AGC_PRKCQ (Protein kinase C theta type)

Total number of chains: 11
Active chains: 11
Uniprot: KPCT_HUMAN
Kinase Domain Residues: 380 - 634
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 11 100.0% AF-Q04759-K1A

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PRKCQ AF-Q04759-K1A Q04759 372 642 706.0 No_ligand No_ligand Active DFGin 5.8884 13.0918 BLAminus -111.47, -161.58 28.49, 81.48 -87.29, 15.51 303.95, 98.21 -58.98, -28.73 in-in in 8.4889 Saltbr-in 2.611 HRD-in -79.51, -46.72 64.6, -6.08 in-in-in SNCiii in-in ActLoopNT-in 2.8802 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.83, 164.71 APE9-dihe-na 120.22, 165.8 APE8-dihe-in -69.46, 133.57 APE8-rot-in 297.66 APE67-dihe-in -68.66, -21.56 -49.68, -45.16 APE12-dist-in 8.6977 APE11-dist-in 12.0451 APE10-dist-in 6.4475 APE9-dist-in 3.5009 None None None AF2 -1.0 1.0 1.0 A 271.0 271.0 0 28 28 0 [[380, 634]] 1.0 AF-Q04759-K1 AGC_PRKCQ_HUMAN AGC 5e-96 326.7 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ AF-Q04759-K3A Q04759 372 642 706.0 No_ligand No_ligand Active DFGin 5.719 13.1124 BLAminus -115.41, 178.48 45.7, 90.34 -95.22, 12.74 305.99, 102.65 -59.82, -31.49 in-in in 8.3953 Saltbr-in 2.6304 HRD-in -80.31, -47.4 66.14, 1.97 in-in-in SNCiii in-in ActLoopNT-in 2.837 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.38, 163.76 APE9-dihe-na 124.04, 165.42 APE8-dihe-in -77.47, 131.1 APE8-rot-in 294.41 APE67-dihe-in -61.12, -22.91 -45.2, -50.91 APE12-dist-in 8.8337 APE11-dist-in 11.7017 APE10-dist-in 6.1405 APE9-dist-in 3.3316 None None None AF2 -1.0 1.0 1.0 A 271.0 271.0 0 28 28 0 [[380, 634]] 1.0 AF-Q04759-K3 AGC_PRKCQ_HUMAN AGC 5e-96 326.7 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ 4Q9ZA Q04759 375 706 706.0 PZW:60801 Type1 Active DFGin 6.4983 13.9835 BLAminus -129.62, 170.17 59.89, 78.05 -94.48, 11.49 301.06, 109.09 -65.66, -19.81 in-in in 8.8664 Saltbr-in 2.5882 HRD-in -84.02, -47.96 72.84, -13.44 in-in-in SNCiii in-in ActLoopNT-in 2.9307 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.72, 164.65 APE9-dihe-na 122.97, 176.49 APE8-dihe-in -90.21, 130.45 APE8-rot-in 303.85 APE67-dihe-in -60.12, -27.82 -40.48, -49.54 APE12-dist-in 9.8733 APE11-dist-in 11.9531 APE10-dist-in 6.3671 APE9-dist-in 3.6301 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.6 0.22 0.256 A 334.0 332.0 0 28 28 0 [[380, 634]] 1.0 4q9z AGC_PRKCQ_HUMAN AGC 5.3e-96 326.6 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ 4Q9ZB Q04759 374 704 706.0 PZW:60801 Type1 Active DFGin 6.4596 14.069 BLAminus -122.43, 171.24 60.71, 80.12 -96.99, 17.44 300.93, 103.53 -66.22, -22.55 in-in in 9.0422 Saltbr-in 3.222 HRD-in -78.02, -50.1 71.67, -5.88 in-in-in SNCiii in-in ActLoopNT-in 3.0454 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.73, 161.59 APE9-dihe-na 120.2, 169.91 APE8-dihe-in -85.09, 127.51 APE8-rot-in 308.63 APE67-dihe-in -57.39, -28.45 -39.09, -50.47 APE12-dist-in 9.5485 APE11-dist-in 11.8187 APE10-dist-in 6.2945 APE9-dist-in 3.5507 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.6 0.22 0.256 B 334.0 309.0 0 28 28 0 [[380, 634]] 1.0 4q9z AGC_PRKCQ_HUMAN AGC 5.3e-96 326.6 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ 4RA5A Q04759 374 706 706.0 3L0:60801 Type1 Active DFGin 6.502 13.7063 BLAminus -130.8, 165.47 60.37, 80.63 -96.28, 13.82 305.06, 108.57 -65.07, -21.73 in-in in 8.6895 Saltbr-in 2.7057 HRD-in -81.4, -52.17 72.03, -7.02 in-in-in SNCiii in-in ActLoopNT-in 2.8945 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.29, 168.72 APE9-dihe-na 122.43, 171.49 APE8-dihe-in -88.88, 125.08 APE8-rot-in 316.66 APE67-dihe-in -56.04, -31.31 -40.84, -48.14 APE12-dist-in 8.8649 APE11-dist-in 12.0862 APE10-dist-in 6.5061 APE9-dist-in 3.4777 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.61 0.23 0.277 A 334.0 333.0 0 28 28 0 [[380, 634]] 1.0 4ra5 AGC_PRKCQ_HUMAN AGC 5.3e-96 326.6 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ 4RA5B Q04759 375 701 706.0 3L0:60801 Type1 Active DFGin 6.4995 13.9579 BLAminus -124.58, 172.11 61.76, 74.37 -91.68, 16.04 298.23, 101.99 -61.29, -29.96 in-in in 8.8135 Saltbr-in 2.7679 HRD-in -76.54, -51.94 71.71, -2.05 in-in-in SNCiii in-in ActLoopNT-in 3.094 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.62, 162.67 APE9-dihe-na 133.57, -170.02 APE8-dihe-in -109.6, 121.98 APE8-rot-in 311.54 APE67-dihe-in -60.14, -31.4 -32.49, -52.6 APE12-dist-in 8.7326 APE11-dist-in 12.0188 APE10-dist-in 6.4921 APE9-dist-in 3.5754 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.61 0.23 0.277 B 334.0 312.0 0 28 28 0 [[380, 634]] 1.0 4ra5 AGC_PRKCQ_HUMAN AGC 5.3e-96 326.6 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ 2JEDA Q04759 375 700 706.0 LG8:61701 Type1 Active DFGin 6.6135 13.6674 BLAminus -113.39, 165.43 67.55, 92.49 -102.81, 25.08 299.09, 96.04 -77.76, -4.74 in-in in 8.6977 Saltbr-in 3.2014 HRD-in -82.61, -46.83 69.15, -8.62 in-in-in SNCiii in-in ActLoopNT-in 2.842 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.64, 141.45 APE9-dihe-na 144.48, -176.42 APE8-dihe-in -112.96, 132.15 APE8-rot-in 286.91 APE67-dihe-in -65.19, -26.4 -40.31, -53.61 APE12-dist-in 8.797 APE11-dist-in 11.7497 APE10-dist-in 5.9618 APE9-dist-in 3.8827 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.32 0.188 0.221 A 352.0 326.0 0 28 28 0 [[380, 634]] 1.0 2jed AGC_PRKCQ_HUMAN AGC 6.3e-96 326.4 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ 2JEDB Q04759 375 706 706.0 LG8:61712 Type1 Active DFGin 6.4774 13.7752 BLAminus -116.9, 164.62 69.71, 89.68 -101.74, 24.61 303.13, 88.06 -65.56, -17.66 in-in in 8.9098 Saltbr-in 3.0201 HRD-in -77.46, -49.1 72.97, -12.75 in-in-in SNCiii in-in ActLoopNT-in 2.9394 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.05, 132.52 APE9-dihe-na 123.41, 168.41 APE8-dihe-in -74.67, 129.81 APE8-rot-in 290.27 APE67-dihe-in -53.63, -32.33 -43.76, -48.79 APE12-dist-in 8.7728 APE11-dist-in 11.6804 APE10-dist-in 6.647 APE9-dist-in 4.1 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.32 0.188 0.221 B 352.0 317.0 0 28 28 0 [[380, 634]] 1.0 2jed AGC_PRKCQ_HUMAN AGC 6.3e-96 326.4 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ 5F9EA Q04759 374 706 706.0 5VS:61001 Type1 Active DFGin 6.4755 13.8521 BLAminus -124.47, 161.09 72.18, 90.67 -101.4, 15.51 297.35, 95.13 -63.75, -26.0 in-in in 9.058 Saltbr-in 2.7166 HRD-in -81.15, -47.98 73.24, -5.11 in-in-in SNCiii in-in ActLoopNT-in 2.8522 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.97, 169.63 APE9-dihe-na 131.49, -173.01 APE8-dihe-in -109.76, 129.84 APE8-rot-in 295.69 APE67-dihe-in -61.77, -26.26 -46.68, -44.42 APE12-dist-in 8.9537 APE11-dist-in 12.0173 APE10-dist-in 6.5605 APE9-dist-in 3.6595 None SEP676,SEP695 SEP676,SEP695 XRAY 2.0 0.199 0.233 A 353.0 333.0 0 28 28 0 [[380, 634]] 1.0 5f9e AGC_PRKCQ_HUMAN AGC 6.4e-96 326.4 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ 5F9EB Q04759 375 700 706.0 5VS:61001 Type1 Active DFGin 6.583 13.8849 BLAminus -118.45, 165.26 62.54, 88.94 -98.52, 15.46 302.93, 89.41 -59.36, -22.06 in-in in 9.2672 Saltbr-in 2.5897 HRD-in -84.26, -45.13 71.76, -7.56 in-in-in SNCiii in-in ActLoopNT-in 2.9056 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -170.19, 135.47 APE9-dihe-na 127.82, -166.17 APE8-dihe-in -112.12, 133.27 APE8-rot-in 297.56 APE67-dihe-in -57.44, -27.74 -44.31, -54.84 APE12-dist-in 8.7675 APE11-dist-in 12.0459 APE10-dist-in 7.3231 APE9-dist-in 3.5782 None SEP676,SEP695 SEP676,SEP695 XRAY 2.0 0.199 0.233 B 353.0 294.0 0 28 28 0 [[380, 634]] 1.0 5f9e AGC_PRKCQ_HUMAN AGC 6.4e-96 326.4 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ 1XJDA Q04759 377 696 706.0 STU:200 Type1 Active DFGin 5.8284 13.1925 BLAminus -132.69, 162.8 69.28, 95.13 -109.8, 21.13 305.67, 104.94 -64.79, -17.76 in-in in 8.0639 Saltbr-in 2.5131 HRD-in -67.27, -48.59 64.56, -1.72 in-in-in SNCiii in-in ActLoopNT-in 2.9684 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.73, 166.78 APE9-dihe-na 120.3, 163.8 APE8-dihe-in -75.86, 125.98 APE8-rot-in 298.87 APE67-dihe-in -57.15, -29.94 -38.43, -48.34 APE12-dist-in 9.0296 APE11-dist-in 12.2938 APE10-dist-in 6.8961 APE9-dist-in 3.7669 None TPO538,SEP695 TPO538,SEP695 XRAY 2.0 0.201 0.216 A 345.0 282.0 0 28 28 0 [[380, 634]] 1.0 1xjd AGC_PRKCQ_HUMAN AGC 1.2e-95 325.5 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type

AGC_PRKCQ (Protein kinase C theta type)

Total number of chains: 11
Active chains: 11
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 11 100.0% AF-Q04759-K1A

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PRKCQ KPCT_HUMAN AF-Q04759-K1A Q04759 372 642 706.0 No_ligand No_ligand Active DFGin 5.8884 13.0918 BLAminus -111.47, -161.58 28.49, 81.48 -87.29, 15.51 303.95, 98.21 -58.98, -28.73 in-in in 8.4889 Saltbr-in 2.611 HRD-in -79.51, -46.72 64.6, -6.08 in-in-in SNCiii in-in ActLoopNT-in 2.8802 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -158.83, 164.71 APE9-dihe-na 120.22, 165.8 APE8-dihe-in -69.46, 133.57 APE8-rot-in 297.66 APE67-dihe-in -68.66, -21.56 -49.68, -45.16 APE12-dist-in 8.6977 APE11-dist-in 12.0451 APE10-dist-in 6.4475 APE9-dist-in 3.5009 None None None AF2 -1.0 1.0 1.0 A 271.0 271.0 0 28 28 0 [[380, 634]] 1.0 AF-Q04759-K1 Homo sapiens AGC_PRKCQ_HUMAN AGC 5e-96 326.7 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ KPCT_HUMAN AF-Q04759-K3A Q04759 372 642 706.0 No_ligand No_ligand Active DFGin 5.719 13.1124 BLAminus -115.41, 178.48 45.7, 90.34 -95.22, 12.74 305.99, 102.65 -59.82, -31.49 in-in in 8.3953 Saltbr-in 2.6304 HRD-in -80.31, -47.4 66.14, 1.97 in-in-in SNCiii in-in ActLoopNT-in 2.837 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.38, 163.76 APE9-dihe-na 124.04, 165.42 APE8-dihe-in -77.47, 131.1 APE8-rot-in 294.41 APE67-dihe-in -61.12, -22.91 -45.2, -50.91 APE12-dist-in 8.8337 APE11-dist-in 11.7017 APE10-dist-in 6.1405 APE9-dist-in 3.3316 None None None AF2 -1.0 1.0 1.0 A 271.0 271.0 0 28 28 0 [[380, 634]] 1.0 AF-Q04759-K3 Homo sapiens AGC_PRKCQ_HUMAN AGC 5e-96 326.7 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ KPCT_HUMAN 4Q9ZA Q04759 375 706 706.0 PZW:60801 Type1 Active DFGin 6.4983 13.9835 BLAminus -129.62, 170.17 59.89, 78.05 -94.48, 11.49 301.06, 109.09 -65.66, -19.81 in-in in 8.8664 Saltbr-in 2.5882 HRD-in -84.02, -47.96 72.84, -13.44 in-in-in SNCiii in-in ActLoopNT-in 2.9307 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -157.72, 164.65 APE9-dihe-na 122.97, 176.49 APE8-dihe-in -90.21, 130.45 APE8-rot-in 303.85 APE67-dihe-in -60.12, -27.82 -40.48, -49.54 APE12-dist-in 9.8733 APE11-dist-in 11.9531 APE10-dist-in 6.3671 APE9-dist-in 3.6301 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.6 0.22 0.256 A 334.0 332.0 0 28 28 0 [[380, 634]] 1.0 4q9z Homo sapiens AGC_PRKCQ_HUMAN AGC 5.3e-96 326.6 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ KPCT_HUMAN 4Q9ZB Q04759 374 704 706.0 PZW:60801 Type1 Active DFGin 6.4596 14.069 BLAminus -122.43, 171.24 60.71, 80.12 -96.99, 17.44 300.93, 103.53 -66.22, -22.55 in-in in 9.0422 Saltbr-in 3.222 HRD-in -78.02, -50.1 71.67, -5.88 in-in-in SNCiii in-in ActLoopNT-in 3.0454 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -164.73, 161.59 APE9-dihe-na 120.2, 169.91 APE8-dihe-in -85.09, 127.51 APE8-rot-in 308.63 APE67-dihe-in -57.39, -28.45 -39.09, -50.47 APE12-dist-in 9.5485 APE11-dist-in 11.8187 APE10-dist-in 6.2945 APE9-dist-in 3.5507 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.6 0.22 0.256 B 334.0 309.0 0 28 28 0 [[380, 634]] 1.0 4q9z Homo sapiens AGC_PRKCQ_HUMAN AGC 5.3e-96 326.6 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ KPCT_HUMAN 4RA5A Q04759 374 706 706.0 3L0:60801 Type1 Active DFGin 6.502 13.7063 BLAminus -130.8, 165.47 60.37, 80.63 -96.28, 13.82 305.06, 108.57 -65.07, -21.73 in-in in 8.6895 Saltbr-in 2.7057 HRD-in -81.4, -52.17 72.03, -7.02 in-in-in SNCiii in-in ActLoopNT-in 2.8945 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -155.29, 168.72 APE9-dihe-na 122.43, 171.49 APE8-dihe-in -88.88, 125.08 APE8-rot-in 316.66 APE67-dihe-in -56.04, -31.31 -40.84, -48.14 APE12-dist-in 8.8649 APE11-dist-in 12.0862 APE10-dist-in 6.5061 APE9-dist-in 3.4777 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.61 0.23 0.277 A 334.0 333.0 0 28 28 0 [[380, 634]] 1.0 4ra5 Homo sapiens AGC_PRKCQ_HUMAN AGC 5.3e-96 326.6 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ KPCT_HUMAN 4RA5B Q04759 375 701 706.0 3L0:60801 Type1 Active DFGin 6.4995 13.9579 BLAminus -124.58, 172.11 61.76, 74.37 -91.68, 16.04 298.23, 101.99 -61.29, -29.96 in-in in 8.8135 Saltbr-in 2.7679 HRD-in -76.54, -51.94 71.71, -2.05 in-in-in SNCiii in-in ActLoopNT-in 3.094 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.62, 162.67 APE9-dihe-na 133.57, -170.02 APE8-dihe-in -109.6, 121.98 APE8-rot-in 311.54 APE67-dihe-in -60.14, -31.4 -32.49, -52.6 APE12-dist-in 8.7326 APE11-dist-in 12.0188 APE10-dist-in 6.4921 APE9-dist-in 3.5754 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.61 0.23 0.277 B 334.0 312.0 0 28 28 0 [[380, 634]] 1.0 4ra5 Homo sapiens AGC_PRKCQ_HUMAN AGC 5.3e-96 326.6 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ KPCT_HUMAN 2JEDA Q04759 375 700 706.0 LG8:61701 Type1 Active DFGin 6.6135 13.6674 BLAminus -113.39, 165.43 67.55, 92.49 -102.81, 25.08 299.09, 96.04 -77.76, -4.74 in-in in 8.6977 Saltbr-in 3.2014 HRD-in -82.61, -46.83 69.15, -8.62 in-in-in SNCiii in-in ActLoopNT-in 2.842 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -128.64, 141.45 APE9-dihe-na 144.48, -176.42 APE8-dihe-in -112.96, 132.15 APE8-rot-in 286.91 APE67-dihe-in -65.19, -26.4 -40.31, -53.61 APE12-dist-in 8.797 APE11-dist-in 11.7497 APE10-dist-in 5.9618 APE9-dist-in 3.8827 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.32 0.188 0.221 A 352.0 326.0 0 28 28 0 [[380, 634]] 1.0 2jed Homo sapiens AGC_PRKCQ_HUMAN AGC 6.3e-96 326.4 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ KPCT_HUMAN 2JEDB Q04759 375 706 706.0 LG8:61712 Type1 Active DFGin 6.4774 13.7752 BLAminus -116.9, 164.62 69.71, 89.68 -101.74, 24.61 303.13, 88.06 -65.56, -17.66 in-in in 8.9098 Saltbr-in 3.0201 HRD-in -77.46, -49.1 72.97, -12.75 in-in-in SNCiii in-in ActLoopNT-in 2.9394 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -143.05, 132.52 APE9-dihe-na 123.41, 168.41 APE8-dihe-in -74.67, 129.81 APE8-rot-in 290.27 APE67-dihe-in -53.63, -32.33 -43.76, -48.79 APE12-dist-in 8.7728 APE11-dist-in 11.6804 APE10-dist-in 6.647 APE9-dist-in 4.1 I381E,T538E SEP676,SEP695 SEP676,SEP695 XRAY 2.32 0.188 0.221 B 352.0 317.0 0 28 28 0 [[380, 634]] 1.0 2jed Homo sapiens AGC_PRKCQ_HUMAN AGC 6.3e-96 326.4 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ KPCT_HUMAN 5F9EA Q04759 374 706 706.0 5VS:61001 Type1 Active DFGin 6.4755 13.8521 BLAminus -124.47, 161.09 72.18, 90.67 -101.4, 15.51 297.35, 95.13 -63.75, -26.0 in-in in 9.058 Saltbr-in 2.7166 HRD-in -81.15, -47.98 73.24, -5.11 in-in-in SNCiii in-in ActLoopNT-in 2.8522 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -162.97, 169.63 APE9-dihe-na 131.49, -173.01 APE8-dihe-in -109.76, 129.84 APE8-rot-in 295.69 APE67-dihe-in -61.77, -26.26 -46.68, -44.42 APE12-dist-in 8.9537 APE11-dist-in 12.0173 APE10-dist-in 6.5605 APE9-dist-in 3.6595 None SEP676,SEP695 SEP676,SEP695 XRAY 2.0 0.199 0.233 A 353.0 333.0 0 28 28 0 [[380, 634]] 1.0 5f9e Homo sapiens AGC_PRKCQ_HUMAN AGC 6.4e-96 326.4 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ KPCT_HUMAN 5F9EB Q04759 375 700 706.0 5VS:61001 Type1 Active DFGin 6.583 13.8849 BLAminus -118.45, 165.26 62.54, 88.94 -98.52, 15.46 302.93, 89.41 -59.36, -22.06 in-in in 9.2672 Saltbr-in 2.5897 HRD-in -84.26, -45.13 71.76, -7.56 in-in-in SNCiii in-in ActLoopNT-in 2.9056 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -170.19, 135.47 APE9-dihe-na 127.82, -166.17 APE8-dihe-in -112.12, 133.27 APE8-rot-in 297.56 APE67-dihe-in -57.44, -27.74 -44.31, -54.84 APE12-dist-in 8.7675 APE11-dist-in 12.0459 APE10-dist-in 7.3231 APE9-dist-in 3.5782 None SEP676,SEP695 SEP676,SEP695 XRAY 2.0 0.199 0.233 B 353.0 294.0 0 28 28 0 [[380, 634]] 1.0 5f9e Homo sapiens AGC_PRKCQ_HUMAN AGC 6.4e-96 326.4 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type
PRKCQ KPCT_HUMAN 1XJDA Q04759 377 696 706.0 STU:200 Type1 Active DFGin 5.8284 13.1925 BLAminus -132.69, 162.8 69.28, 95.13 -109.8, 21.13 305.67, 104.94 -64.79, -17.76 in-in in 8.0639 Saltbr-in 2.5131 HRD-in -67.27, -48.59 64.56, -1.72 in-in-in SNCiii in-in ActLoopNT-in 2.9684 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -163.73, 166.78 APE9-dihe-na 120.3, 163.8 APE8-dihe-in -75.86, 125.98 APE8-rot-in 298.87 APE67-dihe-in -57.15, -29.94 -38.43, -48.34 APE12-dist-in 9.0296 APE11-dist-in 12.2938 APE10-dist-in 6.8961 APE9-dist-in 3.7669 None TPO538,SEP695 TPO538,SEP695 XRAY 2.0 0.201 0.216 A 345.0 282.0 0 28 28 0 [[380, 634]] 1.0 1xjd Homo sapiens AGC_PRKCQ_HUMAN AGC 1.2e-95 325.5 1.0 260.0 260.0 521 522 523 525 527 409 428 432 501 503 502 504.0 561 549 544 543 542 541 540 539 538 459 Protein kinase C theta type

AGC_PRKCQ (Protein kinase C theta type)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name