Ligand: 7GV

Total number of chains: 2
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin ABAminus 2 100.0% 5TQ6A

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein
TYR JAK2-2 JAK2_HUMAN 5TQ6A 2.06 Inactive DFGin‑ABAminus in-in in-none TYR APEdihe_niiai APEdist_aaai 7GV Type1 843 - 1132 0 PTR1007,PTR1008 M1073S,F1076T Tyrosine-protein kinase JAK2
TYR JAK2-2 JAK2_HUMAN 5TQ6B 2.06 Inactive DFGin‑ABAminus in-in in-none TYR APEdihe_nniai APEdist_aaai 7GV Type1 843 - 1130 0 PTR1007,PTR1008 M1073S,F1076T Tyrosine-protein kinase JAK2

Ligand: 7GV

Total number of chains: 2
Active chains: 0
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin ABAminus 2 100.0% 5TQ6A

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism
TYR JAK2-2 JAK2_HUMAN 5TQ6A 2.06 Inactive DFGin‑ABAminus in-in in-none TYR APEdihe_niiai APEdist_aaai 7GV Type1 843 - 1132 0 PTR1007,PTR1008 M1073S,F1076T Tyrosine-protein kinase JAK2 Homo sapiens
TYR JAK2-2 JAK2_HUMAN 5TQ6B 2.06 Inactive DFGin‑ABAminus in-in in-none TYR APEdihe_nniai APEdist_aaai 7GV Type1 843 - 1130 0 PTR1007,PTR1008 M1073S,F1076T Tyrosine-protein kinase JAK2 Homo sapiens

Ligand: 7GV

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Family Gene UniprotID PDB Resolution Activity Spatial-Dihedral Chelix-SaltBridge ActLoopNT-ActLoopCT APEtype APEdihe APEdist Ligand Ligand Type Residues in structure Unresolved residues in A-loop Phosphorylation Mutation Protein Organism