Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | CDKL1 | CDKL1_HUMAN | 4AGUA | Q00532 | 2 | 291 | 357.0 | D15:500 | Type1 | None | DFGin | 6.926 | 15.225 | BLAminus | -125.36, -173.19 | 61.0, 84.36 | -106.79, 0.32 | 274.19, 82.71 | -54.94, -33.89 | in-in | in | 8.329 | Saltbr-in | 2.668 | HRD-in | -62.63, -48.4 | 73.42, -8.74 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.806 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 138.22 | APE8-rot-in | 301.17 | APE67-dihe-in | -58.09, -27.23 | -56.92, -32.3 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | T159D,Y161E | None | None | XRAY | 2.4 | 0.189 | 0.226 | A | 311 | 277 | 13 | 0 | 0 | 12 | [[4, 287]] | 1.0 | 4agu | CMGC_CDKL1_HUMAN | CMGC | 2.9e-80 | 275.7 | 1 | 301 | 301 | 143 | 144 | 145 | 147 | 149 | 33 | 51 | 55 | 123 | 125 | 124 | 126 | 184 | 171 | 166 | 165 | 164 | 163 | 162 | 161 | 160 | 81 | Cyclin-dependent kinase-like 1 |
| CMGC | CDKL1 | CDKL1_HUMAN | 4AGUB | Q00532 | 3 | 292 | 357.0 | D15:500 | Type1 | None | DFGin | 6.911 | 15.242 | BLAminus | -123.13, -174.59 | 61.67, 77.11 | -99.83, 8.36 | 278.04, 80.77 | -62.15, -31.07 | in-in | in | 8.312 | Saltbr-in | 2.668 | HRD-in | -65.94, -47.41 | 70.79, -7.65 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.762 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 133.96 | APE8-rot-in | 300.0 | APE67-dihe-in | -56.83, -27.96 | -64.83, -28.69 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | T159D,Y161E | None | None | XRAY | 2.4 | 0.189 | 0.226 | B | 311 | 276 | 14 | 0 | 0 | 12 | [[4, 287]] | 1.0 | 4agu | CMGC_CDKL1_HUMAN | CMGC | 2.9e-80 | 275.7 | 1 | 301 | 301 | 143 | 144 | 145 | 147 | 149 | 33 | 51 | 55 | 123 | 125 | 124 | 126 | 184 | 171 | 166 | 165 | 164 | 163 | 162 | 161 | 160 | 81 | Cyclin-dependent kinase-like 1 |
| CMGC | CDKL1 | CDKL1_HUMAN | 4AGUC | Q00532 | 2 | 291 | 357.0 | D15:500 | Type1 | None | DFGin | 7.076 | 15.076 | BLAminus | -126.2, -170.17 | 57.04, 81.0 | -105.59, 6.66 | 281.53, 85.88 | -54.99, -37.13 | in-in | in | 8.283 | Saltbr-in | 2.658 | HRD-in | -56.25, -49.02 | 74.36, -3.78 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.791 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 127.06 | APE8-rot-in | 293.41 | APE67-dihe-in | -52.47, -36.63 | -43.96, -43.49 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | T159D,Y161E | None | None | XRAY | 2.4 | 0.189 | 0.226 | C | 311 | 278 | 12 | 0 | 0 | 12 | [[4, 287]] | 1.0 | 4agu | CMGC_CDKL1_HUMAN | CMGC | 2.9e-80 | 275.7 | 1 | 301 | 301 | 143 | 144 | 145 | 147 | 149 | 33 | 51 | 55 | 123 | 125 | 124 | 126 | 184 | 171 | 166 | 165 | 164 | 163 | 162 | 161 | 160 | 81 | Cyclin-dependent kinase-like 1 |
| CMGC | DYRK1A | DYR1A_HUMAN | 2VX3A | Q13627 | 135 | 481 | 763.0 | D15:600 | Type1 | Active | DFGin | 7.177 | 14.936 | BLAminus | -117.81, 179.58 | 65.92, 72.63 | -91.66, 22.61 | 288.71, 80.01 | -64.63, -16.68 | in-in | in | 9.357 | Saltbr-in | 2.613 | HRD-in | -69.18, -45.26 | 74.92, -7.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.827 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.77, 169.88 | APE9-dihe-na | 74.29, 146.1 | APE8-dihe-in | -68.67, 142.33 | APE8-rot-in | 277.43 | APE67-dihe-in | -61.53, -28.29 | -54.62, -46.41 | APE12-dist-in | 12.499 | APE11-dist-in | 11.435 | APE10-dist-in | 6.965 | APE9-dist-in | 3.064 | None | PTR321 | PTR321 | XRAY | 2.4 | 0.186 | 0.23 | A | 382 | 347 | 0 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2vx3 | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 2VX3B | Q13627 | 135 | 480 | 763.0 | D15:600 | Type1 | Active | DFGin | 7.264 | 15.037 | BLAminus | -122.56, -178.04 | 63.15, 68.41 | -88.18, 26.58 | 286.19, 82.05 | -63.3, -25.27 | in-in | in | 9.323 | Saltbr-in | 2.487 | HRD-in | -63.29, -48.28 | 78.74, -5.5 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.884 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.98, 169.63 | APE9-dihe-na | 73.35, 142.01 | APE8-dihe-in | -64.13, 145.91 | APE8-rot-in | 293.73 | APE67-dihe-in | -61.18, -25.64 | -59.75, -45.87 | APE12-dist-in | 12.788 | APE11-dist-in | 11.481 | APE10-dist-in | 7.216 | APE9-dist-in | 3.173 | None | PTR321 | PTR321 | XRAY | 2.4 | 0.186 | 0.23 | B | 382 | 341 | 5 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2vx3 | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 2VX3C | Q13627 | 135 | 480 | 763.0 | D15:600 | Type1 | Active | DFGin | 7.171 | 15.076 | BLAminus | -121.44, 178.92 | 62.09, 79.8 | -99.68, 23.42 | 286.42, 75.22 | -71.85, -9.09 | in-in | in | 9.284 | Saltbr-in | 2.559 | HRD-in | -69.05, -51.28 | 81.08, -2.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.848 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.91, 169.36 | APE9-dihe-na | 73.6, 142.61 | APE8-dihe-in | -69.05, 142.27 | APE8-rot-in | 289.71 | APE67-dihe-in | -57.92, -27.82 | -52.31, -50.36 | APE12-dist-in | 12.693 | APE11-dist-in | 11.469 | APE10-dist-in | 7.054 | APE9-dist-in | 3.198 | None | PTR321 | PTR321 | XRAY | 2.4 | 0.186 | 0.23 | C | 382 | 339 | 7 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2vx3 | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 2VX3D | Q13627 | 135 | 480 | 763.0 | D15:600 | Type1 | Active | DFGin | 7.127 | 15.124 | BLAminus | -119.03, 173.28 | 66.12, 79.97 | -97.89, 24.65 | 287.18, 77.93 | -62.52, -22.35 | in-in | in | 9.434 | Saltbr-in | 2.837 | HRD-in | -59.24, -53.5 | 80.78, -1.27 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.821 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.8, 170.17 | APE9-dihe-na | 73.1, 153.08 | APE8-dihe-in | -81.31, 142.62 | APE8-rot-in | 292.88 | APE67-dihe-in | -60.26, -27.62 | -52.95, -48.14 | APE12-dist-in | 12.928 | APE11-dist-in | 11.48 | APE10-dist-in | 7.18 | APE9-dist-in | 3.148 | None | PTR321 | PTR321 | XRAY | 2.4 | 0.186 | 0.23 | D | 382 | 343 | 3 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2vx3 | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 2WO6A | Q13627 | 133 | 481 | 763.0 | D15:60600 | Type1 | Active | DFGin | 7.448 | 15.138 | BLAminus | -113.71, 170.1 | 69.22, 79.01 | -93.27, 30.89 | 281.47, 79.67 | -74.92, -25.98 | in-in | in | 8.538 | Saltbr-in | 2.478 | HRD-in | -60.74, -47.85 | 77.07, -4.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.791 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -109.22, 165.87 | APE9-dihe-na | 75.78, 143.18 | APE8-dihe-in | -71.63, 143.35 | APE8-rot-in | 298.65 | APE67-dihe-in | -54.81, -27.06 | -54.61, -51.13 | APE12-dist-in | 13.979 | APE11-dist-in | 11.967 | APE10-dist-in | 7.387 | APE9-dist-in | 3.275 | None | PTR321 | PTR321 | XRAY | 2.5 | 0.19 | 0.229 | A | 382 | 345 | 4 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2wo6 | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 2WO6B | Q13627 | 136 | 480 | 763.0 | D15:60600 | Type1 | Active | DFGin | 7.392 | 15.045 | BLAminus | -114.82, 170.21 | 64.99, 84.74 | -96.3, 34.41 | 283.13, 77.19 | -78.24, -22.43 | in-in | in | 9.207 | Saltbr-in | 2.725 | HRD-in | -63.58, -44.58 | 74.08, -1.57 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.791 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.01, 169.27 | APE9-dihe-na | 76.89, 144.45 | APE8-dihe-in | -76.49, 136.75 | APE8-rot-in | 283.78 | APE67-dihe-in | -66.31, -25.74 | -49.43, -39.9 | APE12-dist-in | 12.633 | APE11-dist-in | 11.105 | APE10-dist-in | 6.823 | APE9-dist-in | 3.096 | None | PTR321 | PTR321 | XRAY | 2.5 | 0.19 | 0.229 | B | 382 | 340 | 5 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2wo6 | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| CMGC | CDKL1 | CDKL1_HUMAN | 4AGUA | Q00532 | 2 | 291 | 357.0 | D15:500 | Type1 | None | DFGin | 6.926 | 15.225 | BLAminus | -125.36, -173.19 | 61.0, 84.36 | -106.79, 0.32 | 274.19, 82.71 | -54.94, -33.89 | in-in | in | 8.329 | Saltbr-in | 2.668 | HRD-in | -62.63, -48.4 | 73.42, -8.74 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.806 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 138.22 | APE8-rot-in | 301.17 | APE67-dihe-in | -58.09, -27.23 | -56.92, -32.3 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | T159D,Y161E | None | None | XRAY | 2.4 | 0.189 | 0.226 | A | 311 | 277 | 13 | 0 | 0 | 12 | [[4, 287]] | 1.0 | 4agu | Homo sapiens | CMGC_CDKL1_HUMAN | CMGC | 2.9e-80 | 275.7 | 1 | 301 | 301 | 143 | 144 | 145 | 147 | 149 | 33 | 51 | 55 | 123 | 125 | 124 | 126 | 184 | 171 | 166 | 165 | 164 | 163 | 162 | 161 | 160 | 81 | Cyclin-dependent kinase-like 1 |
| CMGC | CDKL1 | CDKL1_HUMAN | 4AGUB | Q00532 | 3 | 292 | 357.0 | D15:500 | Type1 | None | DFGin | 6.911 | 15.242 | BLAminus | -123.13, -174.59 | 61.67, 77.11 | -99.83, 8.36 | 278.04, 80.77 | -62.15, -31.07 | in-in | in | 8.312 | Saltbr-in | 2.668 | HRD-in | -65.94, -47.41 | 70.79, -7.65 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.762 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 133.96 | APE8-rot-in | 300.0 | APE67-dihe-in | -56.83, -27.96 | -64.83, -28.69 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | T159D,Y161E | None | None | XRAY | 2.4 | 0.189 | 0.226 | B | 311 | 276 | 14 | 0 | 0 | 12 | [[4, 287]] | 1.0 | 4agu | Homo sapiens | CMGC_CDKL1_HUMAN | CMGC | 2.9e-80 | 275.7 | 1 | 301 | 301 | 143 | 144 | 145 | 147 | 149 | 33 | 51 | 55 | 123 | 125 | 124 | 126 | 184 | 171 | 166 | 165 | 164 | 163 | 162 | 161 | 160 | 81 | Cyclin-dependent kinase-like 1 |
| CMGC | CDKL1 | CDKL1_HUMAN | 4AGUC | Q00532 | 2 | 291 | 357.0 | D15:500 | Type1 | None | DFGin | 7.076 | 15.076 | BLAminus | -126.2, -170.17 | 57.04, 81.0 | -105.59, 6.66 | 281.53, 85.88 | -54.99, -37.13 | in-in | in | 8.283 | Saltbr-in | 2.658 | HRD-in | -56.25, -49.02 | 74.36, -3.78 | in-in-none | SNCiin | in-none | ActLoopNT-in | 2.791 | ActLoopCT-none | nonTYR | APEdihe_aanii | APEdist_nnnn | APE10-dihe-na | 999.0, 999.0 | APE9-dihe-na | 999.0, 999.0 | APE8-dihe-none | 999.0, 127.06 | APE8-rot-in | 293.41 | APE67-dihe-in | -52.47, -36.63 | -43.96, -43.49 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-none | 999.0 | APE9-dist-none | 999.0 | T159D,Y161E | None | None | XRAY | 2.4 | 0.189 | 0.226 | C | 311 | 278 | 12 | 0 | 0 | 12 | [[4, 287]] | 1.0 | 4agu | Homo sapiens | CMGC_CDKL1_HUMAN | CMGC | 2.9e-80 | 275.7 | 1 | 301 | 301 | 143 | 144 | 145 | 147 | 149 | 33 | 51 | 55 | 123 | 125 | 124 | 126 | 184 | 171 | 166 | 165 | 164 | 163 | 162 | 161 | 160 | 81 | Cyclin-dependent kinase-like 1 |
| CMGC | DYRK1A | DYR1A_HUMAN | 2VX3A | Q13627 | 135 | 481 | 763.0 | D15:600 | Type1 | Active | DFGin | 7.177 | 14.936 | BLAminus | -117.81, 179.58 | 65.92, 72.63 | -91.66, 22.61 | 288.71, 80.01 | -64.63, -16.68 | in-in | in | 9.357 | Saltbr-in | 2.613 | HRD-in | -69.18, -45.26 | 74.92, -7.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.827 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.77, 169.88 | APE9-dihe-na | 74.29, 146.1 | APE8-dihe-in | -68.67, 142.33 | APE8-rot-in | 277.43 | APE67-dihe-in | -61.53, -28.29 | -54.62, -46.41 | APE12-dist-in | 12.499 | APE11-dist-in | 11.435 | APE10-dist-in | 6.965 | APE9-dist-in | 3.064 | None | PTR321 | PTR321 | XRAY | 2.4 | 0.186 | 0.23 | A | 382 | 347 | 0 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2vx3 | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 2VX3B | Q13627 | 135 | 480 | 763.0 | D15:600 | Type1 | Active | DFGin | 7.264 | 15.037 | BLAminus | -122.56, -178.04 | 63.15, 68.41 | -88.18, 26.58 | 286.19, 82.05 | -63.3, -25.27 | in-in | in | 9.323 | Saltbr-in | 2.487 | HRD-in | -63.29, -48.28 | 78.74, -5.5 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.884 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.98, 169.63 | APE9-dihe-na | 73.35, 142.01 | APE8-dihe-in | -64.13, 145.91 | APE8-rot-in | 293.73 | APE67-dihe-in | -61.18, -25.64 | -59.75, -45.87 | APE12-dist-in | 12.788 | APE11-dist-in | 11.481 | APE10-dist-in | 7.216 | APE9-dist-in | 3.173 | None | PTR321 | PTR321 | XRAY | 2.4 | 0.186 | 0.23 | B | 382 | 341 | 5 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2vx3 | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 2VX3C | Q13627 | 135 | 480 | 763.0 | D15:600 | Type1 | Active | DFGin | 7.171 | 15.076 | BLAminus | -121.44, 178.92 | 62.09, 79.8 | -99.68, 23.42 | 286.42, 75.22 | -71.85, -9.09 | in-in | in | 9.284 | Saltbr-in | 2.559 | HRD-in | -69.05, -51.28 | 81.08, -2.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.848 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -141.91, 169.36 | APE9-dihe-na | 73.6, 142.61 | APE8-dihe-in | -69.05, 142.27 | APE8-rot-in | 289.71 | APE67-dihe-in | -57.92, -27.82 | -52.31, -50.36 | APE12-dist-in | 12.693 | APE11-dist-in | 11.469 | APE10-dist-in | 7.054 | APE9-dist-in | 3.198 | None | PTR321 | PTR321 | XRAY | 2.4 | 0.186 | 0.23 | C | 382 | 339 | 7 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2vx3 | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 2VX3D | Q13627 | 135 | 480 | 763.0 | D15:600 | Type1 | Active | DFGin | 7.127 | 15.124 | BLAminus | -119.03, 173.28 | 66.12, 79.97 | -97.89, 24.65 | 287.18, 77.93 | -62.52, -22.35 | in-in | in | 9.434 | Saltbr-in | 2.837 | HRD-in | -59.24, -53.5 | 80.78, -1.27 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.821 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -128.8, 170.17 | APE9-dihe-na | 73.1, 153.08 | APE8-dihe-in | -81.31, 142.62 | APE8-rot-in | 292.88 | APE67-dihe-in | -60.26, -27.62 | -52.95, -48.14 | APE12-dist-in | 12.928 | APE11-dist-in | 11.48 | APE10-dist-in | 7.18 | APE9-dist-in | 3.148 | None | PTR321 | PTR321 | XRAY | 2.4 | 0.186 | 0.23 | D | 382 | 343 | 3 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2vx3 | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 2WO6A | Q13627 | 133 | 481 | 763.0 | D15:60600 | Type1 | Active | DFGin | 7.448 | 15.138 | BLAminus | -113.71, 170.1 | 69.22, 79.01 | -93.27, 30.89 | 281.47, 79.67 | -74.92, -25.98 | in-in | in | 8.538 | Saltbr-in | 2.478 | HRD-in | -60.74, -47.85 | 77.07, -4.65 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.791 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -109.22, 165.87 | APE9-dihe-na | 75.78, 143.18 | APE8-dihe-in | -71.63, 143.35 | APE8-rot-in | 298.65 | APE67-dihe-in | -54.81, -27.06 | -54.61, -51.13 | APE12-dist-in | 13.979 | APE11-dist-in | 11.967 | APE10-dist-in | 7.387 | APE9-dist-in | 3.275 | None | PTR321 | PTR321 | XRAY | 2.5 | 0.19 | 0.229 | A | 382 | 345 | 4 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2wo6 | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| CMGC | DYRK1A | DYR1A_HUMAN | 2WO6B | Q13627 | 136 | 480 | 763.0 | D15:60600 | Type1 | Active | DFGin | 7.392 | 15.045 | BLAminus | -114.82, 170.21 | 64.99, 84.74 | -96.3, 34.41 | 283.13, 77.19 | -78.24, -22.43 | in-in | in | 9.207 | Saltbr-in | 2.725 | HRD-in | -63.58, -44.58 | 74.08, -1.57 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.791 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.01, 169.27 | APE9-dihe-na | 76.89, 144.45 | APE8-dihe-in | -76.49, 136.75 | APE8-rot-in | 283.78 | APE67-dihe-in | -66.31, -25.74 | -49.43, -39.9 | APE12-dist-in | 12.633 | APE11-dist-in | 11.105 | APE10-dist-in | 6.823 | APE9-dist-in | 3.096 | None | PTR321 | PTR321 | XRAY | 2.5 | 0.19 | 0.229 | B | 382 | 340 | 5 | 0 | 0 | 0 | [[159, 479]] | 1.0 | 2wo6 | Homo sapiens | CMGC_DYRK1A_HUMAN | CMGC | 1e-90 | 310.0 | 1 | 301 | 301 | 306 | 307 | 308 | 310 | 312 | 188 | 203 | 207 | 284 | 286 | 285 | 287 | 343 | 331 | 326 | 325 | 324 | 323 | 322 | 321 | 320 | 239 | Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
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