Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | ABL1 | ABL1_HUMAN | 2HZ4A | P00519 | 234 | 500 | 1130.0 | 4ST:501 | Allosteric | Inactive | DFGin | 6.899 | 13.314 | BLAminus | -141.07, -179.05 | 61.44, 74.68 | -93.23, 11.06 | 298.48, 103.02 | -47.37, -45.58 | in-out | in | 8.043 | Saltbr-out | 4.199 | HRD-in | -73.48, -44.6 | 66.11, 2.51 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.136 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -110.55, 127.23 | APE9-dihe-in | -112.0, 154.72 | APE8-dihe-in | -73.75, 92.13 | APE8-rot-na | 28.06 | APE67-dihe-in | -62.73, -9.15 | -43.63, -56.72 | APE12-dist-na | 15.433 | APE11-dist-na | 10.608 | APE10-dist-na | 12.472 | APE9-dist-in | 7.423 | None | None | None | XRAY | 2.8 | 0.22 | 0.285 | A | 273 | 262 | 5 | 0 | 0 | 0 | [[242, 495]] | 1.0 | 2hz4 | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1 | 260 | 260 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 2HZ4C | P00519 | 234 | 500 | 1130.0 | 4ST:501 | Allosteric | Active | DFGin | 7.109 | 13.517 | BLAminus | -106.9, 179.4 | 68.82, 76.0 | -90.83, 7.94 | 295.39, 93.15 | -43.83, -23.1 | in-in | in | 7.878 | Saltbr-in | 2.737 | HRD-in | -90.54, -43.68 | 68.76, 3.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -120.98, 153.91 | APE9-dihe-in | -143.05, 161.74 | APE8-dihe-in | -62.63, 109.18 | APE8-rot-na | 10.02 | APE67-dihe-in | -54.86, -29.12 | -56.69, -54.75 | APE12-dist-na | 14.951 | APE11-dist-na | 10.157 | APE10-dist-na | 13.134 | APE9-dist-in | 7.41 | None | None | None | XRAY | 2.8 | 0.22 | 0.285 | C | 273 | 259 | 8 | 0 | 0 | 0 | [[242, 495]] | 1.0 | 2hz4 | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1 | 260 | 260 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 2HZ4B | P00519 | 233 | 498 | 1130.0 | 4ST:501 | Type1 | Active | DFGin | 6.781 | 12.906 | BLAminus | -136.29, 178.03 | 62.62, 92.29 | -99.12, 17.06 | 306.64, 102.22 | -49.71, -38.7 | in-in | in | 8.114 | Saltbr-in | 2.713 | HRD-in | -96.51, -47.12 | 66.31, -5.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.105 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -93.77, 139.94 | APE9-dihe-in | -124.12, 153.4 | APE8-dihe-in | -60.98, 117.48 | APE8-rot-na | 25.18 | APE67-dihe-in | -77.16, -10.29 | -56.55, -40.66 | APE12-dist-na | 14.733 | APE11-dist-na | 10.004 | APE10-dist-na | 12.996 | APE9-dist-in | 7.129 | None | None | None | XRAY | 2.8 | 0.22 | 0.285 | B | 273 | 261 | 5 | 0 | 0 | 0 | [[242, 495]] | 1.0 | 2hz4 | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1 | 260 | 260 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | JAK3-2 | JAK3_HUMAN | 1YVJA | P52333 | 814 | 1103 | 1124.0 | 4ST:2000 | Type1 | Inactive | DFGin | 6.505 | 14.005 | BLAminus | -117.35, -176.34 | 48.83, 98.04 | -113.48, 29.61 | 287.79, 84.73 | -71.88, -20.61 | in-in | in | 8.618 | Saltbr-in | 2.837 | HRD-in | -75.54, -39.16 | 74.88, -34.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.832 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -96.81, -5.63 | APE9-dihe-in | -95.15, 159.49 | APE8-dihe-in | -47.0, 152.52 | APE8-rot-na | 325.56 | APE67-dihe-in | -77.97, 4.18 | -53.16, -16.76 | APE12-dist-na | 9.806 | APE11-dist-na | 6.854 | APE10-dist-na | 8.778 | APE9-dist-out | 8.2 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.55 | 0.204 | 0.254 | A | 290 | 290 | 0 | 0 | 0 | 0 | [[521, 779], [822, 1097]] | 2.0 | 1yvj | TYR_JAK3-2_HUMAN | TYR | 5.4e-81 | 277.7 | 1 | 260 | 260 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | PTK2 | FAK1_CHICK | 2J0MB | Q00944 | 414 | 686 | 1053.0 | 4ST:1687 | Type1 | Inactive | DFGin | 6.972 | 14.287 | None | -122.76, 167.67 | 145.4, -137.08 | -124.29, 100.35 | 290.36, 64.77 | -132.69, 154.11 | in-in | in | 7.468 | Saltbr-in | 2.443 | HRD-in | -71.25, -49.34 | 81.19, -3.46 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 132.23 | APE8-dihe-in | -85.72, 66.92 | APE8-rot-na | 31.09 | APE67-dihe-in | -64.84, -11.69 | -52.92, -44.76 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.379 | None | None | None | XRAY | 2.8 | 0.224 | 0.282 | B | 276 | 257 | 16 | 0 | 0 | 16 | [[422, 678]] | 1.0 | 2j0m | Gallus gallus | TYR_PTK2_CHICK | TYR | 3.3e-93 | 317.7 | 1 | 260 | 260 | 563 | 564 | 565 | 567 | 569 | 454 | 471 | 475 | 543 | 545 | 544 | 546 | 604 | 592 | 587 | 586 | 585 | 584 | 583 | 582 | 581 | 500 | Focal adhesion kinase 1 |
| TYR | PTK2 | FAK1_CHICK | 2J0JA | Q00944 | 35 | 686 | 1053.0 | 4ST:1687 | Type1 | Inactive | DFGin | 6.918 | 14.385 | None | -123.19, 169.5 | 101.29, -103.63 | 66.49, 28.41 | 317.16, 97.31 | -90.27, 177.52 | in-in | in | 8.119 | Saltbr-in | 2.703 | HRD-in | -78.32, -40.43 | 79.32, -8.22 | in-out-out | SNCioo | out-out | ActLoopNT-out | 12.463 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 124.84 | APE8-dihe-in | -80.69, 57.63 | APE8-rot-na | 26.07 | APE67-dihe-in | -61.42, -10.9 | -40.75, -50.86 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.849 | None | None | None | XRAY | 2.8 | 0.22 | 0.274 | A | 656 | 611 | 10 | 0 | 0 | 10 | [[422, 678]] | 1.0 | 2j0j | Gallus gallus | TYR_PTK2_CHICK | TYR | 3.1e-92 | 314.9 | 1 | 260 | 260 | 563 | 564 | 565 | 567 | 569 | 454 | 471 | 475 | 543 | 545 | 544 | 546 | 604 | 592 | 587 | 586 | 585 | 584 | 583 | 582 | 581 | 500 | Focal adhesion kinase 1 |
| TYR | PTK2 | FAK1_CHICK | 2J0KA | Q00944 | 35 | 686 | 1053.0 | 4ST:1687 | Type1 | Inactive | DFGin | 6.84 | 14.522 | None | -94.55, -93.91 | -78.14, -58.62 | 58.67, 36.74 | 310.17, 120.14 | -115.82, 158.23 | in-in | in | 8.167 | Saltbr-in | 2.834 | HRD-in | -98.8, -33.31 | 77.39, -21.17 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 52.29 | APE9-dihe-in | -82.72, 133.73 | APE8-dihe-in | -69.87, 64.39 | APE8-rot-na | 25.61 | APE67-dihe-in | -58.59, -19.95 | -50.1, -51.91 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.019 | APE9-dist-out | 8.81 | None | None | None | XRAY | 3.0 | 0.237 | 0.299 | A | 656 | 598 | 15 | 0 | 0 | 15 | [[422, 678]] | 1.0 | 2j0k | Gallus gallus | TYR_PTK2_CHICK | TYR | 1.5e-91 | 312.7 | 1 | 260 | 260 | 563 | 564 | 565 | 567 | 569 | 454 | 471 | 475 | 543 | 545 | 544 | 546 | 604 | 592 | 587 | 586 | 585 | 584 | 583 | 582 | 581 | 500 | Focal adhesion kinase 1 |
| TYR | PTK2 | FAK1_CHICK | 2J0KB | Q00944 | 35 | 686 | 1053.0 | 4ST:1687 | Type1 | Inactive | DFGin | 6.8 | 13.944 | None | -96.91, -85.38 | -80.15, -63.34 | 50.19, 5.1 | 328.51, 122.72 | -57.61, 145.44 | in-in | in | 8.042 | Saltbr-in | 3.114 | HRD-in | -78.83, -42.91 | 75.23, -10.09 | in-out-out | SNCioo | out-out | ActLoopNT-out | 10.513 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 135.8 | APE8-dihe-in | -80.14, 57.93 | APE8-rot-na | 30.91 | APE67-dihe-in | -67.94, -7.65 | -42.39, -46.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.247 | None | None | None | XRAY | 3.0 | 0.237 | 0.299 | B | 656 | 612 | 14 | 0 | 0 | 14 | [[422, 678]] | 1.0 | 2j0k | Gallus gallus | TYR_PTK2_CHICK | TYR | 1.5e-91 | 312.7 | 1 | 260 | 260 | 563 | 564 | 565 | 567 | 569 | 454 | 471 | 475 | 543 | 545 | 544 | 546 | 604 | 592 | 587 | 586 | 585 | 584 | 583 | 582 | 581 | 500 | Focal adhesion kinase 1 |
| TYR | ABL1 | ABL1_HUMAN | 2HZ4A | P00519 | 234 | 500 | 1130.0 | 4ST:501 | Allosteric | Inactive | DFGin | 6.899 | 13.314 | BLAminus | -141.07, -179.05 | 61.44, 74.68 | -93.23, 11.06 | 298.48, 103.02 | -47.37, -45.58 | in-out | in | 8.043 | Saltbr-out | 4.199 | HRD-in | -73.48, -44.6 | 66.11, 2.51 | out-in-in | SNCoii | in-in | ActLoopNT-in | 3.136 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -110.55, 127.23 | APE9-dihe-in | -112.0, 154.72 | APE8-dihe-in | -73.75, 92.13 | APE8-rot-na | 28.06 | APE67-dihe-in | -62.73, -9.15 | -43.63, -56.72 | APE12-dist-na | 15.433 | APE11-dist-na | 10.608 | APE10-dist-na | 12.472 | APE9-dist-in | 7.423 | None | None | None | XRAY | 2.8 | 0.22 | 0.285 | A | 273 | 262 | 5 | 0 | 0 | 0 | [[242, 495]] | 1.0 | 2hz4 | Homo sapiens | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1 | 260 | 260 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 2HZ4C | P00519 | 234 | 500 | 1130.0 | 4ST:501 | Allosteric | Active | DFGin | 7.109 | 13.517 | BLAminus | -106.9, 179.4 | 68.82, 76.0 | -90.83, 7.94 | 295.39, 93.15 | -43.83, -23.1 | in-in | in | 7.878 | Saltbr-in | 2.737 | HRD-in | -90.54, -43.68 | 68.76, 3.22 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.0 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -120.98, 153.91 | APE9-dihe-in | -143.05, 161.74 | APE8-dihe-in | -62.63, 109.18 | APE8-rot-na | 10.02 | APE67-dihe-in | -54.86, -29.12 | -56.69, -54.75 | APE12-dist-na | 14.951 | APE11-dist-na | 10.157 | APE10-dist-na | 13.134 | APE9-dist-in | 7.41 | None | None | None | XRAY | 2.8 | 0.22 | 0.285 | C | 273 | 259 | 8 | 0 | 0 | 0 | [[242, 495]] | 1.0 | 2hz4 | Homo sapiens | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1 | 260 | 260 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | ABL1 | ABL1_HUMAN | 2HZ4B | P00519 | 233 | 498 | 1130.0 | 4ST:501 | Type1 | Active | DFGin | 6.781 | 12.906 | BLAminus | -136.29, 178.03 | 62.62, 92.29 | -99.12, 17.06 | 306.64, 102.22 | -49.71, -38.7 | in-in | in | 8.114 | Saltbr-in | 2.713 | HRD-in | -96.51, -47.12 | 66.31, -5.28 | in-in-in | SNCiii | in-in | ActLoopNT-in | 3.105 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -93.77, 139.94 | APE9-dihe-in | -124.12, 153.4 | APE8-dihe-in | -60.98, 117.48 | APE8-rot-na | 25.18 | APE67-dihe-in | -77.16, -10.29 | -56.55, -40.66 | APE12-dist-na | 14.733 | APE11-dist-na | 10.004 | APE10-dist-na | 12.996 | APE9-dist-in | 7.129 | None | None | None | XRAY | 2.8 | 0.22 | 0.285 | B | 273 | 261 | 5 | 0 | 0 | 0 | [[242, 495]] | 1.0 | 2hz4 | Homo sapiens | TYR_ABL1_HUMAN | TYR | 2.2e-100 | 341.2 | 1 | 260 | 260 | 380 | 381 | 382 | 384 | 386 | 271 | 286 | 290 | 360 | 362 | 361 | 363 | 421 | 409 | 404 | 403 | 402 | 401 | 400 | 399 | 398 | 316 | Tyrosine-protein kinase ABL1 |
| TYR | JAK3-2 | JAK3_HUMAN | 1YVJA | P52333 | 814 | 1103 | 1124.0 | 4ST:2000 | Type1 | Inactive | DFGin | 6.505 | 14.005 | BLAminus | -117.35, -176.34 | 48.83, 98.04 | -113.48, 29.61 | 287.79, 84.73 | -71.88, -20.61 | in-in | in | 8.618 | Saltbr-in | 2.837 | HRD-in | -75.54, -39.16 | 74.88, -34.81 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.832 | ActLoopCT-out | TYR | APEdihe_oiiai | APEdist_aaao | APE10-dihe-out | -96.81, -5.63 | APE9-dihe-in | -95.15, 159.49 | APE8-dihe-in | -47.0, 152.52 | APE8-rot-na | 325.56 | APE67-dihe-in | -77.97, 4.18 | -53.16, -16.76 | APE12-dist-na | 9.806 | APE11-dist-na | 6.854 | APE10-dist-na | 8.778 | APE9-dist-out | 8.2 | None | PTR980,PTR981 | PTR980,PTR981 | XRAY | 2.55 | 0.204 | 0.254 | A | 290 | 290 | 0 | 0 | 0 | 0 | [[521, 779], [822, 1097]] | 2.0 | 1yvj | Homo sapiens | TYR_JAK3-2_HUMAN | TYR | 5.4e-81 | 277.7 | 1 | 260 | 260 | 966 | 967 | 968 | 970 | 972 | 855 | 871 | 875 | 946 | 948 | 947 | 949 | 1009 | 997 | 992 | 991 | 990 | 989 | 988 | 987 | 986 | 903 | Tyrosine-protein kinase JAK3 |
Hover over column headers for tooltip help
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | PTK2 | FAK1_CHICK | 2J0MB | Q00944 | 414 | 686 | 1053.0 | 4ST:1687 | Type1 | Inactive | DFGin | 6.972 | 14.287 | None | -122.76, 167.67 | 145.4, -137.08 | -124.29, 100.35 | 290.36, 64.77 | -132.69, 154.11 | in-in | in | 7.468 | Saltbr-in | 2.443 | HRD-in | -71.25, -49.34 | 81.19, -3.46 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 132.23 | APE8-dihe-in | -85.72, 66.92 | APE8-rot-na | 31.09 | APE67-dihe-in | -64.84, -11.69 | -52.92, -44.76 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.379 | None | None | None | XRAY | 2.8 | 0.224 | 0.282 | B | 276 | 257 | 16 | 0 | 0 | 16 | [[422, 678]] | 1.0 | 2j0m | Gallus gallus | TYR_PTK2_CHICK | TYR | 3.3e-93 | 317.7 | 1 | 260 | 260 | 563 | 564 | 565 | 567 | 569 | 454 | 471 | 475 | 543 | 545 | 544 | 546 | 604 | 592 | 587 | 586 | 585 | 584 | 583 | 582 | 581 | 500 | Focal adhesion kinase 1 |
| TYR | PTK2 | FAK1_CHICK | 2J0JA | Q00944 | 35 | 686 | 1053.0 | 4ST:1687 | Type1 | Inactive | DFGin | 6.918 | 14.385 | None | -123.19, 169.5 | 101.29, -103.63 | 66.49, 28.41 | 317.16, 97.31 | -90.27, 177.52 | in-in | in | 8.119 | Saltbr-in | 2.703 | HRD-in | -78.32, -40.43 | 79.32, -8.22 | in-out-out | SNCioo | out-out | ActLoopNT-out | 12.463 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 124.84 | APE8-dihe-in | -80.69, 57.63 | APE8-rot-na | 26.07 | APE67-dihe-in | -61.42, -10.9 | -40.75, -50.86 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.849 | None | None | None | XRAY | 2.8 | 0.22 | 0.274 | A | 656 | 611 | 10 | 0 | 0 | 10 | [[422, 678]] | 1.0 | 2j0j | Gallus gallus | TYR_PTK2_CHICK | TYR | 3.1e-92 | 314.9 | 1 | 260 | 260 | 563 | 564 | 565 | 567 | 569 | 454 | 471 | 475 | 543 | 545 | 544 | 546 | 604 | 592 | 587 | 586 | 585 | 584 | 583 | 582 | 581 | 500 | Focal adhesion kinase 1 |
| TYR | PTK2 | FAK1_CHICK | 2J0KA | Q00944 | 35 | 686 | 1053.0 | 4ST:1687 | Type1 | Inactive | DFGin | 6.84 | 14.522 | None | -94.55, -93.91 | -78.14, -58.62 | 58.67, 36.74 | 310.17, 120.14 | -115.82, 158.23 | in-in | in | 8.167 | Saltbr-in | 2.834 | HRD-in | -98.8, -33.31 | 77.39, -21.17 | in-none-out | SNCino | none-out | ActLoopNT-none | 999.0 | ActLoopCT-out | TYR | APEdihe_niiai | APEdist_aaao | APE10-dihe-none | 999.0, 52.29 | APE9-dihe-in | -82.72, 133.73 | APE8-dihe-in | -69.87, 64.39 | APE8-rot-na | 25.61 | APE67-dihe-in | -58.59, -19.95 | -50.1, -51.91 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 13.019 | APE9-dist-out | 8.81 | None | None | None | XRAY | 3.0 | 0.237 | 0.299 | A | 656 | 598 | 15 | 0 | 0 | 15 | [[422, 678]] | 1.0 | 2j0k | Gallus gallus | TYR_PTK2_CHICK | TYR | 1.5e-91 | 312.7 | 1 | 260 | 260 | 563 | 564 | 565 | 567 | 569 | 454 | 471 | 475 | 543 | 545 | 544 | 546 | 604 | 592 | 587 | 586 | 585 | 584 | 583 | 582 | 581 | 500 | Focal adhesion kinase 1 |
| TYR | PTK2 | FAK1_CHICK | 2J0KB | Q00944 | 35 | 686 | 1053.0 | 4ST:1687 | Type1 | Inactive | DFGin | 6.8 | 13.944 | None | -96.91, -85.38 | -80.15, -63.34 | 50.19, 5.1 | 328.51, 122.72 | -57.61, 145.44 | in-in | in | 8.042 | Saltbr-in | 3.114 | HRD-in | -78.83, -42.91 | 75.23, -10.09 | in-out-out | SNCioo | out-out | ActLoopNT-out | 10.513 | ActLoopCT-out | TYR | APEdihe_nniai | APEdist_aaao | APE10-dihe-none | 999.0, 999.0 | APE9-dihe-none | 999.0, 135.8 | APE8-dihe-in | -80.14, 57.93 | APE8-rot-na | 30.91 | APE67-dihe-in | -67.94, -7.65 | -42.39, -46.82 | APE12-dist-na | 999.0 | APE11-dist-na | 999.0 | APE10-dist-na | 999.0 | APE9-dist-out | 8.247 | None | None | None | XRAY | 3.0 | 0.237 | 0.299 | B | 656 | 612 | 14 | 0 | 0 | 14 | [[422, 678]] | 1.0 | 2j0k | Gallus gallus | TYR_PTK2_CHICK | TYR | 1.5e-91 | 312.7 | 1 | 260 | 260 | 563 | 564 | 565 | 567 | 569 | 454 | 471 | 475 | 543 | 545 | 544 | 546 | 604 | 592 | 587 | 586 | 585 | 584 | 583 | 582 | 581 | 500 | Focal adhesion kinase 1 |