbr-in | 2.748 | HRD-in | -73.34, -48.14 | 69.22, 2.13 | in-in-none | SNCiin | in-none | ActLoopNT-in | 3.018 | ActLoopCT-none | TYR | APEdihe_niiai | APEdist_aaai | APE10-dihe-none | 999.0, 121.75 | APE9-dihe-in | -146.0, 163.38 | APE8-dihe-in | -89.43, 103.15 | APE8-rot-na | 22.0 | APE67-dihe-in | -71.22, -17.13 | -66.77, -37.78 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 10.554 | APE9-dist-in | 6.798 | None | None | None | XRAY | 2.5 | 0.216 | 0.244 | A | 333 | 312 | 6 | 0 | 0 | 2 | [[712, 970]] | 1.0 | 7b85 | Homo sapiens | TYR_EGFR_HUMAN | TYR | 1.1e-87 | 299.7 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7T4JA | P00533 | 701 | 984 | 1210.0 | R28:61101 | Type1 | Inactive | DFGin | 6.008 | 14.415 | BLAminus | -144.5, 169.5 | 68.77, 85.47 | -96.42, 20.57 | 291.54, 77.61 | -59.75, -25.89 | in-in | in | 8.017 | Saltbr-in | 2.568 | HRD-in | -76.71, -52.5 | 81.16, 2.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.877 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaai | APE10-dihe-out | 45.96, 61.38 | APE9-dihe-in | -145.01, 131.44 | APE8-dihe-in | -84.06, 121.96 | APE8-rot-na | 31.03 | APE67-dihe-in | -61.46, 1.98 | -82.97, -44.13 | APE12-dist-na | 11.773 | APE11-dist-na | 11.055 | APE10-dist-na | 8.533 | APE9-dist-in | 6.334 | V948R | None | None | XRAY | 2.2 | 0.227 | 0.278 | A | 331 | 276 | 8 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7t4j | Homo sapiens | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7T4JB | P00533 | 701 | 984 | 1210.0 | R28:61101 | Type1 | Active | DFGin | 6.154 | 14.095 | BLAminus | -144.13, 179.52 | 58.61, 83.85 | -92.13, 21.8 | 294.24, 75.73 | -54.65, -26.76 | in-in | in | 7.881 | Saltbr-in | 2.775 | HRD-in | -69.57, -54.49 | 84.7, -3.58 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.806 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -117.5, 142.26 | APE9-dihe-in | -155.99, 150.11 | APE8-dihe-in | -82.77, 101.36 | APE8-rot-na | 36.83 | APE67-dihe-in | -75.7, -4.6 | -67.21, -37.02 | APE12-dist-na | 11.913 | APE11-dist-na | 10.71 | APE10-dist-na | 10.255 | APE9-dist-in | 6.477 | V948R | None | None | XRAY | 2.2 | 0.227 | 0.278 | B | 331 | 275 | 9 | 0 | 0 | 0 | [[712, 970]] | 1.0 | 7t4j | Homo sapiens | TYR_EGFR_HUMAN | TYR | 1.2e-85 | 293.0 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7A6KA | P00533 | 700 | 984 | 1210.0 | R28:1101 | Type1 | Inactive | DFGin | 5.672 | 16.532 | BLBtrans | -113.38, -178.74 | 66.45, 17.22 | -70.85, 135.38 | 162.57, 71.95 | 93.0, -13.33 | out-out | out | 13.46 | Saltbr-out | 13.73 | HRD-in | -79.28, -53.26 | 81.06, -6.15 | out-out-out | SNCooo | out-out | ActLoopNT-out | 7.541 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 9.43 | APE9-dihe-in | -71.11, 126.54 | APE8-dihe-in | -79.69, 67.98 | APE8-rot-na | 32.03 | APE67-dihe-in | -70.72, -4.33 | -56.41, -46.0 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 11.919 | APE9-dist-out | 8.412 | T790M,V948R | None | None | XRAY | 2.0 | 0.193 | 0.22 | A | 333 | 266 | 19 | 0 | 0 | 14 | [[712, 970]] | 1.0 | 7a6k | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7A6KB | P00533 | 700 | 982 | 1210.0 | R28:1101 | Type1 | Inactive | DFGin | 5.343 | 15.868 | BLBtrans | -129.04, -178.67 | 62.57, 21.81 | -71.79, 126.77 | 154.84, 72.08 | 83.61, 999.0 | out-none | out | 13.481 | Saltbr-none | 999.0 | HRD-in | -76.88, -46.01 | 73.74, -7.71 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 133.51 | APE9-dihe-in | -84.9, 130.78 | APE8-dihe-in | -77.41, 66.48 | APE8-rot-na | 31.07 | APE67-dihe-in | -72.33, -5.85 | -61.23, -39.01 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.682 | T790M,V948R | None | None | XRAY | 2.0 | 0.193 | 0.22 | B | 333 | 260 | 23 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7a6k | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7A6KC | P00533 | 700 | 984 | 1210.0 | R28:1101 | Type1 | Inactive | DFGin | 5.484 | 15.789 | BLBtrans | -131.64, -174.72 | 61.99, 29.43 | -91.7, 131.8 | 164.71, 64.61 | 141.03, 999.0 | out-none | out | 13.417 | Saltbr-none | 999.0 | HRD-in | -76.77, -47.52 | 68.03, -0.55 | none-none-out | SNCnno | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, -68.19 | APE9-dihe-in | -103.13, 125.01 | APE8-dihe-in | -86.91, 68.74 | APE8-rot-na | 26.28 | APE67-dihe-in | -74.92, -1.32 | -57.04, -40.43 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.556 | T790M,V948R | None | None | XRAY | 2.0 | 0.193 | 0.22 | C | 333 | 262 | 23 | 0 | 0 | 17 | [[712, 970]] | 1.0 | 7a6k | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| TYR | EGFR | EGFR_HUMAN | 7A6KD | P00533 | 702 | 984 | 1210.0 | R28:1101 | Type1 | Inactive | DFGin | 5.163 | 15.725 | BLBtrans | -125.34, -177.59 | 58.43, 37.54 | -98.25, 128.03 | 151.98, 71.88 | 111.44, 999.0 | out-out | out | 13.356 | Saltbr-out | 9.148 | HRD-in | -91.6, -48.16 | 65.02, 0.98 | out-none-out | SNCono | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 116.46 | APE8-dihe-in | -80.89, 70.4 | APE8-rot-na | 24.1 | APE67-dihe-in | -72.66, -6.51 | -57.4, -40.86 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.69 | T790M,V948R | None | None | XRAY | 2.0 | 0.193 | 0.22 | D | 333 | 255 | 28 | 0 | 0 | 18 | [[712, 970]] | 1.0 | 7a6k | Homo sapiens | TYR_EGFR_HUMAN | TYR | 6.4e-88 | 300.5 | 3 | 259 | 257 | 854 | 855 | 856 | 858 | 860 | 745 | 762 | 766 | 834 | 836 | 835 | 837 | 896 | 884 | 879 | 878 | 877 | 876 | 875 | 874 | 873 | 791 | Epidermal growth factor receptor |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|