| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | CLK1 | CLK1_HUMAN | 6Z4ZA | P49759 | 148 | 482 | 484.0 | PQ5:60505 | Type1 | Active | DFGin | 7.046 | 14.2363 | BLAminus | -126.68, 179.24 | 66.69, 82.0 | -103.33, 19.73 | 297.68, 94.61 | -71.59, -13.97 | in-in | in | 8.4611 | Saltbr-in | 2.7642 | HRD-in | -69.38, -51.98 | 76.89, -13.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9245 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.91, 169.84 | APE9-dihe-na | 70.81, 154.45 | APE8-dihe-in | -79.18, 136.44 | APE8-rot-in | 295.15 | APE67-dihe-in | -64.16, -17.67 | -45.6, -49.57 | APE12-dist-in | 13.5127 | APE11-dist-in | 11.3594 | APE10-dist-in | 7.327 | APE9-dist-in | 3.0405 | None | None | None | XRAY | 2.07 | 0.177 | 0.213 | A | 339.0 | 335.0 | 0 | 25 | 25 | 0 | [[161, 477]] | 1.0 | 6z4z | CMGC_CLK1_HUMAN | CMGC | 2.5e-93 | 318.5 | 1.0 | 301.0 | 301.0 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288.0 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6Z4ZB | P49759 | 148 | 484 | 484.0 | PQ5:60501 | Type1 | Active | DFGin | 7.0483 | 14.168 | BLAminus | -127.78, 179.44 | 66.36, 84.49 | -106.02, 23.22 | 298.83, 96.06 | -73.86, -11.97 | in-in | in | 8.4214 | Saltbr-in | 2.7252 | HRD-in | -70.61, -51.12 | 77.5, -15.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9096 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.17, 168.57 | APE9-dihe-na | 73.19, 152.9 | APE8-dihe-in | -77.75, 136.06 | APE8-rot-in | 294.47 | APE67-dihe-in | -61.42, -18.21 | -47.63, -47.77 | APE12-dist-in | 13.4848 | APE11-dist-in | 11.247 | APE10-dist-in | 7.2192 | APE9-dist-in | 3.0518 | None | None | None | XRAY | 2.07 | 0.177 | 0.213 | B | 339.0 | 337.0 | 0 | 25 | 25 | 0 | [[161, 477]] | 1.0 | 6z4z | CMGC_CLK1_HUMAN | CMGC | 2.5e-93 | 318.5 | 1.0 | 301.0 | 301.0 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288.0 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6Z4ZC | P49759 | 148 | 482 | 484.0 | PQ5:60502 | Type1 | Active | DFGin | 7.1081 | 14.2491 | BLAminus | -126.87, 178.82 | 67.48, 81.17 | -101.74, 18.48 | 298.94, 95.28 | -65.75, -17.47 | in-in | in | 8.5666 | Saltbr-in | 2.7627 | HRD-in | -67.93, -52.14 | 78.08, -12.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8763 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.01, 169.28 | APE9-dihe-na | 73.05, 151.25 | APE8-dihe-in | -74.69, 135.04 | APE8-rot-in | 294.69 | APE67-dihe-in | -63.57, -18.13 | -46.66, -45.93 | APE12-dist-in | 13.7076 | APE11-dist-in | 11.4576 | APE10-dist-in | 7.407 | APE9-dist-in | 3.0276 | None | None | None | XRAY | 2.07 | 0.177 | 0.213 | C | 339.0 | 335.0 | 0 | 25 | 25 | 0 | [[161, 477]] | 1.0 | 6z4z | CMGC_CLK1_HUMAN | CMGC | 2.5e-93 | 318.5 | 1.0 | 301.0 | 301.0 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288.0 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK3 | CLK3_HUMAN | 6Z55A | P49761 | 127 | 482 | 490.0 | PQ5:60519 | Type1 | Active | DFGin | 7.3991 | 15.5451 | BLAminus | -114.58, 173.98 | 75.12, 75.81 | -96.97, 17.81 | 291.53, 88.35 | -70.47, -12.03 | in-in | in | 8.8932 | Saltbr-in | 2.6425 | HRD-in | -73.34, -50.13 | 78.35, -13.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9074 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.62, 168.42 | APE9-dihe-na | 71.12, 154.19 | APE8-dihe-in | -74.72, 147.13 | APE8-rot-in | 286.47 | APE67-dihe-in | -63.58, -22.91 | -38.61, -57.63 | APE12-dist-in | 13.1402 | APE11-dist-in | 11.9251 | APE10-dist-in | 7.4483 | APE9-dist-in | 3.0436 | None | None | None | XRAY | 1.7 | 0.158 | 0.195 | A | 360.0 | 356.0 | 2 | 25 | 25 | 0 | [[156, 472]] | 1.0 | 6z55 | CMGC_CLK3_HUMAN | CMGC | 1.2e-90 | 309.6 | 1.0 | 301.0 | 301.0 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283.0 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | CLK3 | CLK3_HUMAN | 6Z55B | P49761 | 128 | 484 | 490.0 | PQ5:60516 | Type1 | Active | DFGin | 7.3569 | 15.5257 | BLAminus | -113.15, 172.16 | 75.56, 76.57 | -97.3, 14.76 | 289.76, 90.56 | -61.38, -19.22 | in-in | in | 8.8957 | Saltbr-in | 2.7048 | HRD-in | -73.58, -49.98 | 78.81, -11.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8934 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.67, 168.41 | APE9-dihe-na | 68.9, 153.38 | APE8-dihe-in | -74.53, 145.27 | APE8-rot-in | 288.03 | APE67-dihe-in | -60.23, -27.92 | -39.2, -58.45 | APE12-dist-in | 13.1278 | APE11-dist-in | 11.8254 | APE10-dist-in | 7.3801 | APE9-dist-in | 3.0549 | None | None | None | XRAY | 1.7 | 0.158 | 0.195 | B | 360.0 | 357.0 | 0 | 25 | 25 | 0 | [[156, 472]] | 1.0 | 6z55 | CMGC_CLK3_HUMAN | CMGC | 1.2e-90 | 309.6 | 1.0 | 301.0 | 301.0 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283.0 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | CSNK2A1 | CSK21_HUMAN | 6YULAAA | P68400 | 3 | 333 | 391.0 | PQ5:403 | Type1 | Active | DFGin | 7.4108 | 16.6374 | BLAminus | -119.76, 177.88 | 54.4, 77.49 | -88.72, 16.75 | 296.13, 83.32 | -68.07, -20.02 | in-in | in | 9.5741 | Saltbr-in | 2.5954 | HRD-in | -71.56, -51.98 | 70.9, 15.42 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8823 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.14, 159.08 | APE9-dihe-na | 80.59, 170.52 | APE8-dihe-in | -82.75, 140.87 | APE8-rot-in | 297.23 | APE67-dihe-in | -69.04, -16.25 | -40.76, -51.06 | APE12-dist-in | 12.8354 | APE11-dist-in | 10.9234 | APE10-dist-in | 6.3551 | APE9-dist-in | 3.7331 | None | None | None | XRAY | 2.4 | 0.218 | 0.232 | AAA | 391.0 | 331.0 | 0 | 27 | 27 | 0 | [[39, 324]] | 1.0 | 6yul | CMGC_CSNK2A1_HUMAN | CMGC | 2.2e-69 | 239.9 | 1.0 | 301.0 | 301.0 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156.0 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 6YULGGG | P68400 | 3 | 333 | 391.0 | PQ5:404 | Type1 | Active | DFGin | 7.5082 | 16.5432 | BLAminus | -117.8, 176.89 | 56.9, 76.16 | -89.82, 20.37 | 297.24, 85.22 | -71.56, -18.77 | in-in | in | 9.4598 | Saltbr-in | 3.0029 | HRD-in | -71.33, -53.46 | 70.0, 16.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8803 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.91, 158.86 | APE9-dihe-na | 75.12, 171.78 | APE8-dihe-in | -91.15, 146.0 | APE8-rot-in | 309.69 | APE67-dihe-in | -67.12, -19.35 | -39.65, -53.16 | APE12-dist-in | 12.6916 | APE11-dist-in | 10.235 | APE10-dist-in | 6.3547 | APE9-dist-in | 3.4374 | None | None | None | XRAY | 2.4 | 0.218 | 0.232 | GGG | 391.0 | 331.0 | 0 | 27 | 27 | 0 | [[39, 324]] | 1.0 | 6yul | CMGC_CSNK2A1_HUMAN | CMGC | 2.2e-69 | 239.9 | 1.0 | 301.0 | 301.0 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156.0 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| OTHER | HASPIN | HASP_HUMAN | 6Z5CA | Q8TF76 | 470 | 798 | 798.0 | PQ5:805 | Type1 | Inactive | DFGin | 4.7306 | 13.1081 | BLAminus | -133.84, 170.31 | 75.72, 94.52 | -110.21, 19.19 | 311.37, 116.86 | -61.87, -31.19 | out-out | out | 10.462 | Saltbr-out | 3.7004 | HRD-naN | -70.06, -50.84 | 74.01, -0.31 | out-in-na | SNCoia | in-na | ActLoopNT-in | 2.9311 | ActLoopCT-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | APE10-dihe-na | -116.88, 20.45 | APE9-dihe-na | -80.43, 159.13 | APE8-dihe-na | -144.39, 165.92 | APE8-rot-na | 214.89 | APE67-dihe-na | -162.19, 147.1 | 97.48, -3.07 | APE12-dist-na | 9.4878 | APE11-dist-na | 13.5203 | APE10-dist-na | 17.0497 | APE9-dist-na | 13.1004 | None | None | None | XRAY | 1.75 | 0.16 | 0.188 | A | 357.0 | 329.0 | 0 | 35 | 35 | 0 | [[484, 797]] | 1.0 | 6z5c | OTHER_HASPIN_HUMAN | HASP | 1.4e-226 | 756.6 | 1.0 | 314.0 | 314.0 | 686 | 687 | 688 | 690 | 692 | 511 | 535 | 539 | 646 | 648 | 647 | 649.0 | 741 | 721 | 716 | 715 | 714 | 713 | 712 | 711 | 710 | 604 | Serine/threonine-protein kinase haspin |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | CLK1 | CLK1_HUMAN | 6Z4ZA | P49759 | 148 | 482 | 484.0 | PQ5:60505 | Type1 | Active | DFGin | 7.046 | 14.2363 | BLAminus | -126.68, 179.24 | 66.69, 82.0 | -103.33, 19.73 | 297.68, 94.61 | -71.59, -13.97 | in-in | in | 8.4611 | Saltbr-in | 2.7642 | HRD-in | -69.38, -51.98 | 76.89, -13.79 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9245 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -138.91, 169.84 | APE9-dihe-na | 70.81, 154.45 | APE8-dihe-in | -79.18, 136.44 | APE8-rot-in | 295.15 | APE67-dihe-in | -64.16, -17.67 | -45.6, -49.57 | APE12-dist-in | 13.5127 | APE11-dist-in | 11.3594 | APE10-dist-in | 7.327 | APE9-dist-in | 3.0405 | None | None | None | XRAY | 2.07 | 0.177 | 0.213 | A | 339.0 | 335.0 | 0 | 25 | 25 | 0 | [[161, 477]] | 1.0 | 6z4z | Homo sapiens | CMGC_CLK1_HUMAN | CMGC | 2.5e-93 | 318.5 | 1.0 | 301.0 | 301.0 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288.0 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6Z4ZB | P49759 | 148 | 484 | 484.0 | PQ5:60501 | Type1 | Active | DFGin | 7.0483 | 14.168 | BLAminus | -127.78, 179.44 | 66.36, 84.49 | -106.02, 23.22 | 298.83, 96.06 | -73.86, -11.97 | in-in | in | 8.4214 | Saltbr-in | 2.7252 | HRD-in | -70.61, -51.12 | 77.5, -15.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9096 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -137.17, 168.57 | APE9-dihe-na | 73.19, 152.9 | APE8-dihe-in | -77.75, 136.06 | APE8-rot-in | 294.47 | APE67-dihe-in | -61.42, -18.21 | -47.63, -47.77 | APE12-dist-in | 13.4848 | APE11-dist-in | 11.247 | APE10-dist-in | 7.2192 | APE9-dist-in | 3.0518 | None | None | None | XRAY | 2.07 | 0.177 | 0.213 | B | 339.0 | 337.0 | 0 | 25 | 25 | 0 | [[161, 477]] | 1.0 | 6z4z | Homo sapiens | CMGC_CLK1_HUMAN | CMGC | 2.5e-93 | 318.5 | 1.0 | 301.0 | 301.0 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288.0 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK1 | CLK1_HUMAN | 6Z4ZC | P49759 | 148 | 482 | 484.0 | PQ5:60502 | Type1 | Active | DFGin | 7.1081 | 14.2491 | BLAminus | -126.87, 178.82 | 67.48, 81.17 | -101.74, 18.48 | 298.94, 95.28 | -65.75, -17.47 | in-in | in | 8.5666 | Saltbr-in | 2.7627 | HRD-in | -67.93, -52.14 | 78.08, -12.45 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8763 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -140.01, 169.28 | APE9-dihe-na | 73.05, 151.25 | APE8-dihe-in | -74.69, 135.04 | APE8-rot-in | 294.69 | APE67-dihe-in | -63.57, -18.13 | -46.66, -45.93 | APE12-dist-in | 13.7076 | APE11-dist-in | 11.4576 | APE10-dist-in | 7.407 | APE9-dist-in | 3.0276 | None | None | None | XRAY | 2.07 | 0.177 | 0.213 | C | 339.0 | 335.0 | 0 | 25 | 25 | 0 | [[161, 477]] | 1.0 | 6z4z | Homo sapiens | CMGC_CLK1_HUMAN | CMGC | 2.5e-93 | 318.5 | 1.0 | 301.0 | 301.0 | 324 | 325 | 326 | 328 | 330 | 191 | 206 | 210 | 285 | 287 | 286 | 288.0 | 361 | 349 | 344 | 343 | 342 | 341 | 340 | 339 | 338 | 242 | Dual specificity protein kinase CLK1 |
| CMGC | CLK3 | CLK3_HUMAN | 6Z55A | P49761 | 127 | 482 | 490.0 | PQ5:60519 | Type1 | Active | DFGin | 7.3991 | 15.5451 | BLAminus | -114.58, 173.98 | 75.12, 75.81 | -96.97, 17.81 | 291.53, 88.35 | -70.47, -12.03 | in-in | in | 8.8932 | Saltbr-in | 2.6425 | HRD-in | -73.34, -50.13 | 78.35, -13.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9074 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -122.62, 168.42 | APE9-dihe-na | 71.12, 154.19 | APE8-dihe-in | -74.72, 147.13 | APE8-rot-in | 286.47 | APE67-dihe-in | -63.58, -22.91 | -38.61, -57.63 | APE12-dist-in | 13.1402 | APE11-dist-in | 11.9251 | APE10-dist-in | 7.4483 | APE9-dist-in | 3.0436 | None | None | None | XRAY | 1.7 | 0.158 | 0.195 | A | 360.0 | 356.0 | 2 | 25 | 25 | 0 | [[156, 472]] | 1.0 | 6z55 | Homo sapiens | CMGC_CLK3_HUMAN | CMGC | 1.2e-90 | 309.6 | 1.0 | 301.0 | 301.0 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283.0 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | CLK3 | CLK3_HUMAN | 6Z55B | P49761 | 128 | 484 | 490.0 | PQ5:60516 | Type1 | Active | DFGin | 7.3569 | 15.5257 | BLAminus | -113.15, 172.16 | 75.56, 76.57 | -97.3, 14.76 | 289.76, 90.56 | -61.38, -19.22 | in-in | in | 8.8957 | Saltbr-in | 2.7048 | HRD-in | -73.58, -49.98 | 78.81, -11.77 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8934 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -125.67, 168.41 | APE9-dihe-na | 68.9, 153.38 | APE8-dihe-in | -74.53, 145.27 | APE8-rot-in | 288.03 | APE67-dihe-in | -60.23, -27.92 | -39.2, -58.45 | APE12-dist-in | 13.1278 | APE11-dist-in | 11.8254 | APE10-dist-in | 7.3801 | APE9-dist-in | 3.0549 | None | None | None | XRAY | 1.7 | 0.158 | 0.195 | B | 360.0 | 357.0 | 0 | 25 | 25 | 0 | [[156, 472]] | 1.0 | 6z55 | Homo sapiens | CMGC_CLK3_HUMAN | CMGC | 1.2e-90 | 309.6 | 1.0 | 301.0 | 301.0 | 319 | 320 | 321 | 323 | 325 | 186 | 201 | 205 | 280 | 282 | 281 | 283.0 | 356 | 344 | 339 | 338 | 337 | 336 | 335 | 334 | 333 | 237 | Dual specificity protein kinase CLK3 |
| CMGC | CSNK2A1 | CSK21_HUMAN | 6YULAAA | P68400 | 3 | 333 | 391.0 | PQ5:403 | Type1 | Active | DFGin | 7.4108 | 16.6374 | BLAminus | -119.76, 177.88 | 54.4, 77.49 | -88.72, 16.75 | 296.13, 83.32 | -68.07, -20.02 | in-in | in | 9.5741 | Saltbr-in | 2.5954 | HRD-in | -71.56, -51.98 | 70.9, 15.42 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8823 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -131.14, 159.08 | APE9-dihe-na | 80.59, 170.52 | APE8-dihe-in | -82.75, 140.87 | APE8-rot-in | 297.23 | APE67-dihe-in | -69.04, -16.25 | -40.76, -51.06 | APE12-dist-in | 12.8354 | APE11-dist-in | 10.9234 | APE10-dist-in | 6.3551 | APE9-dist-in | 3.7331 | None | None | None | XRAY | 2.4 | 0.218 | 0.232 | AAA | 391.0 | 331.0 | 0 | 27 | 27 | 0 | [[39, 324]] | 1.0 | 6yul | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 2.2e-69 | 239.9 | 1.0 | 301.0 | 301.0 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156.0 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| CMGC | CSNK2A1 | CSK21_HUMAN | 6YULGGG | P68400 | 3 | 333 | 391.0 | PQ5:404 | Type1 | Active | DFGin | 7.5082 | 16.5432 | BLAminus | -117.8, 176.89 | 56.9, 76.16 | -89.82, 20.37 | 297.24, 85.22 | -71.56, -18.77 | in-in | in | 9.4598 | Saltbr-in | 3.0029 | HRD-in | -71.33, -53.46 | 70.0, 16.13 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8803 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -133.91, 158.86 | APE9-dihe-na | 75.12, 171.78 | APE8-dihe-in | -91.15, 146.0 | APE8-rot-in | 309.69 | APE67-dihe-in | -67.12, -19.35 | -39.65, -53.16 | APE12-dist-in | 12.6916 | APE11-dist-in | 10.235 | APE10-dist-in | 6.3547 | APE9-dist-in | 3.4374 | None | None | None | XRAY | 2.4 | 0.218 | 0.232 | GGG | 391.0 | 331.0 | 0 | 27 | 27 | 0 | [[39, 324]] | 1.0 | 6yul | Homo sapiens | CMGC_CSNK2A1_HUMAN | CMGC | 2.2e-69 | 239.9 | 1.0 | 301.0 | 301.0 | 174 | 175 | 176 | 178 | 180 | 68 | 81 | 85 | 153 | 155 | 154 | 156.0 | 214 | 201 | 196 | 195 | 194 | 193 | 192 | 191 | 190 | 114 | Casein kinase II subunit alpha |
| OTHER | HASPIN | HASP_HUMAN | 6Z5CA | Q8TF76 | 470 | 798 | 798.0 | PQ5:805 | Type1 | Inactive | DFGin | 4.7306 | 13.1081 | BLAminus | -133.84, 170.31 | 75.72, 94.52 | -110.21, 19.19 | 311.37, 116.86 | -61.87, -31.19 | out-out | out | 10.462 | Saltbr-out | 3.7004 | HRD-naN | -70.06, -50.84 | 74.01, -0.31 | out-in-na | SNCoia | in-na | ActLoopNT-in | 2.9311 | ActLoopCT-na | noAPE | APEdihe_aaaaa | APEdist_aaaa | APE10-dihe-na | -116.88, 20.45 | APE9-dihe-na | -80.43, 159.13 | APE8-dihe-na | -144.39, 165.92 | APE8-rot-na | 214.89 | APE67-dihe-na | -162.19, 147.1 | 97.48, -3.07 | APE12-dist-na | 9.4878 | APE11-dist-na | 13.5203 | APE10-dist-na | 17.0497 | APE9-dist-na | 13.1004 | None | None | None | XRAY | 1.75 | 0.16 | 0.188 | A | 357.0 | 329.0 | 0 | 35 | 35 | 0 | [[484, 797]] | 1.0 | 6z5c | Homo sapiens | OTHER_HASPIN_HUMAN | HASP | 1.4e-226 | 756.6 | 1.0 | 314.0 | 314.0 | 686 | 687 | 688 | 690 | 692 | 511 | 535 | 539 | 646 | 648 | 647 | 649.0 | 741 | 721 | 716 | 715 | 714 | 713 | 712 | 711 | 710 | 604 | Serine/threonine-protein kinase haspin |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|