CAMK_STK17A (Serine/threonine-protein kinase 17A)

Total number of chains: 6
Active chains: 2
Family: CAMK
Uniprot: ST17A_HUMAN
Kinase Domain Residues: 59 - 321
Spatial label Dihedral label Number of Chains Percent Representative
DFGin ABAminus 3 50.0% 7QUFA
DFGin BLAminus 3 50.0% AF-Q9UEE5-K1A

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PDB First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
AF-Q9UEE5-K1A 51 329 414.0 No_ligand No_ligand Active DFGin 6.159 14.099 BLAminus -129.27, 170.92 64.97, 64.55 -75.43, 21.24 291.56, 83.12 -65.43, -24.67 in-in in 9.002 Saltbr-in 2.633 HRD-in -80.88, -43.24 65.02, -3.61 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.49, 177.42 APE9-dihe-na 89.95, -178.48 APE8-dihe-in -91.88, 126.45 APE8-rot-in 302.18 APE67-dihe-in -76.05, -22.22 -46.99, -32.12 APE12-dist-in 9.005 APE11-dist-in 12.14 APE10-dist-in 6.485 APE9-dist-in 4.683 None None None AF2 -1.0 1.0 1.0 A 279 279 0 0 0 0 [[59, 321]] 1.0 AF-Q9UEE5-K1 CAMK_STK17A_HUMAN CAMK 1.4e-86 295.9 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A
AF-Q9UEE5-K3A 51 329 414.0 No_ligand No_ligand Active DFGin 5.918 13.901 BLAminus -132.98, 171.56 63.24, 63.04 -72.48, 15.51 295.77, 90.58 -64.92, -20.79 in-in in 8.778 Saltbr-in 2.595 HRD-in -84.59, -41.6 65.53, 5.87 in-in-in SNCiii in-in ActLoopNT-in 2.9 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.79, -176.51 APE9-dihe-na 92.4, 171.63 APE8-dihe-in -81.96, 126.41 APE8-rot-in 298.66 APE67-dihe-in -72.42, -21.04 -47.99, -41.58 APE12-dist-in 8.97 APE11-dist-in 12.044 APE10-dist-in 6.293 APE9-dist-in 3.632 None None None AF2 -1.0 1.0 1.0 A 279 279 0 0 0 0 [[59, 321]] 1.0 AF-Q9UEE5-K3 CAMK_STK17A_HUMAN CAMK 1.4e-86 295.9 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A
7QUEB 59 322 414.0 F7I:60401 Type1 Inactive DFGin 6.097 14.438 ABAminus -112.52, -32.9 -122.41, 133.23 -125.43, 20.39 297.06, 88.08 -55.17, -31.91 in-out in 9.139 Saltbr-out 3.913 HRD-out 55.74, 49.22 -83.59, 137.61 out-in-out SNCoio in-out ActLoopNT-in 3.1 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -84.31, 1.38 APE9-dihe-na -74.9, -3.54 APE8-dihe-in -123.33, 68.17 APE8-rot-none 999.0 APE67-dihe-in -55.47, -30.5 -62.56, -34.53 APE12-dist-out 25.219 APE11-dist-out 23.781 APE10-dist-out 26.756 APE9-dist-out 32.206 None None None XRAY 2.4 0.235 0.266 B 275 239 25 0 0 6 [[59, 321]] 1.0 7que CAMK_STK17A_HUMAN CAMK 1.3e-86 296.0 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A
7QUFA 50 322 414.0 F8I:60401 Type1 Inactive DFGin 5.726 13.875 ABAminus -122.57, -17.7 -129.74, 145.86 -137.48, 25.23 294.61, 85.2 -65.55, -25.05 in-in in 8.676 Saltbr-in 3.525 HRD-in -74.09, -51.85 70.16, 11.74 in-in-out SNCiio in-out ActLoopNT-in 2.895 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -60.31, -42.78 APE9-dihe-na 87.11, -170.08 APE8-dihe-in -60.31, 123.62 APE8-rot-in 278.22 APE67-dihe-in -71.85, -10.66 -61.07, -29.38 APE12-dist-out 24.271 APE11-dist-out 20.62 APE10-dist-out 24.621 APE9-dist-out 27.51 None None None XRAY 2.6 0.235 0.294 A 275 268 5 0 0 0 [[59, 321]] 1.0 7quf CAMK_STK17A_HUMAN CAMK 1.3e-86 296.0 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A
7QUFB 55 322 414.0 F8I:60401 Type1 Inactive DFGin 6.63 14.579 ABAminus -109.96, -28.04 -133.72, 141.49 -139.5, 24.01 294.67, 82.9 -63.63, -25.63 in-none in 9.168 Saltbr-none 999.0 HRD-out 62.58, 55.6 -87.85, 137.63 none-in-out SNCnio in-out ActLoopNT-in 2.736 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -89.23, -3.61 APE9-dihe-na -63.23, -9.98 APE8-dihe-in -131.17, 74.63 APE8-rot-out 36.39 APE67-dihe-in -50.75, -37.34 -59.6, -41.11 APE12-dist-out 24.845 APE11-dist-out 23.538 APE10-dist-out 26.592 APE9-dist-out 32.17 None None None XRAY 2.6 0.235 0.294 B 275 249 19 0 0 0 [[59, 321]] 1.0 7quf CAMK_STK17A_HUMAN CAMK 1.3e-86 296.0 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A
7QUEA 50 322 414.0 F7I:60401 Type1 Inactive DFGin 5.94 14.508 BLAminus -123.87, 169.48 73.3, 84.52 -97.37, 24.76 291.76, 92.48 -60.06, -34.52 in-in in 8.739 Saltbr-in 2.554 HRD-in -67.47, -57.59 81.18, 10.24 in-in-out SNCiio in-out ActLoopNT-in 2.853 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -63.29, -50.03 APE9-dihe-na 84.76, 176.19 APE8-dihe-in -65.0, 132.13 APE8-rot-out 35.79 APE67-dihe-in -64.45, -4.9 -63.94, -42.06 APE12-dist-out 24.676 APE11-dist-out 20.706 APE10-dist-out 24.464 APE9-dist-out 27.588 None None None XRAY 2.4 0.235 0.266 A 275 264 9 0 0 0 [[59, 321]] 1.0 7que CAMK_STK17A_HUMAN CAMK 1.3e-86 296.0 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A

CAMK_STK17A (Serine/threonine-protein kinase 17A)

Total number of chains: 6
Active chains: 2
Family: CAMK
Spatial label Dihedral label Number of Chains Percent Representative
DFGin ABAminus 3 50.0% 7QUFA
DFGin BLAminus 3 50.0% AF-Q9UEE5-K1A

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
ST17A_HUMAN AF-Q9UEE5-K1A Q9UEE5 51 329 414.0 No_ligand No_ligand Active DFGin 6.159 14.099 BLAminus -129.27, 170.92 64.97, 64.55 -75.43, 21.24 291.56, 83.12 -65.43, -24.67 in-in in 9.002 Saltbr-in 2.633 HRD-in -80.88, -43.24 65.02, -3.61 in-in-in SNCiii in-in ActLoopNT-in 2.921 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.49, 177.42 APE9-dihe-na 89.95, -178.48 APE8-dihe-in -91.88, 126.45 APE8-rot-in 302.18 APE67-dihe-in -76.05, -22.22 -46.99, -32.12 APE12-dist-in 9.005 APE11-dist-in 12.14 APE10-dist-in 6.485 APE9-dist-in 4.683 None None None AF2 -1.0 1.0 1.0 A 279 279 0 0 0 0 [[59, 321]] 1.0 AF-Q9UEE5-K1 Homo sapiens CAMK_STK17A_HUMAN CAMK 1.4e-86 295.9 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A
ST17A_HUMAN AF-Q9UEE5-K3A Q9UEE5 51 329 414.0 No_ligand No_ligand Active DFGin 5.918 13.901 BLAminus -132.98, 171.56 63.24, 63.04 -72.48, 15.51 295.77, 90.58 -64.92, -20.79 in-in in 8.778 Saltbr-in 2.595 HRD-in -84.59, -41.6 65.53, 5.87 in-in-in SNCiii in-in ActLoopNT-in 2.9 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -145.79, -176.51 APE9-dihe-na 92.4, 171.63 APE8-dihe-in -81.96, 126.41 APE8-rot-in 298.66 APE67-dihe-in -72.42, -21.04 -47.99, -41.58 APE12-dist-in 8.97 APE11-dist-in 12.044 APE10-dist-in 6.293 APE9-dist-in 3.632 None None None AF2 -1.0 1.0 1.0 A 279 279 0 0 0 0 [[59, 321]] 1.0 AF-Q9UEE5-K3 Homo sapiens CAMK_STK17A_HUMAN CAMK 1.4e-86 295.9 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A
ST17A_HUMAN 7QUEB Q9UEE5 59 322 414.0 F7I:60401 Type1 Inactive DFGin 6.097 14.438 ABAminus -112.52, -32.9 -122.41, 133.23 -125.43, 20.39 297.06, 88.08 -55.17, -31.91 in-out in 9.139 Saltbr-out 3.913 HRD-out 55.74, 49.22 -83.59, 137.61 out-in-out SNCoio in-out ActLoopNT-in 3.1 ActLoopCT-out nonTYR APEdihe_aaini APEdist_oooo APE10-dihe-na -84.31, 1.38 APE9-dihe-na -74.9, -3.54 APE8-dihe-in -123.33, 68.17 APE8-rot-none 999.0 APE67-dihe-in -55.47, -30.5 -62.56, -34.53 APE12-dist-out 25.219 APE11-dist-out 23.781 APE10-dist-out 26.756 APE9-dist-out 32.206 None None None XRAY 2.4 0.235 0.266 B 275 239 25 0 0 6 [[59, 321]] 1.0 7que Homo sapiens CAMK_STK17A_HUMAN CAMK 1.3e-86 296.0 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A
ST17A_HUMAN 7QUFA Q9UEE5 50 322 414.0 F8I:60401 Type1 Inactive DFGin 5.726 13.875 ABAminus -122.57, -17.7 -129.74, 145.86 -137.48, 25.23 294.61, 85.2 -65.55, -25.05 in-in in 8.676 Saltbr-in 3.525 HRD-in -74.09, -51.85 70.16, 11.74 in-in-out SNCiio in-out ActLoopNT-in 2.895 ActLoopCT-out nonTYR APEdihe_aaiii APEdist_oooo APE10-dihe-na -60.31, -42.78 APE9-dihe-na 87.11, -170.08 APE8-dihe-in -60.31, 123.62 APE8-rot-in 278.22 APE67-dihe-in -71.85, -10.66 -61.07, -29.38 APE12-dist-out 24.271 APE11-dist-out 20.62 APE10-dist-out 24.621 APE9-dist-out 27.51 None None None XRAY 2.6 0.235 0.294 A 275 268 5 0 0 0 [[59, 321]] 1.0 7quf Homo sapiens CAMK_STK17A_HUMAN CAMK 1.3e-86 296.0 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A
ST17A_HUMAN 7QUFB Q9UEE5 55 322 414.0 F8I:60401 Type1 Inactive DFGin 6.63 14.579 ABAminus -109.96, -28.04 -133.72, 141.49 -139.5, 24.01 294.67, 82.9 -63.63, -25.63 in-none in 9.168 Saltbr-none 999.0 HRD-out 62.58, 55.6 -87.85, 137.63 none-in-out SNCnio in-out ActLoopNT-in 2.736 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -89.23, -3.61 APE9-dihe-na -63.23, -9.98 APE8-dihe-in -131.17, 74.63 APE8-rot-out 36.39 APE67-dihe-in -50.75, -37.34 -59.6, -41.11 APE12-dist-out 24.845 APE11-dist-out 23.538 APE10-dist-out 26.592 APE9-dist-out 32.17 None None None XRAY 2.6 0.235 0.294 B 275 249 19 0 0 0 [[59, 321]] 1.0 7quf Homo sapiens CAMK_STK17A_HUMAN CAMK 1.3e-86 296.0 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A
ST17A_HUMAN 7QUEA Q9UEE5 50 322 414.0 F7I:60401 Type1 Inactive DFGin 5.94 14.508 BLAminus -123.87, 169.48 73.3, 84.52 -97.37, 24.76 291.76, 92.48 -60.06, -34.52 in-in in 8.739 Saltbr-in 2.554 HRD-in -67.47, -57.59 81.18, 10.24 in-in-out SNCiio in-out ActLoopNT-in 2.853 ActLoopCT-out nonTYR APEdihe_aaioi APEdist_oooo APE10-dihe-na -63.29, -50.03 APE9-dihe-na 84.76, 176.19 APE8-dihe-in -65.0, 132.13 APE8-rot-out 35.79 APE67-dihe-in -64.45, -4.9 -63.94, -42.06 APE12-dist-out 24.676 APE11-dist-out 20.706 APE10-dist-out 24.464 APE9-dist-out 27.588 None None None XRAY 2.4 0.235 0.266 A 275 264 9 0 0 0 [[59, 321]] 1.0 7que Homo sapiens CAMK_STK17A_HUMAN CAMK 1.3e-86 296.0 4 256 253 206 207 208 210 212 90 108 112 183 185 184 186 245 233 228 227 226 225 224 223 222 139 Serine/threonine-protein kinase 17A

CAMK_STK17A (Serine/threonine-protein kinase 17A)

Total number of chains: 0
Active chains: 0
Family: CAMK
Spatial label Dihedral label Number of Chains Percent Representative

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name