OTHER_PKMYT1 (Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase)

Total number of chains: 35
Active chains: 2
Family: OTHER
Uniprot: PMYT1_HUMAN
Kinase Domain Residues: 110 - 359
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 35 100.0% AF-Q99640-K3A

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PDB First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
AF-Q99640-K3A 102 367 499.0 No_ligand No_ligand Active DFGin 6.236 13.701 BLAminus -143.13, -168.07 58.28, 61.82 -75.8, 25.38 307.25, 116.63 -66.88, -23.15 in-in in 8.561 Saltbr-in 2.634 HRD-in -79.61, -40.06 65.08, -14.15 in-in-in SNCiii in-in ActLoopNT-in 2.894 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na -115.86, 147.43 APE9-dihe-na 131.87, 175.12 APE8-dihe-in -90.14, 114.63 APE8-rot-na 184.92 APE67-dihe-in -64.0, -37.49 -58.22, -20.46 APE12-dist-in 8.015 APE11-dist-in 11.205 APE10-dist-in 6.6 APE9-dist-in 5.014 None None None AF2 -1.0 1.0 1.0 A 266 266 0 0 0 0 [[110, 359]] 1.0 AF-Q99640-K3 OTHER_PKMYT1_HUMAN STE 5.6e-39 140.2 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
9M6PBBB 78 361 499.0 A1EMX:401 Type1.5_Back Active DFGin 5.669 14.666 BLAminus -131.55, -170.33 48.66, 72.13 -83.6, 27.49 299.21, 115.57 -58.85, -40.14 in-in in 9.083 Saltbr-in 2.939 HRD-in -81.31, -52.85 67.1, 16.58 in-in-in SNCiii in-in ActLoopNT-in 2.689 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na -92.01, 34.89 APE9-dihe-na -82.85, 167.58 APE8-dihe-in -98.1, 112.26 APE8-rot-na 199.29 APE67-dihe-in -67.7, -28.82 -66.94, -18.17 APE12-dist-in 8.01 APE11-dist-in 10.161 APE10-dist-in 7.317 APE9-dist-in 4.909 None None None XRAY 2.383 0.207 0.29 BBB 311 284 0 0 0 0 [[110, 359]] 1.0 9m6p OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
AF-Q99640-K1A 102 367 499.0 No_ligand No_ligand Inactive DFGin 6.42 13.937 BLAminus -142.18, -168.0 57.83, 63.32 -78.3, 23.73 306.23, 113.15 -65.54, -24.78 in-in in 8.716 Saltbr-in 2.674 HRD-in -78.23, -43.04 64.8, -8.81 in-in-out SNCiio in-out ActLoopNT-in 2.867 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -68.82, 139.71 APE9-dihe-na -79.9, -156.35 APE8-dihe-in -68.58, 121.44 APE8-rot-na 183.21 APE67-dihe-in -65.02, -28.9 -56.4, -24.44 APE12-dist-in 8.19 APE11-dist-out 5.909 APE10-dist-out 9.449 APE9-dist-in 3.898 None None None AF2 -1.0 1.0 1.0 A 266 266 0 0 0 0 [[110, 359]] 1.0 AF-Q99640-K1 OTHER_PKMYT1_HUMAN STE 5.6e-39 140.2 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
3P1AA 76 362 499.0 No_ligand No_ligand Inactive DFGin 6.216 14.644 BLAminus -133.67, -162.14 57.49, 68.87 -85.75, 17.71 301.5, 112.21 -60.51, -27.31 in-in in 8.853 Saltbr-in 2.883 HRD-in -65.08, -43.54 71.41, -3.49 in-in-out SNCiio in-out ActLoopNT-in 2.914 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_oooi APE10-dihe-na -94.27, 138.82 APE9-dihe-na -76.85, 177.99 APE8-dihe-in -60.09, 127.98 APE8-rot-na 184.73 APE67-dihe-in -58.71, -32.77 -62.35, -24.18 APE12-dist-out 6.772 APE11-dist-out 5.446 APE10-dist-out 8.988 APE9-dist-in 3.515 None None None XRAY 1.7 0.152 0.195 A 311 281 6 0 0 6 [[110, 359]] 1.0 3p1a OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8ZTXA 75 361 499.0 A1D83:401 Type1 Inactive DFGin 6.445 14.436 BLAminus -137.85, -159.22 59.85, 66.88 -90.63, 11.4 293.03, 126.73 -73.26, -10.59 in-in in 9.068 Saltbr-in 2.83 HRD-out -87.92, 121.21 -96.15, 14.43 in-in-out SNCiio in-out ActLoopNT-in 2.85 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_oooi APE10-dihe-na -73.57, 129.4 APE9-dihe-na -75.5, 167.07 APE8-dihe-in -68.16, 128.19 APE8-rot-na 189.14 APE67-dihe-in -58.79, -32.8 -64.52, -23.06 APE12-dist-out 5.34 APE11-dist-out 6.439 APE10-dist-out 9.664 APE9-dist-in 3.651 None None None XRAY 1.7 0.183 0.216 A 288 276 4 0 0 3 [[110, 359]] 1.0 8ztx OTHER_PKMYT1_HUMAN STE 7.6e-39 139.7 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
9LGVB 77 361 499.0 A1EJV:403 Type1 Inactive DFGin 6.358 14.519 BLAminus -139.58, -160.2 51.05, 71.76 -89.99, 26.16 301.47, 116.48 -66.83, -24.64 in-in in 8.844 Saltbr-in 2.746 HRD-in -67.6, -49.72 69.87, 5.57 in-in-out SNCiio in-out ActLoopNT-in 2.949 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -66.13, 126.77 APE9-dihe-na -93.12, 179.57 APE8-dihe-in -80.66, 111.84 APE8-rot-na 194.83 APE67-dihe-in -61.91, -33.86 -60.46, -22.61 APE12-dist-in 8.039 APE11-dist-out 5.587 APE10-dist-out 9.595 APE9-dist-in 4.725 None None None XRAY 2.041 0.194 0.234 B 288 279 6 0 0 6 [[110, 359]] 1.0 9lgv OTHER_PKMYT1_HUMAN STE 7.6e-39 139.7 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8ZU2A 75 361 499.0 A1D85:502 Type1 Inactive DFGin 6.426 14.164 BLAminus -143.18, -161.94 58.06, 72.03 -94.83, 14.01 296.25, 122.75 -74.58, -10.24 in-in in 9.031 Saltbr-in 2.807 HRD-out -88.49, 117.25 -97.58, 15.79 in-in-out SNCiio in-out ActLoopNT-in 2.817 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_oooi APE10-dihe-na -77.33, 131.47 APE9-dihe-na -75.94, 168.29 APE8-dihe-in -67.63, 125.44 APE8-rot-na 189.07 APE67-dihe-in -58.12, -32.81 -63.45, -25.22 APE12-dist-out 5.373 APE11-dist-out 6.476 APE10-dist-out 9.654 APE9-dist-in 3.587 None None None XRAY 1.799 0.181 0.222 A 287 273 7 0 0 5 [[110, 359]] 1.0 8zu2 OTHER_PKMYT1_HUMAN STE 7.5e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8ZUDA 75 361 499.0 A1D82:401 Type1 Inactive DFGin 6.321 14.353 BLAminus -140.04, -162.56 63.44, 68.43 -90.94, 13.24 294.38, 121.99 -65.79, -18.98 in-in in 9.069 Saltbr-in 2.789 HRD-out -84.37, 118.24 -94.57, 15.46 in-in-out SNCiio in-out ActLoopNT-in 2.852 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_oooi APE10-dihe-na -73.12, 115.52 APE9-dihe-na -67.77, 166.87 APE8-dihe-in -72.47, 122.64 APE8-rot-na 187.82 APE67-dihe-in -58.53, -33.84 -61.09, -24.42 APE12-dist-out 5.036 APE11-dist-out 6.204 APE10-dist-out 9.679 APE9-dist-in 3.923 None None None XRAY 1.505 0.204 0.238 A 287 280 4 0 0 3 [[110, 359]] 1.0 8zud OTHER_PKMYT1_HUMAN STE 7.5e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8ZULA 75 361 499.0 A1D84:401 Type1 Inactive DFGin 6.412 14.179 BLAminus -138.34, -163.13 57.44, 78.97 -95.66, 20.39 298.61, 119.83 -65.91, -22.49 in-in in 9.119 Saltbr-in 2.878 HRD-out -86.65, 118.04 -96.94, 17.18 in-in-out SNCiio in-out ActLoopNT-in 2.804 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_oooi APE10-dihe-na -86.92, 115.88 APE9-dihe-na -65.84, 161.03 APE8-dihe-in -64.68, 125.13 APE8-rot-na 189.07 APE67-dihe-in -58.22, -33.63 -66.01, -22.62 APE12-dist-out 5.224 APE11-dist-out 6.317 APE10-dist-out 9.704 APE9-dist-in 3.797 None None None XRAY 1.8 0.188 0.219 A 287 278 4 0 0 3 [[110, 359]] 1.0 8zul OTHER_PKMYT1_HUMAN STE 7.5e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
9LGLA 78 361 499.0 A1EJW:401 Type1 Inactive DFGin 6.071 14.461 BLAminus -136.52, -168.54 55.02, 82.28 -98.77, 26.36 303.21, 105.93 -68.53, -22.91 in-in in 9.07 Saltbr-in 2.774 HRD-in -72.0, -47.88 68.59, 9.6 in-in-out SNCiio in-out ActLoopNT-in 2.973 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -72.07, 123.35 APE9-dihe-na -90.71, 177.99 APE8-dihe-in -76.33, 121.78 APE8-rot-na 199.0 APE67-dihe-in -62.44, -32.83 -69.35, -22.28 APE12-dist-in 7.552 APE11-dist-out 6.056 APE10-dist-out 9.809 APE9-dist-in 4.604 None None None XRAY 2.17 0.199 0.234 A 287 269 7 0 0 7 [[110, 359]] 1.0 9lgl OTHER_PKMYT1_HUMAN STE 7.5e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
9LGLB 75 361 499.0 A1EJW:602 Type1 Inactive DFGin 6.19 14.659 BLAminus -138.78, -167.73 53.99, 80.56 -97.13, 31.13 301.33, 106.64 -70.92, -24.39 in-in in 8.979 Saltbr-in 2.604 HRD-in -71.57, -47.46 69.81, 5.38 in-in-out SNCiio in-out ActLoopNT-in 2.937 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -71.5, 123.2 APE9-dihe-na -90.52, 177.91 APE8-dihe-in -75.73, 120.5 APE8-rot-na 196.52 APE67-dihe-in -66.74, -28.94 -66.51, -21.84 APE12-dist-in 7.779 APE11-dist-out 5.745 APE10-dist-out 9.557 APE9-dist-in 4.476 None None None XRAY 2.17 0.199 0.234 B 287 276 3 0 0 3 [[110, 359]] 1.0 9lgl OTHER_PKMYT1_HUMAN STE 7.5e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
5VCVA 75 361 499.0 1N1:60404 Type1 Inactive DFGin 6.173 14.468 BLAminus -133.17, -164.16 53.7, 76.36 -96.77, 22.58 298.04, 107.44 -64.77, -25.22 in-in in 8.918 Saltbr-in 2.826 HRD-in -73.66, -44.65 68.1, -0.34 in-in-out SNCiio in-out ActLoopNT-in 2.893 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -65.91, 159.0 APE9-dihe-na -91.66, -157.73 APE8-dihe-in -52.29, 123.12 APE8-rot-na 188.83 APE67-dihe-in -60.44, -30.04 -60.97, -24.44 APE12-dist-in 7.945 APE11-dist-out 6.449 APE10-dist-out 9.08 APE9-dist-in 3.179 None TPO260 TPO260 XRAY 1.92 0.157 0.197 A 311 287 0 0 0 0 [[110, 359]] 1.0 5vcv OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
5VCWA 77 361 499.0 93J:401 Type1 Inactive DFGin 5.753 14.403 BLAminus -140.89, -170.02 65.17, 65.71 -80.17, 44.69 310.3, 111.94 -72.85, -37.75 in-in in 8.674 Saltbr-in 2.692 HRD-in -65.93, -47.94 69.86, -0.01 in-in-out SNCiio in-out ActLoopNT-in 2.895 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -70.16, 136.95 APE9-dihe-na -95.11, -179.89 APE8-dihe-in -74.56, 119.43 APE8-rot-na 190.69 APE67-dihe-in -62.5, -29.66 -60.78, -22.9 APE12-dist-in 7.636 APE11-dist-out 5.401 APE10-dist-out 9.233 APE9-dist-in 4.514 None None None XRAY 2.25 0.196 0.246 A 311 285 0 0 0 0 [[110, 359]] 1.0 5vcw OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
5VCWB 77 361 499.0 93J:401 Type1 Inactive DFGin 6.174 14.753 BLAminus -145.87, -171.97 60.37, 74.58 -84.49, 28.86 300.8, 108.65 -60.24, -45.91 in-out in 8.991 Saltbr-out 3.796 HRD-in -67.52, -46.64 69.7, -6.0 out-in-out SNCoio in-out ActLoopNT-in 2.905 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -83.37, 139.87 APE9-dihe-na -94.4, -171.94 APE8-dihe-in -64.72, 123.4 APE8-rot-na 193.82 APE67-dihe-in -58.05, -32.99 -66.08, -23.26 APE12-dist-in 8.122 APE11-dist-out 5.498 APE10-dist-out 9.225 APE9-dist-in 4.375 None None None XRAY 2.25 0.196 0.246 B 311 285 0 0 0 0 [[110, 359]] 1.0 5vcw OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
5VCXA 75 361 499.0 H8H:401 Type1 Inactive DFGin 5.945 14.566 BLAminus -133.1, -159.74 56.06, 76.15 -98.03, 28.4 300.17, 108.44 -60.31, -33.85 in-in in 8.996 Saltbr-in 3.063 HRD-in -70.1, -45.94 70.27, -2.25 in-in-out SNCiio in-out ActLoopNT-in 3.051 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -72.13, 165.11 APE9-dihe-na -95.53, -151.65 APE8-dihe-in -59.58, 124.62 APE8-rot-na 194.34 APE67-dihe-in -61.23, -27.43 -59.74, -28.49 APE12-dist-in 7.851 APE11-dist-out 6.313 APE10-dist-out 9.373 APE9-dist-in 3.304 None None None XRAY 2.7 0.201 0.244 A 311 287 0 0 0 0 [[110, 359]] 1.0 5vcx OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
5VCYA 77 362 499.0 DB8:60401 Type1 Inactive DFGin 5.969 14.359 BLAminus -127.91, -168.29 70.38, 72.35 -96.64, 23.14 300.41, 119.28 -68.58, -24.5 in-in in 8.714 Saltbr-in 2.719 HRD-in -69.32, -46.71 70.97, 0.9 in-in-out SNCiio in-out ActLoopNT-in 2.888 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -97.27, 135.17 APE9-dihe-na -76.61, -179.9 APE8-dihe-in -57.88, 126.16 APE8-rot-na 189.14 APE67-dihe-in -62.75, -28.84 -62.08, -23.7 APE12-dist-in 8.015 APE11-dist-out 5.197 APE10-dist-out 9.02 APE9-dist-in 3.47 None None None XRAY 1.56 0.14 0.178 A 311 286 0 0 0 0 [[110, 359]] 1.0 5vcy OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
5VCZA 78 361 499.0 XZN:60401 Type1 Inactive DFGin 6.225 14.363 BLAminus -132.39, -165.29 58.87, 84.05 -99.27, 22.38 300.75, 125.52 -66.24, -24.02 in-in in 8.752 Saltbr-in 2.82 HRD-in -66.5, -47.19 72.05, -1.84 in-in-out SNCiio in-out ActLoopNT-in 2.865 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -98.79, 140.56 APE9-dihe-na -80.46, -177.58 APE8-dihe-in -60.96, 126.51 APE8-rot-na 185.51 APE67-dihe-in -59.29, -30.37 -61.35, -26.02 APE12-dist-in 8.031 APE11-dist-out 5.671 APE10-dist-out 9.053 APE9-dist-in 3.572 None None None XRAY 1.5 0.148 0.181 A 311 284 0 0 0 0 [[110, 359]] 1.0 5vcz OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
5VD0A 77 361 499.0 8X7:60401 Type1 Inactive DFGin 5.962 14.355 BLAminus -141.72, -158.67 59.97, 64.91 -92.35, 27.87 296.04, 115.37 -71.23, -25.83 in-in in 8.585 Saltbr-in 2.96 HRD-in -71.7, -46.16 66.6, 10.57 in-in-out SNCiio in-out ActLoopNT-in 2.798 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -105.71, 140.12 APE9-dihe-na -72.16, -168.22 APE8-dihe-in -65.78, 129.44 APE8-rot-na 186.07 APE67-dihe-in -65.63, -30.01 -61.48, -23.1 APE12-dist-in 7.891 APE11-dist-out 6.337 APE10-dist-out 9.159 APE9-dist-in 3.413 None None None XRAY 2.13 0.195 0.231 A 311 285 0 0 0 0 [[110, 359]] 1.0 5vd0 OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
5VD1A 77 361 499.0 P48:60401 Type1 Inactive DFGin 5.996 14.265 BLAminus -132.04, -170.59 60.28, 78.86 -90.66, 20.44 292.47, 159.81 -62.59, -30.61 in-in in 8.633 Saltbr-in 2.718 HRD-in -67.73, -45.78 69.79, 0.1 in-in-out SNCiio in-out ActLoopNT-in 2.858 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -100.09, 132.84 APE9-dihe-na -80.03, -175.61 APE8-dihe-in -61.66, 124.95 APE8-rot-na 190.14 APE67-dihe-in -61.12, -28.84 -63.37, -24.36 APE12-dist-in 10.437 APE11-dist-out 4.987 APE10-dist-out 9.009 APE9-dist-in 3.507 None None None XRAY 1.7 0.146 0.194 A 311 285 0 0 0 0 [[110, 359]] 1.0 5vd1 OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
5VD3A 78 360 499.0 H8H:60401 Type1 Inactive DFGin 5.988 14.425 BLAminus -136.31, -163.22 68.56, 66.31 -95.1, 21.81 295.33, 125.87 -68.4, -23.33 in-in in 8.495 Saltbr-in 2.673 HRD-in -69.52, -49.09 74.0, 4.67 in-in-out SNCiio in-out ActLoopNT-in 2.908 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -97.34, 136.82 APE9-dihe-na -76.5, -172.94 APE8-dihe-in -60.8, 125.68 APE8-rot-na 188.67 APE67-dihe-in -61.07, -31.05 -63.33, -22.08 APE12-dist-in 7.69 APE11-dist-out 5.948 APE10-dist-out 9.338 APE9-dist-in 3.59 None None None XRAY 1.8 0.167 0.204 A 311 283 0 0 0 0 [[110, 359]] 1.0 5vd3 OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8D6CA 78 362 499.0 QGR:404 Type1 Inactive DFGin 6.172 14.665 BLAminus -138.72, -172.18 56.12, 81.66 -98.6, 28.37 305.05, 105.89 -67.69, -35.68 in-in in 9.223 Saltbr-in 2.867 HRD-in -68.86, -47.17 68.84, 2.61 in-in-out SNCiio in-out ActLoopNT-in 3.043 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -68.71, 138.8 APE9-dihe-na -112.82, 177.1 APE8-dihe-in -70.21, 118.66 APE8-rot-na 199.55 APE67-dihe-in -65.27, -28.23 -67.62, -21.84 APE12-dist-in 7.994 APE11-dist-out 5.138 APE10-dist-out 9.147 APE9-dist-in 4.417 None None None XRAY 2.2 0.243 0.267 A 311 276 4 0 0 4 [[110, 359]] 1.0 8d6c OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8D6CB 77 360 499.0 QGR:405 Type1 Inactive DFGin 6.108 14.617 BLAminus -137.16, -171.57 55.86, 81.51 -98.43, 27.78 304.23, 105.4 -67.24, -36.0 in-in in 9.1 Saltbr-in 2.634 HRD-in -69.35, -47.2 69.11, 3.07 in-in-out SNCiio in-out ActLoopNT-in 2.993 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -68.45, 139.33 APE9-dihe-na -113.05, 178.09 APE8-dihe-in -69.89, 119.27 APE8-rot-na 200.33 APE67-dihe-in -65.97, -28.13 -67.77, -22.03 APE12-dist-in 7.79 APE11-dist-out 5.408 APE10-dist-out 9.568 APE9-dist-in 4.624 None None None XRAY 2.2 0.243 0.267 B 311 279 3 0 0 3 [[110, 359]] 1.0 8d6c OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8D6DB 77 361 499.0 QGY:404 Type1 Inactive DFGin 6.147 14.603 BLAminus -147.14, -174.0 60.06, 69.22 -88.07, 31.47 303.72, 105.86 -72.48, -40.72 in-in in 8.999 Saltbr-in 2.772 HRD-in -71.49, -51.39 74.57, -2.28 in-in-out SNCiio in-out ActLoopNT-in 2.95 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -86.53, 143.01 APE9-dihe-na -115.07, 178.0 APE8-dihe-in -63.78, 124.17 APE8-rot-na 190.84 APE67-dihe-in -58.21, -31.84 -62.0, -28.89 APE12-dist-in 8.114 APE11-dist-out 5.203 APE10-dist-out 9.25 APE9-dist-in 4.199 None None None XRAY 2.35 0.242 0.272 B 311 274 6 0 0 6 [[110, 359]] 1.0 8d6d OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8D6EB 77 361 499.0 QGI:402 Type1 Inactive DFGin 6.114 14.465 BLAminus -132.8, -171.53 58.57, 80.76 -95.11, 24.5 304.2, 110.2 -64.56, -30.79 in-in in 8.951 Saltbr-in 2.628 HRD-in -73.41, -48.43 71.29, 4.33 in-in-out SNCiio in-out ActLoopNT-in 2.998 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -71.04, 132.61 APE9-dihe-na -98.92, -179.59 APE8-dihe-in -79.2, 116.58 APE8-rot-na 195.17 APE67-dihe-in -57.38, -35.46 -62.14, -27.07 APE12-dist-in 7.932 APE11-dist-out 5.296 APE10-dist-out 9.4 APE9-dist-in 4.697 None None None XRAY 2.15 0.192 0.218 B 311 281 0 0 0 0 [[110, 359]] 1.0 8d6e OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8WJYA 76 361 499.0 W9X:60401 Type1 Inactive DFGin 5.935 14.221 BLAminus -135.65, -170.95 60.01, 76.07 -89.46, 18.35 301.57, 113.76 -59.15, -32.82 in-in in 8.832 Saltbr-in 2.806 HRD-in -66.07, -46.85 67.06, 2.44 in-in-out SNCiio in-out ActLoopNT-in 2.772 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nooi APE10-dihe-na -114.14, 142.3 APE9-dihe-na -71.54, 178.2 APE8-dihe-in -61.77, 125.41 APE8-rot-na 182.9 APE67-dihe-in -64.92, -26.73 -59.54, -24.39 APE12-dist-none 999.0 APE11-dist-out 5.785 APE10-dist-out 8.923 APE9-dist-in 3.225 None None None XRAY 1.88 0.174 0.217 A 311 281 5 0 0 5 [[110, 359]] 1.0 8wjy OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
9M6PAAA 78 361 499.0 A1EMX:401 Type1 Inactive DFGin 5.882 14.502 BLAminus -134.53, -168.45 48.74, 78.92 -95.7, 22.92 299.91, 114.53 -64.04, -30.22 in-in in 8.791 Saltbr-in 2.932 HRD-in -72.24, -50.49 83.32, -3.18 in-in-out SNCiio in-out ActLoopNT-in 2.896 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnoi APE10-dihe-na 999.0, 174.25 APE9-dihe-na -61.97, 170.52 APE8-dihe-in -68.14, 121.24 APE8-rot-na 192.46 APE67-dihe-in -58.03, -44.1 -54.7, -32.79 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 8.286 APE9-dist-in 3.496 None None None XRAY 2.383 0.207 0.29 AAA 311 274 7 0 0 7 [[110, 359]] 1.0 9m6p OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
9LGVA 77 361 499.0 A1EJV:403 Type1.5_Back Inactive DFGin 6.247 14.441 BLAminus -138.6, -160.29 51.54, 71.26 -89.36, 26.39 302.35, 116.07 -67.62, -25.64 in-in in 8.813 Saltbr-in 2.72 HRD-in -66.78, -49.09 69.76, 4.94 in-in-out SNCiio in-out ActLoopNT-in 2.923 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -64.33, 125.9 APE9-dihe-na -92.9, 178.41 APE8-dihe-in -82.16, 111.58 APE8-rot-na 195.81 APE67-dihe-in -61.81, -34.11 -61.17, -22.76 APE12-dist-in 7.729 APE11-dist-out 5.577 APE10-dist-out 9.531 APE9-dist-in 4.737 None None None XRAY 2.041 0.194 0.234 A 288 277 7 0 0 7 [[110, 359]] 1.0 9lgv OTHER_PKMYT1_HUMAN STE 7.6e-39 139.7 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
9LIDA 77 361 499.0 A1EJX:401 Type1.5_Back Inactive DFGin 6.147 14.664 BLAminus -141.57, -159.93 44.66, 82.65 -96.79, 25.45 296.42, 128.92 -69.09, -25.86 in-in in 8.914 Saltbr-in 2.78 HRD-in -71.98, -50.6 73.9, 10.26 in-in-out SNCiio in-out ActLoopNT-in 2.986 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -65.91, 118.73 APE9-dihe-na -84.87, 178.55 APE8-dihe-in -75.21, 121.23 APE8-rot-na 199.89 APE67-dihe-in -56.46, -34.28 -66.08, -29.38 APE12-dist-in 7.934 APE11-dist-out 5.555 APE10-dist-out 9.424 APE9-dist-in 4.289 None None None XRAY 2.06 0.205 0.231 A 288 272 5 0 0 5 [[110, 359]] 1.0 9lid OTHER_PKMYT1_HUMAN STE 7.6e-39 139.7 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
9LIDB 77 361 499.0 A1EJX:401 Type1.5_Back Inactive DFGin 6.109 14.623 BLAminus -138.92, -162.74 50.8, 79.94 -95.85, 31.4 299.01, 122.08 -70.56, -35.67 in-in in 8.837 Saltbr-in 2.739 HRD-in -63.43, -48.29 66.83, 6.87 in-in-out SNCiio in-out ActLoopNT-in 3.014 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -70.06, 130.49 APE9-dihe-na -98.3, 177.7 APE8-dihe-in -71.64, 117.04 APE8-rot-na 198.93 APE67-dihe-in -59.05, -34.81 -63.57, -26.6 APE12-dist-in 7.886 APE11-dist-out 5.525 APE10-dist-out 9.483 APE9-dist-in 4.637 None None None XRAY 2.06 0.205 0.231 B 288 279 0 0 0 0 [[110, 359]] 1.0 9lid OTHER_PKMYT1_HUMAN STE 7.6e-39 139.7 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
9LGNA 77 361 499.0 A1EJU:60401 Type1.5_Back Inactive DFGin 6.296 14.466 BLAminus -145.99, -171.4 50.86, 84.26 -97.86, 29.36 304.36, 111.52 -72.91, -21.87 in-in in 8.887 Saltbr-in 2.795 HRD-in -66.21, -46.68 65.26, 16.91 in-in-out SNCiio in-out ActLoopNT-in 3.082 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -68.54, 120.07 APE9-dihe-na -90.78, -176.48 APE8-dihe-in -82.34, 121.43 APE8-rot-na 199.89 APE67-dihe-in -63.02, -34.9 -65.92, -23.54 APE12-dist-in 7.833 APE11-dist-out 5.486 APE10-dist-out 9.422 APE9-dist-in 4.545 None None None XRAY 2.03 0.196 0.241 A 286 280 5 0 0 5 [[110, 359]] 1.0 9lgn OTHER_PKMYT1_HUMAN STE 7.4e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
9LGNB 77 361 499.0 A1EJU:60401 Type1.5_Back Inactive DFGin 6.068 14.404 BLAminus -142.39, -165.96 54.01, 79.86 -92.24, 28.67 300.8, 134.57 -69.88, -31.54 in-in in 8.842 Saltbr-in 2.621 HRD-in -68.45, -46.04 66.53, 9.81 in-in-out SNCiio in-out ActLoopNT-in 3.009 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -64.59, 124.38 APE9-dihe-na -93.34, -179.18 APE8-dihe-in -77.16, 120.0 APE8-rot-na 200.38 APE67-dihe-in -63.03, -36.01 -66.03, -24.01 APE12-dist-in 7.864 APE11-dist-out 5.611 APE10-dist-out 9.357 APE9-dist-in 4.519 None None None XRAY 2.03 0.196 0.241 B 286 281 4 0 0 4 [[110, 359]] 1.0 9lgn OTHER_PKMYT1_HUMAN STE 7.4e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8D6DA 78 361 499.0 QGY:405 Type1.5_Back Inactive DFGin 6.211 14.538 BLAminus -148.07, -173.76 61.71, 69.04 -87.4, 33.63 306.09, 107.4 -73.23, -43.69 in-in in 8.979 Saltbr-in 2.792 HRD-in -70.41, -52.13 74.56, -0.66 in-in-out SNCiio in-out ActLoopNT-in 3.042 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -82.14, 144.34 APE9-dihe-na -114.82, 178.25 APE8-dihe-in -66.9, 123.15 APE8-rot-na 195.13 APE67-dihe-in -58.55, -32.2 -61.02, -29.72 APE12-dist-in 7.901 APE11-dist-out 5.216 APE10-dist-out 9.078 APE9-dist-in 4.364 None None None XRAY 2.35 0.242 0.272 A 311 270 5 0 0 5 [[110, 359]] 1.0 8d6d OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8D6EA 77 361 499.0 QGI:1303 Type1.5_Back Inactive DFGin 5.964 14.172 BLAminus -132.85, -170.23 57.02, 82.01 -94.72, 23.46 304.19, 110.84 -65.02, -29.08 in-in in 8.87 Saltbr-in 2.717 HRD-in -75.21, -49.23 71.68, 5.95 in-in-out SNCiio in-out ActLoopNT-in 2.94 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -70.02, 134.68 APE9-dihe-na -98.58, -177.84 APE8-dihe-in -78.94, 114.38 APE8-rot-na 196.53 APE67-dihe-in -55.24, -36.47 -61.38, -25.28 APE12-dist-in 7.804 APE11-dist-out 5.579 APE10-dist-out 9.69 APE9-dist-in 4.697 None None None XRAY 2.15 0.192 0.218 A 311 278 3 0 0 3 [[110, 359]] 1.0 8d6e OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8D6FA 78 361 499.0 QG5:402 Type1.5_Back Inactive DFGin 5.934 14.393 BLAminus -137.99, -170.0 54.51, 81.69 -95.67, 27.93 303.43, 112.84 -67.3, -27.64 in-in in 8.927 Saltbr-in 2.693 HRD-in -64.05, -49.24 70.41, 3.13 in-in-out SNCiio in-out ActLoopNT-in 2.974 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -70.94, 136.66 APE9-dihe-na -111.83, 176.77 APE8-dihe-in -71.13, 118.43 APE8-rot-na 201.17 APE67-dihe-in -57.59, -30.74 -64.31, -29.06 APE12-dist-in 7.268 APE11-dist-out 5.262 APE10-dist-out 9.373 APE9-dist-in 4.633 None None None XRAY 2.49 0.216 0.239 A 311 270 6 0 0 6 [[110, 359]] 1.0 8d6f OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
8D6FB 76 361 499.0 QG5:402 Type1.5_Back Inactive DFGin 6.014 14.327 BLAminus -137.52, -169.84 54.56, 81.42 -96.27, 27.52 303.69, 112.72 -67.62, -27.32 in-in in 8.86 Saltbr-in 2.731 HRD-in -63.86, -48.97 70.29, 4.03 in-in-out SNCiio in-out ActLoopNT-in 3.061 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -70.91, 136.32 APE9-dihe-na -112.58, 175.93 APE8-dihe-in -71.78, 118.97 APE8-rot-na 200.9 APE67-dihe-in -57.56, -31.19 -64.02, -28.04 APE12-dist-in 7.294 APE11-dist-out 5.136 APE10-dist-out 9.236 APE9-dist-in 4.543 None None None XRAY 2.49 0.216 0.239 B 311 272 6 0 0 6 [[110, 359]] 1.0 8d6f OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase

OTHER_PKMYT1 (Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase)

Total number of chains: 35
Active chains: 2
Family: OTHER
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 35 100.0% AF-Q99640-K3A

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
PMYT1_HUMAN AF-Q99640-K3A Q99640 102 367 499.0 No_ligand No_ligand Active DFGin 6.236 13.701 BLAminus -143.13, -168.07 58.28, 61.82 -75.8, 25.38 307.25, 116.63 -66.88, -23.15 in-in in 8.561 Saltbr-in 2.634 HRD-in -79.61, -40.06 65.08, -14.15 in-in-in SNCiii in-in ActLoopNT-in 2.894 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na -115.86, 147.43 APE9-dihe-na 131.87, 175.12 APE8-dihe-in -90.14, 114.63 APE8-rot-na 184.92 APE67-dihe-in -64.0, -37.49 -58.22, -20.46 APE12-dist-in 8.015 APE11-dist-in 11.205 APE10-dist-in 6.6 APE9-dist-in 5.014 None None None AF2 -1.0 1.0 1.0 A 266 266 0 0 0 0 [[110, 359]] 1.0 AF-Q99640-K3 Homo sapiens OTHER_PKMYT1_HUMAN STE 5.6e-39 140.2 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 9M6PBBB Q99640 78 361 499.0 A1EMX:401 Type1.5_Back Active DFGin 5.669 14.666 BLAminus -131.55, -170.33 48.66, 72.13 -83.6, 27.49 299.21, 115.57 -58.85, -40.14 in-in in 9.083 Saltbr-in 2.939 HRD-in -81.31, -52.85 67.1, 16.58 in-in-in SNCiii in-in ActLoopNT-in 2.689 ActLoopCT-in nonTYR APEdihe_aaiai APEdist_iiii APE10-dihe-na -92.01, 34.89 APE9-dihe-na -82.85, 167.58 APE8-dihe-in -98.1, 112.26 APE8-rot-na 199.29 APE67-dihe-in -67.7, -28.82 -66.94, -18.17 APE12-dist-in 8.01 APE11-dist-in 10.161 APE10-dist-in 7.317 APE9-dist-in 4.909 None None None XRAY 2.383 0.207 0.29 BBB 311 284 0 0 0 0 [[110, 359]] 1.0 9m6p Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN AF-Q99640-K1A Q99640 102 367 499.0 No_ligand No_ligand Inactive DFGin 6.42 13.937 BLAminus -142.18, -168.0 57.83, 63.32 -78.3, 23.73 306.23, 113.15 -65.54, -24.78 in-in in 8.716 Saltbr-in 2.674 HRD-in -78.23, -43.04 64.8, -8.81 in-in-out SNCiio in-out ActLoopNT-in 2.867 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -68.82, 139.71 APE9-dihe-na -79.9, -156.35 APE8-dihe-in -68.58, 121.44 APE8-rot-na 183.21 APE67-dihe-in -65.02, -28.9 -56.4, -24.44 APE12-dist-in 8.19 APE11-dist-out 5.909 APE10-dist-out 9.449 APE9-dist-in 3.898 None None None AF2 -1.0 1.0 1.0 A 266 266 0 0 0 0 [[110, 359]] 1.0 AF-Q99640-K1 Homo sapiens OTHER_PKMYT1_HUMAN STE 5.6e-39 140.2 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 3P1AA Q99640 76 362 499.0 No_ligand No_ligand Inactive DFGin 6.216 14.644 BLAminus -133.67, -162.14 57.49, 68.87 -85.75, 17.71 301.5, 112.21 -60.51, -27.31 in-in in 8.853 Saltbr-in 2.883 HRD-in -65.08, -43.54 71.41, -3.49 in-in-out SNCiio in-out ActLoopNT-in 2.914 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_oooi APE10-dihe-na -94.27, 138.82 APE9-dihe-na -76.85, 177.99 APE8-dihe-in -60.09, 127.98 APE8-rot-na 184.73 APE67-dihe-in -58.71, -32.77 -62.35, -24.18 APE12-dist-out 6.772 APE11-dist-out 5.446 APE10-dist-out 8.988 APE9-dist-in 3.515 None None None XRAY 1.7 0.152 0.195 A 311 281 6 0 0 6 [[110, 359]] 1.0 3p1a Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8ZTXA Q99640 75 361 499.0 A1D83:401 Type1 Inactive DFGin 6.445 14.436 BLAminus -137.85, -159.22 59.85, 66.88 -90.63, 11.4 293.03, 126.73 -73.26, -10.59 in-in in 9.068 Saltbr-in 2.83 HRD-out -87.92, 121.21 -96.15, 14.43 in-in-out SNCiio in-out ActLoopNT-in 2.85 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_oooi APE10-dihe-na -73.57, 129.4 APE9-dihe-na -75.5, 167.07 APE8-dihe-in -68.16, 128.19 APE8-rot-na 189.14 APE67-dihe-in -58.79, -32.8 -64.52, -23.06 APE12-dist-out 5.34 APE11-dist-out 6.439 APE10-dist-out 9.664 APE9-dist-in 3.651 None None None XRAY 1.7 0.183 0.216 A 288 276 4 0 0 3 [[110, 359]] 1.0 8ztx Homo sapiens OTHER_PKMYT1_HUMAN STE 7.6e-39 139.7 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 9LGVB Q99640 77 361 499.0 A1EJV:403 Type1 Inactive DFGin 6.358 14.519 BLAminus -139.58, -160.2 51.05, 71.76 -89.99, 26.16 301.47, 116.48 -66.83, -24.64 in-in in 8.844 Saltbr-in 2.746 HRD-in -67.6, -49.72 69.87, 5.57 in-in-out SNCiio in-out ActLoopNT-in 2.949 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -66.13, 126.77 APE9-dihe-na -93.12, 179.57 APE8-dihe-in -80.66, 111.84 APE8-rot-na 194.83 APE67-dihe-in -61.91, -33.86 -60.46, -22.61 APE12-dist-in 8.039 APE11-dist-out 5.587 APE10-dist-out 9.595 APE9-dist-in 4.725 None None None XRAY 2.041 0.194 0.234 B 288 279 6 0 0 6 [[110, 359]] 1.0 9lgv Homo sapiens OTHER_PKMYT1_HUMAN STE 7.6e-39 139.7 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8ZU2A Q99640 75 361 499.0 A1D85:502 Type1 Inactive DFGin 6.426 14.164 BLAminus -143.18, -161.94 58.06, 72.03 -94.83, 14.01 296.25, 122.75 -74.58, -10.24 in-in in 9.031 Saltbr-in 2.807 HRD-out -88.49, 117.25 -97.58, 15.79 in-in-out SNCiio in-out ActLoopNT-in 2.817 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_oooi APE10-dihe-na -77.33, 131.47 APE9-dihe-na -75.94, 168.29 APE8-dihe-in -67.63, 125.44 APE8-rot-na 189.07 APE67-dihe-in -58.12, -32.81 -63.45, -25.22 APE12-dist-out 5.373 APE11-dist-out 6.476 APE10-dist-out 9.654 APE9-dist-in 3.587 None None None XRAY 1.799 0.181 0.222 A 287 273 7 0 0 5 [[110, 359]] 1.0 8zu2 Homo sapiens OTHER_PKMYT1_HUMAN STE 7.5e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8ZUDA Q99640 75 361 499.0 A1D82:401 Type1 Inactive DFGin 6.321 14.353 BLAminus -140.04, -162.56 63.44, 68.43 -90.94, 13.24 294.38, 121.99 -65.79, -18.98 in-in in 9.069 Saltbr-in 2.789 HRD-out -84.37, 118.24 -94.57, 15.46 in-in-out SNCiio in-out ActLoopNT-in 2.852 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_oooi APE10-dihe-na -73.12, 115.52 APE9-dihe-na -67.77, 166.87 APE8-dihe-in -72.47, 122.64 APE8-rot-na 187.82 APE67-dihe-in -58.53, -33.84 -61.09, -24.42 APE12-dist-out 5.036 APE11-dist-out 6.204 APE10-dist-out 9.679 APE9-dist-in 3.923 None None None XRAY 1.505 0.204 0.238 A 287 280 4 0 0 3 [[110, 359]] 1.0 8zud Homo sapiens OTHER_PKMYT1_HUMAN STE 7.5e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8ZULA Q99640 75 361 499.0 A1D84:401 Type1 Inactive DFGin 6.412 14.179 BLAminus -138.34, -163.13 57.44, 78.97 -95.66, 20.39 298.61, 119.83 -65.91, -22.49 in-in in 9.119 Saltbr-in 2.878 HRD-out -86.65, 118.04 -96.94, 17.18 in-in-out SNCiio in-out ActLoopNT-in 2.804 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_oooi APE10-dihe-na -86.92, 115.88 APE9-dihe-na -65.84, 161.03 APE8-dihe-in -64.68, 125.13 APE8-rot-na 189.07 APE67-dihe-in -58.22, -33.63 -66.01, -22.62 APE12-dist-out 5.224 APE11-dist-out 6.317 APE10-dist-out 9.704 APE9-dist-in 3.797 None None None XRAY 1.8 0.188 0.219 A 287 278 4 0 0 3 [[110, 359]] 1.0 8zul Homo sapiens OTHER_PKMYT1_HUMAN STE 7.5e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 9LGLA Q99640 78 361 499.0 A1EJW:401 Type1 Inactive DFGin 6.071 14.461 BLAminus -136.52, -168.54 55.02, 82.28 -98.77, 26.36 303.21, 105.93 -68.53, -22.91 in-in in 9.07 Saltbr-in 2.774 HRD-in -72.0, -47.88 68.59, 9.6 in-in-out SNCiio in-out ActLoopNT-in 2.973 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -72.07, 123.35 APE9-dihe-na -90.71, 177.99 APE8-dihe-in -76.33, 121.78 APE8-rot-na 199.0 APE67-dihe-in -62.44, -32.83 -69.35, -22.28 APE12-dist-in 7.552 APE11-dist-out 6.056 APE10-dist-out 9.809 APE9-dist-in 4.604 None None None XRAY 2.17 0.199 0.234 A 287 269 7 0 0 7 [[110, 359]] 1.0 9lgl Homo sapiens OTHER_PKMYT1_HUMAN STE 7.5e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 9LGLB Q99640 75 361 499.0 A1EJW:602 Type1 Inactive DFGin 6.19 14.659 BLAminus -138.78, -167.73 53.99, 80.56 -97.13, 31.13 301.33, 106.64 -70.92, -24.39 in-in in 8.979 Saltbr-in 2.604 HRD-in -71.57, -47.46 69.81, 5.38 in-in-out SNCiio in-out ActLoopNT-in 2.937 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -71.5, 123.2 APE9-dihe-na -90.52, 177.91 APE8-dihe-in -75.73, 120.5 APE8-rot-na 196.52 APE67-dihe-in -66.74, -28.94 -66.51, -21.84 APE12-dist-in 7.779 APE11-dist-out 5.745 APE10-dist-out 9.557 APE9-dist-in 4.476 None None None XRAY 2.17 0.199 0.234 B 287 276 3 0 0 3 [[110, 359]] 1.0 9lgl Homo sapiens OTHER_PKMYT1_HUMAN STE 7.5e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 5VCVA Q99640 75 361 499.0 1N1:60404 Type1 Inactive DFGin 6.173 14.468 BLAminus -133.17, -164.16 53.7, 76.36 -96.77, 22.58 298.04, 107.44 -64.77, -25.22 in-in in 8.918 Saltbr-in 2.826 HRD-in -73.66, -44.65 68.1, -0.34 in-in-out SNCiio in-out ActLoopNT-in 2.893 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -65.91, 159.0 APE9-dihe-na -91.66, -157.73 APE8-dihe-in -52.29, 123.12 APE8-rot-na 188.83 APE67-dihe-in -60.44, -30.04 -60.97, -24.44 APE12-dist-in 7.945 APE11-dist-out 6.449 APE10-dist-out 9.08 APE9-dist-in 3.179 None TPO260 TPO260 XRAY 1.92 0.157 0.197 A 311 287 0 0 0 0 [[110, 359]] 1.0 5vcv Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 5VCWA Q99640 77 361 499.0 93J:401 Type1 Inactive DFGin 5.753 14.403 BLAminus -140.89, -170.02 65.17, 65.71 -80.17, 44.69 310.3, 111.94 -72.85, -37.75 in-in in 8.674 Saltbr-in 2.692 HRD-in -65.93, -47.94 69.86, -0.01 in-in-out SNCiio in-out ActLoopNT-in 2.895 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -70.16, 136.95 APE9-dihe-na -95.11, -179.89 APE8-dihe-in -74.56, 119.43 APE8-rot-na 190.69 APE67-dihe-in -62.5, -29.66 -60.78, -22.9 APE12-dist-in 7.636 APE11-dist-out 5.401 APE10-dist-out 9.233 APE9-dist-in 4.514 None None None XRAY 2.25 0.196 0.246 A 311 285 0 0 0 0 [[110, 359]] 1.0 5vcw Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 5VCWB Q99640 77 361 499.0 93J:401 Type1 Inactive DFGin 6.174 14.753 BLAminus -145.87, -171.97 60.37, 74.58 -84.49, 28.86 300.8, 108.65 -60.24, -45.91 in-out in 8.991 Saltbr-out 3.796 HRD-in -67.52, -46.64 69.7, -6.0 out-in-out SNCoio in-out ActLoopNT-in 2.905 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -83.37, 139.87 APE9-dihe-na -94.4, -171.94 APE8-dihe-in -64.72, 123.4 APE8-rot-na 193.82 APE67-dihe-in -58.05, -32.99 -66.08, -23.26 APE12-dist-in 8.122 APE11-dist-out 5.498 APE10-dist-out 9.225 APE9-dist-in 4.375 None None None XRAY 2.25 0.196 0.246 B 311 285 0 0 0 0 [[110, 359]] 1.0 5vcw Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 5VCXA Q99640 75 361 499.0 H8H:401 Type1 Inactive DFGin 5.945 14.566 BLAminus -133.1, -159.74 56.06, 76.15 -98.03, 28.4 300.17, 108.44 -60.31, -33.85 in-in in 8.996 Saltbr-in 3.063 HRD-in -70.1, -45.94 70.27, -2.25 in-in-out SNCiio in-out ActLoopNT-in 3.051 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -72.13, 165.11 APE9-dihe-na -95.53, -151.65 APE8-dihe-in -59.58, 124.62 APE8-rot-na 194.34 APE67-dihe-in -61.23, -27.43 -59.74, -28.49 APE12-dist-in 7.851 APE11-dist-out 6.313 APE10-dist-out 9.373 APE9-dist-in 3.304 None None None XRAY 2.7 0.201 0.244 A 311 287 0 0 0 0 [[110, 359]] 1.0 5vcx Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 5VCYA Q99640 77 362 499.0 DB8:60401 Type1 Inactive DFGin 5.969 14.359 BLAminus -127.91, -168.29 70.38, 72.35 -96.64, 23.14 300.41, 119.28 -68.58, -24.5 in-in in 8.714 Saltbr-in 2.719 HRD-in -69.32, -46.71 70.97, 0.9 in-in-out SNCiio in-out ActLoopNT-in 2.888 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -97.27, 135.17 APE9-dihe-na -76.61, -179.9 APE8-dihe-in -57.88, 126.16 APE8-rot-na 189.14 APE67-dihe-in -62.75, -28.84 -62.08, -23.7 APE12-dist-in 8.015 APE11-dist-out 5.197 APE10-dist-out 9.02 APE9-dist-in 3.47 None None None XRAY 1.56 0.14 0.178 A 311 286 0 0 0 0 [[110, 359]] 1.0 5vcy Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 5VCZA Q99640 78 361 499.0 XZN:60401 Type1 Inactive DFGin 6.225 14.363 BLAminus -132.39, -165.29 58.87, 84.05 -99.27, 22.38 300.75, 125.52 -66.24, -24.02 in-in in 8.752 Saltbr-in 2.82 HRD-in -66.5, -47.19 72.05, -1.84 in-in-out SNCiio in-out ActLoopNT-in 2.865 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -98.79, 140.56 APE9-dihe-na -80.46, -177.58 APE8-dihe-in -60.96, 126.51 APE8-rot-na 185.51 APE67-dihe-in -59.29, -30.37 -61.35, -26.02 APE12-dist-in 8.031 APE11-dist-out 5.671 APE10-dist-out 9.053 APE9-dist-in 3.572 None None None XRAY 1.5 0.148 0.181 A 311 284 0 0 0 0 [[110, 359]] 1.0 5vcz Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 5VD0A Q99640 77 361 499.0 8X7:60401 Type1 Inactive DFGin 5.962 14.355 BLAminus -141.72, -158.67 59.97, 64.91 -92.35, 27.87 296.04, 115.37 -71.23, -25.83 in-in in 8.585 Saltbr-in 2.96 HRD-in -71.7, -46.16 66.6, 10.57 in-in-out SNCiio in-out ActLoopNT-in 2.798 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -105.71, 140.12 APE9-dihe-na -72.16, -168.22 APE8-dihe-in -65.78, 129.44 APE8-rot-na 186.07 APE67-dihe-in -65.63, -30.01 -61.48, -23.1 APE12-dist-in 7.891 APE11-dist-out 6.337 APE10-dist-out 9.159 APE9-dist-in 3.413 None None None XRAY 2.13 0.195 0.231 A 311 285 0 0 0 0 [[110, 359]] 1.0 5vd0 Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 5VD1A Q99640 77 361 499.0 P48:60401 Type1 Inactive DFGin 5.996 14.265 BLAminus -132.04, -170.59 60.28, 78.86 -90.66, 20.44 292.47, 159.81 -62.59, -30.61 in-in in 8.633 Saltbr-in 2.718 HRD-in -67.73, -45.78 69.79, 0.1 in-in-out SNCiio in-out ActLoopNT-in 2.858 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -100.09, 132.84 APE9-dihe-na -80.03, -175.61 APE8-dihe-in -61.66, 124.95 APE8-rot-na 190.14 APE67-dihe-in -61.12, -28.84 -63.37, -24.36 APE12-dist-in 10.437 APE11-dist-out 4.987 APE10-dist-out 9.009 APE9-dist-in 3.507 None None None XRAY 1.7 0.146 0.194 A 311 285 0 0 0 0 [[110, 359]] 1.0 5vd1 Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 5VD3A Q99640 78 360 499.0 H8H:60401 Type1 Inactive DFGin 5.988 14.425 BLAminus -136.31, -163.22 68.56, 66.31 -95.1, 21.81 295.33, 125.87 -68.4, -23.33 in-in in 8.495 Saltbr-in 2.673 HRD-in -69.52, -49.09 74.0, 4.67 in-in-out SNCiio in-out ActLoopNT-in 2.908 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -97.34, 136.82 APE9-dihe-na -76.5, -172.94 APE8-dihe-in -60.8, 125.68 APE8-rot-na 188.67 APE67-dihe-in -61.07, -31.05 -63.33, -22.08 APE12-dist-in 7.69 APE11-dist-out 5.948 APE10-dist-out 9.338 APE9-dist-in 3.59 None None None XRAY 1.8 0.167 0.204 A 311 283 0 0 0 0 [[110, 359]] 1.0 5vd3 Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8D6CA Q99640 78 362 499.0 QGR:404 Type1 Inactive DFGin 6.172 14.665 BLAminus -138.72, -172.18 56.12, 81.66 -98.6, 28.37 305.05, 105.89 -67.69, -35.68 in-in in 9.223 Saltbr-in 2.867 HRD-in -68.86, -47.17 68.84, 2.61 in-in-out SNCiio in-out ActLoopNT-in 3.043 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -68.71, 138.8 APE9-dihe-na -112.82, 177.1 APE8-dihe-in -70.21, 118.66 APE8-rot-na 199.55 APE67-dihe-in -65.27, -28.23 -67.62, -21.84 APE12-dist-in 7.994 APE11-dist-out 5.138 APE10-dist-out 9.147 APE9-dist-in 4.417 None None None XRAY 2.2 0.243 0.267 A 311 276 4 0 0 4 [[110, 359]] 1.0 8d6c Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8D6CB Q99640 77 360 499.0 QGR:405 Type1 Inactive DFGin 6.108 14.617 BLAminus -137.16, -171.57 55.86, 81.51 -98.43, 27.78 304.23, 105.4 -67.24, -36.0 in-in in 9.1 Saltbr-in 2.634 HRD-in -69.35, -47.2 69.11, 3.07 in-in-out SNCiio in-out ActLoopNT-in 2.993 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -68.45, 139.33 APE9-dihe-na -113.05, 178.09 APE8-dihe-in -69.89, 119.27 APE8-rot-na 200.33 APE67-dihe-in -65.97, -28.13 -67.77, -22.03 APE12-dist-in 7.79 APE11-dist-out 5.408 APE10-dist-out 9.568 APE9-dist-in 4.624 None None None XRAY 2.2 0.243 0.267 B 311 279 3 0 0 3 [[110, 359]] 1.0 8d6c Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8D6DB Q99640 77 361 499.0 QGY:404 Type1 Inactive DFGin 6.147 14.603 BLAminus -147.14, -174.0 60.06, 69.22 -88.07, 31.47 303.72, 105.86 -72.48, -40.72 in-in in 8.999 Saltbr-in 2.772 HRD-in -71.49, -51.39 74.57, -2.28 in-in-out SNCiio in-out ActLoopNT-in 2.95 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -86.53, 143.01 APE9-dihe-na -115.07, 178.0 APE8-dihe-in -63.78, 124.17 APE8-rot-na 190.84 APE67-dihe-in -58.21, -31.84 -62.0, -28.89 APE12-dist-in 8.114 APE11-dist-out 5.203 APE10-dist-out 9.25 APE9-dist-in 4.199 None None None XRAY 2.35 0.242 0.272 B 311 274 6 0 0 6 [[110, 359]] 1.0 8d6d Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8D6EB Q99640 77 361 499.0 QGI:402 Type1 Inactive DFGin 6.114 14.465 BLAminus -132.8, -171.53 58.57, 80.76 -95.11, 24.5 304.2, 110.2 -64.56, -30.79 in-in in 8.951 Saltbr-in 2.628 HRD-in -73.41, -48.43 71.29, 4.33 in-in-out SNCiio in-out ActLoopNT-in 2.998 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -71.04, 132.61 APE9-dihe-na -98.92, -179.59 APE8-dihe-in -79.2, 116.58 APE8-rot-na 195.17 APE67-dihe-in -57.38, -35.46 -62.14, -27.07 APE12-dist-in 7.932 APE11-dist-out 5.296 APE10-dist-out 9.4 APE9-dist-in 4.697 None None None XRAY 2.15 0.192 0.218 B 311 281 0 0 0 0 [[110, 359]] 1.0 8d6e Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8WJYA Q99640 76 361 499.0 W9X:60401 Type1 Inactive DFGin 5.935 14.221 BLAminus -135.65, -170.95 60.01, 76.07 -89.46, 18.35 301.57, 113.76 -59.15, -32.82 in-in in 8.832 Saltbr-in 2.806 HRD-in -66.07, -46.85 67.06, 2.44 in-in-out SNCiio in-out ActLoopNT-in 2.772 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nooi APE10-dihe-na -114.14, 142.3 APE9-dihe-na -71.54, 178.2 APE8-dihe-in -61.77, 125.41 APE8-rot-na 182.9 APE67-dihe-in -64.92, -26.73 -59.54, -24.39 APE12-dist-none 999.0 APE11-dist-out 5.785 APE10-dist-out 8.923 APE9-dist-in 3.225 None None None XRAY 1.88 0.174 0.217 A 311 281 5 0 0 5 [[110, 359]] 1.0 8wjy Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 9M6PAAA Q99640 78 361 499.0 A1EMX:401 Type1 Inactive DFGin 5.882 14.502 BLAminus -134.53, -168.45 48.74, 78.92 -95.7, 22.92 299.91, 114.53 -64.04, -30.22 in-in in 8.791 Saltbr-in 2.932 HRD-in -72.24, -50.49 83.32, -3.18 in-in-out SNCiio in-out ActLoopNT-in 2.896 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_nnoi APE10-dihe-na 999.0, 174.25 APE9-dihe-na -61.97, 170.52 APE8-dihe-in -68.14, 121.24 APE8-rot-na 192.46 APE67-dihe-in -58.03, -44.1 -54.7, -32.79 APE12-dist-none 999.0 APE11-dist-none 999.0 APE10-dist-out 8.286 APE9-dist-in 3.496 None None None XRAY 2.383 0.207 0.29 AAA 311 274 7 0 0 7 [[110, 359]] 1.0 9m6p Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 9LGVA Q99640 77 361 499.0 A1EJV:403 Type1.5_Back Inactive DFGin 6.247 14.441 BLAminus -138.6, -160.29 51.54, 71.26 -89.36, 26.39 302.35, 116.07 -67.62, -25.64 in-in in 8.813 Saltbr-in 2.72 HRD-in -66.78, -49.09 69.76, 4.94 in-in-out SNCiio in-out ActLoopNT-in 2.923 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -64.33, 125.9 APE9-dihe-na -92.9, 178.41 APE8-dihe-in -82.16, 111.58 APE8-rot-na 195.81 APE67-dihe-in -61.81, -34.11 -61.17, -22.76 APE12-dist-in 7.729 APE11-dist-out 5.577 APE10-dist-out 9.531 APE9-dist-in 4.737 None None None XRAY 2.041 0.194 0.234 A 288 277 7 0 0 7 [[110, 359]] 1.0 9lgv Homo sapiens OTHER_PKMYT1_HUMAN STE 7.6e-39 139.7 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 9LIDA Q99640 77 361 499.0 A1EJX:401 Type1.5_Back Inactive DFGin 6.147 14.664 BLAminus -141.57, -159.93 44.66, 82.65 -96.79, 25.45 296.42, 128.92 -69.09, -25.86 in-in in 8.914 Saltbr-in 2.78 HRD-in -71.98, -50.6 73.9, 10.26 in-in-out SNCiio in-out ActLoopNT-in 2.986 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -65.91, 118.73 APE9-dihe-na -84.87, 178.55 APE8-dihe-in -75.21, 121.23 APE8-rot-na 199.89 APE67-dihe-in -56.46, -34.28 -66.08, -29.38 APE12-dist-in 7.934 APE11-dist-out 5.555 APE10-dist-out 9.424 APE9-dist-in 4.289 None None None XRAY 2.06 0.205 0.231 A 288 272 5 0 0 5 [[110, 359]] 1.0 9lid Homo sapiens OTHER_PKMYT1_HUMAN STE 7.6e-39 139.7 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 9LIDB Q99640 77 361 499.0 A1EJX:401 Type1.5_Back Inactive DFGin 6.109 14.623 BLAminus -138.92, -162.74 50.8, 79.94 -95.85, 31.4 299.01, 122.08 -70.56, -35.67 in-in in 8.837 Saltbr-in 2.739 HRD-in -63.43, -48.29 66.83, 6.87 in-in-out SNCiio in-out ActLoopNT-in 3.014 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -70.06, 130.49 APE9-dihe-na -98.3, 177.7 APE8-dihe-in -71.64, 117.04 APE8-rot-na 198.93 APE67-dihe-in -59.05, -34.81 -63.57, -26.6 APE12-dist-in 7.886 APE11-dist-out 5.525 APE10-dist-out 9.483 APE9-dist-in 4.637 None None None XRAY 2.06 0.205 0.231 B 288 279 0 0 0 0 [[110, 359]] 1.0 9lid Homo sapiens OTHER_PKMYT1_HUMAN STE 7.6e-39 139.7 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 9LGNA Q99640 77 361 499.0 A1EJU:60401 Type1.5_Back Inactive DFGin 6.296 14.466 BLAminus -145.99, -171.4 50.86, 84.26 -97.86, 29.36 304.36, 111.52 -72.91, -21.87 in-in in 8.887 Saltbr-in 2.795 HRD-in -66.21, -46.68 65.26, 16.91 in-in-out SNCiio in-out ActLoopNT-in 3.082 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -68.54, 120.07 APE9-dihe-na -90.78, -176.48 APE8-dihe-in -82.34, 121.43 APE8-rot-na 199.89 APE67-dihe-in -63.02, -34.9 -65.92, -23.54 APE12-dist-in 7.833 APE11-dist-out 5.486 APE10-dist-out 9.422 APE9-dist-in 4.545 None None None XRAY 2.03 0.196 0.241 A 286 280 5 0 0 5 [[110, 359]] 1.0 9lgn Homo sapiens OTHER_PKMYT1_HUMAN STE 7.4e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 9LGNB Q99640 77 361 499.0 A1EJU:60401 Type1.5_Back Inactive DFGin 6.068 14.404 BLAminus -142.39, -165.96 54.01, 79.86 -92.24, 28.67 300.8, 134.57 -69.88, -31.54 in-in in 8.842 Saltbr-in 2.621 HRD-in -68.45, -46.04 66.53, 9.81 in-in-out SNCiio in-out ActLoopNT-in 3.009 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -64.59, 124.38 APE9-dihe-na -93.34, -179.18 APE8-dihe-in -77.16, 120.0 APE8-rot-na 200.38 APE67-dihe-in -63.03, -36.01 -66.03, -24.01 APE12-dist-in 7.864 APE11-dist-out 5.611 APE10-dist-out 9.357 APE9-dist-in 4.519 None None None XRAY 2.03 0.196 0.241 B 286 281 4 0 0 4 [[110, 359]] 1.0 9lgn Homo sapiens OTHER_PKMYT1_HUMAN STE 7.4e-39 139.8 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8D6DA Q99640 78 361 499.0 QGY:405 Type1.5_Back Inactive DFGin 6.211 14.538 BLAminus -148.07, -173.76 61.71, 69.04 -87.4, 33.63 306.09, 107.4 -73.23, -43.69 in-in in 8.979 Saltbr-in 2.792 HRD-in -70.41, -52.13 74.56, -0.66 in-in-out SNCiio in-out ActLoopNT-in 3.042 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -82.14, 144.34 APE9-dihe-na -114.82, 178.25 APE8-dihe-in -66.9, 123.15 APE8-rot-na 195.13 APE67-dihe-in -58.55, -32.2 -61.02, -29.72 APE12-dist-in 7.901 APE11-dist-out 5.216 APE10-dist-out 9.078 APE9-dist-in 4.364 None None None XRAY 2.35 0.242 0.272 A 311 270 5 0 0 5 [[110, 359]] 1.0 8d6d Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8D6EA Q99640 77 361 499.0 QGI:1303 Type1.5_Back Inactive DFGin 5.964 14.172 BLAminus -132.85, -170.23 57.02, 82.01 -94.72, 23.46 304.19, 110.84 -65.02, -29.08 in-in in 8.87 Saltbr-in 2.717 HRD-in -75.21, -49.23 71.68, 5.95 in-in-out SNCiio in-out ActLoopNT-in 2.94 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -70.02, 134.68 APE9-dihe-na -98.58, -177.84 APE8-dihe-in -78.94, 114.38 APE8-rot-na 196.53 APE67-dihe-in -55.24, -36.47 -61.38, -25.28 APE12-dist-in 7.804 APE11-dist-out 5.579 APE10-dist-out 9.69 APE9-dist-in 4.697 None None None XRAY 2.15 0.192 0.218 A 311 278 3 0 0 3 [[110, 359]] 1.0 8d6e Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8D6FA Q99640 78 361 499.0 QG5:402 Type1.5_Back Inactive DFGin 5.934 14.393 BLAminus -137.99, -170.0 54.51, 81.69 -95.67, 27.93 303.43, 112.84 -67.3, -27.64 in-in in 8.927 Saltbr-in 2.693 HRD-in -64.05, -49.24 70.41, 3.13 in-in-out SNCiio in-out ActLoopNT-in 2.974 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -70.94, 136.66 APE9-dihe-na -111.83, 176.77 APE8-dihe-in -71.13, 118.43 APE8-rot-na 201.17 APE67-dihe-in -57.59, -30.74 -64.31, -29.06 APE12-dist-in 7.268 APE11-dist-out 5.262 APE10-dist-out 9.373 APE9-dist-in 4.633 None None None XRAY 2.49 0.216 0.239 A 311 270 6 0 0 6 [[110, 359]] 1.0 8d6f Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase
PMYT1_HUMAN 8D6FB Q99640 76 361 499.0 QG5:402 Type1.5_Back Inactive DFGin 6.014 14.327 BLAminus -137.52, -169.84 54.56, 81.42 -96.27, 27.52 303.69, 112.72 -67.62, -27.32 in-in in 8.86 Saltbr-in 2.731 HRD-in -63.86, -48.97 70.29, 4.03 in-in-out SNCiio in-out ActLoopNT-in 3.061 ActLoopCT-out nonTYR APEdihe_aaiai APEdist_iooi APE10-dihe-na -70.91, 136.32 APE9-dihe-na -112.58, 175.93 APE8-dihe-in -71.78, 118.97 APE8-rot-na 200.9 APE67-dihe-in -57.56, -31.19 -64.02, -28.04 APE12-dist-in 7.294 APE11-dist-out 5.136 APE10-dist-out 9.236 APE9-dist-in 4.543 None None None XRAY 2.49 0.216 0.239 B 311 272 6 0 0 6 [[110, 359]] 1.0 8d6f Homo sapiens OTHER_PKMYT1_HUMAN STE 9.9e-39 139.4 1 255 255 250 251 252 254 256 139 157 161 230 232 231 233 288 277 272 271 270 269 268 267 266 188 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase

OTHER_PKMYT1 (Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase)

Total number of chains: 0
Active chains: 0
Family: OTHER
Spatial label Dihedral label Number of Chains Percent Representative

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SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name