| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| VRK2 | AF-Q86Y07-K1A | Q86Y07 | 21 | 323 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.9476 | 14.7984 | BLAminus | -119.05, 177.71 | 65.11, 69.16 | -80.5, 23.83 | 289.5, 88.67 | -62.34, -29.88 | in-in | in | 8.0198 | Saltbr-in | 2.6572 | HRD-in | -84.77, -50.44 | 77.78, 0.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.909 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -61.7, 143.45 | APE9-dihe-na | 96.44, -172.51 | APE8-dihe-in | -74.74, 115.77 | APE8-rot-in | 298.71 | APE67-dihe-in | -66.17, -30.1 | -53.98, -39.95 | APE12-dist-in | 13.6026 | APE11-dist-in | 13.4404 | APE10-dist-in | 7.7494 | APE9-dist-in | 4.3637 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 303.0 | 303.0 | 0 | 35 | 35 | 0 | [[29, 315]] | 1.0 | AF-Q86Y07-K1 | CK1_VRK2_HUMAN | CK1 | 1.2e-103 | 352.0 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | AF-Q86Y07-K3A | Q86Y07 | 21 | 323 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.8466 | 14.4688 | BLAminus | -115.0, 179.72 | 63.98, 65.55 | -78.94, 22.97 | 296.3, 84.35 | -64.97, -24.45 | in-in | in | 7.6164 | Saltbr-in | 2.7356 | HRD-in | -82.47, -50.04 | 76.81, -12.36 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.935 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -64.52, 146.14 | APE9-dihe-na | 93.49, -170.52 | APE8-dihe-in | -75.59, 116.8 | APE8-rot-in | 299.91 | APE67-dihe-in | -57.82, -37.72 | -53.79, -34.98 | APE12-dist-in | 13.7844 | APE11-dist-in | 13.5251 | APE10-dist-in | 7.937 | APE9-dist-in | 4.3311 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 303.0 | 303.0 | 0 | 35 | 35 | 0 | [[29, 315]] | 1.0 | AF-Q86Y07-K3 | CK1_VRK2_HUMAN | CK1 | 1.2e-103 | 352.0 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | 2V62A | Q86Y07 | 15 | 330 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.5216 | 14.2783 | BLAminus | -126.42, 177.81 | 61.4, 82.15 | -97.89, 25.94 | 290.77, 86.68 | -60.53, -27.7 | in-in | in | 7.4688 | Saltbr-in | 2.6513 | HRD-in | -85.44, -49.42 | 78.82, -6.43 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -77.49, 164.36 | APE9-dihe-na | 100.65, -175.4 | APE8-dihe-in | -81.64, 115.53 | APE8-rot-in | 300.97 | APE67-dihe-in | -58.37, -37.59 | -55.92, -37.43 | APE12-dist-in | 13.8351 | APE11-dist-in | 13.7728 | APE10-dist-in | 7.9511 | APE9-dist-in | 4.5825 | None | None | None | XRAY | 1.7 | 0.203 | 0.236 | A | 345.0 | 309.0 | 7 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 2v62 | CK1_VRK2_HUMAN | CK1 | 2e-103 | 351.3 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | 2V62B | Q86Y07 | 15 | 330 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.6633 | 14.235 | BLAminus | -125.07, 178.48 | 58.38, 82.78 | -95.02, 25.08 | 292.21, 85.61 | -65.49, -19.52 | in-in | in | 7.4809 | Saltbr-in | 3.1122 | HRD-in | -84.77, -51.43 | 82.43, -6.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8814 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -78.49, 164.48 | APE9-dihe-na | 105.42, -177.12 | APE8-dihe-in | -82.14, 116.45 | APE8-rot-in | 302.32 | APE67-dihe-in | -58.69, -38.25 | -56.97, -36.01 | APE12-dist-in | 13.7404 | APE11-dist-in | 13.6627 | APE10-dist-in | 7.977 | APE9-dist-in | 4.6212 | None | None | None | XRAY | 1.7 | 0.203 | 0.236 | B | 345.0 | 310.0 | 6 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 2v62 | CK1_VRK2_HUMAN | CK1 | 2e-103 | 351.3 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | 8Q1ZA | Q86Y07 | 15 | 330 | 508.0 | IKD:401 | Type1 | Active | DFGin | 7.6395 | 14.2844 | BLAminus | -121.18, 178.27 | 65.89, 75.15 | -84.6, 26.91 | 299.19, 79.94 | -58.07, -32.45 | in-in | in | 7.7906 | Saltbr-in | 2.8066 | HRD-in | -86.89, -55.74 | 82.47, 4.18 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8389 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -79.8, 160.18 | APE9-dihe-na | 103.61, -173.61 | APE8-dihe-in | -78.9, 112.93 | APE8-rot-in | 304.74 | APE67-dihe-in | -56.6, -35.59 | -54.54, -39.51 | APE12-dist-in | 13.7009 | APE11-dist-in | 13.7658 | APE10-dist-in | 7.9891 | APE9-dist-in | 4.5705 | None | None | None | XRAY | 1.85 | 0.203 | 0.251 | A | 324.0 | 311.0 | 5 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 8q1z | CK1_VRK2_HUMAN | CK1 | 1.6e-103 | 351.6 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | 9FETA | Q86Y07 | 15 | 330 | 508.0 | REB:401 | Type1.5_Back | Active | DFGin | 7.7569 | 14.1775 | BLAminus | -126.51, -179.88 | 62.99, 75.15 | -90.88, 34.72 | 299.05, 76.11 | -73.88, -23.01 | in-in | in | 7.4719 | Saltbr-in | 3.1195 | HRD-in | -79.75, -50.35 | 72.0, 10.87 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8102 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.38, 169.25 | APE9-dihe-na | 101.33, -175.93 | APE8-dihe-in | -76.93, 108.74 | APE8-rot-in | 301.77 | APE67-dihe-in | -59.32, -37.67 | -45.84, -39.32 | APE12-dist-in | 13.5609 | APE11-dist-in | 13.6582 | APE10-dist-in | 7.9227 | APE9-dist-in | 4.6041 | None | None | None | XRAY | 2.4 | 0.224 | 0.269 | A | 324.0 | 313.0 | 3 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 9fet | CK1_VRK2_HUMAN | CK1 | 1.6e-103 | 351.6 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | 5UU1A | Q86Y07 | 14 | 328 | 508.0 | 7DZ:401 | Type1.5_Back | Inactive | DFGin | 8.4017 | 14.1464 | ABAminus | -105.17, 5.91 | -139.93, 132.89 | -129.79, 29.75 | 298.27, 85.6 | -64.07, -29.29 | in-in | in | 8.3215 | Saltbr-in | 2.7413 | HRD-in | -72.24, -51.92 | 73.83, 1.33 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8062 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -81.98, 168.28 | APE9-dihe-na | 87.0, -169.82 | APE8-dihe-in | -84.32, 117.18 | APE8-rot-in | 301.27 | APE67-dihe-in | -54.03, -35.31 | -55.55, -41.02 | APE12-dist-in | 13.8145 | APE11-dist-out | 14.1872 | APE10-dist-out | 8.3917 | APE9-dist-in | 4.5395 | None | None | None | XRAY | 2.0 | 0.184 | 0.221 | A | 324.0 | 315.0 | 0 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 5uu1 | CK1_VRK2_HUMAN | CK1 | 1.6e-103 | 351.6 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | 6NCGA | Q86Y07 | 14 | 326 | 508.0 | KJD:401 | Type1.5_Back | Inactive | DFGin | 7.8329 | 14.3362 | BLAminus | -125.61, 178.62 | 60.55, 62.42 | -76.78, 23.63 | 300.3, 88.18 | -58.42, -42.6 | in-none | in | 8.0111 | Saltbr-none | 999.0 | HRD-in | -72.05, -54.32 | 82.86, -13.02 | none-in-out | SNCnio | in-out | ActLoopNT-in | 2.9459 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -78.98, 159.16 | APE9-dihe-na | 90.01, -173.25 | APE8-dihe-in | -74.1, 126.42 | APE8-rot-in | 306.94 | APE67-dihe-in | -58.12, -40.54 | -65.34, -36.48 | APE12-dist-in | 13.6753 | APE11-dist-out | 14.0275 | APE10-dist-out | 8.2529 | APE9-dist-in | 5.0774 | None | None | None | XRAY | 2.45 | 0.224 | 0.297 | A | 324.0 | 308.0 | 5 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 6ncg | CK1_VRK2_HUMAN | CK1 | 1.6e-103 | 351.6 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | 6NCGB | Q86Y07 | 16 | 326 | 508.0 | KJD:600 | Type1.5_Back | Inactive | DFGin | 8.0938 | 14.469 | BLAminus | -139.64, 179.69 | 67.8, 54.79 | -86.31, 18.42 | 302.17, 88.4 | -59.83, -52.96 | in-out | in | 8.1729 | Saltbr-out | 3.7674 | HRD-in | -73.43, -54.05 | 79.99, 3.47 | out-in-none | SNCoin | in-none | ActLoopNT-in | 2.7683 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnii | APE10-dihe-na | 999.0, -0.09 | APE9-dihe-na | -98.27, -160.94 | APE8-dihe-in | -91.38, 128.96 | APE8-rot-in | 317.51 | APE67-dihe-in | -56.32, -42.58 | -60.83, -41.47 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-in | 6.891 | APE9-dist-in | 4.2111 | None | None | None | XRAY | 2.45 | 0.224 | 0.297 | B | 324.0 | 287.0 | 24 | 35 | 20 | 15 | [[29, 315]] | 1.0 | 6ncg | CK1_VRK2_HUMAN | CK1 | 1.6e-103 | 351.6 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| VRK2 | VRK2_HUMAN | AF-Q86Y07-K1A | Q86Y07 | 21 | 323 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.9476 | 14.7984 | BLAminus | -119.05, 177.71 | 65.11, 69.16 | -80.5, 23.83 | 289.5, 88.67 | -62.34, -29.88 | in-in | in | 8.0198 | Saltbr-in | 2.6572 | HRD-in | -84.77, -50.44 | 77.78, 0.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.909 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -61.7, 143.45 | APE9-dihe-na | 96.44, -172.51 | APE8-dihe-in | -74.74, 115.77 | APE8-rot-in | 298.71 | APE67-dihe-in | -66.17, -30.1 | -53.98, -39.95 | APE12-dist-in | 13.6026 | APE11-dist-in | 13.4404 | APE10-dist-in | 7.7494 | APE9-dist-in | 4.3637 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 303.0 | 303.0 | 0 | 35 | 35 | 0 | [[29, 315]] | 1.0 | AF-Q86Y07-K1 | Homo sapiens | CK1_VRK2_HUMAN | CK1 | 1.2e-103 | 352.0 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | VRK2_HUMAN | AF-Q86Y07-K3A | Q86Y07 | 21 | 323 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.8466 | 14.4688 | BLAminus | -115.0, 179.72 | 63.98, 65.55 | -78.94, 22.97 | 296.3, 84.35 | -64.97, -24.45 | in-in | in | 7.6164 | Saltbr-in | 2.7356 | HRD-in | -82.47, -50.04 | 76.81, -12.36 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.935 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -64.52, 146.14 | APE9-dihe-na | 93.49, -170.52 | APE8-dihe-in | -75.59, 116.8 | APE8-rot-in | 299.91 | APE67-dihe-in | -57.82, -37.72 | -53.79, -34.98 | APE12-dist-in | 13.7844 | APE11-dist-in | 13.5251 | APE10-dist-in | 7.937 | APE9-dist-in | 4.3311 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 303.0 | 303.0 | 0 | 35 | 35 | 0 | [[29, 315]] | 1.0 | AF-Q86Y07-K3 | Homo sapiens | CK1_VRK2_HUMAN | CK1 | 1.2e-103 | 352.0 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | VRK2_HUMAN | 2V62A | Q86Y07 | 15 | 330 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.5216 | 14.2783 | BLAminus | -126.42, 177.81 | 61.4, 82.15 | -97.89, 25.94 | 290.77, 86.68 | -60.53, -27.7 | in-in | in | 7.4688 | Saltbr-in | 2.6513 | HRD-in | -85.44, -49.42 | 78.82, -6.43 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.93 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -77.49, 164.36 | APE9-dihe-na | 100.65, -175.4 | APE8-dihe-in | -81.64, 115.53 | APE8-rot-in | 300.97 | APE67-dihe-in | -58.37, -37.59 | -55.92, -37.43 | APE12-dist-in | 13.8351 | APE11-dist-in | 13.7728 | APE10-dist-in | 7.9511 | APE9-dist-in | 4.5825 | None | None | None | XRAY | 1.7 | 0.203 | 0.236 | A | 345.0 | 309.0 | 7 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 2v62 | Homo sapiens | CK1_VRK2_HUMAN | CK1 | 2e-103 | 351.3 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | VRK2_HUMAN | 2V62B | Q86Y07 | 15 | 330 | 508.0 | No_ligand | No_ligand | Active | DFGin | 7.6633 | 14.235 | BLAminus | -125.07, 178.48 | 58.38, 82.78 | -95.02, 25.08 | 292.21, 85.61 | -65.49, -19.52 | in-in | in | 7.4809 | Saltbr-in | 3.1122 | HRD-in | -84.77, -51.43 | 82.43, -6.15 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8814 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -78.49, 164.48 | APE9-dihe-na | 105.42, -177.12 | APE8-dihe-in | -82.14, 116.45 | APE8-rot-in | 302.32 | APE67-dihe-in | -58.69, -38.25 | -56.97, -36.01 | APE12-dist-in | 13.7404 | APE11-dist-in | 13.6627 | APE10-dist-in | 7.977 | APE9-dist-in | 4.6212 | None | None | None | XRAY | 1.7 | 0.203 | 0.236 | B | 345.0 | 310.0 | 6 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 2v62 | Homo sapiens | CK1_VRK2_HUMAN | CK1 | 2e-103 | 351.3 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | VRK2_HUMAN | 8Q1ZA | Q86Y07 | 15 | 330 | 508.0 | IKD:401 | Type1 | Active | DFGin | 7.6395 | 14.2844 | BLAminus | -121.18, 178.27 | 65.89, 75.15 | -84.6, 26.91 | 299.19, 79.94 | -58.07, -32.45 | in-in | in | 7.7906 | Saltbr-in | 2.8066 | HRD-in | -86.89, -55.74 | 82.47, 4.18 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8389 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -79.8, 160.18 | APE9-dihe-na | 103.61, -173.61 | APE8-dihe-in | -78.9, 112.93 | APE8-rot-in | 304.74 | APE67-dihe-in | -56.6, -35.59 | -54.54, -39.51 | APE12-dist-in | 13.7009 | APE11-dist-in | 13.7658 | APE10-dist-in | 7.9891 | APE9-dist-in | 4.5705 | None | None | None | XRAY | 1.85 | 0.203 | 0.251 | A | 324.0 | 311.0 | 5 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 8q1z | Homo sapiens | CK1_VRK2_HUMAN | CK1 | 1.6e-103 | 351.6 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | VRK2_HUMAN | 9FETA | Q86Y07 | 15 | 330 | 508.0 | REB:401 | Type1.5_Back | Active | DFGin | 7.7569 | 14.1775 | BLAminus | -126.51, -179.88 | 62.99, 75.15 | -90.88, 34.72 | 299.05, 76.11 | -73.88, -23.01 | in-in | in | 7.4719 | Saltbr-in | 3.1195 | HRD-in | -79.75, -50.35 | 72.0, 10.87 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8102 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -84.38, 169.25 | APE9-dihe-na | 101.33, -175.93 | APE8-dihe-in | -76.93, 108.74 | APE8-rot-in | 301.77 | APE67-dihe-in | -59.32, -37.67 | -45.84, -39.32 | APE12-dist-in | 13.5609 | APE11-dist-in | 13.6582 | APE10-dist-in | 7.9227 | APE9-dist-in | 4.6041 | None | None | None | XRAY | 2.4 | 0.224 | 0.269 | A | 324.0 | 313.0 | 3 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 9fet | Homo sapiens | CK1_VRK2_HUMAN | CK1 | 1.6e-103 | 351.6 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | VRK2_HUMAN | 5UU1A | Q86Y07 | 14 | 328 | 508.0 | 7DZ:401 | Type1.5_Back | Inactive | DFGin | 8.4017 | 14.1464 | ABAminus | -105.17, 5.91 | -139.93, 132.89 | -129.79, 29.75 | 298.27, 85.6 | -64.07, -29.29 | in-in | in | 8.3215 | Saltbr-in | 2.7413 | HRD-in | -72.24, -51.92 | 73.83, 1.33 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8062 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -81.98, 168.28 | APE9-dihe-na | 87.0, -169.82 | APE8-dihe-in | -84.32, 117.18 | APE8-rot-in | 301.27 | APE67-dihe-in | -54.03, -35.31 | -55.55, -41.02 | APE12-dist-in | 13.8145 | APE11-dist-out | 14.1872 | APE10-dist-out | 8.3917 | APE9-dist-in | 4.5395 | None | None | None | XRAY | 2.0 | 0.184 | 0.221 | A | 324.0 | 315.0 | 0 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 5uu1 | Homo sapiens | CK1_VRK2_HUMAN | CK1 | 1.6e-103 | 351.6 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | VRK2_HUMAN | 6NCGA | Q86Y07 | 14 | 326 | 508.0 | KJD:401 | Type1.5_Back | Inactive | DFGin | 7.8329 | 14.3362 | BLAminus | -125.61, 178.62 | 60.55, 62.42 | -76.78, 23.63 | 300.3, 88.18 | -58.42, -42.6 | in-none | in | 8.0111 | Saltbr-none | 999.0 | HRD-in | -72.05, -54.32 | 82.86, -13.02 | none-in-out | SNCnio | in-out | ActLoopNT-in | 2.9459 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -78.98, 159.16 | APE9-dihe-na | 90.01, -173.25 | APE8-dihe-in | -74.1, 126.42 | APE8-rot-in | 306.94 | APE67-dihe-in | -58.12, -40.54 | -65.34, -36.48 | APE12-dist-in | 13.6753 | APE11-dist-out | 14.0275 | APE10-dist-out | 8.2529 | APE9-dist-in | 5.0774 | None | None | None | XRAY | 2.45 | 0.224 | 0.297 | A | 324.0 | 308.0 | 5 | 35 | 35 | 0 | [[29, 315]] | 1.0 | 6ncg | Homo sapiens | CK1_VRK2_HUMAN | CK1 | 1.6e-103 | 351.6 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| VRK2 | VRK2_HUMAN | 6NCGB | Q86Y07 | 16 | 326 | 508.0 | KJD:600 | Type1.5_Back | Inactive | DFGin | 8.0938 | 14.469 | BLAminus | -139.64, 179.69 | 67.8, 54.79 | -86.31, 18.42 | 302.17, 88.4 | -59.83, -52.96 | in-out | in | 8.1729 | Saltbr-out | 3.7674 | HRD-in | -73.43, -54.05 | 79.99, 3.47 | out-in-none | SNCoin | in-none | ActLoopNT-in | 2.7683 | ActLoopCT-none | nonTYR | APEdihe_aaiii | APEdist_nnii | APE10-dihe-na | 999.0, -0.09 | APE9-dihe-na | -98.27, -160.94 | APE8-dihe-in | -91.38, 128.96 | APE8-rot-in | 317.51 | APE67-dihe-in | -56.32, -42.58 | -60.83, -41.47 | APE12-dist-none | 999.0 | APE11-dist-none | 999.0 | APE10-dist-in | 6.891 | APE9-dist-in | 4.2111 | None | None | None | XRAY | 2.45 | 0.224 | 0.297 | B | 324.0 | 287.0 | 24 | 35 | 20 | 15 | [[29, 315]] | 1.0 | 6ncg | Homo sapiens | CK1_VRK2_HUMAN | CK1 | 1.6e-103 | 351.6 | 1.0 | 261.0 | 261.0 | 185 | 186 | 187 | 189 | 191 | 61 | 73 | 77 | 163 | 165 | 164 | 166.0 | 232 | 220 | 215 | 214 | 213 | 212 | 211 | 210 | 209 | 122 | Serine/threonine-protein kinase VRK2 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|