| Gene | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| ACVR2A | AF-P27037-K1A | P27037 | 184 | 489 | 513.0 | No_ligand | No_ligand | Active | DFGin | 7.269 | 13.7003 | BLAminus | -137.45, 169.69 | 67.25, 68.52 | -84.71, 16.97 | 304.39, 108.34 | -63.28, -19.76 | in-in | in | 7.8867 | Saltbr-in | 2.6721 | HRD-in | -85.43, -41.28 | 66.31, 6.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8788 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -99.89, 156.32 | APE9-dihe-na | 105.55, -169.46 | APE8-dihe-in | -93.07, 118.12 | APE8-rot-in | 303.12 | APE67-dihe-in | -59.36, -25.82 | -49.75, -42.86 | APE12-dist-in | 10.7018 | APE11-dist-in | 12.4807 | APE10-dist-in | 6.3872 | APE9-dist-in | 3.4511 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306.0 | 306.0 | 0 | 30 | 30 | 0 | [[192, 481]] | 1.0 | AF-P27037-K1 | TKL_ACVR2A_HUMAN | TKL | 2.9e-83 | 285.4 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | AF-P27037-K3A | P27037 | 184 | 489 | 513.0 | No_ligand | No_ligand | Active | DFGin | 6.7063 | 13.9826 | BLAminus | -138.42, 173.36 | 68.77, 61.7 | -77.85, 18.77 | 302.81, 110.47 | -60.19, -21.37 | in-in | in | 7.8878 | Saltbr-in | 2.7307 | HRD-in | -81.7, -38.65 | 63.48, 6.34 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8396 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.93, 163.23 | APE9-dihe-na | 97.04, -163.98 | APE8-dihe-in | -90.36, 115.81 | APE8-rot-in | 304.87 | APE67-dihe-in | -57.74, -26.76 | -42.5, -46.12 | APE12-dist-in | 10.3774 | APE11-dist-in | 12.1036 | APE10-dist-in | 6.1819 | APE9-dist-in | 3.6194 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306.0 | 306.0 | 0 | 30 | 30 | 0 | [[192, 481]] | 1.0 | AF-P27037-K3 | TKL_ACVR2A_HUMAN | TKL | 2.9e-83 | 285.4 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | 3Q4TB | P27037 | 191 | 485 | 513.0 | TAK:60001 | Type1 | Active | DFGin | 7.5844 | 13.7734 | BLAminus | -128.74, 167.36 | 69.0, 93.18 | -108.05, 19.83 | 304.44, 108.16 | -60.68, -27.36 | in-in | in | 8.091 | Saltbr-in | 2.7887 | HRD-in | -87.27, -46.41 | 76.78, -1.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8357 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -109.89, -26.02 | APE9-dihe-na | -85.65, -161.16 | APE8-dihe-in | -82.47, 131.09 | APE8-rot-in | 297.46 | APE67-dihe-in | -64.09, -26.22 | -62.33, -41.13 | APE12-dist-in | 10.9477 | APE11-dist-in | 12.4473 | APE10-dist-in | 6.4709 | APE9-dist-in | 3.4539 | None | None | None | XRAY | 1.96 | 0.171 | 0.223 | B | 322.0 | 293.0 | 2 | 30 | 28 | 2 | [[192, 481]] | 1.0 | 3q4t | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | 3SOCB | P27037 | 191 | 486 | 513.0 | GVD:60001 | Type1 | Active | DFGin | 7.5819 | 13.8829 | BLAminus | -125.19, 161.27 | 74.66, 92.72 | -105.52, 25.82 | 308.76, 104.61 | -59.88, -27.57 | in-in | in | 7.9875 | Saltbr-in | 2.6813 | HRD-in | -86.72, -48.71 | 80.27, -0.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8822 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -95.59, -20.99 | APE9-dihe-na | -82.69, -168.74 | APE8-dihe-in | -77.8, 127.48 | APE8-rot-in | 301.33 | APE67-dihe-in | -68.64, -19.61 | -61.12, -39.03 | APE12-dist-in | 10.9898 | APE11-dist-in | 12.4011 | APE10-dist-in | 6.3732 | APE9-dist-in | 3.3677 | None | None | None | XRAY | 1.95 | 0.165 | 0.211 | B | 322.0 | 294.0 | 2 | 30 | 28 | 2 | [[192, 481]] | 1.0 | 3soc | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | 4ASXA | P27037 | 191 | 486 | 513.0 | 6OJ:61487 | Type1 | Active | DFGin | 7.5848 | 13.7119 | BLAminus | -124.23, 158.41 | 76.6, 95.75 | -110.56, 27.08 | 303.84, 107.63 | -64.07, -28.35 | in-in | in | 8.1512 | Saltbr-in | 2.681 | HRD-in | -83.4, -48.78 | 80.27, 1.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9143 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -98.14, -19.06 | APE9-dihe-na | -92.2, -158.06 | APE8-dihe-in | -89.26, 125.94 | APE8-rot-in | 297.71 | APE67-dihe-in | -63.22, -23.86 | -54.78, -47.48 | APE12-dist-in | 10.9349 | APE11-dist-in | 12.4424 | APE10-dist-in | 6.3997 | APE9-dist-in | 3.4817 | None | None | None | XRAY | 2.05 | 0.188 | 0.225 | A | 322.0 | 295.0 | 1 | 30 | 29 | 1 | [[192, 481]] | 1.0 | 4asx | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | 3Q4TA | P27037 | 191 | 484 | 513.0 | TAK:60002 | Type1 | Inactive | DFGin | 7.5736 | 14.0966 | BLAminus | -123.56, 165.6 | 68.53, 85.67 | -104.01, 23.68 | 300.6, 98.11 | -61.19, -27.21 | in-in | in | 8.2168 | Saltbr-in | 2.797 | HRD-in | -88.26, -44.7 | 74.99, 6.75 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8743 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -135.25, 165.71 | APE9-dihe-na | -78.55, -169.19 | APE8-dihe-in | -70.65, 121.11 | APE8-rot-in | 308.48 | APE67-dihe-in | -46.78, -36.2 | -40.9, -55.96 | APE12-dist-in | 10.3422 | APE11-dist-out | 6.2827 | APE10-dist-out | 8.8817 | APE9-dist-in | 3.5295 | None | None | None | XRAY | 1.96 | 0.171 | 0.223 | A | 322.0 | 294.0 | 0 | 30 | 30 | 0 | [[192, 481]] | 1.0 | 3q4t | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | 3SOCA | P27037 | 191 | 486 | 513.0 | GVD:60001 | Type1 | Inactive | DFGin | 7.6273 | 14.1199 | BLAminus | -129.53, 162.94 | 71.26, 89.98 | -103.8, 24.98 | 302.16, 98.96 | -63.88, -23.66 | in-in | in | 8.1095 | Saltbr-in | 2.6616 | HRD-in | -79.15, -50.46 | 79.66, 5.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9044 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -135.71, 167.82 | APE9-dihe-na | -85.17, -168.04 | APE8-dihe-in | -72.04, 119.11 | APE8-rot-in | 310.28 | APE67-dihe-in | -43.46, -38.05 | -39.83, -55.04 | APE12-dist-in | 9.9819 | APE11-dist-out | 5.797 | APE10-dist-out | 8.9398 | APE9-dist-in | 3.5905 | None | None | None | XRAY | 1.95 | 0.165 | 0.211 | A | 322.0 | 296.0 | 0 | 30 | 30 | 0 | [[192, 481]] | 1.0 | 3soc | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | 4ASXB | P27037 | 191 | 486 | 513.0 | 6OJ:61487 | Type1 | Inactive | DFGin | 7.649 | 13.9339 | BLAminus | -125.14, 162.25 | 70.64, 90.86 | -105.86, 23.27 | 300.55, 102.55 | -60.78, -32.52 | in-in | in | 8.1876 | Saltbr-in | 2.8127 | HRD-in | -76.15, -47.44 | 73.25, 3.45 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9141 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -130.56, 171.14 | APE9-dihe-na | -89.41, -155.19 | APE8-dihe-in | -83.7, 128.51 | APE8-rot-in | 306.98 | APE67-dihe-in | -59.4, -19.9 | -51.63, -52.75 | APE12-dist-in | 10.1183 | APE11-dist-out | 5.9218 | APE10-dist-out | 8.9293 | APE9-dist-in | 3.6405 | None | None | None | XRAY | 2.05 | 0.188 | 0.225 | B | 322.0 | 296.0 | 0 | 30 | 30 | 0 | [[192, 481]] | 1.0 | 4asx | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| ACVR2A | AVR2A_HUMAN | AF-P27037-K1A | P27037 | 184 | 489 | 513.0 | No_ligand | No_ligand | Active | DFGin | 7.269 | 13.7003 | BLAminus | -137.45, 169.69 | 67.25, 68.52 | -84.71, 16.97 | 304.39, 108.34 | -63.28, -19.76 | in-in | in | 7.8867 | Saltbr-in | 2.6721 | HRD-in | -85.43, -41.28 | 66.31, 6.96 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8788 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -99.89, 156.32 | APE9-dihe-na | 105.55, -169.46 | APE8-dihe-in | -93.07, 118.12 | APE8-rot-in | 303.12 | APE67-dihe-in | -59.36, -25.82 | -49.75, -42.86 | APE12-dist-in | 10.7018 | APE11-dist-in | 12.4807 | APE10-dist-in | 6.3872 | APE9-dist-in | 3.4511 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306.0 | 306.0 | 0 | 30 | 30 | 0 | [[192, 481]] | 1.0 | AF-P27037-K1 | Homo sapiens | TKL_ACVR2A_HUMAN | TKL | 2.9e-83 | 285.4 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | AVR2A_HUMAN | AF-P27037-K3A | P27037 | 184 | 489 | 513.0 | No_ligand | No_ligand | Active | DFGin | 6.7063 | 13.9826 | BLAminus | -138.42, 173.36 | 68.77, 61.7 | -77.85, 18.77 | 302.81, 110.47 | -60.19, -21.37 | in-in | in | 7.8878 | Saltbr-in | 2.7307 | HRD-in | -81.7, -38.65 | 63.48, 6.34 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8396 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -127.93, 163.23 | APE9-dihe-na | 97.04, -163.98 | APE8-dihe-in | -90.36, 115.81 | APE8-rot-in | 304.87 | APE67-dihe-in | -57.74, -26.76 | -42.5, -46.12 | APE12-dist-in | 10.3774 | APE11-dist-in | 12.1036 | APE10-dist-in | 6.1819 | APE9-dist-in | 3.6194 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 306.0 | 306.0 | 0 | 30 | 30 | 0 | [[192, 481]] | 1.0 | AF-P27037-K3 | Homo sapiens | TKL_ACVR2A_HUMAN | TKL | 2.9e-83 | 285.4 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | AVR2A_HUMAN | 3Q4TB | P27037 | 191 | 485 | 513.0 | TAK:60001 | Type1 | Active | DFGin | 7.5844 | 13.7734 | BLAminus | -128.74, 167.36 | 69.0, 93.18 | -108.05, 19.83 | 304.44, 108.16 | -60.68, -27.36 | in-in | in | 8.091 | Saltbr-in | 2.7887 | HRD-in | -87.27, -46.41 | 76.78, -1.51 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8357 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -109.89, -26.02 | APE9-dihe-na | -85.65, -161.16 | APE8-dihe-in | -82.47, 131.09 | APE8-rot-in | 297.46 | APE67-dihe-in | -64.09, -26.22 | -62.33, -41.13 | APE12-dist-in | 10.9477 | APE11-dist-in | 12.4473 | APE10-dist-in | 6.4709 | APE9-dist-in | 3.4539 | None | None | None | XRAY | 1.96 | 0.171 | 0.223 | B | 322.0 | 293.0 | 2 | 30 | 28 | 2 | [[192, 481]] | 1.0 | 3q4t | Homo sapiens | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | AVR2A_HUMAN | 3SOCB | P27037 | 191 | 486 | 513.0 | GVD:60001 | Type1 | Active | DFGin | 7.5819 | 13.8829 | BLAminus | -125.19, 161.27 | 74.66, 92.72 | -105.52, 25.82 | 308.76, 104.61 | -59.88, -27.57 | in-in | in | 7.9875 | Saltbr-in | 2.6813 | HRD-in | -86.72, -48.71 | 80.27, -0.88 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8822 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -95.59, -20.99 | APE9-dihe-na | -82.69, -168.74 | APE8-dihe-in | -77.8, 127.48 | APE8-rot-in | 301.33 | APE67-dihe-in | -68.64, -19.61 | -61.12, -39.03 | APE12-dist-in | 10.9898 | APE11-dist-in | 12.4011 | APE10-dist-in | 6.3732 | APE9-dist-in | 3.3677 | None | None | None | XRAY | 1.95 | 0.165 | 0.211 | B | 322.0 | 294.0 | 2 | 30 | 28 | 2 | [[192, 481]] | 1.0 | 3soc | Homo sapiens | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | AVR2A_HUMAN | 4ASXA | P27037 | 191 | 486 | 513.0 | 6OJ:61487 | Type1 | Active | DFGin | 7.5848 | 13.7119 | BLAminus | -124.23, 158.41 | 76.6, 95.75 | -110.56, 27.08 | 303.84, 107.63 | -64.07, -28.35 | in-in | in | 8.1512 | Saltbr-in | 2.681 | HRD-in | -83.4, -48.78 | 80.27, 1.37 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9143 | ActLoopCT-in | nonTYR | APEdihe_aaiii | APEdist_iiii | APE10-dihe-na | -98.14, -19.06 | APE9-dihe-na | -92.2, -158.06 | APE8-dihe-in | -89.26, 125.94 | APE8-rot-in | 297.71 | APE67-dihe-in | -63.22, -23.86 | -54.78, -47.48 | APE12-dist-in | 10.9349 | APE11-dist-in | 12.4424 | APE10-dist-in | 6.3997 | APE9-dist-in | 3.4817 | None | None | None | XRAY | 2.05 | 0.188 | 0.225 | A | 322.0 | 295.0 | 1 | 30 | 29 | 1 | [[192, 481]] | 1.0 | 4asx | Homo sapiens | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | AVR2A_HUMAN | 3Q4TA | P27037 | 191 | 484 | 513.0 | TAK:60002 | Type1 | Inactive | DFGin | 7.5736 | 14.0966 | BLAminus | -123.56, 165.6 | 68.53, 85.67 | -104.01, 23.68 | 300.6, 98.11 | -61.19, -27.21 | in-in | in | 8.2168 | Saltbr-in | 2.797 | HRD-in | -88.26, -44.7 | 74.99, 6.75 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.8743 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -135.25, 165.71 | APE9-dihe-na | -78.55, -169.19 | APE8-dihe-in | -70.65, 121.11 | APE8-rot-in | 308.48 | APE67-dihe-in | -46.78, -36.2 | -40.9, -55.96 | APE12-dist-in | 10.3422 | APE11-dist-out | 6.2827 | APE10-dist-out | 8.8817 | APE9-dist-in | 3.5295 | None | None | None | XRAY | 1.96 | 0.171 | 0.223 | A | 322.0 | 294.0 | 0 | 30 | 30 | 0 | [[192, 481]] | 1.0 | 3q4t | Homo sapiens | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | AVR2A_HUMAN | 3SOCA | P27037 | 191 | 486 | 513.0 | GVD:60001 | Type1 | Inactive | DFGin | 7.6273 | 14.1199 | BLAminus | -129.53, 162.94 | 71.26, 89.98 | -103.8, 24.98 | 302.16, 98.96 | -63.88, -23.66 | in-in | in | 8.1095 | Saltbr-in | 2.6616 | HRD-in | -79.15, -50.46 | 79.66, 5.28 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9044 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -135.71, 167.82 | APE9-dihe-na | -85.17, -168.04 | APE8-dihe-in | -72.04, 119.11 | APE8-rot-in | 310.28 | APE67-dihe-in | -43.46, -38.05 | -39.83, -55.04 | APE12-dist-in | 9.9819 | APE11-dist-out | 5.797 | APE10-dist-out | 8.9398 | APE9-dist-in | 3.5905 | None | None | None | XRAY | 1.95 | 0.165 | 0.211 | A | 322.0 | 296.0 | 0 | 30 | 30 | 0 | [[192, 481]] | 1.0 | 3soc | Homo sapiens | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| ACVR2A | AVR2A_HUMAN | 4ASXB | P27037 | 191 | 486 | 513.0 | 6OJ:61487 | Type1 | Inactive | DFGin | 7.649 | 13.9339 | BLAminus | -125.14, 162.25 | 70.64, 90.86 | -105.86, 23.27 | 300.55, 102.55 | -60.78, -32.52 | in-in | in | 8.1876 | Saltbr-in | 2.8127 | HRD-in | -76.15, -47.44 | 73.25, 3.45 | in-in-out | SNCiio | in-out | ActLoopNT-in | 2.9141 | ActLoopCT-out | nonTYR | APEdihe_aaiii | APEdist_iooi | APE10-dihe-na | -130.56, 171.14 | APE9-dihe-na | -89.41, -155.19 | APE8-dihe-in | -83.7, 128.51 | APE8-rot-in | 306.98 | APE67-dihe-in | -59.4, -19.9 | -51.63, -52.75 | APE12-dist-in | 10.1183 | APE11-dist-out | 5.9218 | APE10-dist-out | 8.9293 | APE9-dist-in | 3.6405 | None | None | None | XRAY | 2.05 | 0.188 | 0.225 | B | 322.0 | 296.0 | 0 | 30 | 30 | 0 | [[192, 481]] | 1.0 | 4asx | Homo sapiens | TKL_ACVR2A_HUMAN | TKL | 3.5e-83 | 285.1 | 2.0 | 266.0 | 265.0 | 339 | 340 | 341 | 343 | 345 | 219 | 232 | 236 | 319 | 321 | 320 | 322.0 | 386 | 369 | 364 | 363 | 362 | 361 | 360 | 359 | 358 | 268 | Activin receptor type-2A |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|