AGC_CDC42BPB (Serine/threonine-protein kinase MRCK beta)

Total number of chains: 10
Active chains: 10
Family: AGC
Uniprot: MRCKB_HUMAN
Kinase Domain Residues: 76 - 342
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 10 100.0% AF-Q9Y5S2-K1A

Hover over column headers for tooltip help

PDB First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
4UAKA 2 417 1711.0 ADP:60501 ATPlike Active DFGin 6.536 13.389 BLAminus -126.67, 169.91 71.43, 81.15 -99.11, 14.11 300.02, 102.96 -73.12, -5.53 in-in in 8.635 Saltbr-in 2.748 HRD-in -78.82, -49.28 69.95, 4.01 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.28, 157.85 APE9-dihe-na 87.21, -164.86 APE8-dihe-in -127.15, 132.61 APE8-rot-in 302.21 APE67-dihe-in -64.23, -20.61 -57.86, -36.49 APE12-dist-in 10.511 APE11-dist-in 11.151 APE10-dist-in 6.313 APE9-dist-in 3.548 None None None XRAY 1.73 0.198 0.243 A 419 401 0 0 0 0 [[76, 342]] 1.0 4uak AGC_CDC42BPB_HUMAN AGC 6.5e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
AF-Q9Y5S2-K1A 68 350 1711.0 No_ligand No_ligand Active DFGin 6.286 13.418 BLAminus -138.11, 175.86 52.03, 73.16 -82.88, 16.9 300.82, 95.68 -61.27, -18.14 in-in in 8.67 Saltbr-in 2.619 HRD-in -80.82, -44.33 65.35, 6.41 in-in-in SNCiii in-in ActLoopNT-in 2.885 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.32, 151.0 APE9-dihe-na 118.31, 170.33 APE8-dihe-in -66.77, 129.62 APE8-rot-in 287.64 APE67-dihe-in -77.39, -20.44 -51.73, -36.54 APE12-dist-in 9.843 APE11-dist-in 10.942 APE10-dist-in 5.188 APE9-dist-in 3.788 None None None AF2 -1.0 1.0 1.0 A 283 283 0 0 0 0 [[76, 342]] 1.0 AF-Q9Y5S2-K1 AGC_CDC42BPB_HUMAN AGC 1.7e-96 328.2 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
AF-Q9Y5S2-K3A 68 350 1711.0 No_ligand No_ligand Active DFGin 6.165 13.252 BLAminus -140.87, 174.27 54.93, 67.41 -77.14, 15.47 302.2, 109.63 -60.94, -17.3 in-in in 8.594 Saltbr-in 2.681 HRD-in -80.0, -45.38 64.95, 8.05 in-in-in SNCiii in-in ActLoopNT-in 2.873 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.11, 160.14 APE9-dihe-na 106.26, -177.58 APE8-dihe-in -89.7, 125.56 APE8-rot-in 303.52 APE67-dihe-in -69.05, -20.8 -47.75, -44.36 APE12-dist-in 9.53 APE11-dist-in 10.952 APE10-dist-in 5.151 APE9-dist-in 3.627 None None None AF2 -1.0 1.0 1.0 A 283 283 0 0 0 0 [[76, 342]] 1.0 AF-Q9Y5S2-K3 AGC_CDC42BPB_HUMAN AGC 1.7e-96 328.2 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
3QFVA 2 415 1711.0 NM7:416 Type1 Active DFGin 6.652 13.483 BLAminus -155.19, -177.74 51.28, 74.91 -100.44, 20.96 290.95, 120.41 -84.8, 1.24 in-in in 8.66 Saltbr-in 3.586 HRD-in -68.56, -55.63 80.26, 2.79 in-in-in SNCiii in-in ActLoopNT-in 3.062 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.25, 145.57 APE9-dihe-na 95.66, -174.68 APE8-dihe-in -88.83, 133.9 APE8-rot-in 320.1 APE67-dihe-in -63.11, -25.9 -60.21, -35.51 APE12-dist-in 10.616 APE11-dist-in 11.198 APE10-dist-in 5.501 APE9-dist-in 4.17 None None None XRAY 2.65 0.196 0.268 A 415 395 0 0 0 0 [[76, 342]] 1.0 3qfv AGC_CDC42BPB_HUMAN AGC 6.3e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
3QFVB 2 415 1711.0 NM7:416 Type1 Active DFGin 6.357 13.248 BLAminus -146.98, -178.33 51.23, 77.88 -102.57, 32.33 302.88, 111.63 -92.77, 5.32 in-in in 8.692 Saltbr-in 2.619 HRD-in -65.12, -52.57 79.81, -7.22 in-in-in SNCiii in-in ActLoopNT-in 3.139 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.96, 150.13 APE9-dihe-na 114.47, 164.94 APE8-dihe-in -66.67, 141.54 APE8-rot-in 317.58 APE67-dihe-in -60.07, -38.36 -60.72, -35.72 APE12-dist-in 10.736 APE11-dist-in 11.342 APE10-dist-in 5.667 APE9-dist-in 4.087 None None None XRAY 2.65 0.196 0.268 B 415 396 0 0 0 0 [[76, 342]] 1.0 3qfv AGC_CDC42BPB_HUMAN AGC 6.3e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
4UALA 2 417 1711.0 3FV:60501 Type1 Active DFGin 6.57 13.343 BLAminus -128.09, 170.47 58.99, 78.49 -90.49, 11.57 302.61, 102.02 -65.54, -5.61 in-in in 8.675 Saltbr-in 2.909 HRD-in -76.1, -52.24 74.17, 2.64 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -119.7, -165.94 APE9-dihe-na 97.69, -165.3 APE8-dihe-in -123.13, 127.49 APE8-rot-in 312.99 APE67-dihe-in -64.7, -21.04 -49.2, -41.29 APE12-dist-in 10.401 APE11-dist-in 10.706 APE10-dist-in 5.458 APE9-dist-in 3.725 None None None XRAY 1.71 0.206 0.236 A 419 400 5 0 0 3 [[76, 342]] 1.0 4ual AGC_CDC42BPB_HUMAN AGC 6.5e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
5OTEA 2 417 1711.0 AQE:60501 Type1 Active DFGin 6.44 13.538 BLAminus -132.86, 172.8 58.15, 78.6 -89.88, 11.87 305.96, 106.7 -64.89, -6.52 in-in in 8.637 Saltbr-in 2.717 HRD-in -76.88, -48.31 73.79, 2.14 in-in-in SNCiii in-in ActLoopNT-in 2.96 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.88, 152.67 APE9-dihe-na 86.33, -167.63 APE8-dihe-in -120.1, 130.3 APE8-rot-in 304.26 APE67-dihe-in -60.96, -19.55 -48.3, -43.83 APE12-dist-in 10.442 APE11-dist-in 11.319 APE10-dist-in 6.425 APE9-dist-in 3.469 None None None XRAY 1.68 0.197 0.218 A 419 404 2 0 0 0 [[76, 342]] 1.0 5ote AGC_CDC42BPB_HUMAN AGC 6.5e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
5OTFA 2 417 1711.0 AQ5:60504 Type1 Active DFGin 6.474 13.836 BLAminus -138.71, 166.8 56.15, 77.62 -87.94, 13.12 305.59, 108.27 -63.54, -12.28 in-in in 8.966 Saltbr-in 2.633 HRD-in -69.74, -49.73 69.82, 11.73 in-in-in SNCiii in-in ActLoopNT-in 2.93 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.82, 174.96 APE9-dihe-na 90.86, 165.77 APE8-dihe-in -78.76, 136.08 APE8-rot-in 311.34 APE67-dihe-in -61.08, -29.98 -51.0, -40.22 APE12-dist-in 10.501 APE11-dist-in 10.889 APE10-dist-in 5.774 APE9-dist-in 4.003 None None None XRAY 2.0 0.201 0.227 A 419 408 0 0 0 0 [[76, 342]] 1.0 5otf AGC_CDC42BPB_HUMAN AGC 6.5e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
3TKUA 2 415 1711.0 M77:418,M77:419 Type1,Allosteric Active DFGin 6.602 13.355 BLAminus -143.03, 175.94 52.02, 80.01 -94.23, 18.83 305.33, 99.72 -66.85, -0.48 in-in in 8.858 Saltbr-in 2.916 HRD-in -68.08, -55.01 75.95, 5.48 in-in-in SNCiii in-in ActLoopNT-in 3.044 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.43, 163.82 APE9-dihe-na 93.99, -165.51 APE8-dihe-in -114.48, 131.1 APE8-rot-in 310.89 APE67-dihe-in -54.25, -25.55 -45.59, -49.4 APE12-dist-in 11.04 APE11-dist-in 11.04 APE10-dist-in 5.176 APE9-dist-in 3.762 None None None XRAY 2.15 0.223 0.273 A 433 395 0 0 0 0 [[76, 342]] 1.0 3tku AGC_CDC42BPB_HUMAN AGC 7.2e-96 326.3 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
3TKUB 2 415 1711.0 M77:418,M77:419 Type1,Allosteric Active DFGin 6.7 13.42 BLAminus -146.47, 178.95 50.88, 78.82 -93.25, 17.64 304.13, 100.62 -66.46, -1.59 in-in in 8.934 Saltbr-in 2.849 HRD-in -79.08, -52.56 75.39, 5.44 in-in-in SNCiii in-in ActLoopNT-in 3.022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.41, 166.49 APE9-dihe-na 89.07, -163.52 APE8-dihe-in -118.0, 134.6 APE8-rot-in 310.18 APE67-dihe-in -54.07, -25.9 -51.37, -47.08 APE12-dist-in 11.06 APE11-dist-in 11.053 APE10-dist-in 5.192 APE9-dist-in 3.746 None None None XRAY 2.15 0.223 0.273 B 433 395 0 0 0 0 [[76, 342]] 1.0 3tku AGC_CDC42BPB_HUMAN AGC 7.2e-96 326.3 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta

AGC_CDC42BPB (Serine/threonine-protein kinase MRCK beta)

Total number of chains: 10
Active chains: 10
Family: AGC
Spatial label Dihedral label Number of Chains Percent Representative
DFGin BLAminus 10 100.0% AF-Q9Y5S2-K1A

Hover over column headers for tooltip help

SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name
MRCKB_HUMAN 4UAKA Q9Y5S2 2 417 1711.0 ADP:60501 ATPlike Active DFGin 6.536 13.389 BLAminus -126.67, 169.91 71.43, 81.15 -99.11, 14.11 300.02, 102.96 -73.12, -5.53 in-in in 8.635 Saltbr-in 2.748 HRD-in -78.82, -49.28 69.95, 4.01 in-in-in SNCiii in-in ActLoopNT-in 2.977 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -131.28, 157.85 APE9-dihe-na 87.21, -164.86 APE8-dihe-in -127.15, 132.61 APE8-rot-in 302.21 APE67-dihe-in -64.23, -20.61 -57.86, -36.49 APE12-dist-in 10.511 APE11-dist-in 11.151 APE10-dist-in 6.313 APE9-dist-in 3.548 None None None XRAY 1.73 0.198 0.243 A 419 401 0 0 0 0 [[76, 342]] 1.0 4uak Homo sapiens AGC_CDC42BPB_HUMAN AGC 6.5e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
MRCKB_HUMAN AF-Q9Y5S2-K1A Q9Y5S2 68 350 1711.0 No_ligand No_ligand Active DFGin 6.286 13.418 BLAminus -138.11, 175.86 52.03, 73.16 -82.88, 16.9 300.82, 95.68 -61.27, -18.14 in-in in 8.67 Saltbr-in 2.619 HRD-in -80.82, -44.33 65.35, 6.41 in-in-in SNCiii in-in ActLoopNT-in 2.885 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -121.32, 151.0 APE9-dihe-na 118.31, 170.33 APE8-dihe-in -66.77, 129.62 APE8-rot-in 287.64 APE67-dihe-in -77.39, -20.44 -51.73, -36.54 APE12-dist-in 9.843 APE11-dist-in 10.942 APE10-dist-in 5.188 APE9-dist-in 3.788 None None None AF2 -1.0 1.0 1.0 A 283 283 0 0 0 0 [[76, 342]] 1.0 AF-Q9Y5S2-K1 Homo sapiens AGC_CDC42BPB_HUMAN AGC 1.7e-96 328.2 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
MRCKB_HUMAN AF-Q9Y5S2-K3A Q9Y5S2 68 350 1711.0 No_ligand No_ligand Active DFGin 6.165 13.252 BLAminus -140.87, 174.27 54.93, 67.41 -77.14, 15.47 302.2, 109.63 -60.94, -17.3 in-in in 8.594 Saltbr-in 2.681 HRD-in -80.0, -45.38 64.95, 8.05 in-in-in SNCiii in-in ActLoopNT-in 2.873 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -124.11, 160.14 APE9-dihe-na 106.26, -177.58 APE8-dihe-in -89.7, 125.56 APE8-rot-in 303.52 APE67-dihe-in -69.05, -20.8 -47.75, -44.36 APE12-dist-in 9.53 APE11-dist-in 10.952 APE10-dist-in 5.151 APE9-dist-in 3.627 None None None AF2 -1.0 1.0 1.0 A 283 283 0 0 0 0 [[76, 342]] 1.0 AF-Q9Y5S2-K3 Homo sapiens AGC_CDC42BPB_HUMAN AGC 1.7e-96 328.2 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
MRCKB_HUMAN 3QFVA Q9Y5S2 2 415 1711.0 NM7:416 Type1 Active DFGin 6.652 13.483 BLAminus -155.19, -177.74 51.28, 74.91 -100.44, 20.96 290.95, 120.41 -84.8, 1.24 in-in in 8.66 Saltbr-in 3.586 HRD-in -68.56, -55.63 80.26, 2.79 in-in-in SNCiii in-in ActLoopNT-in 3.062 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -127.25, 145.57 APE9-dihe-na 95.66, -174.68 APE8-dihe-in -88.83, 133.9 APE8-rot-in 320.1 APE67-dihe-in -63.11, -25.9 -60.21, -35.51 APE12-dist-in 10.616 APE11-dist-in 11.198 APE10-dist-in 5.501 APE9-dist-in 4.17 None None None XRAY 2.65 0.196 0.268 A 415 395 0 0 0 0 [[76, 342]] 1.0 3qfv Homo sapiens AGC_CDC42BPB_HUMAN AGC 6.3e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
MRCKB_HUMAN 3QFVB Q9Y5S2 2 415 1711.0 NM7:416 Type1 Active DFGin 6.357 13.248 BLAminus -146.98, -178.33 51.23, 77.88 -102.57, 32.33 302.88, 111.63 -92.77, 5.32 in-in in 8.692 Saltbr-in 2.619 HRD-in -65.12, -52.57 79.81, -7.22 in-in-in SNCiii in-in ActLoopNT-in 3.139 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -126.96, 150.13 APE9-dihe-na 114.47, 164.94 APE8-dihe-in -66.67, 141.54 APE8-rot-in 317.58 APE67-dihe-in -60.07, -38.36 -60.72, -35.72 APE12-dist-in 10.736 APE11-dist-in 11.342 APE10-dist-in 5.667 APE9-dist-in 4.087 None None None XRAY 2.65 0.196 0.268 B 415 396 0 0 0 0 [[76, 342]] 1.0 3qfv Homo sapiens AGC_CDC42BPB_HUMAN AGC 6.3e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
MRCKB_HUMAN 4UALA Q9Y5S2 2 417 1711.0 3FV:60501 Type1 Active DFGin 6.57 13.343 BLAminus -128.09, 170.47 58.99, 78.49 -90.49, 11.57 302.61, 102.02 -65.54, -5.61 in-in in 8.675 Saltbr-in 2.909 HRD-in -76.1, -52.24 74.17, 2.64 in-in-in SNCiii in-in ActLoopNT-in 2.963 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -119.7, -165.94 APE9-dihe-na 97.69, -165.3 APE8-dihe-in -123.13, 127.49 APE8-rot-in 312.99 APE67-dihe-in -64.7, -21.04 -49.2, -41.29 APE12-dist-in 10.401 APE11-dist-in 10.706 APE10-dist-in 5.458 APE9-dist-in 3.725 None None None XRAY 1.71 0.206 0.236 A 419 400 5 0 0 3 [[76, 342]] 1.0 4ual Homo sapiens AGC_CDC42BPB_HUMAN AGC 6.5e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
MRCKB_HUMAN 5OTEA Q9Y5S2 2 417 1711.0 AQE:60501 Type1 Active DFGin 6.44 13.538 BLAminus -132.86, 172.8 58.15, 78.6 -89.88, 11.87 305.96, 106.7 -64.89, -6.52 in-in in 8.637 Saltbr-in 2.717 HRD-in -76.88, -48.31 73.79, 2.14 in-in-in SNCiii in-in ActLoopNT-in 2.96 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -150.88, 152.67 APE9-dihe-na 86.33, -167.63 APE8-dihe-in -120.1, 130.3 APE8-rot-in 304.26 APE67-dihe-in -60.96, -19.55 -48.3, -43.83 APE12-dist-in 10.442 APE11-dist-in 11.319 APE10-dist-in 6.425 APE9-dist-in 3.469 None None None XRAY 1.68 0.197 0.218 A 419 404 2 0 0 0 [[76, 342]] 1.0 5ote Homo sapiens AGC_CDC42BPB_HUMAN AGC 6.5e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
MRCKB_HUMAN 5OTFA Q9Y5S2 2 417 1711.0 AQ5:60504 Type1 Active DFGin 6.474 13.836 BLAminus -138.71, 166.8 56.15, 77.62 -87.94, 13.12 305.59, 108.27 -63.54, -12.28 in-in in 8.966 Saltbr-in 2.633 HRD-in -69.74, -49.73 69.82, 11.73 in-in-in SNCiii in-in ActLoopNT-in 2.93 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -144.82, 174.96 APE9-dihe-na 90.86, 165.77 APE8-dihe-in -78.76, 136.08 APE8-rot-in 311.34 APE67-dihe-in -61.08, -29.98 -51.0, -40.22 APE12-dist-in 10.501 APE11-dist-in 10.889 APE10-dist-in 5.774 APE9-dist-in 4.003 None None None XRAY 2.0 0.201 0.227 A 419 408 0 0 0 0 [[76, 342]] 1.0 5otf Homo sapiens AGC_CDC42BPB_HUMAN AGC 6.5e-96 326.4 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
MRCKB_HUMAN 3TKUA Q9Y5S2 2 415 1711.0 M77:418,M77:419 Type1,Allosteric Active DFGin 6.602 13.355 BLAminus -143.03, 175.94 52.02, 80.01 -94.23, 18.83 305.33, 99.72 -66.85, -0.48 in-in in 8.858 Saltbr-in 2.916 HRD-in -68.08, -55.01 75.95, 5.48 in-in-in SNCiii in-in ActLoopNT-in 3.044 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -125.43, 163.82 APE9-dihe-na 93.99, -165.51 APE8-dihe-in -114.48, 131.1 APE8-rot-in 310.89 APE67-dihe-in -54.25, -25.55 -45.59, -49.4 APE12-dist-in 11.04 APE11-dist-in 11.04 APE10-dist-in 5.176 APE9-dist-in 3.762 None None None XRAY 2.15 0.223 0.273 A 433 395 0 0 0 0 [[76, 342]] 1.0 3tku Homo sapiens AGC_CDC42BPB_HUMAN AGC 7.2e-96 326.3 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta
MRCKB_HUMAN 3TKUB Q9Y5S2 2 415 1711.0 M77:418,M77:419 Type1,Allosteric Active DFGin 6.7 13.42 BLAminus -146.47, 178.95 50.88, 78.82 -93.25, 17.64 304.13, 100.62 -66.46, -1.59 in-in in 8.934 Saltbr-in 2.849 HRD-in -79.08, -52.56 75.39, 5.44 in-in-in SNCiii in-in ActLoopNT-in 3.022 ActLoopCT-in nonTYR APEdihe_aaiii APEdist_iiii APE10-dihe-na -129.41, 166.49 APE9-dihe-na 89.07, -163.52 APE8-dihe-in -118.0, 134.6 APE8-rot-in 310.18 APE67-dihe-in -54.07, -25.9 -51.37, -47.08 APE12-dist-in 11.06 APE11-dist-in 11.053 APE10-dist-in 5.192 APE9-dist-in 3.746 None None None XRAY 2.15 0.223 0.273 B 433 395 0 0 0 0 [[76, 342]] 1.0 3tku Homo sapiens AGC_CDC42BPB_HUMAN AGC 7.2e-96 326.3 1 260 260 217 218 219 221 223 105 124 128 197 199 198 200 263 246 241 240 239 238 237 236 235 154 Serine/threonine-protein kinase MRCK beta

AGC_CDC42BPB (Serine/threonine-protein kinase MRCK beta)

Total number of chains: 0
Active chains: 0
Family: AGC
Spatial label Dihedral label Number of Chains Percent Representative

Hover over column headers for tooltip help

SwissprotID PDB UniprotID First_obs_res Last_obs_res Length_Unp Ligand Ligand_type Activity_label Spatial_label Phe_Glu4_dis Phe_Lys_dis Dihedral_label XDFG
φ,ψ
DFG-Asp
φ,ψ
DFG-Phe
φ,ψ
DFG-Phe
χ1,χ2
DFG-Gly
φ,ψ
ChelixSaltbr_label Chelix_label Lys_Glu_dis Saltbr_label LysNZ_GluOE_dis HRD_label His φ,ψ Arg φ,ψ SNC_label SNCpymol_label ActLoop_label ActLoopNT_label DFG6_XHRD_dis ActLoopCT_label APEtype APEdihe_label APEdist_label APE10_dihe_label APE10 φ,ψ APE9_dihe_label APE9 φ,ψ APE8_dihe_label APE8 φ,ψ APE8_rotamer_label APE8 χ1 APE67_label APE6 φ,ψ APE7 φ,ψ APE12_dist_label APE12_DFG4_dis APE11_dist_label APE11_DFG4_dis APE10_dist_label APE10_DFG4_dis APE9_dist_label APE9_Arg_dis Chain_mut Chain_phos Modified_aa Method Resolution Rvalue FreeRvalue Chain_id ChainLen Ordered_residues DomainBreak ActLoopLength ActLoopResolvedResidues ActLoopDisorderedResidues Kinase_domains_Unp N_Kinase_domains_Unp pdb Species Kincore_name hmm Evalue Score hmmbeg hmmend hmmlen XDFGnum DFGnum PHEnum DFG4num DFG6num LYSnum GLUnum GLU4num XHRDnum ARGnum HRDnum HRDaspnum aFaspnum APEnum APE6num APE7num APE8num APE9num APE10num APE11num APE12num Hinge1num Protein_name