TYR_EPHB1 (Ephrin type-B receptor 1)

Total number of chains: 18
Active chains: 4
Uniprot: EPHB1_HUMAN
Kinase Domain Residues: 619 - 880
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 15 83.3% AF-P54762-K1A
DFGin None 3 16.7% 6UMWA

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Gene PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
EPHB1 AF-P54762-K1A P54762 611 888 984.0 No_ligand No_ligand Active DFGin 6.0425 14.032 BLAminus -131.01, -178.54 62.42, 60.04 -77.93, 10.0 300.47, 94.81 -59.93, -32.36 in-in in 8.0298 Saltbr-in 2.7647 HRD-in -80.21, -45.62 66.24, -9.55 in-in-in SNCiii in-in ActLoopNT-in 2.9226 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -61.53, 127.64 APE9-dihe-in -128.31, 141.79 APE8-dihe-in -78.18, 81.97 APE8-rot-na 35.95 APE67-dihe-in -69.22, -12.87 -42.28, -52.19 APE12-dist-na 13.8521 APE11-dist-na 10.0204 APE10-dist-na 9.5403 APE9-dist-in 5.8975 None None None AF2 -1.0 1.0 1.0 A 278.0 278.0 0 33 33 0 [[619, 880]] 1.0 AF-P54762-K1 TYR_EPHB1_HUMAN TYR 2.2e-109 370.7 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 AF-P54762-K3A P54762 611 888 984.0 No_ligand No_ligand Active DFGin 5.9191 14.1485 BLAminus -144.43, -176.57 56.86, 68.35 -80.03, 12.67 292.38, 96.35 -58.87, -32.19 in-in in 8.382 Saltbr-in 2.744 HRD-in -80.65, -47.86 68.16, -8.24 in-in-in SNCiii in-in ActLoopNT-in 2.9551 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -59.39, 136.1 APE9-dihe-in -130.38, 143.82 APE8-dihe-in -79.65, 76.31 APE8-rot-na 35.71 APE67-dihe-in -63.6, -21.92 -42.82, -45.82 APE12-dist-na 13.1105 APE11-dist-na 9.3315 APE10-dist-na 9.2572 APE9-dist-in 5.9217 None None None AF2 -1.0 1.0 1.0 A 278.0 278.0 0 33 33 0 [[619, 880]] 1.0 AF-P54762-K3 TYR_EPHB1_HUMAN TYR 2.2e-109 370.7 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 5MJAB P54762 609 890 984.0 7O3:901 Type1 Active DFGin 6.083 14.0535 BLAminus -141.24, -171.2 58.22, 72.67 -91.84, 11.93 298.24, 99.38 -53.11, -46.2 in-in in 7.8716 Saltbr-in 2.8065 HRD-in -76.6, -50.2 73.12, -6.86 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -71.9, 136.79 APE9-dihe-in -131.04, 157.79 APE8-dihe-in -83.23, 87.47 APE8-rot-na 26.22 APE67-dihe-in -75.23, -7.99 -41.53, -51.14 APE12-dist-na 15.035 APE11-dist-na 11.2696 APE10-dist-na 11.1128 APE9-dist-in 6.3542 None PTR647,PTR778 PTR647,PTR778 XRAY 2.14 0.202 0.236 B 305.0 276.0 6 33 27 6 [[619, 880]] 1.0 5mja TYR_EPHB1_HUMAN TYR 5.3e-109 369.5 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 5MJBB P54762 608 890 984.0 7O3:901 Type1 Active DFGin 6.0945 13.9285 BLAminus -144.01, -170.2 57.06, 72.11 -90.61, 7.86 298.99, 102.19 -51.34, -41.82 in-in in 7.9276 Saltbr-in 2.8313 HRD-in -77.06, -51.4 72.88, -5.4 in-in-in SNCiii in-in ActLoopNT-in 2.9434 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -64.28, 141.56 APE9-dihe-in -138.81, 153.61 APE8-dihe-in -82.83, 91.49 APE8-rot-na 25.93 APE67-dihe-in -72.9, -9.32 -44.37, -51.53 APE12-dist-na 15.1158 APE11-dist-na 11.3642 APE10-dist-na 10.9972 APE9-dist-in 6.3188 None PTR647,PTR778 PTR647,PTR778 XRAY 2.23 0.199 0.214 B 305.0 280.0 3 33 30 3 [[619, 880]] 1.0 5mjb TYR_EPHB1_HUMAN TYR 8.1e-108 365.6 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 3ZFXA P54762 611 893 984.0 No_ligand No_ligand Inactive DFGin 5.65 14.5402 BLAminus -137.28, 176.34 70.3, 72.85 -91.87, 22.74 297.85, 83.96 -73.04, -25.82 in-in in 8.2641 Saltbr-in 2.7627 HRD-in -74.92, -55.25 81.01, -3.92 in-in-out SNCiio in-out ActLoopNT-in 2.9474 ActLoopCT-out TYR APEdihe_iiiai APEdist_aaao APE10-dihe-in -62.12, 104.75 APE9-dihe-in -69.4, 128.33 APE8-dihe-in -64.25, 173.31 APE8-rot-na 33.55 APE67-dihe-in -79.3, 6.2 -139.5, -29.76 APE12-dist-na 999.0 APE11-dist-na 12.149 APE10-dist-na 14.7777 APE9-dist-out 8.9587 None None None XRAY 2.5 0.19 0.217 A 298.0 267.0 16 33 20 13 [[619, 880]] 1.0 3zfx TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 3ZFXD P54762 611 893 984.0 No_ligand No_ligand Inactive DFGin 5.7057 14.6339 BLAminus -140.75, 172.17 74.92, 66.44 -93.4, 30.36 297.9, 86.18 -75.9, -27.4 in-in in 8.3153 Saltbr-in 2.0915 HRD-in -69.91, -59.77 85.71, -11.32 in-in-out SNCiio in-out ActLoopNT-in 2.8002 ActLoopCT-out TYR APEdihe_iiiai APEdist_aaao APE10-dihe-in -111.5, 128.09 APE9-dihe-in -84.51, 112.07 APE8-dihe-in -58.31, 178.25 APE8-rot-na 350.35 APE67-dihe-in -71.14, 2.25 -140.4, -34.58 APE12-dist-na 999.0 APE11-dist-na 12.7602 APE10-dist-na 14.343 APE9-dist-out 8.9516 None None None XRAY 2.5 0.19 0.217 D 298.0 265.0 18 33 20 13 [[619, 880]] 1.0 3zfx TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 3ZFXE P54762 611 893 984.0 No_ligand No_ligand Inactive DFGin 5.8207 14.4641 BLAminus -138.13, 178.47 66.78, 71.49 -93.93, 20.13 295.76, 113.75 -66.41, -32.63 in-in in 8.2561 Saltbr-in 3.3893 HRD-in -74.16, -50.25 78.75, -8.09 in-in-out SNCiio in-out ActLoopNT-in 2.9184 ActLoopCT-out TYR APEdihe_iiiai APEdist_aaao APE10-dihe-in -62.16, 94.27 APE9-dihe-in -52.71, 111.04 APE8-dihe-in -58.17, 174.33 APE8-rot-na 11.84 APE67-dihe-in -79.05, -2.46 -147.97, -24.49 APE12-dist-na 999.0 APE11-dist-na 11.7655 APE10-dist-na 14.2019 APE9-dist-out 8.8298 None None None XRAY 2.5 0.19 0.217 E 298.0 262.0 21 33 19 14 [[619, 880]] 1.0 3zfx TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 3ZFXH P54762 611 892 984.0 No_ligand No_ligand Inactive DFGin 5.6085 14.7076 BLAminus -137.94, 177.39 70.52, 70.48 -91.79, 19.67 293.87, 95.22 -66.32, -32.05 in-in in 8.4193 Saltbr-in 2.4198 HRD-in -66.01, -56.98 82.79, -2.13 in-in-out SNCiio in-out ActLoopNT-in 2.874 ActLoopCT-out TYR APEdihe_iiiai APEdist_aaao APE10-dihe-in -90.32, 129.98 APE9-dihe-in -81.42, 123.05 APE8-dihe-in -69.76, 172.99 APE8-rot-na 21.61 APE67-dihe-in -73.91, 2.65 -141.66, -31.27 APE12-dist-na 999.0 APE11-dist-na 12.3697 APE10-dist-na 14.4798 APE9-dist-out 8.9107 None None None XRAY 2.5 0.19 0.217 H 298.0 266.0 16 33 19 14 [[619, 880]] 1.0 3zfx TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 3ZFXI P54762 611 891 984.0 No_ligand No_ligand Inactive DFGin 5.7526 14.4832 BLAminus -139.17, 176.15 66.64, 74.45 -93.15, 18.83 295.38, 84.8 -62.38, -38.47 in-in in 8.3056 Saltbr-in 2.8139 HRD-in -71.01, -51.08 79.54, -7.87 in-in-out SNCiio in-out ActLoopNT-in 2.9869 ActLoopCT-out TYR APEdihe_iioai APEdist_aaao APE10-dihe-in -62.99, 134.6 APE9-dihe-in -93.24, 134.04 APE8-dihe-out -75.13, -179.06 APE8-rot-na 15.06 APE67-dihe-in -78.21, 4.42 -143.86, -33.88 APE12-dist-na 999.0 APE11-dist-na 11.6734 APE10-dist-na 14.0366 APE9-dist-out 8.6392 None None None XRAY 2.5 0.19 0.217 I 298.0 263.0 18 33 19 14 [[619, 880]] 1.0 3zfx TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 5MJBA P54762 608 891 984.0 7O3:901 Type1.5_Back Inactive DFGin 6.0019 13.7853 BLAminus -133.67, -168.42 59.63, 70.74 -90.66, 8.06 299.37, 101.12 -49.79, -42.85 in-in in 7.9171 Saltbr-in 2.8126 HRD-in -76.18, -50.21 70.23, -5.93 in-in-out SNCiio in-out ActLoopNT-in 2.9333 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -109.93, -30.04 APE9-dihe-in -66.85, 139.16 APE8-dihe-in -90.86, 97.78 APE8-rot-na 25.99 APE67-dihe-in -71.64, -10.32 -44.79, -51.82 APE12-dist-na 12.1701 APE11-dist-na 12.3619 APE10-dist-na 7.7046 APE9-dist-in 5.5946 None PTR647,PTR778 PTR647,PTR778 XRAY 2.23 0.199 0.214 A 305.0 278.0 6 33 27 6 [[619, 880]] 1.0 5mjb TYR_EPHB1_HUMAN TYR 8.1e-108 365.6 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 7KPMA P54762 611 888 984.0 ADP:901 ATPlike Inactive DFGin 6.1477 15.077 None -129.01, -161.15 68.81, 56.56 -103.91, 999.0 293.32, 103.77 999.0, 999.0 in-in in 7.7435 Saltbr-in 2.7086 HRD-in -77.02, -45.59 75.58, -13.35 in-none-none SNCinn none-none ActLoopNT-none 999.0 ActLoopCT-none TYR APEdihe_nnnai APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 76.94 APE8-rot-na 30.04 APE67-dihe-in -77.93, -6.39 -53.89, -41.84 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None PTR647 PTR647 XRAY 1.608 0.169 0.197 A 279.0 255.0 23 33 10 23 [[619, 880]] 1.0 7kpm TYR_EPHB1_HUMAN TYR 2.3e-109 370.6 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 7KPLA P54762 611 888 984.0 No_ligand No_ligand Inactive DFGin 6.1167 14.504 None -122.5, -147.19 60.66, 72.8 -110.8, 999.0 285.53, 126.95 999.0, 999.0 in-in in 8.7776 Saltbr-in 3.1106 HRD-in -81.07, -50.31 62.2, -0.14 in-none-none SNCinn none-none ActLoopNT-none 999.0 ActLoopCT-none TYR APEdihe_nniai APEdist_aaai APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 120.78 APE8-dihe-in -69.07, 87.68 APE8-rot-na 25.45 APE67-dihe-in -71.96, -7.05 -54.45, -46.98 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-in 6.6029 None PTR647 PTR647 XRAY 2.705 0.202 0.25 A 279.0 256.0 22 33 11 22 [[619, 880]] 1.0 7kpl TYR_EPHB1_HUMAN TYR 2.3e-109 370.6 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 6UMWA P54762 611 889 984.0 CTC:901 Type1.5_Back Inactive DFGin 6.0667 14.8859 None -130.77, -142.58 52.4, 64.34 -100.65, 999.0 280.28, 134.37 999.0, 999.0 in-out in 8.9314 Saltbr-out 5.9984 HRD-in -72.73, -48.51 73.38, -14.75 out-none-none SNConn none-none ActLoopNT-none 999.0 ActLoopCT-none TYR APEdihe_nniai APEdist_aaai APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 118.46 APE8-dihe-in -70.84, 88.26 APE8-rot-na 28.98 APE67-dihe-in -78.1, -4.96 -58.23, -45.11 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-in 6.7503 None PTR647 PTR647 XRAY 1.982 0.184 0.221 A 301.0 257.0 22 33 11 22 [[619, 880]] 1.0 6umw TYR_EPHB1_HUMAN TYR 3e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 3ZFXB P54762 611 892 984.0 No_ligand No_ligand None DFGin 5.8171 14.5127 BLAminus -140.84, 175.74 70.16, 66.52 -88.36, 22.51 296.61, 82.06 -65.86, -37.4 in-in in 8.3613 Saltbr-in 2.7446 HRD-in -73.6, -53.87 82.61, -12.27 in-in-none SNCiin in-none ActLoopNT-in 2.9825 ActLoopCT-none TYR APEdihe_nnnan APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-na 999.0 APE67-dihe-none -68.46, -4.35 999.0, -41.26 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None None None XRAY 2.5 0.19 0.217 B 298.0 254.0 28 33 15 18 [[619, 880]] 1.0 3zfx TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 3ZFXC P54762 614 892 984.0 No_ligand No_ligand None DFGin 5.7379 14.5606 BLAminus -137.69, 173.75 69.1, 70.2 -91.34, 24.03 296.14, 85.79 -69.43, -30.67 in-none in 8.3875 Saltbr-none 999.0 HRD-in -72.86, -47.73 75.93, -10.98 none-in-none SNCnin in-none ActLoopNT-in 3.0033 ActLoopCT-none TYR APEdihe_nnnai APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 119.99 APE8-rot-na 23.72 APE67-dihe-in -76.29, 1.22 -135.32, -30.63 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None None None XRAY 2.5 0.19 0.217 C 298.0 248.0 31 33 14 19 [[619, 880]] 1.0 3zfx TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 3ZFXF P54762 612 893 984.0 No_ligand No_ligand None DFGin 5.7509 14.4499 BLAminus -141.17, 174.54 70.47, 73.51 -96.07, 25.2 298.87, 86.22 -68.13, -33.68 in-none in 8.2624 Saltbr-none 999.0 HRD-in -76.22, -51.77 80.7, -11.45 none-in-none SNCnin in-none ActLoopNT-in 2.9076 ActLoopCT-none TYR APEdihe_nnnan APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-na 999.0 APE67-dihe-none -75.22, -1.35 999.0, -38.52 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None None None XRAY 2.5 0.19 0.217 F 298.0 254.0 28 33 15 18 [[619, 880]] 1.0 3zfx TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 3ZFXG P54762 611 892 984.0 No_ligand No_ligand None DFGin 5.7178 14.5195 BLAminus -137.41, 174.48 70.94, 70.55 -95.84, 25.71 297.3, 82.59 -71.73, -27.91 in-in in 8.3597 Saltbr-in 2.7612 HRD-in -75.32, -55.18 83.83, -8.92 in-in-none SNCiin in-none ActLoopNT-in 2.9702 ActLoopCT-none TYR APEdihe_nnnan APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-na 999.0 APE67-dihe-none -75.69, 3.79 999.0, -41.74 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None None None XRAY 2.5 0.19 0.217 G 298.0 253.0 29 33 15 18 [[619, 880]] 1.0 3zfx TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 5MJAA P54762 609 892 984.0 7O3:901 Type1.5_Back None DFGin 5.8801 13.9025 BLAminus -139.99, -175.99 56.55, 73.99 -90.49, 10.93 298.25, 99.95 -50.92, -47.24 in-in in 7.8806 Saltbr-in 2.7929 HRD-in -76.83, -50.44 72.7, -6.85 in-in-none SNCiin in-none ActLoopNT-in 2.8638 ActLoopCT-none TYR APEdihe_nnnai APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 37.53 APE8-rot-na 25.39 APE67-dihe-in -70.7, -7.58 -41.98, -56.11 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None PTR647,PTR778 PTR647,PTR778 XRAY 2.14 0.202 0.236 A 305.0 273.0 11 33 22 11 [[619, 880]] 1.0 5mja TYR_EPHB1_HUMAN TYR 5.3e-109 369.5 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1

TYR_EPHB1 (Ephrin type-B receptor 1)

Total number of chains: 18
Active chains: 4
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 15 83.3% AF-P54762-K1A
DFGin None 3 16.7% 6UMWA

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
EPHB1 EPHB1_HUMAN AF-P54762-K1A P54762 611 888 984.0 No_ligand No_ligand Active DFGin 6.0425 14.032 BLAminus -131.01, -178.54 62.42, 60.04 -77.93, 10.0 300.47, 94.81 -59.93, -32.36 in-in in 8.0298 Saltbr-in 2.7647 HRD-in -80.21, -45.62 66.24, -9.55 in-in-in SNCiii in-in ActLoopNT-in 2.9226 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -61.53, 127.64 APE9-dihe-in -128.31, 141.79 APE8-dihe-in -78.18, 81.97 APE8-rot-na 35.95 APE67-dihe-in -69.22, -12.87 -42.28, -52.19 APE12-dist-na 13.8521 APE11-dist-na 10.0204 APE10-dist-na 9.5403 APE9-dist-in 5.8975 None None None AF2 -1.0 1.0 1.0 A 278.0 278.0 0 33 33 0 [[619, 880]] 1.0 AF-P54762-K1 Homo sapiens TYR_EPHB1_HUMAN TYR 2.2e-109 370.7 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN AF-P54762-K3A P54762 611 888 984.0 No_ligand No_ligand Active DFGin 5.9191 14.1485 BLAminus -144.43, -176.57 56.86, 68.35 -80.03, 12.67 292.38, 96.35 -58.87, -32.19 in-in in 8.382 Saltbr-in 2.744 HRD-in -80.65, -47.86 68.16, -8.24 in-in-in SNCiii in-in ActLoopNT-in 2.9551 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -59.39, 136.1 APE9-dihe-in -130.38, 143.82 APE8-dihe-in -79.65, 76.31 APE8-rot-na 35.71 APE67-dihe-in -63.6, -21.92 -42.82, -45.82 APE12-dist-na 13.1105 APE11-dist-na 9.3315 APE10-dist-na 9.2572 APE9-dist-in 5.9217 None None None AF2 -1.0 1.0 1.0 A 278.0 278.0 0 33 33 0 [[619, 880]] 1.0 AF-P54762-K3 Homo sapiens TYR_EPHB1_HUMAN TYR 2.2e-109 370.7 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 5MJAB P54762 609 890 984.0 7O3:901 Type1 Active DFGin 6.083 14.0535 BLAminus -141.24, -171.2 58.22, 72.67 -91.84, 11.93 298.24, 99.38 -53.11, -46.2 in-in in 7.8716 Saltbr-in 2.8065 HRD-in -76.6, -50.2 73.12, -6.86 in-in-in SNCiii in-in ActLoopNT-in 2.856 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -71.9, 136.79 APE9-dihe-in -131.04, 157.79 APE8-dihe-in -83.23, 87.47 APE8-rot-na 26.22 APE67-dihe-in -75.23, -7.99 -41.53, -51.14 APE12-dist-na 15.035 APE11-dist-na 11.2696 APE10-dist-na 11.1128 APE9-dist-in 6.3542 None PTR647,PTR778 PTR647,PTR778 XRAY 2.14 0.202 0.236 B 305.0 276.0 6 33 27 6 [[619, 880]] 1.0 5mja Homo sapiens TYR_EPHB1_HUMAN TYR 5.3e-109 369.5 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 5MJBB P54762 608 890 984.0 7O3:901 Type1 Active DFGin 6.0945 13.9285 BLAminus -144.01, -170.2 57.06, 72.11 -90.61, 7.86 298.99, 102.19 -51.34, -41.82 in-in in 7.9276 Saltbr-in 2.8313 HRD-in -77.06, -51.4 72.88, -5.4 in-in-in SNCiii in-in ActLoopNT-in 2.9434 ActLoopCT-in TYR APEdihe_iiiai APEdist_aaai APE10-dihe-in -64.28, 141.56 APE9-dihe-in -138.81, 153.61 APE8-dihe-in -82.83, 91.49 APE8-rot-na 25.93 APE67-dihe-in -72.9, -9.32 -44.37, -51.53 APE12-dist-na 15.1158 APE11-dist-na 11.3642 APE10-dist-na 10.9972 APE9-dist-in 6.3188 None PTR647,PTR778 PTR647,PTR778 XRAY 2.23 0.199 0.214 B 305.0 280.0 3 33 30 3 [[619, 880]] 1.0 5mjb Homo sapiens TYR_EPHB1_HUMAN TYR 8.1e-108 365.6 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 3ZFXA P54762 611 893 984.0 No_ligand No_ligand Inactive DFGin 5.65 14.5402 BLAminus -137.28, 176.34 70.3, 72.85 -91.87, 22.74 297.85, 83.96 -73.04, -25.82 in-in in 8.2641 Saltbr-in 2.7627 HRD-in -74.92, -55.25 81.01, -3.92 in-in-out SNCiio in-out ActLoopNT-in 2.9474 ActLoopCT-out TYR APEdihe_iiiai APEdist_aaao APE10-dihe-in -62.12, 104.75 APE9-dihe-in -69.4, 128.33 APE8-dihe-in -64.25, 173.31 APE8-rot-na 33.55 APE67-dihe-in -79.3, 6.2 -139.5, -29.76 APE12-dist-na 999.0 APE11-dist-na 12.149 APE10-dist-na 14.7777 APE9-dist-out 8.9587 None None None XRAY 2.5 0.19 0.217 A 298.0 267.0 16 33 20 13 [[619, 880]] 1.0 3zfx Homo sapiens TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 3ZFXD P54762 611 893 984.0 No_ligand No_ligand Inactive DFGin 5.7057 14.6339 BLAminus -140.75, 172.17 74.92, 66.44 -93.4, 30.36 297.9, 86.18 -75.9, -27.4 in-in in 8.3153 Saltbr-in 2.0915 HRD-in -69.91, -59.77 85.71, -11.32 in-in-out SNCiio in-out ActLoopNT-in 2.8002 ActLoopCT-out TYR APEdihe_iiiai APEdist_aaao APE10-dihe-in -111.5, 128.09 APE9-dihe-in -84.51, 112.07 APE8-dihe-in -58.31, 178.25 APE8-rot-na 350.35 APE67-dihe-in -71.14, 2.25 -140.4, -34.58 APE12-dist-na 999.0 APE11-dist-na 12.7602 APE10-dist-na 14.343 APE9-dist-out 8.9516 None None None XRAY 2.5 0.19 0.217 D 298.0 265.0 18 33 20 13 [[619, 880]] 1.0 3zfx Homo sapiens TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 3ZFXE P54762 611 893 984.0 No_ligand No_ligand Inactive DFGin 5.8207 14.4641 BLAminus -138.13, 178.47 66.78, 71.49 -93.93, 20.13 295.76, 113.75 -66.41, -32.63 in-in in 8.2561 Saltbr-in 3.3893 HRD-in -74.16, -50.25 78.75, -8.09 in-in-out SNCiio in-out ActLoopNT-in 2.9184 ActLoopCT-out TYR APEdihe_iiiai APEdist_aaao APE10-dihe-in -62.16, 94.27 APE9-dihe-in -52.71, 111.04 APE8-dihe-in -58.17, 174.33 APE8-rot-na 11.84 APE67-dihe-in -79.05, -2.46 -147.97, -24.49 APE12-dist-na 999.0 APE11-dist-na 11.7655 APE10-dist-na 14.2019 APE9-dist-out 8.8298 None None None XRAY 2.5 0.19 0.217 E 298.0 262.0 21 33 19 14 [[619, 880]] 1.0 3zfx Homo sapiens TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 3ZFXH P54762 611 892 984.0 No_ligand No_ligand Inactive DFGin 5.6085 14.7076 BLAminus -137.94, 177.39 70.52, 70.48 -91.79, 19.67 293.87, 95.22 -66.32, -32.05 in-in in 8.4193 Saltbr-in 2.4198 HRD-in -66.01, -56.98 82.79, -2.13 in-in-out SNCiio in-out ActLoopNT-in 2.874 ActLoopCT-out TYR APEdihe_iiiai APEdist_aaao APE10-dihe-in -90.32, 129.98 APE9-dihe-in -81.42, 123.05 APE8-dihe-in -69.76, 172.99 APE8-rot-na 21.61 APE67-dihe-in -73.91, 2.65 -141.66, -31.27 APE12-dist-na 999.0 APE11-dist-na 12.3697 APE10-dist-na 14.4798 APE9-dist-out 8.9107 None None None XRAY 2.5 0.19 0.217 H 298.0 266.0 16 33 19 14 [[619, 880]] 1.0 3zfx Homo sapiens TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 3ZFXI P54762 611 891 984.0 No_ligand No_ligand Inactive DFGin 5.7526 14.4832 BLAminus -139.17, 176.15 66.64, 74.45 -93.15, 18.83 295.38, 84.8 -62.38, -38.47 in-in in 8.3056 Saltbr-in 2.8139 HRD-in -71.01, -51.08 79.54, -7.87 in-in-out SNCiio in-out ActLoopNT-in 2.9869 ActLoopCT-out TYR APEdihe_iioai APEdist_aaao APE10-dihe-in -62.99, 134.6 APE9-dihe-in -93.24, 134.04 APE8-dihe-out -75.13, -179.06 APE8-rot-na 15.06 APE67-dihe-in -78.21, 4.42 -143.86, -33.88 APE12-dist-na 999.0 APE11-dist-na 11.6734 APE10-dist-na 14.0366 APE9-dist-out 8.6392 None None None XRAY 2.5 0.19 0.217 I 298.0 263.0 18 33 19 14 [[619, 880]] 1.0 3zfx Homo sapiens TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 5MJBA P54762 608 891 984.0 7O3:901 Type1.5_Back Inactive DFGin 6.0019 13.7853 BLAminus -133.67, -168.42 59.63, 70.74 -90.66, 8.06 299.37, 101.12 -49.79, -42.85 in-in in 7.9171 Saltbr-in 2.8126 HRD-in -76.18, -50.21 70.23, -5.93 in-in-out SNCiio in-out ActLoopNT-in 2.9333 ActLoopCT-out TYR APEdihe_oiiai APEdist_aaai APE10-dihe-out -109.93, -30.04 APE9-dihe-in -66.85, 139.16 APE8-dihe-in -90.86, 97.78 APE8-rot-na 25.99 APE67-dihe-in -71.64, -10.32 -44.79, -51.82 APE12-dist-na 12.1701 APE11-dist-na 12.3619 APE10-dist-na 7.7046 APE9-dist-in 5.5946 None PTR647,PTR778 PTR647,PTR778 XRAY 2.23 0.199 0.214 A 305.0 278.0 6 33 27 6 [[619, 880]] 1.0 5mjb Homo sapiens TYR_EPHB1_HUMAN TYR 8.1e-108 365.6 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 7KPMA P54762 611 888 984.0 ADP:901 ATPlike Inactive DFGin 6.1477 15.077 None -129.01, -161.15 68.81, 56.56 -103.91, 999.0 293.32, 103.77 999.0, 999.0 in-in in 7.7435 Saltbr-in 2.7086 HRD-in -77.02, -45.59 75.58, -13.35 in-none-none SNCinn none-none ActLoopNT-none 999.0 ActLoopCT-none TYR APEdihe_nnnai APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 76.94 APE8-rot-na 30.04 APE67-dihe-in -77.93, -6.39 -53.89, -41.84 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None PTR647 PTR647 XRAY 1.608 0.169 0.197 A 279.0 255.0 23 33 10 23 [[619, 880]] 1.0 7kpm Homo sapiens TYR_EPHB1_HUMAN TYR 2.3e-109 370.6 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 7KPLA P54762 611 888 984.0 No_ligand No_ligand Inactive DFGin 6.1167 14.504 None -122.5, -147.19 60.66, 72.8 -110.8, 999.0 285.53, 126.95 999.0, 999.0 in-in in 8.7776 Saltbr-in 3.1106 HRD-in -81.07, -50.31 62.2, -0.14 in-none-none SNCinn none-none ActLoopNT-none 999.0 ActLoopCT-none TYR APEdihe_nniai APEdist_aaai APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 120.78 APE8-dihe-in -69.07, 87.68 APE8-rot-na 25.45 APE67-dihe-in -71.96, -7.05 -54.45, -46.98 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-in 6.6029 None PTR647 PTR647 XRAY 2.705 0.202 0.25 A 279.0 256.0 22 33 11 22 [[619, 880]] 1.0 7kpl Homo sapiens TYR_EPHB1_HUMAN TYR 2.3e-109 370.6 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 6UMWA P54762 611 889 984.0 CTC:901 Type1.5_Back Inactive DFGin 6.0667 14.8859 None -130.77, -142.58 52.4, 64.34 -100.65, 999.0 280.28, 134.37 999.0, 999.0 in-out in 8.9314 Saltbr-out 5.9984 HRD-in -72.73, -48.51 73.38, -14.75 out-none-none SNConn none-none ActLoopNT-none 999.0 ActLoopCT-none TYR APEdihe_nniai APEdist_aaai APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 118.46 APE8-dihe-in -70.84, 88.26 APE8-rot-na 28.98 APE67-dihe-in -78.1, -4.96 -58.23, -45.11 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-in 6.7503 None PTR647 PTR647 XRAY 1.982 0.184 0.221 A 301.0 257.0 22 33 11 22 [[619, 880]] 1.0 6umw Homo sapiens TYR_EPHB1_HUMAN TYR 3e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 3ZFXB P54762 611 892 984.0 No_ligand No_ligand None DFGin 5.8171 14.5127 BLAminus -140.84, 175.74 70.16, 66.52 -88.36, 22.51 296.61, 82.06 -65.86, -37.4 in-in in 8.3613 Saltbr-in 2.7446 HRD-in -73.6, -53.87 82.61, -12.27 in-in-none SNCiin in-none ActLoopNT-in 2.9825 ActLoopCT-none TYR APEdihe_nnnan APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-na 999.0 APE67-dihe-none -68.46, -4.35 999.0, -41.26 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None None None XRAY 2.5 0.19 0.217 B 298.0 254.0 28 33 15 18 [[619, 880]] 1.0 3zfx Homo sapiens TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 3ZFXC P54762 614 892 984.0 No_ligand No_ligand None DFGin 5.7379 14.5606 BLAminus -137.69, 173.75 69.1, 70.2 -91.34, 24.03 296.14, 85.79 -69.43, -30.67 in-none in 8.3875 Saltbr-none 999.0 HRD-in -72.86, -47.73 75.93, -10.98 none-in-none SNCnin in-none ActLoopNT-in 3.0033 ActLoopCT-none TYR APEdihe_nnnai APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 119.99 APE8-rot-na 23.72 APE67-dihe-in -76.29, 1.22 -135.32, -30.63 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None None None XRAY 2.5 0.19 0.217 C 298.0 248.0 31 33 14 19 [[619, 880]] 1.0 3zfx Homo sapiens TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 3ZFXF P54762 612 893 984.0 No_ligand No_ligand None DFGin 5.7509 14.4499 BLAminus -141.17, 174.54 70.47, 73.51 -96.07, 25.2 298.87, 86.22 -68.13, -33.68 in-none in 8.2624 Saltbr-none 999.0 HRD-in -76.22, -51.77 80.7, -11.45 none-in-none SNCnin in-none ActLoopNT-in 2.9076 ActLoopCT-none TYR APEdihe_nnnan APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-na 999.0 APE67-dihe-none -75.22, -1.35 999.0, -38.52 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None None None XRAY 2.5 0.19 0.217 F 298.0 254.0 28 33 15 18 [[619, 880]] 1.0 3zfx Homo sapiens TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 3ZFXG P54762 611 892 984.0 No_ligand No_ligand None DFGin 5.7178 14.5195 BLAminus -137.41, 174.48 70.94, 70.55 -95.84, 25.71 297.3, 82.59 -71.73, -27.91 in-in in 8.3597 Saltbr-in 2.7612 HRD-in -75.32, -55.18 83.83, -8.92 in-in-none SNCiin in-none ActLoopNT-in 2.9702 ActLoopCT-none TYR APEdihe_nnnan APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 999.0 APE8-rot-na 999.0 APE67-dihe-none -75.69, 3.79 999.0, -41.74 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None None None XRAY 2.5 0.19 0.217 G 298.0 253.0 29 33 15 18 [[619, 880]] 1.0 3zfx Homo sapiens TYR_EPHB1_HUMAN TYR 2.9e-109 370.3 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1
EPHB1 EPHB1_HUMAN 5MJAA P54762 609 892 984.0 7O3:901 Type1.5_Back None DFGin 5.8801 13.9025 BLAminus -139.99, -175.99 56.55, 73.99 -90.49, 10.93 298.25, 99.95 -50.92, -47.24 in-in in 7.8806 Saltbr-in 2.7929 HRD-in -76.83, -50.44 72.7, -6.85 in-in-none SNCiin in-none ActLoopNT-in 2.8638 ActLoopCT-none TYR APEdihe_nnnai APEdist_aaan APE10-dihe-none 999.0, 999.0 APE9-dihe-none 999.0, 999.0 APE8-dihe-none 999.0, 37.53 APE8-rot-na 25.39 APE67-dihe-in -70.7, -7.58 -41.98, -56.11 APE12-dist-na 999.0 APE11-dist-na 999.0 APE10-dist-na 999.0 APE9-dist-none 999.0 None PTR647,PTR778 PTR647,PTR778 XRAY 2.14 0.202 0.236 A 305.0 273.0 11 33 22 11 [[619, 880]] 1.0 5mja Homo sapiens TYR_EPHB1_HUMAN TYR 5.3e-109 369.5 2.0 261.0 260.0 761 762 763 765 767 651 668 672 741 743 742 744.0 806 794 789 788 787 786 785 784 783 698 Ephrin type-B receptor 1

TYR_EPHB1 (Ephrin type-B receptor 1)

Total number of chains: 0
Active chains: 0
Spatial label Dihedral label Number of Chains Percent Representative

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Gene SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name