Ligand: 54G

Total number of chains: 6
Active chains: 6
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 6 100.0% 6EHKA

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CMGC CSNK2A1 CSK21_HUMAN 5CU2A P68400 2 329 391.0 551:401,551:402,551:403,54G:404 Allosteric,Allosteric,Allosteric,Type1 Active DFGin 7.519 16.209 BLAminus -113.66, -177.31 51.16, 77.73 -89.83, 18.07 294.61, 78.9 -65.06, -23.44 in-in in 9.4 Saltbr-in 2.726 HRD-in -76.06, -45.19 67.54, 11.18 in-in-in SNCiii in-in ActLoopNT-in 2.952 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.97, 173.4 APE9-dihe-na 61.24, 163.5 APE8-dihe-in -94.92, 144.32 APE8-rot-in 296.75 APE67-dihe-in -65.7, -18.97 -31.9, -56.38 APE12-dist-in 12.602 APE11-dist-in 10.278 APE10-dist-in 6.078 APE9-dist-in 3.217 R21S None None XRAY 1.705 0.184 0.204 A 352 328 0 0 0 0 [[39, 324]] 1.0 5cu2 CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5CU0A P68400 2 328 391.0 54R:401,54R:402,54G:403 Allosteric,Allosteric,Type1 Active DFGin 7.474 16.33 BLAminus -108.17, 179.26 48.97, 78.44 -91.09, 19.74 296.33, 78.99 -64.41, -23.32 in-in in 9.491 Saltbr-in 2.665 HRD-in -71.9, -43.67 60.96, 17.7 in-in-in SNCiii in-in ActLoopNT-in 2.98 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.82, 163.88 APE9-dihe-na 66.04, 164.8 APE8-dihe-in -91.15, 141.16 APE8-rot-in 299.25 APE67-dihe-in -65.84, -25.23 -31.96, -52.91 APE12-dist-in 12.592 APE11-dist-in 10.152 APE10-dist-in 6.04 APE9-dist-in 3.308 R21S None None XRAY 2.18 0.206 0.236 A 352 327 0 0 0 0 [[39, 324]] 1.0 5cu0 CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5CU0B P68400 4 328 391.0 54R:401,54R:402,54G:403 Allosteric,Allosteric,Type1 Active DFGin 7.475 16.485 BLAminus -107.16, 178.28 49.21, 76.61 -87.02, 19.81 295.51, 81.17 -66.45, -22.95 in-in in 9.656 Saltbr-in 2.711 HRD-in -69.69, -44.08 61.46, 15.8 in-in-in SNCiii in-in ActLoopNT-in 2.979 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.17, 165.97 APE9-dihe-na 68.44, 158.46 APE8-dihe-in -87.49, 141.33 APE8-rot-in 294.87 APE67-dihe-in -70.65, -23.28 -32.83, -46.44 APE12-dist-in 12.493 APE11-dist-in 10.149 APE10-dist-in 5.928 APE9-dist-in 3.311 R21S None None XRAY 2.18 0.206 0.236 B 352 325 0 0 0 0 [[39, 324]] 1.0 5cu0 CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5CU2B P68400 3 327 391.0 551:401,551:402,54G:403 Allosteric,Allosteric,Type1 Active DFGin 7.484 16.361 BLAminus -112.75, -177.3 50.36, 74.97 -87.28, 18.57 295.0, 80.7 -65.4, -23.23 in-in in 9.495 Saltbr-in 2.765 HRD-in -74.03, -45.41 67.64, 11.27 in-in-in SNCiii in-in ActLoopNT-in 2.93 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.42, 172.71 APE9-dihe-na 62.21, 161.82 APE8-dihe-in -90.75, 143.8 APE8-rot-in 295.24 APE67-dihe-in -64.1, -19.98 -31.79, -58.09 APE12-dist-in 12.52 APE11-dist-in 10.243 APE10-dist-in 6.028 APE9-dist-in 3.208 R21S None None XRAY 1.705 0.184 0.204 B 352 325 0 0 0 0 [[39, 324]] 1.0 5cu2 CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5CSPA P68400 3 329 391.0 54G:401 Type1 Active DFGin 7.451 16.173 BLAminus -116.64, -179.3 51.58, 76.77 -89.31, 18.46 295.54, 83.4 -67.53, -21.61 in-in in 9.239 Saltbr-in 2.805 HRD-in -73.91, -47.86 69.29, 11.76 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.9, 170.74 APE9-dihe-na 59.4, 161.34 APE8-dihe-in -83.18, 147.47 APE8-rot-in 284.37 APE67-dihe-in -67.93, -17.25 -36.65, -56.55 APE12-dist-in 12.671 APE11-dist-in 10.255 APE10-dist-in 6.112 APE9-dist-in 3.273 R21S,K74A,K75A,K76A None None XRAY 1.5 0.164 0.186 A 328 327 0 0 0 0 [[39, 324]] 1.0 5csp CMGC_CSNK2A1_HUMAN CMGC 8.1e-69 238.0 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 6EHKA P68400 3 329 391.0 AUW:403,54G:404 Type1,Type1 Active DFGin 7.495 16.137 BLAminus -115.01, -177.46 49.41, 78.33 -90.39, 16.63 296.14, 78.36 -64.91, -22.64 in-in in 9.258 Saltbr-in 2.731 HRD-in -74.43, -45.83 68.89, 8.65 in-in-in SNCiii in-in ActLoopNT-in 2.946 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.67, 169.99 APE9-dihe-na 57.78, 156.66 APE8-dihe-in -80.85, 148.35 APE8-rot-in 290.21 APE67-dihe-in -72.54, -10.78 -36.07, -54.95 APE12-dist-in 12.842 APE11-dist-in 10.569 APE10-dist-in 6.403 APE9-dist-in 3.335 R21S,K74A,K75A,K76A None None XRAY 1.4 0.179 0.194 A 342 327 0 0 0 0 [[39, 324]] 1.0 6ehk CMGC_CSNK2A1_HUMAN CMGC 9.4e-69 237.9 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha

Ligand: 54G

Total number of chains: 6
Active chains: 6
Total number of genes: 1
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 6 100.0% 6EHKA

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Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
CMGC CSNK2A1 CSK21_HUMAN 5CU2A P68400 2 329 391.0 551:401,551:402,551:403,54G:404 Allosteric,Allosteric,Allosteric,Type1 Active DFGin 7.519 16.209 BLAminus -113.66, -177.31 51.16, 77.73 -89.83, 18.07 294.61, 78.9 -65.06, -23.44 in-in in 9.4 Saltbr-in 2.726 HRD-in -76.06, -45.19 67.54, 11.18 in-in-in SNCiii in-in ActLoopNT-in 2.952 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -133.97, 173.4 APE9-dihe-na 61.24, 163.5 APE8-dihe-in -94.92, 144.32 APE8-rot-in 296.75 APE67-dihe-in -65.7, -18.97 -31.9, -56.38 APE12-dist-in 12.602 APE11-dist-in 10.278 APE10-dist-in 6.078 APE9-dist-in 3.217 R21S None None XRAY 1.705 0.184 0.204 A 352 328 0 0 0 0 [[39, 324]] 1.0 5cu2 Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5CU0A P68400 2 328 391.0 54R:401,54R:402,54G:403 Allosteric,Allosteric,Type1 Active DFGin 7.474 16.33 BLAminus -108.17, 179.26 48.97, 78.44 -91.09, 19.74 296.33, 78.99 -64.41, -23.32 in-in in 9.491 Saltbr-in 2.665 HRD-in -71.9, -43.67 60.96, 17.7 in-in-in SNCiii in-in ActLoopNT-in 2.98 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.82, 163.88 APE9-dihe-na 66.04, 164.8 APE8-dihe-in -91.15, 141.16 APE8-rot-in 299.25 APE67-dihe-in -65.84, -25.23 -31.96, -52.91 APE12-dist-in 12.592 APE11-dist-in 10.152 APE10-dist-in 6.04 APE9-dist-in 3.308 R21S None None XRAY 2.18 0.206 0.236 A 352 327 0 0 0 0 [[39, 324]] 1.0 5cu0 Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5CU0B P68400 4 328 391.0 54R:401,54R:402,54G:403 Allosteric,Allosteric,Type1 Active DFGin 7.475 16.485 BLAminus -107.16, 178.28 49.21, 76.61 -87.02, 19.81 295.51, 81.17 -66.45, -22.95 in-in in 9.656 Saltbr-in 2.711 HRD-in -69.69, -44.08 61.46, 15.8 in-in-in SNCiii in-in ActLoopNT-in 2.979 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -136.17, 165.97 APE9-dihe-na 68.44, 158.46 APE8-dihe-in -87.49, 141.33 APE8-rot-in 294.87 APE67-dihe-in -70.65, -23.28 -32.83, -46.44 APE12-dist-in 12.493 APE11-dist-in 10.149 APE10-dist-in 5.928 APE9-dist-in 3.311 R21S None None XRAY 2.18 0.206 0.236 B 352 325 0 0 0 0 [[39, 324]] 1.0 5cu0 Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5CU2B P68400 3 327 391.0 551:401,551:402,54G:403 Allosteric,Allosteric,Type1 Active DFGin 7.484 16.361 BLAminus -112.75, -177.3 50.36, 74.97 -87.28, 18.57 295.0, 80.7 -65.4, -23.23 in-in in 9.495 Saltbr-in 2.765 HRD-in -74.03, -45.41 67.64, 11.27 in-in-in SNCiii in-in ActLoopNT-in 2.93 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -134.42, 172.71 APE9-dihe-na 62.21, 161.82 APE8-dihe-in -90.75, 143.8 APE8-rot-in 295.24 APE67-dihe-in -64.1, -19.98 -31.79, -58.09 APE12-dist-in 12.52 APE11-dist-in 10.243 APE10-dist-in 6.028 APE9-dist-in 3.208 R21S None None XRAY 1.705 0.184 0.204 B 352 325 0 0 0 0 [[39, 324]] 1.0 5cu2 Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 1.6e-69 240.4 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 5CSPA P68400 3 329 391.0 54G:401 Type1 Active DFGin 7.451 16.173 BLAminus -116.64, -179.3 51.58, 76.77 -89.31, 18.46 295.54, 83.4 -67.53, -21.61 in-in in 9.239 Saltbr-in 2.805 HRD-in -73.91, -47.86 69.29, 11.76 in-in-in SNCiii in-in ActLoopNT-in 2.938 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -132.9, 170.74 APE9-dihe-na 59.4, 161.34 APE8-dihe-in -83.18, 147.47 APE8-rot-in 284.37 APE67-dihe-in -67.93, -17.25 -36.65, -56.55 APE12-dist-in 12.671 APE11-dist-in 10.255 APE10-dist-in 6.112 APE9-dist-in 3.273 R21S,K74A,K75A,K76A None None XRAY 1.5 0.164 0.186 A 328 327 0 0 0 0 [[39, 324]] 1.0 5csp Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 8.1e-69 238.0 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha
CMGC CSNK2A1 CSK21_HUMAN 6EHKA P68400 3 329 391.0 AUW:403,54G:404 Type1,Type1 Active DFGin 7.495 16.137 BLAminus -115.01, -177.46 49.41, 78.33 -90.39, 16.63 296.14, 78.36 -64.91, -22.64 in-in in 9.258 Saltbr-in 2.731 HRD-in -74.43, -45.83 68.89, 8.65 in-in-in SNCiii in-in ActLoopNT-in 2.946 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -130.67, 169.99 APE9-dihe-na 57.78, 156.66 APE8-dihe-in -80.85, 148.35 APE8-rot-in 290.21 APE67-dihe-in -72.54, -10.78 -36.07, -54.95 APE12-dist-in 12.842 APE11-dist-in 10.569 APE10-dist-in 6.403 APE9-dist-in 3.335 R21S,K74A,K75A,K76A None None XRAY 1.4 0.179 0.194 A 342 327 0 0 0 0 [[39, 324]] 1.0 6ehk Homo sapiens CMGC_CSNK2A1_HUMAN CMGC 9.4e-69 237.9 1 301 301 174 175 176 178 180 68 81 85 153 155 154 156 214 201 196 195 194 193 192 191 190 114 Casein kinase II subunit alpha

Ligand: 54G

Total number of chains: 0
Active chains: 0
Total number of genes: 0
Spatial label Dihedral label Number of Chains Percent Representative

Hover over column headers for tooltip help

Group Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name