| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4RWKA | P11362 | 458 | 764 | 822.0 | 66T:60801 | Type1 | Inactive | DFGin | 5.334 | 13.4485 | BLAplus | -119.61, 171.78 | 43.5, 42.06 | -91.27, -13.97 | 55.41, 85.99 | -97.85, 1.35 | in-in | in | 8.3001 | Saltbr-in | 2.8581 | HRD-in | -72.97, -43.98 | 66.64, 7.94 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.6119 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -132.9, 130.16 | APE9-dihe-in | -81.93, 117.68 | APE8-dihe-out | -73.74, -2.4 | APE8-rot-na | 340.19 | APE67-dihe-in | -78.12, -6.2 | -84.98, -15.3 | APE12-dist-na | 17.0094 | APE11-dist-na | 18.9505 | APE10-dist-na | 16.7093 | APE9-dist-out | 11.0044 | C488A,V561M,C584S | None | None | XRAY | 2.982 | 0.244 | 0.299 | A | 317.0 | 307.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 4rwk | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWKB | P11362 | 459 | 763 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.7367 | 13.232 | BLAplus | -119.15, 169.82 | 41.98, 44.21 | -90.47, -9.61 | 54.08, 84.94 | -94.37, 2.45 | in-in | in | 8.4157 | Saltbr-in | 3.448 | HRD-in | -74.45, -44.2 | 66.06, 8.62 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -133.04, 131.77 | APE9-dihe-in | -79.69, 122.84 | APE8-dihe-out | -69.38, -1.04 | APE8-rot-na | 339.66 | APE67-dihe-in | -75.83, -3.81 | -84.39, -12.82 | APE12-dist-na | 999.0 | APE11-dist-na | 21.9267 | APE10-dist-na | 19.8348 | APE9-dist-out | 11.6466 | C488A,V561M,C584S | None | None | XRAY | 2.982 | 0.244 | 0.299 | B | 317.0 | 282.0 | 23 | 30 | 23 | 7 | [[478, 756]] | 1.0 | 4rwk | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V05A | P11362 | 464 | 765 | 822.0 | 66T:1769 | Type1.5_Back | Inactive | DFGin | 5.4734 | 13.4201 | BLAplus | -110.72, 173.08 | 50.09, 39.57 | -95.62, -19.67 | 60.09, 83.48 | -87.99, 3.34 | in-in | in | 8.0484 | Saltbr-in | 2.7499 | HRD-in | -64.72, -51.32 | 77.65, -23.6 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.3021 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -98.91, 158.86 | APE9-dihe-in | -104.86, 116.5 | APE8-dihe-out | -57.09, -23.19 | APE8-rot-na | 335.63 | APE67-dihe-in | -66.78, -18.31 | -54.95, -24.99 | APE12-dist-na | 20.8412 | APE11-dist-na | 21.8076 | APE10-dist-na | 19.9108 | APE9-dist-out | 11.6016 | None | None | None | XRAY | 2.57 | 0.196 | 0.256 | A | 309.0 | 287.0 | 15 | 30 | 26 | 4 | [[478, 756]] | 1.0 | 4v05 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V05B | P11362 | 459 | 764 | 822.0 | 66T:1767 | Type1.5_Back | Inactive | DFGin | 5.4267 | 13.0724 | BLAplus | -110.08, 173.06 | 48.31, 47.35 | -106.86, -10.85 | 58.74, 86.16 | -77.17, -18.0 | in-in | in | 7.8311 | Saltbr-in | 2.9832 | HRD-in | -65.29, -47.82 | 74.06, -21.09 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.03, 160.1 | APE9-dihe-in | -100.97, 109.95 | APE8-dihe-out | -53.4, -23.19 | APE8-rot-na | 333.98 | APE67-dihe-in | -59.05, -11.55 | -51.93, -35.21 | APE12-dist-na | 21.3913 | APE11-dist-na | 22.0888 | APE10-dist-na | 20.5381 | APE9-dist-out | 11.4653 | None | None | None | XRAY | 2.57 | 0.196 | 0.256 | B | 309.0 | 286.0 | 20 | 30 | 26 | 4 | [[478, 756]] | 1.0 | 4v05 | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4WUNA | P11362 | 465 | 765 | 822.0 | 66T:801 | Type1.5_Back | Inactive | DFGin | 5.3591 | 13.2871 | BLAplus | -114.51, 167.45 | 61.45, 33.19 | -92.75, -3.72 | 56.8, 81.8 | -94.63, -9.82 | in-in | in | 7.9245 | Saltbr-in | 2.9429 | HRD-in | -77.57, -50.47 | 80.03, -11.41 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -31.68 | APE8-rot-na | 335.8 | APE67-dihe-in | -71.2, -7.75 | -54.8, -30.29 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.65 | 0.226 | 0.247 | A | 311.0 | 282.0 | 19 | 30 | 12 | 18 | [[478, 756]] | 1.0 | 4wun | TYR_FGFR1_HUMAN | TYR | 1.5e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4WUNB | P11362 | 461 | 762 | 822.0 | 66T:801 | Type1.5_Back | Inactive | DFGin | 5.2393 | 13.1038 | BLAplus | -116.49, 163.26 | 61.87, 38.6 | -99.56, -5.62 | 55.6, 83.98 | -99.35, -2.08 | in-in | in | 7.7038 | Saltbr-in | 2.6666 | HRD-in | -74.96, -47.89 | 70.35, -11.28 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 81.94 | APE8-dihe-out | -59.03, -20.07 | APE8-rot-na | 4.38 | APE67-dihe-in | -66.47, -11.9 | -63.08, -22.04 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2021 | None | None | None | XRAY | 1.65 | 0.226 | 0.247 | B | 311.0 | 268.0 | 34 | 30 | 13 | 17 | [[478, 756]] | 1.0 | 4wun | TYR_FGFR1_HUMAN | TYR | 1.5e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWJA | P11362 | 458 | 764 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.2638 | 13.5569 | BLAplus | -111.1, 165.72 | 44.3, 59.14 | -104.5, -7.94 | 52.98, 85.2 | -108.93, 18.9 | in-in | in | 8.0637 | Saltbr-in | 3.1247 | HRD-in | -76.03, -43.68 | 72.99, -8.16 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9816 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.41, 138.95 | APE9-dihe-in | -108.01, 100.05 | APE8-dihe-out | -61.04, -14.23 | APE8-rot-na | 22.4 | APE67-dihe-in | -81.18, -2.01 | -65.12, -23.42 | APE12-dist-na | 19.4256 | APE11-dist-na | 20.4566 | APE10-dist-na | 17.046 | APE9-dist-out | 11.3201 | C488A,C584S | None | None | XRAY | 2.489 | 0.204 | 0.25 | A | 317.0 | 306.0 | 1 | 30 | 29 | 1 | [[478, 756]] | 1.0 | 4rwj | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWJB | P11362 | 459 | 763 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.3065 | 13.0754 | BLAplus | -111.81, 166.65 | 44.09, 58.11 | -104.8, -5.62 | 52.57, 84.61 | -105.75, 19.27 | in-in | in | 7.9338 | Saltbr-in | 2.8347 | HRD-in | -75.88, -44.44 | 70.84, -6.0 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.6, 139.99 | APE9-dihe-in | -106.55, 102.92 | APE8-dihe-out | -58.58, -14.6 | APE8-rot-na | 336.03 | APE67-dihe-in | -80.58, -2.45 | -66.06, -21.44 | APE12-dist-na | 999.0 | APE11-dist-na | 21.7066 | APE10-dist-na | 18.4779 | APE9-dist-out | 11.5466 | C488A,C584S | None | None | XRAY | 2.489 | 0.204 | 0.25 | B | 317.0 | 282.0 | 23 | 30 | 20 | 10 | [[478, 756]] | 1.0 | 4rwj | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR1 | FGFR1_HUMAN | 4RWKA | P11362 | 458 | 764 | 822.0 | 66T:60801 | Type1 | Inactive | DFGin | 5.334 | 13.4485 | BLAplus | -119.61, 171.78 | 43.5, 42.06 | -91.27, -13.97 | 55.41, 85.99 | -97.85, 1.35 | in-in | in | 8.3001 | Saltbr-in | 2.8581 | HRD-in | -72.97, -43.98 | 66.64, 7.94 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.6119 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -132.9, 130.16 | APE9-dihe-in | -81.93, 117.68 | APE8-dihe-out | -73.74, -2.4 | APE8-rot-na | 340.19 | APE67-dihe-in | -78.12, -6.2 | -84.98, -15.3 | APE12-dist-na | 17.0094 | APE11-dist-na | 18.9505 | APE10-dist-na | 16.7093 | APE9-dist-out | 11.0044 | C488A,V561M,C584S | None | None | XRAY | 2.982 | 0.244 | 0.299 | A | 317.0 | 307.0 | 0 | 30 | 30 | 0 | [[478, 756]] | 1.0 | 4rwk | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWKB | P11362 | 459 | 763 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.7367 | 13.232 | BLAplus | -119.15, 169.82 | 41.98, 44.21 | -90.47, -9.61 | 54.08, 84.94 | -94.37, 2.45 | in-in | in | 8.4157 | Saltbr-in | 3.448 | HRD-in | -74.45, -44.2 | 66.06, 8.62 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -133.04, 131.77 | APE9-dihe-in | -79.69, 122.84 | APE8-dihe-out | -69.38, -1.04 | APE8-rot-na | 339.66 | APE67-dihe-in | -75.83, -3.81 | -84.39, -12.82 | APE12-dist-na | 999.0 | APE11-dist-na | 21.9267 | APE10-dist-na | 19.8348 | APE9-dist-out | 11.6466 | C488A,V561M,C584S | None | None | XRAY | 2.982 | 0.244 | 0.299 | B | 317.0 | 282.0 | 23 | 30 | 23 | 7 | [[478, 756]] | 1.0 | 4rwk | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 8.4e-105 | 355.7 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V05A | P11362 | 464 | 765 | 822.0 | 66T:1769 | Type1.5_Back | Inactive | DFGin | 5.4734 | 13.4201 | BLAplus | -110.72, 173.08 | 50.09, 39.57 | -95.62, -19.67 | 60.09, 83.48 | -87.99, 3.34 | in-in | in | 8.0484 | Saltbr-in | 2.7499 | HRD-in | -64.72, -51.32 | 77.65, -23.6 | in-out-out | SNCioo | out-out | ActLoopNT-out | 8.3021 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -98.91, 158.86 | APE9-dihe-in | -104.86, 116.5 | APE8-dihe-out | -57.09, -23.19 | APE8-rot-na | 335.63 | APE67-dihe-in | -66.78, -18.31 | -54.95, -24.99 | APE12-dist-na | 20.8412 | APE11-dist-na | 21.8076 | APE10-dist-na | 19.9108 | APE9-dist-out | 11.6016 | None | None | None | XRAY | 2.57 | 0.196 | 0.256 | A | 309.0 | 287.0 | 15 | 30 | 26 | 4 | [[478, 756]] | 1.0 | 4v05 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4V05B | P11362 | 459 | 764 | 822.0 | 66T:1767 | Type1.5_Back | Inactive | DFGin | 5.4267 | 13.0724 | BLAplus | -110.08, 173.06 | 48.31, 47.35 | -106.86, -10.85 | 58.74, 86.16 | -77.17, -18.0 | in-in | in | 7.8311 | Saltbr-in | 2.9832 | HRD-in | -65.29, -47.82 | 74.06, -21.09 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -104.03, 160.1 | APE9-dihe-in | -100.97, 109.95 | APE8-dihe-out | -53.4, -23.19 | APE8-rot-na | 333.98 | APE67-dihe-in | -59.05, -11.55 | -51.93, -35.21 | APE12-dist-na | 21.3913 | APE11-dist-na | 22.0888 | APE10-dist-na | 20.5381 | APE9-dist-out | 11.4653 | None | None | None | XRAY | 2.57 | 0.196 | 0.256 | B | 309.0 | 286.0 | 20 | 30 | 26 | 4 | [[478, 756]] | 1.0 | 4v05 | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.4e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4WUNA | P11362 | 465 | 765 | 822.0 | 66T:801 | Type1.5_Back | Inactive | DFGin | 5.3591 | 13.2871 | BLAplus | -114.51, 167.45 | 61.45, 33.19 | -92.75, -3.72 | 56.8, 81.8 | -94.63, -9.82 | in-in | in | 7.9245 | Saltbr-in | 2.9429 | HRD-in | -77.57, -50.47 | 80.03, -11.41 | in-none-none | SNCinn | none-none | ActLoopNT-none | 999.0 | ActLoopCT-none | TYR | APEdihe_nnnai | APEdist_aaan | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 999.0 | APE8-dihe-none | 999.0, -31.68 | APE8-rot-na | 335.8 | APE67-dihe-in | -71.2, -7.75 | -54.8, -30.29 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-none | 999.0 | None | None | None | XRAY | 1.65 | 0.226 | 0.247 | A | 311.0 | 282.0 | 19 | 30 | 12 | 18 | [[478, 756]] | 1.0 | 4wun | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.5e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4WUNB | P11362 | 461 | 762 | 822.0 | 66T:801 | Type1.5_Back | Inactive | DFGin | 5.2393 | 13.1038 | BLAplus | -116.49, 163.26 | 61.87, 38.6 | -99.56, -5.62 | 55.6, 83.98 | -99.35, -2.08 | in-in | in | 7.7038 | Saltbr-in | 2.6666 | HRD-in | -74.96, -47.89 | 70.35, -11.28 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nnoai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 81.94 | APE8-dihe-out | -59.03, -20.07 | APE8-rot-na | 4.38 | APE67-dihe-in | -66.47, -11.9 | -63.08, -22.04 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 11.2021 | None | None | None | XRAY | 1.65 | 0.226 | 0.247 | B | 311.0 | 268.0 | 34 | 30 | 13 | 17 | [[478, 756]] | 1.0 | 4wun | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.5e-104 | 354.9 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWJA | P11362 | 458 | 764 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.2638 | 13.5569 | BLAplus | -111.1, 165.72 | 44.3, 59.14 | -104.5, -7.94 | 52.98, 85.2 | -108.93, 18.9 | in-in | in | 8.0637 | Saltbr-in | 3.1247 | HRD-in | -76.03, -43.68 | 72.99, -8.16 | in-out-out | SNCioo | out-out | ActLoopNT-out | 7.9816 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.41, 138.95 | APE9-dihe-in | -108.01, 100.05 | APE8-dihe-out | -61.04, -14.23 | APE8-rot-na | 22.4 | APE67-dihe-in | -81.18, -2.01 | -65.12, -23.42 | APE12-dist-na | 19.4256 | APE11-dist-na | 20.4566 | APE10-dist-na | 17.046 | APE9-dist-out | 11.3201 | C488A,C584S | None | None | XRAY | 2.489 | 0.204 | 0.25 | A | 317.0 | 306.0 | 1 | 30 | 29 | 1 | [[478, 756]] | 1.0 | 4rwj | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| TYR | FGFR1 | FGFR1_HUMAN | 4RWJB | P11362 | 459 | 763 | 822.0 | 66T:60801 | Type1.5_Back | Inactive | DFGin | 5.3065 | 13.0754 | BLAplus | -111.81, 166.65 | 44.09, 58.11 | -104.8, -5.62 | 52.57, 84.61 | -105.75, 19.27 | in-in | in | 7.9338 | Saltbr-in | 2.8347 | HRD-in | -75.88, -44.44 | 70.84, -6.0 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_iioai | APEdist_aaao | APE10-dihe-in | -97.6, 139.99 | APE9-dihe-in | -106.55, 102.92 | APE8-dihe-out | -58.58, -14.6 | APE8-rot-na | 336.03 | APE67-dihe-in | -80.58, -2.45 | -66.06, -21.44 | APE12-dist-na | 999.0 | APE11-dist-na | 21.7066 | APE10-dist-na | 18.4779 | APE9-dist-out | 11.5466 | C488A,C584S | None | None | XRAY | 2.489 | 0.204 | 0.25 | B | 317.0 | 282.0 | 23 | 30 | 20 | 10 | [[478, 756]] | 1.0 | 4rwj | Homo sapiens | TYR_FGFR1_HUMAN | TYR | 1.6e-104 | 354.8 | 1.0 | 260.0 | 260.0 | 640 | 641 | 642 | 644 | 646 | 514 | 531 | 535 | 620 | 622 | 621 | 623.0 | 682 | 670 | 665 | 664 | 663 | 662 | 661 | 660 | 659 | 562 | Fibroblast growth factor receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|