|
AGC
|
AKT1
|
AKT1_HUMAN
|
4EKKA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
144 - 477 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4EKKB
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
144 - 477 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
AF-P31749-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
142 - 416 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
AF-P31749-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
142 - 416 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6BUUA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
144 - 478 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6BUUB
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
144 - 477 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6NPZA
|
2.12 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
142 - 478 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6NPZB
|
2.12 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
141 - 477 |
0 |
TPO308,SEP473,SEP477 |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4GV1A
|
1.49 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0XZ |
Type1 |
144 - 477 |
0 |
TPO308 |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3OCBA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XM1 |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3OCBB
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XM1 |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3OW4A
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SMY |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3OW4B
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SMY |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3QKLA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SMR |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3QKMA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SM9 |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4EKLA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0RF |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3CQUA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CQU |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3CQWA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CQW |
Type1 |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3MV5A
|
2.47 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XFE |
Type1 |
144 - 477 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3MVHA
|
2.01 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
WFE |
Type1 |
145 - 476 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6CCYA
|
2.18 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX4 |
Type1 |
144 - 983 |
0 |
TPO308 |
N199S,S396P,E397S,T433V |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3QKKA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SMH |
Type1.5_Front |
144 - 478 |
0 |
TPO308 |
S473D |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UVYA
|
2.11 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
XOO |
Allosteric |
3 - 439 |
0 |
None |
E17K |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW2A
|
2.2 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
XOO |
Allosteric |
4 - 437 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW9A
|
1.9 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
XQ2 |
Allosteric |
3 - 428 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
8UW7A
|
1.972 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
XOO |
Allosteric |
3 - 439 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
3O96A
|
2.7 |
Inactive |
DFGout‑BBAminus |
none-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
IQO |
Allosteric |
2 - 429 |
0 |
None |
None |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHHA
|
2.7 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
G4Q |
Allosteric |
2 - 439 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHJA
|
2.3 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
G4H |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6S9WA
|
2.3 |
Inactive |
DFGout‑BBAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
L1Z |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
4EJNA
|
2.19 |
Inactive |
DFGout‑BBAminus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
0R4 |
Type1 |
4 - 438 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
5KCVA
|
2.7 |
Inactive |
DFGout‑None |
none-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
6S1 |
Allosteric |
6 - 438 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
7APJA
|
2.05 |
Inactive |
DFGout‑None |
none-none |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
3 - 439 |
0 |
None |
S2N |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHFA
|
2.9 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
G4K |
Allosteric |
3 - 439 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHGA
|
2.3 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
G4T |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6HHIA
|
2.7 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
G4N |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
6S9XA
|
2.6 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
L1W |
Allosteric |
3 - 443 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
7NH4A
|
2.3 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
UCE |
Allosteric |
4 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT1
|
AKT1_HUMAN
|
7NH5A
|
1.9 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
UC8 |
Allosteric |
3 - 444 |
0 |
None |
E114A,E115A,E116A |
RAC-alpha serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1O6KA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
146 - 479 |
0 |
TPO309 |
S474D |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1O6LA
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
AF-P31751-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
144 - 417 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
AF-P31751-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
144 - 417 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E87A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G95 |
Type1 |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E87B
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G95 |
Type1 |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2JDOA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I5S |
Type1 |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2JDRA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L20 |
Type1 |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2UW9A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVP |
Type1 |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2X39A
|
1.93 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X39 |
Type1 |
146 - 477 |
0 |
TPO309 |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
2XH5A
|
2.72 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X37 |
Type1 |
146 - 479 |
0 |
TPO309 |
R467Q,T468E,H469M,P471E,Q472D,S474D,S476I,S478D,I479W |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3D0EA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G93 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3D0EB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G93 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E88A
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G96 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E88B
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G96 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E8DA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G98 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
3E8DB
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G98 |
Type1.5_Back |
146 - 480 |
0 |
TPO309,TPO451 |
S474D |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
9C1WA
|
2.0 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
XOO |
Allosteric |
3 - 440 |
0 |
None |
P115A,G116A |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
8Q61A
|
2.32 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
K06 |
Type3 |
1 - 435 |
0 |
None |
N2D |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZKA
|
2.3 |
Inactive |
DFGout‑None |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 441 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZOA
|
2.75 |
Inactive |
DFGout‑None |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 442 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1GZNA
|
2.5 |
Inactive |
DFGout‑None |
in-none |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
146 - 442 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1MRVA
|
2.8 |
Inactive |
DFGout‑None |
none-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
147 - 440 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT2
|
AKT2_HUMAN
|
1MRYA
|
2.8 |
Inactive |
DFGout‑None |
none-none |
none-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnio |
No_ligand |
No_ligand |
146 - 440 |
0 |
None |
None |
RAC-beta serine/threonine-protein kinase |
|
AGC
|
AKT3
|
AKT3_HUMAN
|
AF-Q9Y243-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
140 - 413 |
0 |
None |
None |
RAC-gamma serine/threonine-protein kinase |
|
AGC
|
AKT3
|
AKT3_HUMAN
|
AF-Q9Y243-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
140 - 413 |
0 |
None |
None |
RAC-gamma serine/threonine-protein kinase |
|
AGC
|
CDC42BPA
|
MRCKA_HUMAN
|
AF-Q5VT25-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
69 - 351 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK alpha |
|
AGC
|
CDC42BPA
|
MRCKA_HUMAN
|
AF-Q5VT25-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
69 - 351 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK alpha |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
4UAKA
|
1.73 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
2 - 417 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
AF-Q9Y5S2-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
68 - 350 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
AF-Q9Y5S2-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
68 - 350 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
3QFVA
|
2.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NM7 |
Type1 |
2 - 415 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
3QFVB
|
2.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NM7 |
Type1 |
2 - 415 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
4UALA
|
1.71 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3FV |
Type1 |
2 - 417 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
5OTEA
|
1.68 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AQE |
Type1 |
2 - 417 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
5OTFA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AQ5 |
Type1 |
2 - 417 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
3TKUA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77,
M77
|
Type1,
Allosteric
|
2 - 415 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
|
AGC
|
CDC42BPB
|
MRCKB_HUMAN
|
3TKUB
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77,
M77
|
Type1,
Allosteric
|
2 - 415 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK beta |
|
AGC
|
CDC42BPG
|
MRCKG_HUMAN
|
AF-Q6DT37-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
63 - 345 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK gamma |
|
AGC
|
CDC42BPG
|
MRCKG_HUMAN
|
AF-Q6DT37-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
63 - 345 |
0 |
None |
None |
Serine/threonine-protein kinase MRCK gamma |
|
AGC
|
CIT
|
CTRO_HUMAN
|
AF-O14578-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
89 - 368 |
0 |
None |
None |
Citron Rho-interacting kinase |
|
AGC
|
CIT
|
CTRO_HUMAN
|
AF-O14578-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
89 - 368 |
0 |
None |
None |
Citron Rho-interacting kinase |
|
AGC
|
DMPK
|
DMPK_HUMAN
|
AF-Q09013-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
63 - 347 |
0 |
None |
None |
Myotonin-protein kinase |
|
AGC
|
DMPK
|
DMPK_HUMAN
|
AF-Q09013-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
63 - 347 |
0 |
None |
None |
Myotonin-protein kinase |
|
AGC
|
DMPK
|
DMPK_HUMAN
|
2VD5A
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI8 |
Type1 |
11 - 416 |
0 |
None |
None |
Myotonin-protein kinase |
|
AGC
|
DMPK
|
DMPK_HUMAN
|
2VD5B
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI8 |
Type1 |
11 - 416 |
0 |
None |
None |
Myotonin-protein kinase |
|
AGC
|
GRK1
|
GRK1_HUMAN
|
AF-Q15835-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
182 - 463 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
|
AGC
|
GRK1
|
GRK1_HUMAN
|
AF-Q15835-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
182 - 463 |
0 |
None |
None |
Rhodopsin kinase GRK1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
AF-P25098-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 461 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
AF-P25098-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 461 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5UVCA
|
2.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8PV |
Type1 |
30 - 536 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5UKLA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SIX |
Type1 |
31 - 671 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5HE1A
|
3.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZS2 |
Type1 |
29 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
6C2YA
|
2.74 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EJS |
Type1 |
30 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
4MK0A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
29X |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
7K7LA
|
2.539 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W4D |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
7K7ZA
|
2.606 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W4G |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3V5WA
|
2.07 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8PR |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
4PNKA
|
2.56 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
KZQ |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5WG3A
|
2.896 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFM |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5WG4A
|
2.31 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFV |
Type1 |
31 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5WG5A
|
3.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZSO |
Type1 |
30 - 668 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5UUUA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
QRW |
Type1.5_Front |
31 - 538 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
5UKKA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8DJ |
Type1.5_Front |
30 - 667 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
6U7CA
|
2.44 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Q1Y |
Type1.5_Front |
30 - 669 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3CIKA
|
2.75 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 669 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
7PWDA
|
2.6 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8DS |
Type1 |
27 - 668 |
0 |
None |
S670A |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3KRWA
|
2.9 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BA1 |
Type1 |
30 - 671 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK2
|
ARBK1_HUMAN
|
3KRXA
|
3.1 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BA1 |
Type1 |
30 - 671 |
0 |
None |
None |
Beta-adrenergic receptor kinase 1 |
|
AGC
|
GRK3
|
ARBK2_HUMAN
|
AF-P35626-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 461 |
0 |
None |
None |
G protein-coupled receptor kinase 3 |
|
AGC
|
GRK3
|
ARBK2_HUMAN
|
AF-P35626-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 461 |
0 |
None |
None |
G protein-coupled receptor kinase 3 |
|
AGC
|
GRK4
|
GRK4_HUMAN
|
4YHJA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AN2 |
ATPlike |
25 - 525 |
0 |
None |
C563S,C578S |
G protein-coupled receptor kinase 4 |
|
AGC
|
GRK4
|
GRK4_HUMAN
|
4YHJB
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AN2 |
ATPlike |
25 - 527 |
0 |
None |
C563S,C578S |
G protein-coupled receptor kinase 4 |
|
AGC
|
GRK4
|
GRK4_HUMAN
|
AF-P32298-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
179 - 457 |
0 |
None |
None |
G protein-coupled receptor kinase 4 |
|
AGC
|
GRK4
|
GRK4_HUMAN
|
AF-P32298-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
179 - 457 |
0 |
None |
None |
G protein-coupled receptor kinase 4 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9CKOA
|
2.8 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
1 - 542 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRKA
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARA |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRLA
|
2.73 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARB |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRPA
|
2.8 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARF |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
4TNDA
|
1.802 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
15 - 543 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9CKRA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9CKSA
|
3.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
AF-P34947-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
178 - 456 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
AF-P34947-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
178 - 456 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9CKQA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
4TNBA
|
2.113 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
15 - 543 |
0 |
None |
None |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
8UAPA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W2T |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BREA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W3F |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRGA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ6 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRHA
|
3.69 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ7 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRMA
|
2.73 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARC |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRNA
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARD |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BROA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1ARE |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9CKPA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
1 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9MX2A
|
3.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
1 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
6PJXA
|
1.96 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
1 - 542 |
0 |
None |
E104K,R304H,G438E |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
8UAQA
|
2.8 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W3F |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRFA
|
2.84 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ5 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRIA
|
2.9 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ8 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK5
|
GRK5_HUMAN
|
9BRJA
|
2.8 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQ9 |
Type1 |
25 - 542 |
0 |
None |
D311N |
G protein-coupled receptor kinase 5 |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
2ACXA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
14 - 532 |
0 |
None |
C561S,C562S,C565S |
G protein-coupled receptor kinase 6 |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
2ACXB
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
14 - 535 |
0 |
None |
C561S,C562S,C565S |
G protein-coupled receptor kinase 6 |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
3NYOA
|
2.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
2 - 557 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
3NYOB
|
2.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
2 - 557 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
AF-P43250-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
178 - 456 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
AF-P43250-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
178 - 456 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
3NYNA
|
2.72 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
2 - 557 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
|
AGC
|
GRK6
|
GRK6_HUMAN
|
3NYNB
|
2.72 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SGV |
Type1 |
2 - 557 |
0 |
None |
None |
G protein-coupled receptor kinase 6 |
|
AGC
|
GRK7
|
GRK7_HUMAN
|
AF-Q8WTQ7-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 462 |
0 |
None |
None |
Rhodopsin kinase GRK7 |
|
AGC
|
GRK7
|
GRK7_HUMAN
|
AF-Q8WTQ7-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
183 - 462 |
0 |
None |
None |
Rhodopsin kinase GRK7 |
|
AGC
|
LATS1
|
LATS1_HUMAN
|
AF-O95835-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
697 - 1018 |
0 |
None |
None |
Serine/threonine-protein kinase LATS1 |
|
AGC
|
LATS1
|
LATS1_HUMAN
|
AF-O95835-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
697 - 1018 |
0 |
None |
None |
Serine/threonine-protein kinase LATS1 |
|
AGC
|
LATS2
|
LATS2_HUMAN
|
AF-Q9NRM7-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
660 - 981 |
0 |
None |
None |
Serine/threonine-protein kinase LATS2 |
|
AGC
|
LATS2
|
LATS2_HUMAN
|
AF-Q9NRM7-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
660 - 981 |
0 |
None |
None |
Serine/threonine-protein kinase LATS2 |
|
AGC
|
MAST1
|
MAST1_HUMAN
|
AF-Q9Y2H9-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
366 - 655 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 1 |
|
AGC
|
MAST1
|
MAST1_HUMAN
|
AF-Q9Y2H9-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
366 - 655 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 1 |
|
AGC
|
MAST2
|
MAST2_HUMAN
|
AF-Q6P0Q8-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
504 - 793 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 2 |
|
AGC
|
MAST2
|
MAST2_HUMAN
|
AF-Q6P0Q8-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
504 - 793 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 2 |
|
AGC
|
MAST3
|
MAST3_HUMAN
|
AF-O60307-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
359 - 648 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 3 |
|
AGC
|
MAST3
|
MAST3_HUMAN
|
AF-O60307-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
359 - 648 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 3 |
|
AGC
|
MAST4
|
MAST4_HUMAN
|
AF-O15021-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
562 - 851 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 4 |
|
AGC
|
MAST4
|
MAST4_HUMAN
|
AF-O15021-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
562 - 851 |
0 |
None |
None |
Microtubule-associated serine/threonine-protein kinase 4 |
|
AGC
|
MASTL
|
GWL_HUMAN
|
AF-Q96GX5-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 843 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
|
AGC
|
MASTL
|
GWL_HUMAN
|
AF-Q96GX5-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 843 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
|
AGC
|
MASTL
|
GWL_HUMAN
|
8V5HA
|
2.74 |
Inactive |
DFGin‑BLAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
A1AAE |
Type1 |
29 - 847 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
|
AGC
|
MASTL
|
GWL_HUMAN
|
5LOHA
|
3.1 |
Inactive |
DFGin‑BLAplus |
none-none |
out-out |
nonTYR |
APEdihe_aanon |
APEdist_nnno |
STU |
Type1 |
30 - 854 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
|
AGC
|
MASTL
|
GWL_HUMAN
|
5LOHB
|
3.1 |
Inactive |
None‑None |
none-none |
none-out |
nonTYR |
APEdihe_aannn |
APEdist_nnno |
STU |
Type1 |
30 - 854 |
0 |
None |
None |
Serine/threonine-protein kinase greatwall |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1H1WA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ATP |
ATPlike |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2BIYA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
72 - 359 |
0 |
None |
S241A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3HRCA
|
1.91 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
76 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4RRVA
|
1.412 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
76 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5ACKA
|
1.24 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
73 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVPA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVPB
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
74 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVPC
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVPD
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
74 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4CT2A
|
1.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
75 - 359 |
0 |
SEP241 |
L113V,I118V,I119H,V124I,T128Q,R131K,T148C,F157L,Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5MRDA
|
1.41 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
76 - 359 |
0 |
SEP241 |
K76S,L113V,I118V,I119N,V124I,T128Q,R131K,T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3HRFA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
P47
|
ATPlike,
Allosteric
|
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4A06A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
A06
|
ATPlike,
Allosteric
|
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4AW0A
|
1.43 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
MJF
|
ATPlike,
Allosteric
|
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4AW1A
|
1.68 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
21O
|
ATPlike,
Allosteric
|
66 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4RQKA
|
1.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
R1S
|
ATPlike,
Allosteric
|
74 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4RQVA
|
1.502 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
R2S
|
ATPlike,
Allosteric
|
71 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVOA
|
1.09 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
78W
|
ATPlike,
Allosteric
|
73 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4CT1A
|
1.85 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
31S
|
ATPlike,
Allosteric
|
76 - 359 |
0 |
SEP241 |
L113V,I118V,I119H,V124I,T128Q,R131K,T148C,F157L,Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4XX9A
|
1.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
RF4,
RF4
|
ATPlike,
Allosteric,
Allosteric
|
71 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
4A07A
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP,
AZ7,
AZ7
|
ATPlike,
Allosteric,
Allosteric
|
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXA
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXB
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
77 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXC
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXD
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
76 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXE
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
1F8 |
Allosteric |
76 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXF
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXG
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORXH
|
2.204 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
1F8 |
Allosteric |
75 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
8DQTA
|
1.31 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
U35,
U35,
U35
|
Allosteric,
Allosteric,
Allosteric
|
70 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
74 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZB
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
73 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZC
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
74 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3ORZD
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2A2,
BI4
|
Allosteric,
Type1
|
73 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3OTUA
|
2.101 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J30,
BI4
|
Allosteric,
Type1.5_Front
|
77 - 359 |
0 |
SEP241 |
T148C |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
AF-O15530-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
74 - 350 |
0 |
None |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
AF-O15530-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
74 - 350 |
0 |
None |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1Z5MA
|
2.17 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
LI8 |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2PE0A
|
2.35 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
39Z |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2PE1A
|
2.14 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
517 |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2PE2A
|
2.13 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
464 |
Type1 |
74 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUSA
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JNZ |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUUA
|
1.98 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JOZ |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUYA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JPZ |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU9A
|
1.95 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI3 |
Type1 |
72 - 357 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UVRA
|
2.81 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI8 |
Type1 |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NUNA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
JMZ |
Type1 |
71 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2XCHA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
CKG |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HKMA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
61Y |
Type1 |
76 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HNGA
|
3.01 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
62O |
Type1 |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HO7A
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
63L |
Type1 |
71 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5HO8A
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
63E |
Type1 |
71 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1OKYA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
STU |
Type1 |
72 - 360 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1OKZA
|
2.51 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
UCN |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU3A
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
LY4 |
Type1 |
73 - 360 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU7A
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI2 |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
1UU8A
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
BI1 |
Type1 |
72 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NAYA
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
MP6 |
Type1 |
76 - 362 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NAYB
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
MP6 |
Type1 |
76 - 362 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3RWPA
|
1.92 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ABQ |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3RWQA
|
2.55 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3RW |
Type1 |
72 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3SC1A
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3S1 |
Type1 |
73 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3H9OA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
9BD |
Type1 |
75 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2R7BA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
253 |
Type1 |
75 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3IONA
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
8H1 |
Type1 |
75 - 359 |
0 |
None |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3IOPA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
8I1 |
Type1 |
75 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCQA
|
2.501 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q0 |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCSA
|
2.487 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q1 |
Type1 |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3RCJA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3RC |
Type1 |
77 - 358 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVLA
|
1.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
537 |
Type1 |
74 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVMA
|
1.26 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADE |
Type1 |
76 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
5LVNA
|
1.379 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADN |
Type1 |
75 - 359 |
0 |
SEP241 |
Y288G,Q292A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3PWYA
|
3.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
SYP |
Type1 |
71 - 359 |
0 |
None |
E166C,C260S |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
2XCKA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
MH4 |
Type1 |
76 - 359 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCXA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q2 |
Type1.5_Back |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QCYA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
3Q3 |
Type1.5_Front |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QD0A
|
1.99 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
3Q4 |
Type1.5_Front |
73 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QD3A
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3Q5 |
Type1.5_Front |
71 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QD4A
|
2.3 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
3Q6 |
Type1.5_Front |
71 - 358 |
0 |
SEP241 |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3NAXA
|
1.75 |
Inactive |
DFGout‑BBAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MP7 |
Type2 |
76 - 360 |
0 |
None |
None |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QC4A
|
1.8 |
Inactive |
DFGout‑BBAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MP7 |
Type2 |
76 - 359 |
0 |
SEP241 |
E303A,K304A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PDPK1
|
PDPK1_HUMAN
|
3QC4B
|
1.8 |
Inactive |
DFGout‑None |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MP7 |
Type2 |
51 - 359 |
0 |
SEP241 |
E303A,K304A |
3-phosphoinositide-dependent protein kinase 1 |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTDA
|
2.0 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
605 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTGA
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2V9 |
Type1 |
605 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
AF-Q16512-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
607 - 882 |
0 |
None |
None |
Serine/threonine-protein kinase N1 |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
AF-Q16512-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
607 - 882 |
0 |
None |
None |
Serine/threonine-protein kinase N1 |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTHA
|
1.8 |
Inactive |
DFGin‑BLAplus |
in-in |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
DRN |
Type1 |
606 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
|
AGC
|
PKN1
|
PKN1_HUMAN
|
4OTIA
|
1.93 |
Inactive |
DFGin‑BLAplus |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MI1 |
Type1 |
606 - 940 |
0 |
TPO774,SEP916 |
None |
Serine/threonine-protein kinase N1 |
|
AGC
|
PKN2
|
PKN2_HUMAN
|
4CRSA
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
AGS |
ATPlike |
646 - 984 |
0 |
SEP755,TPO816,TPO958 |
None |
Serine/threonine-protein kinase N2 |
|
AGC
|
PKN2
|
PKN2_HUMAN
|
AF-Q16513-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
649 - 924 |
0 |
None |
None |
Serine/threonine-protein kinase N2 |
|
AGC
|
PKN2
|
PKN2_HUMAN
|
AF-Q16513-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
649 - 924 |
0 |
None |
None |
Serine/threonine-protein kinase N2 |
|
AGC
|
PKN3
|
PKN3_HUMAN
|
AF-Q6P5Z2-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
551 - 826 |
0 |
None |
None |
Serine/threonine-protein kinase N3 |
|
AGC
|
PKN3
|
PKN3_HUMAN
|
AF-Q6P5Z2-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
551 - 826 |
0 |
None |
None |
Serine/threonine-protein kinase N3 |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE6A
|
2.1 |
Inactive |
DFGin‑ABAminus |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE6B
|
2.1 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
17 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE9A
|
2.3 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4AE9B
|
2.3 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
7Y1GB
|
2.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
I5G |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9DC6A
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1A3I |
Type1 |
16 - 351 |
0 |
SEP140,TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9DC6B
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1A3I |
Type1 |
16 - 351 |
0 |
SEP140,TPO198 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3AMBA
|
2.25 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VX6 |
Type1 |
4 - 351 |
0 |
SEP11,TPO198,SEP339 |
K48R,L96Q,M121L,V124A,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8X5LA
|
2.75 |
Inactive |
DFGin‑ABAminus |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
RKD |
Type1 |
17 - 351 |
0 |
SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8X5LB
|
2.75 |
Inactive |
DFGin‑ABAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
RKD |
Type1 |
17 - 334 |
0 |
SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB8A
|
1.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB5A
|
1.641 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6NO7E
|
3.55 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6NO7G
|
3.55 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
15 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB7A
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB7B
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYRA
|
3.661 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYRC
|
3.661 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
2 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9EDCA
|
4.18 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9EDDA
|
6.3 |
Inactive |
DFGin‑BLAminus |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9EDEA
|
5.9 |
Inactive |
DFGin‑BLAminus |
in-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB6A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
14 - 351 |
0 |
SEP11,SEP140,TPO198 |
L206R |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4WB6B
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
9 - 351 |
0 |
SEP11,TPO198,SEP339 |
L206R |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5IZJA
|
1.85 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6J9 |
Allosteric |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5IZJB
|
1.85 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6J9 |
Allosteric |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5J5XA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6J9 |
Allosteric |
10 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
AF-P17612-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
AF-P17612-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSA
|
4.75 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSC
|
4.75 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSE
|
4.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6BYSG
|
4.75 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6NO7A
|
3.55 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6NO7C
|
3.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3AGMA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5IZFA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3MVJB
|
2.49 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3NX8A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJFA
|
7.5 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJFB
|
7.5 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
42 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJGA
|
6.2 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
42 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6WJGB
|
6.2 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
42 - 351 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
9DCDA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1A3J |
Type1 |
14 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3AGLA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A03 |
Type1 |
11 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3AGLB
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A03 |
Type1 |
15 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3L9LA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L9L |
Type1 |
12 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3L9LB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L9L |
Type1 |
13 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3OOGA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YTP |
Type1 |
17 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3OVVA
|
1.58 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1SB |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3OWPA
|
1.88 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2SB |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3OXTA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3SB |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3P0MA
|
2.03 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4SB |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3POOA
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
S69 |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3VQHA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQB |
Type1 |
5 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJ1A
|
1.768 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NVX |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJ2A
|
2.019 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NVV |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJ9A
|
1.87 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
S3N |
Type1 |
11 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJAA
|
1.93 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4L7 |
Type1 |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
4UJBA
|
1.949 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8BQ |
Type1 |
5 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5BX6A
|
1.89 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
495 |
Type1 |
6 - 351 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5BX7A
|
1.89 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4W1 |
Type1 |
6 - 350 |
0 |
SEP11,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5UZKA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
504 |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6QJ7A
|
1.69 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J4B |
Type1 |
14 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
7Y1GA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
I5G |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6C0UA
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
EE4 |
Type1 |
12 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3MVJA
|
2.49 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XFE |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3MVJE
|
2.49 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XFE |
Type1 |
16 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3L9MA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L9M |
Type1 |
12 - 351 |
0 |
TPO198,SEP339 |
V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3L9MB
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L9M |
Type1 |
14 - 351 |
0 |
TPO198,SEP339 |
V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3L9NA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L9N |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
V124A,L174M,Q182K |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FE2A
|
2.34 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XTI |
Type1 |
4 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FE2B
|
2.34 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XTI |
Type1 |
4 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FE5A
|
2.51 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XTT |
Type1 |
3 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FE5B
|
2.51 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XTT |
Type1 |
4 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FECA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XU0 |
Type1 |
3 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
8FECB
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XU0 |
Type1 |
3 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
2GU8A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
796 |
Type1 |
15 - 351 |
0 |
TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
5N23A
|
2.088 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
35R |
Type1 |
9 - 351 |
0 |
SEP11,SEP140,TPO198,SEP339 |
K48R,L96Q,M121L,V124A,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
3AMAA
|
1.75 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SKE |
Type1 |
2 - 351 |
0 |
SEP11,TPO198,SEP339 |
K48R,L96Q,M121L,V124A,Q182K,T184A |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACA
|
KAPCA_HUMAN
|
6FRXA
|
1.88 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E3Z |
Type1 |
13 - 351 |
0 |
SEP140,TPO198,SEP339 |
None |
cAMP-dependent protein kinase catalytic subunit alpha |
|
AGC
|
PRKACB
|
KAPCB_HUMAN
|
AF-P22694-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit beta |
|
AGC
|
PRKACB
|
KAPCB_HUMAN
|
AF-P22694-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit beta |
|
AGC
|
PRKACG
|
KAPCG_HUMAN
|
AF-P22612-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit gamma |
|
AGC
|
PRKACG
|
KAPCG_HUMAN
|
AF-P22612-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 306 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit gamma |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
AF-P17252-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
331 - 605 |
0 |
None |
None |
Protein kinase C alpha type |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
AF-P17252-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
331 - 605 |
0 |
None |
None |
Protein kinase C alpha type |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
4RA4A
|
2.63 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3KZ |
Type1 |
332 - 666 |
0 |
TPO497,TPO638,SEP657 |
C619S |
Protein kinase C alpha type |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
3IW4A
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LW4 |
Type1 |
331 - 669 |
0 |
TPO638,SEP657 |
T497E |
Protein kinase C alpha type |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
3IW4B
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LW4 |
Type1 |
332 - 666 |
0 |
TPO638,SEP657 |
T497E |
Protein kinase C alpha type |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
3IW4C
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LW4 |
Type1 |
330 - 670 |
0 |
TPO638,SEP657 |
T497E |
Protein kinase C alpha type |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
8U37A
|
2.48 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V5U |
Type1 |
332 - 666 |
0 |
TPO497,TPO638 |
D463N,V568I,S657E |
Protein kinase C alpha type |
|
AGC
|
PRKCA
|
KPCA_HUMAN
|
8UAKA
|
2.82 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W39 |
Type1 |
332 - 666 |
0 |
TPO497,TPO638 |
D463N,V568I,S657E |
Protein kinase C alpha type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE2A
|
2.95 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE3A
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
30 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE4A
|
2.68 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE4B
|
2.68 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADN |
Type1 |
30 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE1A
|
3.32 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
19 - 668 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE1B
|
3.32 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
19 - 668 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
8SE2B
|
2.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
30 - 671 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
AF-P05771-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
334 - 608 |
0 |
None |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
AF-P05771-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
334 - 608 |
0 |
None |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
2I0EA
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
PDS |
Type1 |
339 - 668 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
2I0EB
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PDS |
Type1 |
339 - 668 |
0 |
TPO500,TPO642,SEP661 |
None |
Protein kinase C beta type |
|
AGC
|
PRKCB
|
KPCB_HUMAN
|
9S9TA
|
3.425 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LY4 |
Type1 |
340 - 667 |
0 |
TPO500,TPO642,SEP661 |
D427N |
Protein kinase C beta type |
|
AGC
|
PRKCD
|
KPCD_HUMAN
|
AF-Q05655-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
341 - 611 |
0 |
None |
None |
Protein kinase C delta type |
|
AGC
|
PRKCD
|
KPCD_HUMAN
|
AF-Q05655-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
341 - 611 |
0 |
None |
None |
Protein kinase C delta type |
|
AGC
|
PRKCE
|
KPCE_HUMAN
|
AF-Q02156-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
400 - 676 |
0 |
None |
None |
Protein kinase C epsilon type |
|
AGC
|
PRKCE
|
KPCE_HUMAN
|
AF-Q02156-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
400 - 676 |
0 |
None |
None |
Protein kinase C epsilon type |
|
AGC
|
PRKCG
|
KPCG_HUMAN
|
AF-P05129-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
343 - 622 |
0 |
None |
None |
Protein kinase C gamma type |
|
AGC
|
PRKCG
|
KPCG_HUMAN
|
AF-P05129-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
343 - 622 |
0 |
None |
None |
Protein kinase C gamma type |
|
AGC
|
PRKCH
|
KPCL_HUMAN
|
AF-P24723-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
347 - 622 |
0 |
None |
None |
Protein kinase C eta type |
|
AGC
|
PRKCH
|
KPCL_HUMAN
|
AF-P24723-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
347 - 622 |
0 |
None |
None |
Protein kinase C eta type |
|
AGC
|
PRKCH
|
KPCL_HUMAN
|
8FP1A
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XXF |
Type1 |
349 - 676 |
0 |
TPO513,TPO656 |
S675E |
Protein kinase C eta type |
|
AGC
|
PRKCH
|
KPCL_HUMAN
|
8FP3A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Y3I |
Type1 |
349 - 679 |
0 |
TPO513,TPO656 |
S675E |
Protein kinase C eta type |
|
AGC
|
PRKCH
|
KPCL_HUMAN
|
3TXOA
|
2.05 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
07U |
Type1 |
353 - 679 |
0 |
TPO656 |
S675E |
Protein kinase C eta type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
8R3YI
|
3.68 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
248 - 585 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
8R3XA
|
2.591 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
8R3XB
|
2.591 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
6ILZA
|
3.261 |
Inactive |
DFGin‑ABAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFU |
Type1 |
254 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3A8WA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3A8WB
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
5LIHA
|
3.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
248 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
5LIHB
|
3.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
5LI9A
|
1.79 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ACP |
ATPlike |
248 - 589 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
5LI1A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
248 - 589 |
0 |
TPO412,SEP484,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
9EJMB
|
3.33 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
AF-P41743-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
246 - 530 |
0 |
None |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
AF-P41743-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
246 - 530 |
0 |
None |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3A8XA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3A8XB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
9EJKB
|
3.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
9EJLB
|
3.48 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
25 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
6ILZC
|
3.261 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFU |
Type1 |
254 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
6ILZE
|
3.261 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFU |
Type1 |
255 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
6ILZG
|
3.261 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AFU |
Type1 |
254 - 587 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3ZH8A
|
2.739 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C58 |
Type1 |
248 - 590 |
0 |
TPO412,TPO564 |
C595S |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3ZH8B
|
2.739 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C58 |
Type1 |
248 - 589 |
0 |
TPO412,TPO564 |
C595S |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
3ZH8C
|
2.739 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C58 |
Type1 |
248 - 588 |
0 |
TPO412,TPO564 |
C595S |
Protein kinase C iota type |
|
AGC
|
PRKCI
|
KPCI_HUMAN
|
1ZRZA
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI1 |
Type1 |
249 - 588 |
0 |
TPO412,TPO564 |
None |
Protein kinase C iota type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
AF-Q04759-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
372 - 642 |
0 |
None |
None |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
AF-Q04759-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
372 - 642 |
0 |
None |
None |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4Q9ZA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PZW |
Type1 |
375 - 706 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4Q9ZB
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PZW |
Type1 |
374 - 704 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4RA5A
|
2.61 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3L0 |
Type1 |
374 - 706 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
4RA5B
|
2.61 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3L0 |
Type1 |
375 - 701 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
2JEDA
|
2.32 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LG8 |
Type1 |
375 - 700 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
2JEDB
|
2.32 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LG8 |
Type1 |
375 - 706 |
0 |
SEP676,SEP695 |
I381E,T538E |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
5F9EA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5VS |
Type1 |
374 - 706 |
0 |
SEP676,SEP695 |
None |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
5F9EB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5VS |
Type1 |
375 - 700 |
0 |
SEP676,SEP695 |
None |
Protein kinase C theta type |
|
AGC
|
PRKCQ
|
KPCT_HUMAN
|
1XJDA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
377 - 696 |
0 |
TPO538,SEP695 |
None |
Protein kinase C theta type |
|
AGC
|
PRKCZ
|
KPCZ_HUMAN
|
AF-Q05513-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
244 - 526 |
0 |
None |
None |
Protein kinase C zeta type |
|
AGC
|
PRKCZ
|
KPCZ_HUMAN
|
AF-Q05513-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
244 - 526 |
0 |
None |
None |
Protein kinase C zeta type |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4UA
|
1.99 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX6 |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4UB
|
1.99 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX6 |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4WA
|
2.23 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZJ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4WB
|
2.23 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZJ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4TA
|
2.08 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PCG,
ATP
|
Allosteric,
ATPlike
|
204 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4TB
|
2.08 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PCG,
ATP
|
Allosteric,
ATPlike
|
204 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BG2A
|
1.83 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
336 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BG2B
|
1.83 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
346 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BG2C
|
1.83 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
337 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BG2D
|
1.83 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
344 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7LV3A
|
2.41 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
57 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7LV3B
|
2.41 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
58 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4VA
|
2.28 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
EXZ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
7T4VB
|
2.28 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EXZ |
Allosteric |
205 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
AF-Q13976-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
352 - 627 |
0 |
None |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
AF-Q13976-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
352 - 627 |
0 |
None |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BDLA
|
1.96 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_iiio |
No_ligand |
No_ligand |
337 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6BDLB
|
1.96 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_iiii |
No_ligand |
No_ligand |
337 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG1
|
KGP1_HUMAN
|
6C0TA
|
1.98 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
EE4 |
Type1.5_Front |
337 - 671 |
0 |
TPO517 |
None |
cGMP-dependent protein kinase 1 |
|
AGC
|
PRKG2
|
KGP2_HUMAN
|
AF-Q13237-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
445 - 719 |
0 |
None |
None |
cGMP-dependent protein kinase 2 |
|
AGC
|
PRKG2
|
KGP2_HUMAN
|
AF-Q13237-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
445 - 719 |
0 |
None |
None |
cGMP-dependent protein kinase 2 |
|
AGC
|
PRKX
|
PRKX_HUMAN
|
AF-P51817-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 311 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit PRKX |
|
AGC
|
PRKX
|
PRKX_HUMAN
|
AF-P51817-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 311 |
0 |
None |
None |
cAMP-dependent protein kinase catalytic subunit PRKX |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMA
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZA
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3NC |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZB
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoi |
3NC |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZC
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3NC |
Type1 |
6 - 404 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NCZD
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3NC |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMB
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
3ND |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMC
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
3ND |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3NDMD
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3ND |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFA
|
2.45 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4V |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFB
|
2.45 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
B4V |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFC
|
2.45 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4V |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNFD
|
2.45 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4V |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGA
|
2.9 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4Y |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGB
|
2.9 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
B4Y |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGC
|
2.9 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B4Y |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNGD
|
2.9 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4Y |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHA
|
3.1 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B5G |
Type1 |
6 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHB
|
3.1 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
B5G |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHC
|
3.1 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
B5G |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNHD
|
3.1 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B5G |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
6E9WA
|
2.96 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J0P |
Type1 |
9 - 404 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
6E9WB
|
2.96 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
J0P |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2V55A
|
3.705 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
6 - 404 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2V55C
|
3.705 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
6 - 404 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
AF-Q13464-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
68 - 346 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
AF-Q13464-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
68 - 346 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S26D
|
2.744 |
Inactive |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
6 - 399 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
8ZH5A
|
3.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S26A
|
2.744 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
86K |
Type1 |
6 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S26B
|
2.744 |
None |
DFGin‑BLAminus |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
86K |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7A
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iiio |
07Q |
Type1 |
9 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7B
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
07Q |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7C
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iiio |
07Q |
Type1 |
9 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TV7D
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioo |
07Q |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SA
|
2.286 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
0HD |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SB
|
2.286 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
0HD |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SC
|
2.286 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
0HD |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3V8SD
|
2.286 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
0HD |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4W7PA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3J7 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4W7PB
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3J7 |
Type1 |
6 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4W7PC
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3J7 |
Type1 |
6 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4W7PD
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3J7 |
Type1 |
6 - 403 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7JOUA
|
3.318 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFS |
Type1 |
9 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ESMA
|
3.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M77 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ESMB
|
3.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
M77 |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ETKA
|
2.96 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HFS |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ETKB
|
2.96 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
HFS |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ETRA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Y27 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
2ETRB
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
Y27 |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3D9VA
|
3.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H52 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3D9VB
|
3.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
H52 |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4YVCA
|
3.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4KH |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4YVCB
|
3.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
4KH |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4YVEA
|
3.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4KK |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
4YVEB
|
3.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iiio |
4KK |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5BMLA
|
2.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4TW |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5BMLB
|
2.95 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
4TW |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5KKSA
|
3.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6U1 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5KKTA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6U2 |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5UZJA
|
3.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8UV |
Type1 |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5UZJB
|
3.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
8UV |
Type1 |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJA
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
07R |
Type1.5_Back |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5HVUA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
65R |
Type1.5_Front |
6 - 405 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5HVUB
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
65R |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5KKSB
|
3.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
6U1 |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5KKTB
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
6U2 |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNEA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4J |
Type1.5_Front |
14 - 400 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNEB
|
2.6 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
B4J |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNEC
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4J |
Type1.5_Front |
6 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
5WNED
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B4J |
Type1.5_Front |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S26C
|
2.744 |
Inactive |
DFGin‑BLBminus |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
86K |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJC
|
2.9 |
Inactive |
DFGin‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oiio |
07R |
Type1 |
7 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJB
|
2.9 |
Inactive |
DFGinter‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
No_ligand |
No_ligand |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
3TWJD
|
2.9 |
Inactive |
DFGinter‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
No_ligand |
No_ligand |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25A
|
2.337 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
86G |
Type1 |
7 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25B
|
2.337 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
86G |
Type1 |
8 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25C
|
2.337 |
Inactive |
DFGout‑None |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
86G |
Type1 |
13 - 402 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK1
|
ROCK1_HUMAN
|
7S25D
|
2.337 |
Inactive |
None‑None |
in-in |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
9 - 401 |
0 |
None |
None |
Rho-associated protein kinase 1 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MC
|
2.65 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MD
|
2.65 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QA
|
3.15 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QB
|
3.15 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
No_ligand |
No_ligand |
28 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QC
|
3.15 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7QD
|
3.15 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RA
|
3.33 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RC
|
3.33 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiio |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PA
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
O1V |
Type1 |
27 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PB
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnio |
O1V |
Type1 |
27 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PC
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
O1V |
Type1 |
28 - 416 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5PD
|
3.3 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
O1V |
Type1 |
26 - 416 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8YB
|
3.2 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
YEA |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8ZA
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YEI |
Type1 |
31 - 416 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8ZB
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
YEI |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X92A
|
2.2 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YEW |
Type1 |
29 - 416 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X92B
|
2.2 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_noio |
YEW |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTA
|
2.93 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
3SG |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTB
|
2.93 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3SG |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTC
|
2.93 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3SG |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4WOTD
|
2.93 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
3SG |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9HFPA
|
2.92 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1IUI |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4L6QA
|
2.79 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1WU |
Type1 |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
4L6QB
|
2.79 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1WU |
Type1 |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
AF-O75116-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
84 - 362 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
AF-O75116-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
84 - 362 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RB
|
3.33 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MA
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
O1S |
Type1 |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6P5MB
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiio |
O1S |
Type1 |
18 - 417 |
0 |
None |
F270Y |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8XA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YDW |
Type1 |
32 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8XB
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiio |
YDW |
Type1 |
29 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8X8YA
|
3.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
YEA |
Type1 |
31 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVA
|
2.586 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
VFS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVB
|
2.586 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
VFS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVC
|
2.586 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_onno |
VFS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVD
|
2.586 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
VFS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVE
|
2.586 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_innn |
VFS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVF
|
2.586 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVG
|
2.586 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_innn |
VFS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JOVH
|
2.586 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTA
|
2.214 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
VFA |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTB
|
2.214 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
VFA |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTC
|
2.214 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
VFA |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTD
|
2.214 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
VFA |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTE
|
2.214 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
VFA |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTF
|
2.214 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFA |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTG
|
2.214 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_innn |
VFA |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7JNTH
|
2.214 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VFA |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NA
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_niio |
5YS |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NB
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NC
|
3.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
5YS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6ND
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NE
|
3.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
5YS |
Type1 |
23 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NF
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NG
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6NH
|
3.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
5YS |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OA
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
5YK |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OB
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OD
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_inii |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OE
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OF
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5YK |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PA
|
2.82 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_onoo |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PB
|
2.82 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PC
|
2.82 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6PD
|
2.82 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5YV |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QA
|
2.89 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QB
|
2.89 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QC
|
2.89 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnio |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6QD
|
2.89 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5YO |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8A
|
2.63 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
A1H6L |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8B
|
2.63 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1H6L |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8C
|
2.63 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1H6L |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9EP8D
|
2.63 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
A1H6L |
Type1 |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6ED6A
|
2.86 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J0P |
Type1 |
27 - 415 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OC
|
2.75 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
5YK |
Type1.5_Front |
22 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OG
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5YK |
Type1.5_Front |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
7P6OH
|
2.75 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
5YK |
Type1.5_Front |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
6ED6B
|
2.86 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
J0P |
Type1.5_Front |
28 - 416 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
5U7RD
|
3.33 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_onno |
81G |
Type1 |
25 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUA
|
3.02 |
Inactive |
DFGout‑BBAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUC
|
3.02 |
Inactive |
DFGout‑BBAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSA
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSB
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSC
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
Z8O |
Type1 |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
8GDSD
|
2.71 |
Inactive |
DFGout‑BBAminus |
out-none |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
Z8O |
Type1.5_Front |
24 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUB
|
3.02 |
Inactive |
DFGout‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
ROCK2
|
ROCK2_HUMAN
|
9JCUD
|
3.02 |
Inactive |
DFGout‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 417 |
0 |
None |
None |
Rho-associated protein kinase 2 |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
AF-Q15418-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
54 - 329 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
AF-Q15418-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
54 - 329 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
8XOVA
|
2.55 |
Inactive |
DFGin‑BLAplus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
ANP |
ATPlike |
56 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
2Z7QA
|
2.0 |
Inactive |
DFGin‑BLBplus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
ACP |
ATPlike |
56 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
2Z7RA
|
2.0 |
Inactive |
DFGin‑BLBplus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
STU |
Type1 |
53 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
AGC
|
RPS6KA1-1
|
KS6A1_HUMAN
|
2Z7SA
|
2.1 |
Inactive |
DFGin‑BLBplus |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
P01 |
Type1 |
56 - 340 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
AGC
|
RPS6KA2-1
|
KS6A2_HUMAN
|
AF-Q15349-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
51 - 326 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-2 |
|
AGC
|
RPS6KA2-1
|
KS6A2_HUMAN
|
AF-Q15349-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
51 - 326 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-2 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
4NW5A
|
1.94 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2NR |
Type1 |
51 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
4NW6A
|
1.74 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2NS |
Type1 |
51 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
AF-P51812-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
60 - 335 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
AF-P51812-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
60 - 335 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOA
|
2.75 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_oonn |
ANP |
ATPlike |
45 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOE
|
2.75 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_oonn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOI
|
2.75 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_onnn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOK
|
2.75 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_oonn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOC
|
2.75 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ANP |
ATPlike |
46 - 347 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
7OPOG
|
2.75 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanni |
APEdist_oonn |
ANP |
ATPlike |
46 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8EQ5A
|
1.8 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
QCT |
Type1 |
49 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8R58A
|
2.31 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
QCT |
Type1 |
49 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYA
|
3.2 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
A1LU8 |
Type1 |
58 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYB
|
3.2 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
59 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYC
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
A1LU8 |
Type1 |
61 - 358 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYD
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYE
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooi |
A1LU8 |
Type1 |
64 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYF
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 345 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYG
|
3.2 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
A1LU8 |
Type1 |
59 - 346 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYH
|
3.2 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooi |
A1LU8 |
Type1 |
59 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYI
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
A1LU8 |
Type1 |
63 - 348 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
8XFYJ
|
3.2 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
A1LU8 |
Type1 |
65 - 347 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
4NUSA
|
2.39 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2NK |
Type1 |
53 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9LA
|
2.15 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
583 |
Type1 |
49 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9KA
|
2.55 |
Inactive |
DFGout‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
584 |
Type1 |
62 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA3-1
|
KS6A3_HUMAN
|
5D9KB
|
2.55 |
Inactive |
DFGout‑None |
in-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
584 |
Type1 |
62 - 359 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
AGC
|
RPS6KA4-1
|
KS6A4_HUMAN
|
AF-O75676-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
25 - 309 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-4 |
|
AGC
|
RPS6KA4-1
|
KS6A4_HUMAN
|
AF-O75676-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
25 - 309 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-4 |
|
AGC
|
RPS6KA5-1
|
KS6A5_HUMAN
|
AF-O75582-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 326 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
AGC
|
RPS6KA5-1
|
KS6A5_HUMAN
|
AF-O75582-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 326 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
AGC
|
RPS6KA5-1
|
KS6A5_HUMAN
|
1VZOA
|
1.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
No_ligand |
No_ligand |
24 - 345 |
0 |
None |
S212D |
Ribosomal protein S6 kinase alpha-5 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
AF-Q9UK32-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
65 - 338 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
AF-Q9UK32-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
65 - 338 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G77A
|
2.499 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP,
ANP
|
Allosteric,
ATPlike
|
51 - 349 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G77B
|
2.499 |
Inactive |
DFGin‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP,
ANP
|
Allosteric,
ATPlike
|
51 - 349 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G76B
|
3.0 |
Inactive |
DFGinter‑None |
none-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ANP |
ATPlike |
51 - 349 |
0 |
SEP232 |
None |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G78A
|
2.5 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
ANP |
ATPlike |
51 - 349 |
0 |
None |
S232E |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G78B
|
2.5 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
ANP |
ATPlike |
51 - 349 |
0 |
None |
S232E |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KA6-1
|
KS6A6_HUMAN
|
6G76A
|
3.0 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP,
ANP
|
ATPlike,
Allosteric
|
51 - 349 |
0 |
SEP232 |
None |
Ribosomal protein S6 kinase alpha-6 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4RLPA
|
2.79 |
Inactive |
DFGin‑ABAminus |
none-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
72B |
Type1 |
85 - 372 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L3JA
|
2.1 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
85 - 375 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L3LA
|
2.1 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
85 - 375 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N91A
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1RJ |
Type1 |
85 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N91B
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-in |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
1RJ |
Type1 |
85 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N93A
|
2.74 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
1SK |
Type1 |
87 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
7N93B
|
2.74 |
Inactive |
DFGin‑ABAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
1SK |
Type1 |
85 - 418 |
0 |
TPO390,SEP394 |
T412E |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A62A
|
2.35 |
Inactive |
DFGin‑ABAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
STU |
Type1 |
85 - 372 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WE4A
|
1.995 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
85 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF5A
|
2.099 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
FZ8 |
Type1 |
85 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF6A
|
2.031 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
FZ9 |
Type1 |
85 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L45A
|
2.9 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
5FI |
Type1 |
81 - 417 |
0 |
None |
T412E |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L42A
|
2.8 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
5FI |
Type1 |
84 - 417 |
0 |
None |
S403E,A404E,N405Q,Q406E,V407M,L409R,G410D,T412E,V414I,P416D,S417W |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L46A
|
3.01 |
Inactive |
DFGin‑ABAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
80 - 417 |
0 |
TPO412 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
AF-P23443-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
83 - 360 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
AF-P23443-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
83 - 360 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF8A
|
1.975 |
Inactive |
DFGin‑BLAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
F76 |
Type1 |
85 - 372 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF9A
|
2.035 |
Inactive |
DFGin‑BLAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
FS7 |
Type1 |
85 - 372 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L43A
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
5FI |
Type1 |
81 - 417 |
0 |
None |
T412A |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4L44A
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
5FI |
Type1 |
81 - 417 |
0 |
None |
T412A |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4RLOA
|
2.527 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
3T3 |
Type1 |
85 - 371 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A60A
|
2.8 |
Inactive |
DFGin‑None |
in-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
STU |
Type1 |
85 - 371 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A61A
|
3.43 |
Inactive |
DFGin‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
STU |
Type1 |
87 - 371 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3WF7A
|
1.85 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
FS9 |
Type1 |
83 - 374 |
0 |
TPO252 |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
4RLOB
|
2.527 |
Inactive |
None‑None |
none-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
STU |
Type1 |
85 - 372 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB1
|
KS6B1_HUMAN
|
3A60B
|
2.8 |
Inactive |
None‑None |
none-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
STU |
Type1 |
85 - 372 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-1 |
|
AGC
|
RPS6KB2
|
KS6B2_HUMAN
|
AF-Q9UBS0-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
59 - 336 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-2 |
|
AGC
|
RPS6KB2
|
KS6B2_HUMAN
|
AF-Q9UBS0-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
59 - 336 |
0 |
None |
None |
Ribosomal protein S6 kinase beta-2 |
|
AGC
|
RSKR
|
KS6R_HUMAN
|
AF-Q96LW2-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
99 - 367 |
0 |
None |
None |
Ribosomal protein S6 kinase-related protein |
|
AGC
|
RSKR
|
KS6R_HUMAN
|
AF-Q96LW2-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
99 - 367 |
0 |
None |
None |
Ribosomal protein S6 kinase-related protein |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
AF-O00141-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
90 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk1 |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
AF-O00141-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
90 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk1 |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
2R5TA
|
1.9 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
ANP |
ATPlike |
82 - 378 |
0 |
None |
S74A,S78A,S397A,S401A |
Serine/threonine-protein kinase Sgk1 |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
3HDMA
|
2.6 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
MMG |
Type1 |
81 - 378 |
0 |
None |
S74A,S78A,S397A,S401A |
Serine/threonine-protein kinase Sgk1 |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
3HDNA
|
3.1 |
Inactive |
DFGinter‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
GMG |
Type1 |
82 - 374 |
0 |
None |
S74A,S78A,S397A,S401A |
Serine/threonine-protein kinase Sgk1 |
|
AGC
|
SGK1
|
SGK1_HUMAN
|
7PUEA
|
2.506 |
Inactive |
DFGout‑None |
none-none |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
86H |
Type1 |
82 - 376 |
0 |
None |
R192A,S422D |
Serine/threonine-protein kinase Sgk1 |
|
AGC
|
SGK2
|
SGK2_HUMAN
|
AF-Q9HBY8-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 300 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk2 |
|
AGC
|
SGK2
|
SGK2_HUMAN
|
AF-Q9HBY8-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
27 - 300 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk2 |
|
AGC
|
SGK3
|
SGK3_HUMAN
|
AF-Q96BR1-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
154 - 427 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk3 |
|
AGC
|
SGK3
|
SGK3_HUMAN
|
AF-Q96BR1-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
154 - 427 |
0 |
None |
None |
Serine/threonine-protein kinase Sgk3 |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
AF-Q8WU08-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 289 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
AF-Q8WU08-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 289 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4A
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4B
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4C
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4D
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4E
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 372 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32A
|
ST32A_HUMAN
|
4FR4F
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
14 - 373 |
0 |
None |
None |
Serine/threonine-protein kinase 32A |
|
AGC
|
STK32B
|
ST32B_HUMAN
|
AF-Q9NY57-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 291 |
0 |
None |
None |
Serine/threonine-protein kinase 32B |
|
AGC
|
STK32B
|
ST32B_HUMAN
|
AF-Q9NY57-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 291 |
0 |
None |
None |
Serine/threonine-protein kinase 32B |
|
AGC
|
STK32C
|
ST32C_HUMAN
|
AF-Q86UX6-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iiii |
No_ligand |
No_ligand |
85 - 361 |
0 |
None |
None |
Serine/threonine-protein kinase 32C |
|
AGC
|
STK32C
|
ST32C_HUMAN
|
AF-Q86UX6-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
85 - 361 |
0 |
None |
None |
Serine/threonine-protein kinase 32C |
|
AGC
|
STK38
|
STK38_HUMAN
|
AF-Q15208-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
81 - 390 |
0 |
None |
None |
Serine/threonine-protein kinase 38 |
|
AGC
|
STK38
|
STK38_HUMAN
|
AF-Q15208-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
81 - 390 |
0 |
None |
None |
Serine/threonine-protein kinase 38 |
|
AGC
|
STK38
|
STK38_HUMAN
|
6BXIA
|
2.2 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ANP |
ATPlike |
82 - 414 |
0 |
None |
None |
Serine/threonine-protein kinase 38 |
|
AGC
|
STK38
|
STK38_HUMAN
|
6BXIB
|
2.2 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ANP |
ATPlike |
83 - 414 |
0 |
None |
None |
Serine/threonine-protein kinase 38 |
|
AGC
|
STK38L
|
ST38L_HUMAN
|
AF-Q9Y2H1-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
82 - 391 |
0 |
None |
None |
Serine/threonine-protein kinase 38-like |
|
AGC
|
STK38L
|
ST38L_HUMAN
|
AF-Q9Y2H1-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
82 - 391 |
0 |
None |
None |
Serine/threonine-protein kinase 38-like |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4C3PD
|
2.69 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_nooo |
ACP |
ATPlike |
125 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8GUWA
|
2.7 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ADP |
ATPlike |
506 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8GUWB
|
2.7 |
Inactive |
DFGin‑ABAminus |
out-out |
none-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
ADP |
ATPlike |
507 - 390 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8GUWC
|
2.7 |
Inactive |
DFGin‑ABAminus |
out-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
ADP |
ATPlike |
506 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DPVA
|
2.285 |
Inactive |
DFGin‑ABAminus |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
5DN,
SKE
|
Allosteric,
Type1
|
127 - 389 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DR6A
|
2.534 |
Inactive |
DFGin‑ABAminus |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
5E1,
SKE
|
Allosteric,
Type1
|
127 - 390 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WTWA
|
3.302 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
ZZL |
Type1 |
128 - 389 |
0 |
None |
L215R,T217E,R220K |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3E5AA
|
2.3 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VX6 |
Type1 |
125 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2NP8A
|
2.25 |
Inactive |
DFGin‑ABAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
CC3 |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4BYIA
|
2.6 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
FH3 |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ONEA
|
2.6 |
Inactive |
DFGin‑ABAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nooo |
9YQ |
Type1 |
127 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DT0A
|
2.15 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
SKE |
Type1 |
127 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UODA
|
2.5 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
0C3 |
Type1 |
124 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UP2A
|
2.3 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
0C8 |
Type1 |
124 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DEAA
|
2.45 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
NHI |
Type1 |
124 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5AAFA
|
2.78 |
Inactive |
DFGin‑ABAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
NL4 |
Type1 |
126 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5AAGA
|
2.85 |
Inactive |
DFGin‑ABAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
6F2 |
Type1 |
127 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6GRAA
|
2.6 |
Inactive |
DFGin‑ABAminus |
out-out |
none-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
F8Z |
Type1.5_Front |
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4BN1A
|
2.499 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
126 - 388 |
0 |
TPO287,TPO288 |
V174M |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
1MQ4A
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DNRA
|
1.95 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
ATP |
ATPlike |
126 - 390 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DT3A
|
2.33 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ATP |
ATPlike |
127 - 390 |
0 |
TPO287 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
1OL5A
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
123 - 388 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
1OL7A
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
127 - 390 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5G15A
|
2.06 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ACP |
ATPlike |
126 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2DWBA
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ANP |
ATPlike |
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6CPFA
|
2.3 |
Inactive |
DFGin‑BLAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ACP |
ATPlike |
128 - 392 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPGA
|
2.64 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
7 - 389 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DRDA
|
2.13 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
ATP |
ATPlike |
127 - 390 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DEEA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
124 - 394 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPIA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
ANP |
ATPlike |
104 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5LXMA
|
2.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
126 - 392 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4CEGA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
127 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5G1XA
|
1.72 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
126 - 389 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
1OL6A
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-out |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
ATP |
ATPlike |
128 - 388 |
0 |
None |
D274N |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPLA
|
1.86 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ANP,
R7D
|
ATPlike,
Allosteric
|
7 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPLB
|
1.86 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ANP,
R7D
|
ATPlike,
Allosteric
|
7 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPMA
|
1.58 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
AMP,
R74
|
ATPlike,
Allosteric
|
7 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPMB
|
1.58 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
AMP,
R74
|
ATPlike,
Allosteric
|
7 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORLA
|
1.69 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A4W
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORNA
|
2.19 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5E
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OROA
|
2.12 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5H
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORPA
|
2.19 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5K
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORRA
|
2.09 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5Q
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORSA
|
1.98 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5W
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORTA
|
2.56 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A5Z
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORVA
|
1.88 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A65
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORWA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A6E
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORXA
|
1.88 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A6H
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORYA
|
1.99 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
AY4
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ORZA
|
1.92 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A6W
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS0A
|
1.74 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A6Z
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS1A
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A7H
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS2A
|
1.92 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
ADP,
A7K
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS3A
|
1.81 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A7N
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS4A
|
1.88 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A8H
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS6A
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A7Q
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OSEA
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A98
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OSFA
|
1.89 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A9E
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OSDA
|
1.99 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A9B
|
ATPlike,
Allosteric
|
125 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OS5A
|
1.74 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
A8K
|
ATPlike,
Allosteric
|
125 - 392 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6R49A
|
2.209 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ADP,
JSB
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6R4AA
|
1.937 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
JRT
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6R4BA
|
2.15 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
JSN
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6R4CA
|
2.04 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
JRQ
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6R4DA
|
2.009 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP,
JRW
|
ATPlike,
Allosteric
|
127 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
7ZTLA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP,
BCN
|
ATPlike,
Allosteric
|
126 - 389 |
0 |
TPO288 |
C290A,K339C,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8OF5A
|
1.97 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ADP,
MPO
|
ATPlike,
Allosteric
|
126 - 390 |
0 |
None |
C290A,N332A,Q335A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C14A
|
1.93 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
ADP,
T5L,
T0L
|
ATPlike,
Allosteric,
Allosteric
|
126 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C15A
|
2.41 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ADP,
T4C,
T5L
|
ATPlike,
Allosteric,
Allosteric
|
126 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1FA
|
1.924 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ADP,
T5L,
T2O
|
ATPlike,
Allosteric,
Allosteric
|
126 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1IA
|
2.81 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ADP,
T1L,
T5L
|
ATPlike,
Allosteric,
Allosteric
|
126 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DN3A
|
2.05 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
5DN,
ATP
|
Allosteric,
ATPlike
|
125 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1EA
|
2.798 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
T0X,
ATP
|
Allosteric,
ATPlike
|
127 - 388 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DT4A
|
2.86 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
5DN,
ATP
|
Allosteric,
ATPlike
|
127 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1MA
|
2.84 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
T4X,
ADP
|
Allosteric,
ATPlike
|
127 - 389 |
0 |
TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DOSA
|
2.98 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
5DN,
ATP
|
Allosteric,
ATPlike
|
127 - 390 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DR2A
|
2.46 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
5E1,
ATP
|
Allosteric,
ATPlike
|
128 - 390 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1DA
|
2.115 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
T2F,
ADP,
T5L
|
Allosteric,
ATPlike,
Allosteric
|
127 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1GA
|
1.96 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
T3I,
ADP,
T5L
|
Allosteric,
ATPlike,
Allosteric
|
127 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1HA
|
2.233 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
T3U,
ADP,
T5L
|
Allosteric,
ATPlike,
Allosteric
|
127 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8C1KA
|
2.43 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
T4O,
ADP,
T5L
|
Allosteric,
ATPlike,
Allosteric
|
127 - 388 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8SSPA
|
2.6 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PDO,
627
|
Allosteric,
Type1
|
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
AF-O14965-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
125 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
AF-O14965-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
125 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6CPEA
|
2.45 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4J8NA
|
3.135 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iioo |
No_ligand |
No_ligand |
125 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4J8NB
|
3.135 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
No_ligand |
No_ligand |
125 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4J8NC
|
3.135 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
No_ligand |
No_ligand |
125 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4J8ND
|
3.135 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
No_ligand |
No_ligand |
126 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8JG8A
|
2.9 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
C74 |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3HA6A
|
2.36 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2JZ |
Type1 |
125 - 388 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3MYGA
|
2.4 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
EML |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3VAPA
|
2.66 |
Inactive |
DFGin‑BLAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
0FY |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2W1CA
|
3.24 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
L0C |
Type1 |
127 - 389 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2W1DA
|
2.97 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
L0D |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2W1EA
|
2.93 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
L0E |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2W1FA
|
2.85 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
L0F |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2W1GA
|
2.71 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
L0G |
Type1 |
127 - 389 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ZANA
|
2.85 |
Inactive |
DFGin‑BLAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
9A6 |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4O0SA
|
2.5 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADN |
Type1 |
126 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2XNGA
|
2.605 |
Inactive |
DFGin‑BLAminus |
in-out |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
A0H |
Type1 |
127 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4JAJA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
XU1 |
Type1 |
125 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2X6DA
|
2.796 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
X6D |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2X6EA
|
3.35 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
YM4 |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4ZS0A
|
3.0 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
4QV |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6I2UA
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
COA |
Type1 |
127 - 391 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2XRUA
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
400 |
Type1 |
126 - 389 |
0 |
None |
T288E |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UO4A
|
2.45 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
0C0 |
Type1 |
124 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UO5A
|
2.701 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
0BX |
Type1 |
124 - 390 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UP7A
|
3.05 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
0C9 |
Type1 |
124 - 387 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DEBA
|
3.05 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
NHJ |
Type1 |
125 - 388 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DEDA
|
3.05 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
NHU |
Type1 |
124 - 388 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4JBOA
|
2.493 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
WPH |
Type1 |
126 - 391 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3NRMA
|
3.05 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
NRM |
Type1 |
126 - 388 |
0 |
None |
T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3R21A
|
2.9 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nooo |
D36 |
Type1 |
127 - 389 |
0 |
None |
T287D,T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5AADA
|
3.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5GX |
Type1 |
127 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2XNEA
|
2.8 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
ASH |
Type1 |
127 - 388 |
0 |
None |
D274N |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5DR9A
|
2.47 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
SKE,
5E2
|
Type1,
Allosteric
|
127 - 390 |
0 |
None |
T287A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3M11A
|
2.75 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
AKI |
Type1.5_Front |
126 - 391 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4JBPA
|
2.45 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
YPH |
Type1.5_Front |
126 - 390 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4J8MA
|
1.853 |
Inactive |
DFGin‑BLAplus |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
CJ5 |
Type1 |
125 - 390 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8PR7D
|
2.76 |
Inactive |
DFGin‑BLBminus |
out-none |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnoo |
ADP |
ATPlike |
126 - 388 |
0 |
None |
D274N,C290A,N332A,Q335A,T347A,D350A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4C3PA
|
2.69 |
Inactive |
DFGin‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
ACP |
ATPlike |
125 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2C6DA
|
2.2 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ANP |
ATPlike |
126 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5ODTA
|
2.021 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnoo |
ADP |
ATPlike |
126 - 392 |
0 |
None |
D274N,C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OBJA
|
2.901 |
Inactive |
DFGin‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
ATP,
9QK
|
ATPlike,
Allosteric
|
127 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9GUCA
|
2.1 |
Inactive |
DFGin‑None |
out-none |
none-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
ADP,
AMP
|
ATPlike,
Allosteric
|
124 - 391 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8JF4A
|
2.893 |
Inactive |
DFGin‑None |
out-none |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
C0N |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8JMXA
|
2.95 |
Inactive |
DFGin‑None |
out-none |
none-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnno |
E47 |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
7AYIA
|
2.86 |
Inactive |
DFGin‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
S9K |
Type1 |
125 - 392 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2J4ZB
|
2.0 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
626 |
Type1 |
126 - 395 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4O0WA
|
2.6 |
Inactive |
DFGin‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nioo |
ADN |
Type1 |
125 - 391 |
0 |
None |
H254Y |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H0ZA
|
2.92 |
Inactive |
DFGin‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
45B |
Type1 |
128 - 388 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DHFA
|
2.8 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnoo |
0K6 |
Type1 |
128 - 389 |
0 |
None |
T287D,T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4DHFB
|
2.8 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_nnoo |
0K6 |
Type1 |
128 - 389 |
0 |
None |
T287D,T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4PRJA
|
2.8 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnoo |
2VU |
Type1 |
125 - 388 |
0 |
None |
K124A,Q154N,A203S,R251K,T287A,T288A,E336D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5AAEA
|
3.11 |
Inactive |
DFGin‑None |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
7HD |
Type1 |
126 - 388 |
0 |
None |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4O0UA
|
2.6 |
Inactive |
DFGin‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
ADN |
Type1 |
126 - 391 |
0 |
None |
H254R |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4UZDA
|
3.2 |
Inactive |
DFGin‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
QMN |
Type1.5_Front |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4UZDB
|
3.2 |
Inactive |
DFGin‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
QMN |
Type1.5_Front |
125 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4UYNA
|
1.9 |
Inactive |
DFGin‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
Y3M |
Type1.5_Front |
125 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4C3RA
|
2.79 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ACP |
ATPlike |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6C83B
|
2.55 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
ACP |
ATPlike |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5L8JA
|
1.68 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
ADP |
ATPlike |
126 - 391 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5L8KA
|
1.79 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ADP |
ATPlike |
126 - 392 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5L8LA
|
1.67 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
ADP |
ATPlike |
126 - 389 |
0 |
TPO288 |
C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8PR7A
|
2.76 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
ADP |
ATPlike |
124 - 389 |
0 |
None |
D274N,C290A,N332A,Q335A,T347A,D350A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6XKAA
|
2.65 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
No_ligand |
No_ligand |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WTVA
|
2.4 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
ZZL |
Type1 |
125 - 389 |
0 |
TPO287,TPO288 |
L215R,T217E,R220K |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WTVB
|
2.4 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ZZL |
Type1 |
126 - 389 |
0 |
TPO287,TPO288 |
L215R,T217E,R220K |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WTVC
|
2.4 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ZZL |
Type1 |
126 - 389 |
0 |
TPO287,TPO288 |
L215R,T217E,R220K |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WTVD
|
2.4 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
ZZL |
Type1 |
125 - 389 |
0 |
TPO287,TPO288 |
L215R,T217E,R220K |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5EW9A
|
2.181 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
5VC |
Type1 |
127 - 390 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6C2RA
|
1.96 |
Inactive |
DFGinter‑None |
out-none |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
EG7 |
Type1 |
128 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6C2TA
|
1.73 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
EGJ |
Type1 |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W16A
|
2.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnno |
P9J |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2J50A
|
3.0 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
627 |
Type1 |
128 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2J50B
|
3.0 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
627 |
Type1 |
128 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4ZTRA
|
2.85 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
4RJ |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6Z4YA
|
2.25 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
Q7Q |
Type1 |
124 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6CPGA
|
2.8 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnoo |
35R |
Type1 |
127 - 387 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6CPGD
|
2.8 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nooo |
35R |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8SSOA
|
1.97 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nooo |
627 |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
8SSOD
|
1.97 |
Inactive |
DFGinter‑None |
out-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
627 |
Type1 |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
1MUOA
|
2.9 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nooo |
ADN |
Type1 |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2J4ZA
|
2.0 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioo |
626 |
Type1 |
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UNZA
|
2.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0BZ |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UNZB
|
2.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0BZ |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UO6A
|
2.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0BY |
Type1 |
126 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UO6B
|
2.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0BY |
Type1 |
126 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOHA
|
2.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C4 |
Type1 |
126 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOHB
|
2.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C4 |
Type1 |
126 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOJA
|
2.9 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C5 |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOJB
|
2.9 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C5 |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOKA
|
2.951 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C6 |
Type1 |
125 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOKB
|
2.951 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C6 |
Type1 |
125 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOLA
|
2.4 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C7 |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3UOLB
|
2.4 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
0C7 |
Type1 |
127 - 389 |
0 |
None |
T287D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3FDNA
|
1.9 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
MMH |
Type1 |
126 - 394 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3K5UA
|
2.35 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
PFQ |
Type1 |
126 - 394 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4JBQA
|
2.3 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
VX6 |
Type1 |
126 - 391 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3LAUA
|
2.1 |
Inactive |
DFGinter‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
OFI |
Type1 |
125 - 391 |
0 |
None |
T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4UZHA
|
2.0 |
Inactive |
DFGinter‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
JVE |
Type1 |
125 - 392 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H0YA
|
2.5 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
48B |
Type1 |
126 - 388 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H10A
|
2.2 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
97B |
Type1 |
124 - 391 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H10B
|
2.2 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
97B |
Type1 |
125 - 391 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H10D
|
2.2 |
Inactive |
DFGinter‑None |
out-out |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
97B |
Type1 |
126 - 388 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3P9JA
|
2.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
P9J |
Type1 |
126 - 388 |
0 |
None |
T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W10A
|
2.7 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
RO9 |
Type1 |
126 - 388 |
0 |
None |
T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3R22A
|
2.9 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
D37 |
Type1 |
126 - 389 |
0 |
None |
T287D,T288D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9KDSA
|
2.5 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
A1EFT |
Type1 |
126 - 391 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCA
|
2.6 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
127 - 394 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCB
|
2.6 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
125 - 394 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCC
|
2.6 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
125 - 393 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCD
|
2.6 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
127 - 394 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCE
|
2.6 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
127 - 394 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2BMCF
|
2.6 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
MPY |
Type1 |
126 - 394 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
7FICA
|
2.32 |
Inactive |
DFGinter‑None |
out-none |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
5YZ |
Type1 |
127 - 391 |
0 |
None |
C290A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9BZGA
|
1.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
OG0 |
Type1 |
127 - 388 |
0 |
TPO288 |
C290A,C393S |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9BZLB
|
1.81 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
OGR |
Type1 |
127 - 388 |
0 |
TPO288 |
C290A,C393S |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
9KS6A
|
2.75 |
Inactive |
DFGinter‑None |
out-na |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
A1EG1 |
Type1 |
127 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4ZTQA
|
2.8 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
4RM |
Type1.5_Back |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4ZTSA
|
2.9 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
4RK |
Type1.5_Back |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3EFWA
|
2.29 |
Inactive |
DFGinter‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
AK8 |
Type1.5_Front |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3EFWB
|
2.29 |
Inactive |
DFGinter‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
AK8 |
Type1.5_Front |
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3O50A
|
2.0 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
LJE |
Type1.5_Front |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3O50B
|
2.0 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
LJE |
Type1.5_Front |
126 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6HJJA
|
2.13 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
G7T |
Type1.5_Front |
127 - 393 |
0 |
None |
L210C,C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2C6EA
|
2.1 |
Inactive |
DFGout‑BBAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
HPM |
Type1.5_Back |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPJA
|
2.1 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
ANP |
ATPlike |
104 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6VPHA
|
2.14 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
ANP |
ATPlike |
7 - 389 |
0 |
TPO287,TPO288 |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4JAIA
|
3.2 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanno |
APEdist_nnnn |
XU2 |
Type1 |
126 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
7AYHA
|
2.8 |
Inactive |
DFGout‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
S9H |
Type1 |
125 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
7O2VA
|
3.1 |
Inactive |
DFGout‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
V0K |
Type1 |
117 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3O51A
|
3.2 |
Inactive |
DFGout‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
LJF |
Type1.5_Front |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6HJKA
|
2.4 |
Inactive |
DFGout‑None |
out-none |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
G7W |
Type1.5_Front |
127 - 391 |
0 |
None |
L210C,C290A,C393A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
6C83A
|
2.55 |
Inactive |
None‑None |
out-none |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
ACP |
ATPlike |
127 - 389 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2WQEA
|
2.5 |
Inactive |
None‑None |
out-none |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
ADP,
ADP,
ADP
|
ATPlike,
ATPlike,
ATPlike
|
127 - 388 |
0 |
None |
S155R |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
5OBRA
|
2.62 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
9QT,
SKE
|
Allosteric,
Type1
|
126 - 390 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W2CC
|
2.45 |
Inactive |
None‑None |
out-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
N15 |
Type1 |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W2CE
|
2.45 |
Inactive |
None‑None |
out-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
N15 |
Type1 |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2X81A
|
2.91 |
Inactive |
None‑None |
out-none |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
ZZL |
Type1 |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W18A
|
2.5 |
Inactive |
None‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
N13 |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W18B
|
2.5 |
Inactive |
None‑None |
none-none |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
N13 |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4B0GA
|
2.5 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
VEK |
Type1 |
126 - 391 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
4BYJA
|
2.75 |
Inactive |
None‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
FH5 |
Type1 |
126 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H0ZB
|
2.92 |
Inactive |
None‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
45B |
Type1 |
126 - 388 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3H0ZC
|
2.92 |
Inactive |
None‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
45B |
Type1 |
126 - 388 |
0 |
None |
K124A,T287A,T288A |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3COHA
|
2.7 |
Inactive |
None‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
83H |
Type1 |
128 - 388 |
0 |
None |
K124A,Q154N,A203S,R251K,T287A,T288A,E336D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3COHB
|
2.7 |
Inactive |
None‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
83H |
Type1 |
128 - 388 |
0 |
None |
K124A,Q154N,A203S,R251K,T287A,T288A,E336D |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3QBNA
|
3.5 |
Inactive |
None‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
E9Z |
Type1 |
126 - 388 |
0 |
None |
V279C,C290S,C393S |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W2CA
|
2.45 |
Inactive |
None‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
N15 |
Type1.5_Back |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
3W2CG
|
2.45 |
Inactive |
None‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
N15 |
Type1.5_Back |
128 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKA
|
AURKA_HUMAN
|
2C6EB
|
2.1 |
Inactive |
None‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnni |
HPM |
Type1.5_Front |
127 - 388 |
0 |
None |
None |
Aurora kinase A |
|
CAMK
|
AURKB
|
AURKB_HUMAN
|
AF-Q96GD4-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
69 - 335 |
0 |
None |
None |
Aurora kinase B |
|
CAMK
|
AURKB
|
AURKB_HUMAN
|
AF-Q96GD4-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
69 - 335 |
0 |
None |
None |
Aurora kinase B |
|
CAMK
|
AURKB
|
AURKB_HUMAN
|
4AF3A
|
2.75 |
Inactive |
DFGinter‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
VX6 |
Type1 |
70 - 338 |
0 |
None |
None |
Aurora kinase B |
|
CAMK
|
AURKC
|
AURKC_HUMAN
|
9ESAAAA
|
2.8 |
Inactive |
DFGin‑ABAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
32 - 306 |
0 |
None |
R195A,R196A,K197A |
Aurora kinase C |
|
CAMK
|
AURKC
|
AURKC_HUMAN
|
9ESABBB
|
2.8 |
Inactive |
DFGin‑ABAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
No_ligand |
No_ligand |
32 - 306 |
0 |
None |
R195A,R196A,K197A |
Aurora kinase C |
|
CAMK
|
AURKC
|
AURKC_HUMAN
|
6GR9A
|
2.25 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VX6 |
Type1 |
37 - 305 |
0 |
TPO39,TPO198 |
None |
Aurora kinase C |
|
CAMK
|
AURKC
|
AURKC_HUMAN
|
6GR8A
|
1.75 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
F8Z |
Type1.5_Front |
36 - 303 |
0 |
TPO39,TPO198 |
None |
Aurora kinase C |
|
CAMK
|
AURKC
|
AURKC_HUMAN
|
AF-Q9UQB9-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
35 - 301 |
0 |
None |
None |
Aurora kinase C |
|
CAMK
|
AURKC
|
AURKC_HUMAN
|
AF-Q9UQB9-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
35 - 301 |
0 |
None |
None |
Aurora kinase C |
|
CAMK
|
BRSK1
|
BRSK1_HUMAN
|
AF-Q8TDC3-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
26 - 293 |
0 |
None |
None |
Serine/threonine-protein kinase BRSK1 |
|
CAMK
|
BRSK1
|
BRSK1_HUMAN
|
AF-Q8TDC3-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
26 - 293 |
0 |
None |
None |
Serine/threonine-protein kinase BRSK1 |
|
CAMK
|
BRSK2
|
BRSK2_HUMAN
|
AF-Q8IWQ3-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
11 - 278 |
0 |
None |
None |
Serine/threonine-protein kinase BRSK2 |
|
CAMK
|
BRSK2
|
BRSK2_HUMAN
|
AF-Q8IWQ3-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
11 - 278 |
0 |
None |
None |
Serine/threonine-protein kinase BRSK2 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
4FG7A
|
2.7 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
ATP |
ATPlike |
9 - 277 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
AF-Q14012-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 284 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
AF-Q14012-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 284 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
4FG9A
|
2.4 |
Inactive |
DFGinter‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ATP |
ATPlike |
10 - 314 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
4FG9B
|
2.4 |
Inactive |
DFGinter‑None |
out-none |
none-out |
nonTYR |
APEdihe_aaini |
APEdist_nnno |
ATP |
ATPlike |
14 - 314 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
4FGBA
|
2.6 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
No_ligand |
No_ligand |
10 - 299 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
4FG8A
|
2.2 |
Inactive |
None‑None |
out-none |
none-out |
nonTYR |
APEdihe_aanno |
APEdist_nnnn |
ATP |
ATPlike |
10 - 299 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1
|
KCC1A_HUMAN
|
4FG8B
|
2.2 |
Inactive |
None‑None |
out-none |
none-out |
nonTYR |
APEdihe_aaino |
APEdist_nnno |
ATP |
ATPlike |
14 - 299 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1 |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
AF-Q8IU85-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 287 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
AF-Q8IU85-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 287 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
6QP5A
|
1.9 |
Inactive |
DFGin‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
13 - 302 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
6T28AAA
|
1.55 |
Inactive |
DFGin‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
M92 |
Type1 |
12 - 302 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
8BFSA
|
1.95 |
Inactive |
DFGin‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
QNR |
Type1 |
12 - 302 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
8BFMA
|
1.7 |
Inactive |
DFGin‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
QI6,
QI6
|
Type1,
Type3
|
12 - 301 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
6T6FA
|
1.97 |
Inactive |
DFGinter‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MMW |
Type1 |
12 - 329 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
6T6FB
|
1.97 |
Inactive |
DFGinter‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MMW |
Type1 |
12 - 329 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
6T29AAA
|
1.484 |
Inactive |
DFGinter‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
M8Z |
Type1 |
12 - 302 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
2JC6A
|
2.3 |
Inactive |
None‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
QPP |
Type1 |
11 - 313 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1D
|
KCC1D_HUMAN
|
2JC6C
|
2.3 |
Inactive |
None‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
QPP |
Type1 |
11 - 313 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1D |
|
CAMK
|
CAMK1G
|
KCC1G_HUMAN
|
AF-Q96NX5-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 285 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1G |
|
CAMK
|
CAMK1G
|
KCC1G_HUMAN
|
AF-Q96NX5-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 285 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1G |
|
CAMK
|
CAMK1G
|
KCC1G_HUMAN
|
2JAMA
|
1.7 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
J60 |
Type1 |
18 - 302 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1G |
|
CAMK
|
CAMK1G
|
KCC1G_HUMAN
|
2JAMB
|
1.7 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
J60 |
Type1 |
16 - 301 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1G |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UJSA
|
2.75 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
7 - 274 |
0 |
None |
Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UIRA
|
3.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UIRB
|
3.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
7 - 273 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UJPA
|
2.56 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UJPB
|
2.56 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
7 - 273 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UJTA
|
2.1 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
AF-Q9UQM7-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 279 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
AF-Q9UQM7-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 279 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UJRA
|
1.95 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 274 |
0 |
None |
Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
6VZKA
|
2.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
6X5QA
|
2.14 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
8 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7KL1A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7KL1B
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7KL2A
|
2.56 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UIQA
|
3.11 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UIQB
|
3.11 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
8 - 273 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UISA
|
2.58 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 273 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
2VZ6A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
FEF |
Type1 |
9 - 299 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
2VZ6B
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
FEF |
Type1 |
9 - 300 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7KL0A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UZD |
Type1 |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7KL0B
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UZD |
Type1 |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UJQA
|
2.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UZD |
Type1 |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
7UJQB
|
2.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UZD |
Type1 |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
6X5GA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BCN |
Type1.5_Back |
7 - 274 |
0 |
None |
D135N,Q223K |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
6W4OO
|
4.8 |
Inactive |
DFGinter‑None |
in-na |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 301 |
0 |
None |
K42M |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
6W4PH
|
6.6 |
Inactive |
DFGinter‑None |
in-na |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 301 |
0 |
None |
K42M |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2A
|
KCC2A_HUMAN
|
3SOAA
|
3.55 |
Inactive |
DFGinter‑None |
in-na |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DB8 |
Type1 |
7 - 474 |
0 |
None |
K42M,D135N,T306V |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
|
CAMK
|
CAMK2B
|
KCC2B_HUMAN
|
AF-Q13554-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6 - 280 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
|
CAMK
|
CAMK2B
|
KCC2B_HUMAN
|
AF-Q13554-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6 - 280 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
|
CAMK
|
CAMK2B
|
KCC2B_HUMAN
|
3BHHC
|
2.4 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
11 - 300 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
|
CAMK
|
CAMK2B
|
KCC2B_HUMAN
|
3BHHD
|
2.4 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
11 - 301 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
|
CAMK
|
CAMK2B
|
KCC2B_HUMAN
|
3BHHA
|
2.4 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5CP |
Type1 |
11 - 301 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
|
CAMK
|
CAMK2B
|
KCC2B_HUMAN
|
3BHHB
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5CP |
Type1 |
11 - 301 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
AF-Q13557-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6 - 280 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
AF-Q13557-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6 - 280 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK2D
|
D6R938_HUMAN
|
8USOA
|
2.3 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 475 |
0 |
None |
D364C |
calcium/calmodulin-dependent protein kinase |
|
CAMK
|
CAMK2D
|
D6R938_HUMAN
|
8USOB
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6 - 475 |
0 |
None |
D364C |
calcium/calmodulin-dependent protein kinase |
|
CAMK
|
CAMK2D
|
D6R938_HUMAN
|
8USOC
|
2.3 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 477 |
0 |
None |
D364C |
calcium/calmodulin-dependent protein kinase |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
9BLHA
|
2.35 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6ZZ |
Type1 |
11 - 301 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
9BLHB
|
2.35 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6ZZ |
Type1 |
11 - 298 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
2VN9A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVD |
Type1 |
10 - 309 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
2VN9B
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GVD |
Type1 |
10 - 309 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
5VLOA
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9EJ |
Type1 |
8 - 300 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
5VLOB
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9EJ |
Type1 |
7 - 299 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
6AYWA
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C2V |
Type1 |
8 - 300 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
6AYWB
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C2V |
Type1 |
7 - 299 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK2D
|
KCC2D_HUMAN
|
2WELA
|
1.9 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
K88 |
Type1 |
10 - 316 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
|
CAMK
|
CAMK2G
|
KCC2G_HUMAN
|
AF-Q13555-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6 - 280 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
|
CAMK
|
CAMK2G
|
KCC2G_HUMAN
|
AF-Q13555-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6 - 280 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
|
CAMK
|
CAMK2G
|
KCC2G_HUMAN
|
2V7OA
|
2.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DRN |
Type1 |
3 - 302 |
0 |
SEP3 |
None |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
|
CAMK
|
CAMK4
|
KCC4_HUMAN
|
AF-Q16566-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
38 - 308 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type IV |
|
CAMK
|
CAMK4
|
KCC4_HUMAN
|
AF-Q16566-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
38 - 308 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type IV |
|
CAMK
|
CAMK4
|
KCC4_HUMAN
|
2W4OA
|
2.17 |
Inactive |
None‑None |
none-none |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
DKI |
Type1 |
34 - 337 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type IV |
|
CAMK
|
CAMKK1
|
KKCC1_HUMAN
|
AF-Q8N5S9-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
120 - 417 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 1 |
|
CAMK
|
CAMKK1
|
KKCC1_HUMAN
|
AF-Q8N5S9-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
120 - 417 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 1 |
|
CAMK
|
CAMKK1
|
KKCC1_HUMAN
|
6CCFA
|
2.1 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H1N |
Type1 |
124 - 411 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 1 |
|
CAMK
|
CAMKK1
|
KKCC1_HUMAN
|
6CCFB
|
2.1 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H1N |
Type1 |
124 - 411 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 1 |
|
CAMK
|
CAMKK1
|
KKCC1_HUMAN
|
6CD6A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DXV |
Type1 |
125 - 411 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 1 |
|
CAMK
|
CAMKK1
|
KKCC1_HUMAN
|
6CD6B
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DXV |
Type1 |
124 - 411 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 1 |
|
CAMK
|
CAMKK1
|
KKCC1_HUMAN
|
6CD6C
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DXV |
Type1 |
124 - 411 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 1 |
|
CAMK
|
CAMKK1
|
KKCC1_HUMAN
|
6CD6D
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DXV |
Type1 |
124 - 411 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 1 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
AF-Q96RR4-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
157 - 454 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
AF-Q96RR4-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
157 - 454 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
6CMJA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F6J |
Type1 |
161 - 463 |
0 |
SEP345,SEP400,TPO462 |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
6CMJB
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F6J |
Type1 |
161 - 462 |
0 |
SEP345,SEP400,TPO462 |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
5UY6A
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8R4 |
Type1 |
161 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
5UYJA
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8R7 |
Type1 |
161 - 449 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
5VT1A
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9JS |
Type1 |
161 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
6BKUA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DXV |
Type1 |
162 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
6BLEA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
34U |
Type1 |
161 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
6BQLA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI9 |
Type1 |
161 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
6BQPA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6T2 |
Type1 |
161 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
6BQQA
|
1.8 |
Active |
DFGin‑BLAminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R78 |
Type1 |
161 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
6BRCA
|
2.2 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E5J |
Type1 |
161 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
6BRCB
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E5J |
Type1 |
161 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
8TUCA
|
1.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
O7I |
Type1 |
161 - 449 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
2ZV2A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
609 |
Type1 |
160 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
5YV8A
|
1.927 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
91L |
Type1 |
160 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
5YVAA
|
2.574 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
91X |
Type1 |
160 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
5YVBA
|
2.02 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
92C |
Type1 |
160 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
5YVCA
|
2.02 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SU6 |
Type1 |
160 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CAMKK2
|
KKCC2_HUMAN
|
5YV9A
|
2.53 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
91O |
Type1.5_Back |
160 - 448 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase kinase 2 |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
3MFRA
|
2.0 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
5 - 306 |
0 |
None |
P22A,H145E,C146N,G162D |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
3MFSA
|
2.1 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
4 - 306 |
0 |
None |
P22A,H145E,C146N,G162D |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
3MFUA
|
2.3 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
5 - 306 |
0 |
None |
P22A,H145E,C146N,G162D |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
9M6GA
|
1.7 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
5 - 312 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
9M5YA
|
1.8 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
3 - 312 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
3C0HA
|
2.3 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
5 - 304 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
3C0HB
|
2.3 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
5 - 304 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
3MFTA
|
2.2 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 306 |
0 |
None |
P22A,H145E,C146N,G162D |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
6KMHA
|
2.4 |
Pseudo |
DFGin‑BLAminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 318 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
6KMHB
|
2.4 |
Pseudo |
DFGin‑BLAminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 319 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
8Y68A
|
2.2 |
Pseudo |
DFGin‑BLAminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 326 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
8Y68B
|
2.2 |
Pseudo |
DFGin‑BLAminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 326 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
3TACA
|
2.2 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 316 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
3C0GA
|
2.19 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3AM |
Type1 |
6 - 322 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
3C0GB
|
2.19 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3AM |
Type1 |
5 - 324 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
3C0IA
|
1.85 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3AM |
Type1 |
6 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAIA
|
2.3 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V5W |
Type1 |
5 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAIB
|
2.3 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V5W |
Type1 |
5 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAIC
|
2.3 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V5W |
Type1 |
5 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAID
|
2.3 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V5W |
Type1 |
6 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAJA
|
1.93 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V6E |
Type1 |
6 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAJB
|
1.93 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V6E |
Type1 |
6 - 302 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAJC
|
1.93 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V6E |
Type1 |
6 - 302 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAJD
|
1.93 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V6E |
Type1 |
6 - 302 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAKA
|
2.23 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V6B |
Type1 |
6 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAKB
|
2.23 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V6B |
Type1 |
6 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAKC
|
2.23 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V6B |
Type1 |
6 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OAKD
|
2.23 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V6B |
Type1 |
6 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OALA
|
2.17 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V62 |
Type1 |
6 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OALB
|
2.17 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V62 |
Type1 |
6 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OALC
|
2.17 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V62 |
Type1 |
6 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CASK
|
CSKP_HUMAN
|
7OALD
|
2.17 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
V62 |
Type1 |
6 - 303 |
0 |
None |
None |
Peripheral plasma membrane protein CASK |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7AKMA
|
1.93 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AGS |
ATPlike |
2 - 271 |
0 |
None |
D10R |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OOPA
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
5 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3JVRA
|
1.76 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AGX |
Allosteric |
2 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3JVSA
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AGY |
Allosteric |
2 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3F9NA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
38M |
Allosteric |
7 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
AF-O14757-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
AF-O14757-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
1IA8A
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 276 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7AKMB
|
1.93 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 269 |
0 |
None |
D10R |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
1ZYSA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
199 |
Type1 |
3 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2E9VA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
85A |
Type1 |
2 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2E9VB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
85A |
Type1 |
2 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2E9OA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A58 |
Type1 |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2E9PA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
77A |
Type1 |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2E9UA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A25 |
Type1 |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2GHGA
|
3.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A53 |
Type1 |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YWPA
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A42 |
Type1 |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3OT3A
|
1.44 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
22K |
Type1 |
4 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3OT8A
|
1.645 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MI5 |
Type1 |
4 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3PA3A
|
1.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C70 |
Type1 |
4 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3PA4A
|
1.59 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C72 |
Type1 |
6 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3PA5A
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C73 |
Type1 |
3 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3U9NA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
09H |
Type1 |
7 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4JIKA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1KO |
Type1 |
4 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2X8EA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X8E |
Type1 |
9 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YDJA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YDJ |
Type1 |
8 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YDJB
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YDJ |
Type1 |
9 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YDKA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YDK |
Type1 |
3 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YERA
|
1.83 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TQ1 |
Type1 |
2 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YEXA
|
1.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YEX |
Type1 |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
6FC8A
|
1.61 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D4Q |
Type1 |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
6FCFA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D58 |
Type1 |
9 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
6FCKA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D4Z |
Type1 |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FSNA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A58 |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FSMA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HK1 |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FSRA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HKC |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FSWA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HK6 |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FSYA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HK7 |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FSZA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HK8 |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FT0A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HK9 |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FT3A
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H1K |
Type1 |
2 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FT5A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H2K |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FT7A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H3K |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FT9A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H4K |
Type1 |
2 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTAA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H5K |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTCA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H6K |
Type1 |
2 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTIA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H7K |
Type1 |
3 - 279 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTJA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H8K |
Type1 |
3 - 279 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTOA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3HK |
Type1 |
3 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTQA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4HK |
Type1 |
3 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTRA
|
2.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5HK |
Type1 |
3 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTTA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6HK |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTUA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7HK |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4GH2A
|
2.03 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HK0 |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
1NVQA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UCN |
Type1 |
3 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
1NVRA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
3 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
1NVSA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UCM |
Type1 |
3 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2WMQA
|
2.48 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZYQ |
Type1 |
7 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2WMRA
|
2.43 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZYR |
Type1 |
7 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2WMSA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZYS |
Type1 |
7 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2WMTA
|
2.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZYT |
Type1 |
8 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2WMUA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZYU |
Type1 |
9 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2WMVA
|
2.009 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZYV |
Type1 |
7 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2WMWA
|
2.43 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZYW |
Type1 |
7 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2WMXA
|
2.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZY6 |
Type1 |
7 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2X8DA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X8D |
Type1 |
2 - 281 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2X8IA
|
1.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X8I |
Type1 |
2 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2XEYA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YVQ |
Type1 |
6 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2XEZA
|
2.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XEZ |
Type1 |
7 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2XF0A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4UB |
Type1 |
4 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YDIA
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YDI |
Type1 |
2 - 281 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YM3A
|
2.007 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YM3 |
Type1 |
8 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YM4A
|
2.35 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4YM |
Type1 |
4 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YM5A
|
2.03 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YM5 |
Type1 |
8 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YM6A
|
2.01 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YM6 |
Type1 |
7 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YM8A
|
2.07 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YM8 |
Type1 |
8 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4HYHA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1AM |
Type1 |
4 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4HYIA
|
1.399 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1AO |
Type1 |
3 - 274 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
1ZLTA
|
1.74 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HYM |
Type1 |
2 - 276 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2GDOA
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
12C |
Type1 |
1 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2BR1A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PFP |
Type1 |
2 - 276 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2BRBA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PFQ |
Type1 |
2 - 276 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2BRGA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DFY |
Type1 |
7 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2BRHA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DFW |
Type1 |
6 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2BRMA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DFZ |
Type1 |
7 - 274 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2BRNA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DF1 |
Type1 |
6 - 276 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2BROA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DF2 |
Type1 |
2 - 276 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2C3JA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DBQ |
Type1 |
6 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2C3LA
|
2.35 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IDZ |
Type1 |
2 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2CGUA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3A3 |
Type1 |
6 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2CGVA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3B3 |
Type1 |
6 - 272 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2CGWA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3C3 |
Type1 |
6 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2CGXA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3D3 |
Type1 |
6 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3NLBA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5BE |
Type1 |
6 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5DLSA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5CV |
Type1 |
6 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BKNA
|
2.74 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADE |
Type1 |
7 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BKOA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TVW |
Type1 |
7 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4QYEA
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3DL |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4QYFA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3DV |
Type1 |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4QYGA
|
1.75 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3DW |
Type1 |
3 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4QYGB
|
1.75 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3DW |
Type1 |
3 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4QYHA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3DX |
Type1 |
3 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4QYHB
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3DX |
Type1 |
3 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4RVKA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3XK |
Type1 |
3 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4RVLA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3XL |
Type1 |
3 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4RVMA
|
1.86 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3X7 |
Type1 |
3 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7AKOA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
2 - 271 |
0 |
None |
D10R |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7AKOB
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
2 - 271 |
0 |
None |
D10R |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2HOGA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
710 |
Type1 |
2 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2HXLA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
422 |
Type1 |
2 - 276 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2HXQA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
373 |
Type1 |
2 - 276 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2HY0A
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
306 |
Type1 |
2 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2QHMA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7CS |
Type1 |
2 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2QHNA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
582 |
Type1 |
2 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2R0UA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M54 |
Type1 |
2 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3TKHA
|
1.79 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
07S |
Type1 |
2 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
3TKIA
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
S25 |
Type1 |
2 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OQ5A
|
1.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4K4 |
Type1 |
3 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OQ7A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A0Q |
Type1 |
8 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OQ7B
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A0Q |
Type1 |
8 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FSUA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HK5 |
Type1 |
4 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OQ6A
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4K4 |
Type1 |
5 - 270 |
0 |
None |
A19S,Y20F,N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OQ8A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A0Q |
Type1 |
4 - 270 |
0 |
None |
A19S,Y20F,N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
9CE4A
|
1.31 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AV4 |
Type1 |
4 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OORA
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
3 - 283 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OOTA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4K4 |
Type1 |
4 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OP2A
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A0Q |
Type1 |
4 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OP4A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A0T |
Type1 |
3 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OP5A
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3FE |
Type1 |
4 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OP7A
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1K |
Type1 |
4 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OPBA
|
1.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1N |
Type1 |
5 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OPRA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A3E |
Type1 |
4 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OPSA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A3Q |
Type1 |
3 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OPUA
|
1.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A3K |
Type1 |
3 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5OPVA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A3H |
Type1 |
3 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BJDA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TVT |
Type1 |
3 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BJEA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADE |
Type1 |
4 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BJHA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
42C |
Type1 |
3 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BJJA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TVW |
Type1 |
3 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BJMA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TW2 |
Type1 |
5 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BJOA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TWK |
Type1 |
5 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BJRA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TWH |
Type1 |
5 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BJXA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
U0Q |
Type1 |
8 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BJXB
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
U0Q |
Type1 |
8 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BK1A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
U0N |
Type1 |
8 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BK2A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
U0K |
Type1 |
5 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7BK3A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
U0T |
Type1 |
5 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7MCKA
|
1.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YXD |
Type1 |
4 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7SUFA
|
1.48 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BVI |
Type1 |
3 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7SUGA
|
1.48 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BWI |
Type1 |
3 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7SUHA
|
2.46 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BXI |
Type1 |
4 - 270 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7SUIA
|
2.119 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L80 |
Type1 |
4 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7SUJA
|
2.299 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BYL |
Type1 |
9 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
7SUJB
|
2.299 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BYL |
Type1 |
9 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
8E80A
|
1.49 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UUF |
Type1 |
8 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
8E81A
|
1.62 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UU6 |
Type1 |
4 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
8SIVA
|
1.759 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZXH |
Type1 |
4 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
8SIWA
|
1.877 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZXL |
Type1 |
4 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
8SIWB
|
1.877 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZXL |
Type1 |
4 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
8SIXA
|
1.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZXP |
Type1 |
8 - 271 |
0 |
None |
N59L,V68I,L84M,Y86L,C87A,E91S,E134H,S147A,F149Y,G150S |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
5F4NA
|
1.91 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5UY,
5UY
|
Type1,
Allosteric
|
5 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2YM7A
|
1.81 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YM7,
YM7
|
Type1,
Type1
|
7 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2E9NA
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
76A |
Type1.5_Back |
2 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FSTA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HK4 |
Type1.5_Back |
3 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2AYPA
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
43A |
Type1.5_Back |
2 - 269 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FSQA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HK3 |
Type1.5_Back |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTKA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H9K |
Type1.5_Back |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTLA
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
H0K |
Type1.5_Back |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTMA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1HK |
Type1.5_Back |
3 - 280 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
4FTNA
|
2.02 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2HK |
Type1.5_Back |
3 - 271 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK1
|
CHK1_HUMAN
|
2C3KA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ABO |
Type1.5_Back |
6 - 270 |
0 |
None |
None |
Serine/threonine-protein kinase Chk1 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2CN5A
|
2.25 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
ADP |
ATPlike |
209 - 504 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
AF-O96017-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
212 - 494 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
AF-O96017-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
212 - 494 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WB
|
3.25 |
Inactive |
DFGin‑BLAminus |
out-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WD
|
3.25 |
Inactive |
DFGin‑BLAminus |
out-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WF
|
3.25 |
Inactive |
DFGin‑BLAminus |
out-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WH
|
3.25 |
Inactive |
DFGin‑BLAminus |
out-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2XK9A
|
2.35 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
XK9 |
Type1 |
211 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YCFA
|
1.77 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
YCF |
Type1 |
210 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2W0JA
|
2.05 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
ZAT |
Type1 |
210 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2W7XA
|
2.07 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
D1A |
Type1 |
210 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YCQA
|
2.05 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
UPX |
Type1 |
211 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YCSA
|
2.35 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
NXP |
Type1 |
210 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YIQA
|
1.89 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
YIQ |
Type1 |
211 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YIRA
|
2.1 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
YIR |
Type1 |
210 - 509 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YCRA
|
2.2 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
HCW |
Type1 |
211 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2CN8A
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_ooon |
DBQ |
Type1 |
212 - 503 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2WTCA
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
VGM |
Type1 |
211 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2WTDA
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaino |
APEdist_oooo |
ZZK |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2WTIA
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
WTI |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2WTJA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
WTJ |
Type1 |
209 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2XBJA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
XBJ |
Type1 |
211 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2XM8A
|
3.4 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oooo |
B4W |
Type1 |
211 - 503 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2XM9A
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
LWH |
Type1 |
211 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4A9RA
|
2.85 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
RU5 |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4A9SA
|
2.66 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
RU9 |
Type1 |
211 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4A9TA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
A9T |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4A9UA
|
2.48 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
A9U |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDAA
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
VFB |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDBA
|
2.5 |
Inactive |
DFGin‑BLAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
ODO |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDCA
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
ODH |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDDA
|
2.67 |
Inactive |
DFGin‑BLAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
Z0O |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDEA
|
2.55 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
CWS |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDFA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
H3R |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDGA
|
2.84 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
P3J |
Type1 |
210 - 512 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDHA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
WVI |
Type1 |
210 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDIA
|
2.32 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
HAU |
Type1 |
210 - 515 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDJA
|
3.01 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
Z2M |
Type1 |
211 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
4BDKA
|
3.3 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
RQQ |
Type1 |
211 - 513 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
2YITA
|
2.2 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
YIT |
Type1.5_Back |
211 - 510 |
0 |
None |
None |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6UA
|
3.0 |
Inactive |
DFGin‑BLAplus |
out-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
89 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6UB
|
3.0 |
Inactive |
DFGin‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
89 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WA
|
3.25 |
Inactive |
DFGin‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WC
|
3.25 |
Inactive |
DFGin‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WE
|
3.25 |
Inactive |
DFGin‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
CHEK2
|
CHK2_HUMAN
|
3I6WG
|
3.25 |
Inactive |
DFGin‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
92 - 501 |
0 |
None |
K249R |
Serine/threonine-protein kinase Chk2 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1WVYA
|
2.8 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
STU |
Type1 |
4 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9INVA
|
1.61 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
HCC |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9INWA
|
1.52 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1L2V |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2W4JA
|
1.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ADP |
ATPlike |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3ZXTB
|
2.65 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
ACP |
ATPlike |
7 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3ZXTC
|
2.65 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ACP |
ATPlike |
5 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3ZXTD
|
2.65 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
ACP |
ATPlike |
7 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1IG1A
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 294 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1JKKA
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 293 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1JKLA
|
1.62 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 294 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3EH9A
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ADP |
ATPlike |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3EHAA
|
1.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3F5GA
|
1.85 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ADP |
ATPlike |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3F5UA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2W4KA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
2 - 302 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3DFCB
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 277 |
0 |
None |
Q23K |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GU4A
|
1.35 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 277 |
0 |
None |
Q23V |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GU5A
|
1.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
2 - 277 |
0 |
None |
Q23V |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GU6A
|
1.49 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ADP |
ATPlike |
2 - 277 |
0 |
None |
Q23V |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GU7A
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ADP |
ATPlike |
2 - 277 |
0 |
None |
Q23V |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2XUUA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
2 - 302 |
0 |
None |
E182A |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1WVWA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
4PF4A
|
1.13 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
AF-P53355-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 283 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
AF-P53355-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 283 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2Y4PA
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
4 - 275 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2Y4PC
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
2 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AV1A
|
1.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
6IN4A
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1JKSA
|
1.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 294 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1JKTA
|
3.5 |
Inactive |
DFGin‑BLAminus |
in-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1JKTB
|
3.5 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iooo |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3DGKA
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
Q23K |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2XZSA
|
2.0 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 312 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2XZSB
|
2.0 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 302 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
6QMOA
|
1.87 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
4 - 302 |
0 |
None |
S289E,S308A |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
6QN4A
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 277 |
0 |
None |
S289E,S308E |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
4UV0A
|
2.49 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 302 |
0 |
None |
S289C |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2Y0AA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 302 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2X0GA
|
2.2 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
3 - 320 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
4TL0A
|
2.7 |
Active |
DFGin‑BLAminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 301 |
0 |
None |
S289E |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
4B4LA
|
1.75 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 303 |
0 |
None |
R302A |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
6FHAA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
4 - 302 |
0 |
None |
S289A,S308A |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
6FHBA
|
1.75 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 302 |
0 |
None |
S289A,S308E |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1WVXA
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
BD4 |
Type1 |
2 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2YAKA
|
2.2 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
OSV |
Type1 |
2 - 278 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUTA
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
2AN |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUVA
|
1.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
AGI |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUXA
|
1.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KMP |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUZA
|
1.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
GEN |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AV0A
|
1.85 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
47X |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AV2A
|
1.502 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KMP |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AV3A
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KMP |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AV4A
|
1.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
GEN |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
6AARA
|
1.95 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
9TF |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
7CCWA
|
1.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
STL |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
8IE6A
|
1.701 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
8KZ |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
8IE7A
|
1.849 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3RL |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
8IE8A
|
1.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
P5O |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9INXA
|
1.72 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1L2W |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
1P4FA
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
86Q |
Type1 |
2 - 293 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9N1TA
|
1.43 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BU8 |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9N2MA
|
1.35 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BVM |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9N2OA
|
1.49 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BVL |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
4YO4A
|
1.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
4FT |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
4YPDA
|
1.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
DKG |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9DUBA
|
1.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BB7 |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
4TXCA
|
1.951 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
38G |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9MIUA
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BLJ |
Type1 |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GU8A
|
1.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
3GU |
Type1 |
2 - 277 |
0 |
None |
L93G |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3GUBA
|
1.71 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
GUB |
Type1 |
2 - 277 |
0 |
None |
L93G |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
9DUEA
|
1.65 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
A1BB6,
BO3
|
Type1,
Allosteric
|
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUUA
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
LU2 |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUWA
|
1.5 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
QUE |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
5AUYA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
MRI |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
7CCUA
|
1.649 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
STL |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
7CCVA
|
1.753 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
PIT |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
8IE5A
|
1.803 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
EZE |
Type1.5_Back |
2 - 277 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
3ZXTA
|
2.65 |
Inactive |
DFGin‑BLBminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ACP |
ATPlike |
7 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2Y4PB
|
2.65 |
Inactive |
None‑None |
none-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
57 - 275 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK1
|
DAPK1_HUMAN
|
2Y4PD
|
2.65 |
Inactive |
None‑None |
none-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
56 - 276 |
0 |
None |
None |
Death-associated protein kinase 1 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
AF-Q9UIK4-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 293 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
AF-Q9UIK4-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 293 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1ZWSA
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 289 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1ZWSB
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 289 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1ZWSC
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 289 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1ZWSD
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 289 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1ZWSE
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 289 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1ZWSF
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 289 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1ZWSG
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 289 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1ZWSH
|
2.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 289 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1Z9XA
|
3.93 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
W315S,S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1Z9XB
|
3.93 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
W315S,S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1Z9XC
|
3.93 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
W315S,S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A2AA
|
1.47 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
11 - 314 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A2AB
|
1.47 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A2AC
|
1.47 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A2AD
|
1.47 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A27A
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 315 |
0 |
None |
W315S,S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A27B
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
W315S,S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A27C
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
W315S,S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A27D
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 315 |
0 |
None |
W315S,S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A27E
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
W315S,S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A27F
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
W315S,S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A27G
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
W315S,S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2A27H
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 315 |
0 |
None |
W315S,S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKA
|
3.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKB
|
3.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 325 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKC
|
3.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKD
|
3.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 325 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKE
|
3.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 324 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKF
|
3.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 314 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKG
|
3.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 324 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
1WMKH
|
3.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
12 - 315 |
0 |
None |
S318D |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
6PAWA
|
2.953 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 329 |
0 |
None |
S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
6PAWB
|
2.953 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 329 |
0 |
None |
S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
6PAWE
|
2.953 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 318 |
0 |
None |
S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
6PAWF
|
2.953 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 327 |
0 |
None |
S318A |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2CKEA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQU |
Type1 |
11 - 311 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2CKEB
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQU |
Type1 |
12 - 311 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2CKEC
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQU |
Type1 |
12 - 311 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK2
|
DAPK2_HUMAN
|
2CKED
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQU |
Type1 |
12 - 311 |
0 |
None |
None |
Death-associated protein kinase 2 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
AF-O43293-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 283 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
AF-O43293-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
5 - 283 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5A6NB
|
1.7 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
9 - 278 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5A6OA
|
1.6 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
9 - 278 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5A6OB
|
1.6 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
No_ligand |
No_ligand |
9 - 277 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
1YRPA
|
3.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 277 |
0 |
TPO265 |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
1YRPB
|
3.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 277 |
0 |
TPO265 |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
3BHYA
|
1.24 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
7CP |
Type1 |
9 - 283 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
3BQRA
|
1.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
4RB |
Type1 |
9 - 284 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5A6NA
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
U7E |
Type1 |
9 - 278 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5VJAA
|
2.46 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DUK |
Type1 |
9 - 277 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5VJAB
|
2.46 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DUK |
Type1 |
9 - 278 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5VJAC
|
2.46 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DUK |
Type1 |
9 - 278 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
5VJAD
|
2.46 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DUK |
Type1 |
9 - 277 |
0 |
None |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
2J90A
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
IZA |
Type1 |
5 - 278 |
0 |
SEP50,TPO265 |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DAPK3
|
DAPK3_HUMAN
|
2J90B
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
IZA |
Type1 |
12 - 280 |
0 |
SEP50,TPO265 |
None |
Death-associated protein kinase 3 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
7F3GB
|
2.1 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RXT |
Type1 |
383 - 648 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
5JZJA
|
1.71 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AN2 |
ATPlike |
374 - 648 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
5JZJB
|
1.71 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AN2 |
ATPlike |
382 - 648 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
AF-O15075-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
382 - 655 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
AF-O15075-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
382 - 655 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
6KYRA
|
2.206 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
380 - 701 |
0 |
None |
P675L |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
6KYRB
|
2.206 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
380 - 700 |
0 |
None |
P675L |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
6KYQA
|
2.141 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
380 - 701 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
6KYQB
|
2.141 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
380 - 700 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
5JZNA
|
2.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GUI |
Type1 |
379 - 648 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
5JZNB
|
2.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GUI |
Type1 |
380 - 648 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
7KX6A
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X7Y |
Type1 |
381 - 648 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
7KX6B
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X7Y |
Type1 |
382 - 648 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
7KXWA
|
3.002 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XBD |
Type1 |
382 - 648 |
0 |
TPO484 |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
7KXWB
|
3.002 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XBD |
Type1 |
382 - 649 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
7F3GA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RXT |
Type1 |
376 - 648 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
7KX8A
|
3.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X8J |
Type1 |
382 - 669 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK1
|
DCLK1_HUMAN
|
7KX8B
|
3.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
X8J |
Type1 |
380 - 647 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK1 |
|
CAMK
|
DCLK2
|
DCLK2_HUMAN
|
AF-Q8N568-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
386 - 659 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK2 |
|
CAMK
|
DCLK2
|
DCLK2_HUMAN
|
AF-Q8N568-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
386 - 659 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK2 |
|
CAMK
|
DCLK3
|
DCLK3_HUMAN
|
AF-Q9C098-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
348 - 621 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK3 |
|
CAMK
|
DCLK3
|
DCLK3_HUMAN
|
AF-Q9C098-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
348 - 621 |
0 |
None |
None |
Serine/threonine-protein kinase DCLK3 |
|
CAMK
|
HUNK
|
HUNK_HUMAN
|
AF-P57058-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
54 - 328 |
0 |
None |
None |
Hormonally up-regulated neu tumor-associated kinase |
|
CAMK
|
HUNK
|
HUNK_HUMAN
|
AF-P57058-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
54 - 328 |
0 |
None |
None |
Hormonally up-regulated neu tumor-associated kinase |
|
CAMK
|
KALRN
|
KALRN_HUMAN
|
AF-O60229-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiai |
APEdist_iiii |
No_ligand |
No_ligand |
2675 - 2945 |
0 |
None |
None |
Kalirin |
|
CAMK
|
KALRN
|
KALRN_HUMAN
|
AF-O60229-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiai |
APEdist_iiii |
No_ligand |
No_ligand |
2675 - 2945 |
0 |
None |
None |
Kalirin |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4A
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 351 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4B
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 351 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4C
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
48 - 351 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4D
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 349 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4E
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 353 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4F
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 353 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4G
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 348 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4H
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 358 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4I
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 347 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4J
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 350 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4K
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 348 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XU4L
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 354 |
0 |
None |
S216G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
1NY3A
|
3.0 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ADP |
ATPlike |
46 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
AF-P49137-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
55 - 333 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
AF-P49137-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
55 - 333 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BC
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BD
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BE
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BF
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BG
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BH
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BI
|
2.9 |
None |
DFGin‑BLAminus |
in-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BJ
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BK
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BL
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2PZYD
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_nnoo |
No_ligand |
No_ligand |
43 - 342 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3G
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
43 - 342 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPJ
|
3.31 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
48 - 328 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
4TYHA
|
3.0 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 400 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2OZAA
|
2.7 |
Inactive |
DFGin‑BLAminus |
out-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 390 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6TCAA
|
3.7 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 399 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6TCAC
|
3.7 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 397 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6TCAE
|
3.7 |
Inactive |
DFGin‑BLAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 394 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6TCAG
|
3.7 |
Inactive |
DFGin‑BLAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
51 - 397 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
8XX1A
|
2.55 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
47 - 364 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
1KWPA
|
2.8 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
46 - 385 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
1KWPB
|
2.8 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
44 - 378 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2ONLC
|
4.0 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_oooo |
No_ligand |
No_ligand |
46 - 393 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2ONLD
|
4.0 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oooo |
No_ligand |
No_ligand |
46 - 393 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BA
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
05B |
Type1 |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2BB
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
05B |
Type1 |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R2YA
|
3.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3R30A
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
CD2 |
Type1 |
46 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2PZYA
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
B18 |
Type1 |
42 - 346 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2PZYB
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
B18 |
Type1 |
44 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2PZYC
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
STU |
Type1 |
42 - 359 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3A
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK2 |
Type1 |
43 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3B
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK2 |
Type1 |
44 - 349 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3C
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK2 |
Type1 |
41 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3D
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK2 |
Type1 |
46 - 342 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3E
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK2 |
Type1 |
44 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3F
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK2 |
Type1 |
44 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3H
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK2 |
Type1 |
44 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3I
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK2 |
Type1 |
45 - 356 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3J
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK2 |
Type1 |
43 - 348 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3K
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK2 |
Type1 |
44 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KC3L
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK2 |
Type1 |
42 - 348 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6A
|
2.99 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6B
|
2.99 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6C
|
2.99 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6D
|
2.99 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6E
|
2.99 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3WI6F
|
2.99 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
YRZ |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3FPMA
|
3.3 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
793 |
Type1 |
44 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2P3GX
|
3.8 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
F10 |
Type1 |
45 - 364 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3FYJX
|
3.8 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
B97 |
Type1 |
45 - 364 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3FYKX
|
3.5 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
B98 |
Type1 |
45 - 364 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
7NRYX
|
3.8 |
Inactive |
DFGin‑BLAminus |
out-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
B97 |
Type1 |
45 - 366 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBOA
|
3.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
P4O |
Type1 |
44 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPA
|
3.31 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPB
|
3.31 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPC
|
3.31 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPD
|
3.31 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
47 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPE
|
3.31 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
44 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPF
|
3.31 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
45 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPG
|
3.31 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
45 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPH
|
3.31 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 347 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPI
|
3.31 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
45 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPK
|
3.31 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
2JBPL
|
3.31 |
Inactive |
DFGin‑BLAminus |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
44 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKA
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKB
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKC
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKD
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKE
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKF
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKG
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKH
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKI
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKJ
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKK
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3GOKL
|
3.2 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
46 - 350 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KA0A
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
MK3 |
Type1 |
47 - 364 |
0 |
None |
T222E |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
9R59A
|
3.0 |
Inactive |
DFGin‑BLAminus |
out-none |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
A1JH4 |
Type1 |
48 - 364 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
1NXKA
|
2.7 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
STU |
Type1 |
42 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
1NXKB
|
2.7 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
STU |
Type1 |
44 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
1NXKC
|
2.7 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
STU |
Type1 |
41 - 357 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
1NXKD
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_nnoo |
STU |
Type1 |
43 - 342 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3KGAA
|
2.55 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
LX9 |
Type1 |
47 - 364 |
0 |
None |
P237G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3M2WA
|
2.41 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
L8I |
Type1 |
47 - 364 |
0 |
None |
P237G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3M42A
|
2.68 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
HGF |
Type1 |
47 - 364 |
0 |
None |
P237G |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CA
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
47 - 344 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CB
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CC
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 342 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CD
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 344 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CE
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 344 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CF
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
47 - 345 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CG
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 342 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CH
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
47 - 343 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CI
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 343 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CJ
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 343 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CK
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 344 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
3A2CL
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
PDY,
PDY
|
Type1,
Allosteric
|
48 - 344 |
0 |
None |
None |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6T8XA
|
2.81 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
B97,
MW8
|
Type1,
Allosteric
|
44 - 330 |
0 |
None |
T222E,T334E |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6T8XB
|
2.81 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
B97,
MW8
|
Type1,
Allosteric
|
45 - 329 |
0 |
None |
T222E,T334E |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6T8XC
|
2.81 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
B97,
MW8
|
Type1,
Allosteric
|
44 - 329 |
0 |
None |
T222E,T334E |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6T8XD
|
2.81 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
B97,
MW8
|
Type1,
Allosteric
|
44 - 331 |
0 |
None |
T222E,T334E |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6T8XE
|
2.81 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
B97,
MW8
|
Type1,
Allosteric
|
45 - 329 |
0 |
None |
T222E,T334E |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK2
|
MAPK2_HUMAN
|
6T8XF
|
2.81 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
B97,
MW8
|
Type1,
Allosteric
|
45 - 329 |
0 |
None |
T222E,T334E |
MAP kinase-activated protein kinase 2 |
|
CAMK
|
MAPKAPK3
|
MAPK3_HUMAN
|
AF-Q16644-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
No_ligand |
No_ligand |
35 - 312 |
0 |
None |
None |
MAP kinase-activated protein kinase 3 |
|
CAMK
|
MAPKAPK3
|
MAPK3_HUMAN
|
AF-Q16644-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
35 - 312 |
0 |
None |
None |
MAP kinase-activated protein kinase 3 |
|
CAMK
|
MAPKAPK3
|
MAPK3_HUMAN
|
3R1NA
|
2.09 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
05B |
Type1 |
33 - 348 |
0 |
None |
None |
MAP kinase-activated protein kinase 3 |
|
CAMK
|
MAPKAPK3
|
MAPK3_HUMAN
|
3SHEA
|
2.25 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
I85 |
Type1 |
33 - 348 |
0 |
None |
None |
MAP kinase-activated protein kinase 3 |
|
CAMK
|
MAPKAPK3
|
MAPK3_HUMAN
|
3FHRA
|
1.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
33 - 349 |
0 |
None |
None |
MAP kinase-activated protein kinase 3 |
|
CAMK
|
MAPKAPK3
|
MAPK3_HUMAN
|
3FXWA
|
2.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
F10 |
Type1 |
33 - 349 |
0 |
None |
None |
MAP kinase-activated protein kinase 3 |
|
CAMK
|
MAPKAPK3
|
MAPK3_HUMAN
|
7NRBA
|
1.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
P4O |
Type1 |
33 - 349 |
0 |
None |
None |
MAP kinase-activated protein kinase 3 |
|
CAMK
|
MAPKAPK5
|
MAPK5_HUMAN
|
AF-Q8IW41-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 312 |
0 |
None |
None |
MAP kinase-activated protein kinase 5 |
|
CAMK
|
MAPKAPK5
|
MAPK5_HUMAN
|
AF-Q8IW41-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 312 |
0 |
None |
None |
MAP kinase-activated protein kinase 5 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
AF-Q9P0L2-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
52 - 319 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
AF-Q9P0L2-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
52 - 319 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
6C9DA
|
2.499 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
53 - 795 |
0 |
None |
T215E,K761S,R764S |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
6C9DB
|
2.499 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
53 - 795 |
0 |
None |
T215E,K761S,R764S |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKA
|
2.6 |
Inactive |
None‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaioo |
APEdist_nnno |
No_ligand |
No_ligand |
55 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKB
|
2.6 |
Inactive |
None‑None |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
53 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKC
|
2.6 |
Inactive |
None‑None |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
53 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKD
|
2.6 |
Inactive |
None‑None |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
54 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKE
|
2.6 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
54 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKF
|
2.6 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiio |
APEdist_oooo |
No_ligand |
No_ligand |
54 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKG
|
2.6 |
Inactive |
None‑None |
in-out |
out-out |
nonTYR |
APEdihe_aanio |
APEdist_nnnn |
No_ligand |
No_ligand |
55 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK1
|
MARK1_HUMAN
|
2HAKH
|
2.6 |
Inactive |
None‑None |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
54 - 371 |
0 |
None |
None |
Serine/threonine-protein kinase MARK1 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
3IECB
|
2.2 |
Inactive |
DFGin‑ABAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
49 - 363 |
0 |
None |
R146W |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
3IECD
|
2.2 |
Inactive |
DFGin‑ABAminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
49 - 363 |
0 |
None |
R146W |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5EAKB
|
2.8 |
Inactive |
DFGin‑ABAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
24R |
Type1 |
51 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
AF-Q7KZI7-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
45 - 312 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
AF-Q7KZI7-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
45 - 312 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
3IECA
|
2.2 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
49 - 363 |
0 |
None |
R146W |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
3IECC
|
2.2 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
49 - 363 |
0 |
None |
R146W |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5EAKA
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nioo |
24R |
Type1 |
47 - 362 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
8TXYA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
SJ0 |
Type1 |
48 - 363 |
0 |
None |
I59L,K66V,V81I,L97I,V113I,M129T,S133K,G134N,S197G |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
8TXYB
|
2.1 |
Inactive |
DFGin‑BLAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
SJ0 |
Type1 |
47 - 363 |
0 |
None |
I59L,K66V,V81I,L97I,V113I,M129T,S133K,G134N,S197G |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5KZ7A
|
3.2 |
Inactive |
DFGin‑None |
in-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
6Z2 |
Type1 |
48 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5KZ8A
|
3.21 |
Inactive |
DFGin‑None |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
6Z5 |
Type1 |
48 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5KZ8B
|
3.21 |
Inactive |
DFGin‑None |
in-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
6Z5 |
Type1 |
48 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK2
|
MARK2_HUMAN
|
5KZ7B
|
3.2 |
Inactive |
None‑None |
in-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
6Z2 |
Type1 |
48 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase MARK2 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
AF-P27448-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
48 - 315 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
AF-P27448-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
48 - 315 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOIA
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
X3Q |
Type1 |
51 - 368 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E,V205K |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOKA
|
1.85 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
X5N |
Type1 |
51 - 369 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E,V205K |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOKB
|
1.85 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
X5N |
Type1 |
51 - 369 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E,V205K |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
7P1LA
|
1.95 |
Inactive |
DFGin‑BLBminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
V5E |
Type1 |
50 - 365 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOJA
|
1.6 |
Inactive |
DFGin‑BLBtrans |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooi |
X5I,
BEZ
|
Type1,
Allosteric
|
50 - 370 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
2QNJA
|
2.7 |
Inactive |
None‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
No_ligand |
No_ligand |
44 - 366 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
2QNJB
|
2.7 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iooo |
No_ligand |
No_ligand |
44 - 367 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
3FE3A
|
1.9 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoni |
APEdist_iooo |
No_ligand |
No_ligand |
50 - 366 |
0 |
None |
T211A,S215A |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
3FE3B
|
1.9 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoni |
APEdist_iooo |
No_ligand |
No_ligand |
50 - 366 |
0 |
None |
T211A,S215A |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOHA
|
2.15 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
No_ligand |
No_ligand |
48 - 369 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
7P1LB
|
1.95 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
V5E |
Type1 |
50 - 365 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOHB
|
2.15 |
Inactive |
None‑None |
in-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_iooo |
X4W |
Type1 |
48 - 370 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOLA
|
1.9 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
X4H |
Type1 |
51 - 370 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK3
|
MARK3_HUMAN
|
8UOLB
|
1.9 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnni |
X4H |
Type1 |
50 - 367 |
0 |
None |
I62L,L72R,V116I,G137K,F141Y,A146E |
MAP/microtubule affinity-regulating kinase 3 |
|
CAMK
|
MARK4
|
MARK4_HUMAN
|
AF-Q96L34-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
51 - 318 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 4 |
|
CAMK
|
MARK4
|
MARK4_HUMAN
|
AF-Q96L34-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
51 - 318 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 4 |
|
CAMK
|
MARK4
|
MARK4_HUMAN
|
8XFLA
|
3.0 |
Inactive |
DFGin‑BLBtrans |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
54 - 370 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 4 |
|
CAMK
|
MARK4
|
MARK4_HUMAN
|
5ES1A
|
2.8 |
Inactive |
DFGin‑None |
in-in |
in-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
5RC |
Type1 |
54 - 370 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 4 |
|
CAMK
|
MARK4
|
MARK4_HUMAN
|
8XFLB
|
3.0 |
Inactive |
None‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
54 - 370 |
0 |
None |
None |
MAP/microtubule affinity-regulating kinase 4 |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4BL1A
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
ANP |
ATPlike |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TX3A
|
2.9 |
Inactive |
DFGin‑ABAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
7MY |
Type1 |
1 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
AF-Q14680-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 271 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
AF-Q14680-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 271 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWUA
|
2.603 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
No_ligand |
No_ligand |
1 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWUB
|
2.603 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoi |
No_ligand |
No_ligand |
1 - 335 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5IH8A
|
1.85 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
6BJ |
Type1 |
3 - 327 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5IH9A
|
1.79 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
6BF |
Type1 |
3 - 327 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5IHAA
|
1.96 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
6BE |
Type1 |
3 - 327 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWZA
|
2.631 |
Inactive |
DFGin‑BLAminus |
out-none |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
45R |
Type1 |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
6GVXA
|
2.24 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
TAK |
Type1 |
1 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
6GVXB
|
2.24 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
TAK |
Type1 |
1 - 335 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4BKYA
|
1.83 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
82B |
Type1 |
3 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4BKZA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
1WS |
Type1 |
2 - 334 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5M5AA
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
KSA |
Type1 |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5MAGA
|
2.35 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
7KC |
Type1 |
3 - 335 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5MAHA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
7KD |
Type1 |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
9F31A
|
2.0 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
A1H9M |
Type1 |
1 - 335 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2TA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_nooi |
3I7 |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2TB
|
2.7 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnii |
3I7 |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2TC
|
2.7 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
3I7 |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2TD
|
2.7 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
3I7 |
Type1 |
3 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2VA
|
2.45 |
None |
DFGin‑BLAminus |
in-in |
none-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
45R |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2VB
|
2.45 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_nnoi |
45R |
Type1 |
2 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2VC
|
2.45 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
45R |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2VD
|
2.45 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
45R |
Type1 |
3 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2WA
|
1.92 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_nnoi |
NF5 |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2WB
|
1.92 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_nnoi |
NF5 |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2WC
|
1.92 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
NF5 |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2WD
|
1.92 |
Inactive |
DFGin‑BLAminus |
in-out |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnii |
NF5 |
Type1 |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMPD
|
2.3 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
5QM |
Type1 |
2 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMRA
|
3.0 |
Inactive |
DFGin‑BLAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
QBB |
Type1 |
6 - 333 |
0 |
None |
T167A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TVTA
|
2.28 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
7LV |
Type1.5_Back |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWLA
|
2.42 |
Inactive |
DFGin‑BLAminus |
in-in |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
H91 |
Type1.5_Back |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5MAFA
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
XIN |
Type1.5_Back |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2PA
|
2.55 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
6Z7 |
Type1.5_Back |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2PB
|
2.55 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnii |
6Z7 |
Type1.5_Back |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2PC
|
2.55 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
6Z7 |
Type1.5_Back |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4D2PD
|
2.55 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
6Z7 |
Type1.5_Back |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMPA
|
2.3 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
5QM |
Type1.5_Back |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMPB
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_nnoi |
5QM |
Type1.5_Back |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMPC
|
2.3 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_nnni |
5QM |
Type1.5_Back |
1 - 333 |
0 |
None |
T167A,S171A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMQA
|
2.6 |
Inactive |
DFGin‑BLAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
B5S |
Type1.5_Back |
5 - 333 |
0 |
None |
T167A,N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5IHCA
|
2.14 |
Inactive |
DFGin‑BLBminus |
out-out |
none-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
6BB |
Type1 |
3 - 327 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWYA
|
2.91 |
Inactive |
DFGin‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaoni |
APEdist_nnno |
7LY |
Type1 |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5MAIA
|
2.15 |
Inactive |
DFGin‑None |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
5U5 |
Type1 |
2 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4IXPA
|
2.749 |
Inactive |
DFGinter‑BABtrans |
out-none |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
No_ligand |
No_ligand |
2 - 335 |
0 |
None |
K40R,D150A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMTA
|
1.98 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
47W |
Type1 |
3 - 333 |
0 |
None |
N213T,V214A,M215A,Y218V,K219A |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
4UMUA
|
2.02 |
Inactive |
DFGinter‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnoo |
0V0 |
Type1 |
3 - 333 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5K00A
|
1.77 |
Inactive |
DFGout‑None |
out-in |
out-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
6PV |
Type2 |
3 - 327 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
6VXRA
|
2.1 |
Inactive |
None‑None |
out-none |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
F7D |
Type1 |
1 - 332 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TWYB
|
2.91 |
Inactive |
None‑None |
out-none |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
7LY |
Type1 |
2 - 332 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MELK
|
MELK_HUMAN
|
5TX3B
|
2.9 |
Inactive |
None‑None |
out-out |
none-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
7MY |
Type1 |
1 - 334 |
0 |
None |
None |
Maternal embryonic leucine zipper kinase |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
AF-Q9BUB5-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
40 - 382 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
AF-Q9BUB5-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
40 - 382 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
2HW6A
|
2.5 |
Inactive |
DFGout‑BBAminus |
in-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
39 - 376 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
2HW6B
|
2.5 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
40 - 375 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
5WVDA
|
3.0 |
Inactive |
DFGout‑None |
in-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
7UX |
Type1 |
41 - 375 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
|
CAMK
|
MKNK1
|
MKNK1_HUMAN
|
5WVDB
|
3.0 |
Inactive |
DFGout‑None |
in-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
7UX |
Type1 |
41 - 374 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 1 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
AF-Q9HBH9-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
75 - 376 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
AF-Q9HBH9-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
75 - 376 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
8XFMA
|
2.6 |
Inactive |
DFGin‑BLBminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
A1LU6 |
Type1 |
73 - 372 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
2HW7A
|
2.71 |
Inactive |
DFGin‑BLBplus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
STU |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CJ5A
|
2.8 |
Inactive |
DFGin‑BLBplus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
F4G |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CJEA
|
3.36 |
Inactive |
DFGin‑BLBplus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
F4A |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CJHA
|
3.6 |
Inactive |
DFGin‑BLBplus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
ET8 |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CJWA
|
3.38 |
Inactive |
DFGin‑BLBplus |
out-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
FYV |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CJYA
|
3.05 |
Inactive |
DFGin‑BLBplus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
F4J |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CK3A
|
2.9 |
Inactive |
DFGin‑BLBplus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
F67 |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CK6A
|
3.32 |
Inactive |
DFGin‑BLBplus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
N45 |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6CKIA
|
2.95 |
Inactive |
DFGin‑BLBplus |
in-in |
none-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
FZJ |
Type1 |
72 - 371 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
9HRCA
|
3.161 |
Inactive |
DFGin‑BLBplus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_oooo |
A1IWO |
Type1 |
72 - 375 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
2AC5A
|
3.2 |
Inactive |
DFGin‑None |
in-in |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
No_ligand |
No_ligand |
72 - 370 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
8P9BA
|
2.59 |
Inactive |
DFGin‑None |
in-in |
none-none |
nonTYR |
APEdihe_aanni |
APEdist_nnnn |
X8K |
Type1 |
72 - 369 |
0 |
None |
D228G |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
2AC3A
|
2.1 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnoo |
No_ligand |
No_ligand |
72 - 369 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MKNK2
|
MKNK2_HUMAN
|
6JLRA
|
2.901 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
BV9 |
Type1 |
72 - 369 |
0 |
None |
None |
MAP kinase-interacting serine/threonine-protein kinase 2 |
|
CAMK
|
MYLK
|
MYLK_HUMAN
|
AF-Q15746-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1456 - 1727 |
0 |
None |
None |
Myosin light chain kinase, smooth muscle |
|
CAMK
|
MYLK
|
MYLK_HUMAN
|
AF-Q15746-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1456 - 1727 |
0 |
None |
None |
Myosin light chain kinase, smooth muscle |
|
CAMK
|
MYLK2
|
MYLK2_HUMAN
|
AF-Q9H1R3-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
275 - 548 |
0 |
None |
None |
Myosin light chain kinase 2, skeletal/cardiac muscle |
|
CAMK
|
MYLK2
|
MYLK2_HUMAN
|
AF-Q9H1R3-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
275 - 548 |
0 |
None |
None |
Myosin light chain kinase 2, skeletal/cardiac muscle |
|
CAMK
|
MYLK3
|
MYLK3_HUMAN
|
AF-Q32MK0-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
505 - 778 |
0 |
None |
None |
Myosin light chain kinase 3 |
|
CAMK
|
MYLK3
|
MYLK3_HUMAN
|
AF-Q32MK0-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
505 - 778 |
0 |
None |
None |
Myosin light chain kinase 3 |
|
CAMK
|
MYLK4
|
MYLK4_HUMAN
|
2X4FA
|
2.67 |
Inactive |
DFGin‑ABAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
16X |
Type1 |
80 - 373 |
0 |
None |
None |
Myosin light chain kinase family member 4 |
|
CAMK
|
MYLK4
|
MYLK4_HUMAN
|
2X4FB
|
2.67 |
Inactive |
DFGin‑ABAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
16X |
Type1 |
81 - 370 |
0 |
None |
None |
Myosin light chain kinase family member 4 |
|
CAMK
|
MYLK4
|
MYLK4_HUMAN
|
AF-Q86YV6-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
96 - 369 |
0 |
None |
None |
Myosin light chain kinase family member 4 |
|
CAMK
|
MYLK4
|
MYLK4_HUMAN
|
AF-Q86YV6-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
96 - 369 |
0 |
None |
None |
Myosin light chain kinase family member 4 |
|
CAMK
|
NIM1K
|
NIM1_HUMAN
|
AF-Q8IY84-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
66 - 333 |
0 |
None |
None |
Serine/threonine-protein kinase NIM1 |
|
CAMK
|
NIM1K
|
NIM1_HUMAN
|
AF-Q8IY84-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
66 - 333 |
0 |
None |
None |
Serine/threonine-protein kinase NIM1 |
|
CAMK
|
NUAK1
|
NUAK1_HUMAN
|
AF-O60285-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
47 - 314 |
0 |
None |
None |
NUAK family SNF1-like kinase 1 |
|
CAMK
|
NUAK1
|
NUAK1_HUMAN
|
AF-O60285-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
47 - 314 |
0 |
None |
None |
NUAK family SNF1-like kinase 1 |
|
CAMK
|
NUAK2
|
NUAK2_HUMAN
|
AF-Q9H093-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
45 - 311 |
0 |
None |
None |
NUAK family SNF1-like kinase 2 |
|
CAMK
|
NUAK2
|
NUAK2_HUMAN
|
AF-Q9H093-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
45 - 311 |
0 |
None |
None |
NUAK family SNF1-like kinase 2 |
|
CAMK
|
OBSCN-1
|
OBSCN_HUMAN
|
AF-Q5VST9-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6460 - 6729 |
0 |
None |
None |
Obscurin |
|
CAMK
|
OBSCN-1
|
OBSCN_HUMAN
|
AF-Q5VST9-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
6460 - 6729 |
0 |
None |
None |
Obscurin |
|
CAMK
|
OBSCN-2
|
OBSCN_HUMAN
|
AF-Q5VST9-K2A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiai |
APEdist_iioi |
No_ligand |
No_ligand |
7664 - 7932 |
0 |
None |
None |
Obscurin |
|
CAMK
|
OBSCN-2
|
OBSCN_HUMAN
|
AF-Q5VST9-K4A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiai |
APEdist_iiii |
No_ligand |
No_ligand |
7664 - 7932 |
0 |
None |
None |
Obscurin |
|
CAMK
|
PASK
|
PASK_HUMAN
|
3DLSA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
982 - 1266 |
0 |
None |
None |
PAS domain-containing serine/threonine-protein kinase |
|
CAMK
|
PASK
|
PASK_HUMAN
|
3DLSB
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
982 - 1267 |
0 |
None |
None |
PAS domain-containing serine/threonine-protein kinase |
|
CAMK
|
PASK
|
PASK_HUMAN
|
3DLSC
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
982 - 1267 |
0 |
None |
None |
PAS domain-containing serine/threonine-protein kinase |
|
CAMK
|
PASK
|
PASK_HUMAN
|
3DLSD
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
982 - 1266 |
0 |
None |
None |
PAS domain-containing serine/threonine-protein kinase |
|
CAMK
|
PASK
|
PASK_HUMAN
|
3DLSE
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
982 - 1267 |
0 |
None |
None |
PAS domain-containing serine/threonine-protein kinase |
|
CAMK
|
PASK
|
PASK_HUMAN
|
3DLSF
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
982 - 1266 |
0 |
None |
None |
PAS domain-containing serine/threonine-protein kinase |
|
CAMK
|
PASK
|
PASK_HUMAN
|
AF-Q96RG2-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
991 - 1259 |
0 |
None |
None |
PAS domain-containing serine/threonine-protein kinase |
|
CAMK
|
PASK
|
PASK_HUMAN
|
AF-Q96RG2-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
991 - 1259 |
0 |
None |
None |
PAS domain-containing serine/threonine-protein kinase |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5RC
|
3.52 |
Inactive |
DFGin‑BLAminus |
out-none |
out-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
12 - 383 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5TC
|
3.74 |
Inactive |
DFGin‑BLAminus |
out-none |
out-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
12 - 383 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5TG
|
3.74 |
Inactive |
DFGin‑BLAminus |
out-none |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ATP |
ATPlike |
12 - 383 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5TK
|
3.74 |
Inactive |
DFGin‑BLAminus |
out-none |
out-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
12 - 383 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5TO
|
3.74 |
Inactive |
DFGin‑BLAminus |
out-none |
out-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
12 - 383 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
AF-Q16816-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 296 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
AF-Q16816-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 296 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8JFKC
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8JFKG
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8JFKK
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8JFKO
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8XYAC
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8XYBC
|
3.1 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 382 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5MC
|
3.66 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5PC
|
3.41 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5PG
|
3.41 |
Inactive |
DFGin‑BLAminus |
out-out |
out-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5QC
|
4.24 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5QG
|
4.24 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5QK
|
4.24 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG1
|
PHKG1_HUMAN
|
8Z5QO
|
4.24 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
10 - 385 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
|
CAMK
|
PHKG2
|
PHKG2_HUMAN
|
AF-P15735-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 299 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
|
CAMK
|
PHKG2
|
PHKG2_HUMAN
|
AF-P15735-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
16 - 299 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
|
CAMK
|
PHKG2
|
PHKG2_HUMAN
|
2Y7JA
|
2.5 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B49 |
Type1 |
10 - 293 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
|
CAMK
|
PHKG2
|
PHKG2_HUMAN
|
2Y7JB
|
2.5 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B49 |
Type1 |
10 - 293 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
|
CAMK
|
PHKG2
|
PHKG2_HUMAN
|
2Y7JC
|
2.5 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B49 |
Type1 |
10 - 293 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
|
CAMK
|
PHKG2
|
PHKG2_HUMAN
|
2Y7JD
|
2.5 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
B49 |
Type1 |
10 - 293 |
0 |
None |
None |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4RBLA
|
2.55 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3O7 |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4RC2A
|
2.096 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3O8 |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4RC3A
|
2.338 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3OA |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4RC4A
|
2.651 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3OK |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4I41A
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
MIX,
MIX
|
Type1,
Allosteric
|
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YXTA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YXUA
|
2.24 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YXUB
|
2.24 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YXUC
|
2.24 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
34 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YXUD
|
2.24 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1XR1A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
32 - 308 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3A99A
|
1.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2BZKB
|
2.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YXSA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
33 - 306 |
0 |
None |
P123M |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
AF-P11309-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
30 - 298 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
AF-P11309-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
30 - 298 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YWVA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1XQZA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
32 - 308 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
7VSYA
|
2.141 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
33 - 305 |
0 |
None |
N82K |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4JX3A
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
7OOVA
|
1.96 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
7OOWA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
7OOXA
|
1.97 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5TOEA
|
2.301 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7GK |
Type1 |
34 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YHSA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YI3A
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LY2 |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YI4A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADN |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3C4EA
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C4E |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3C4EB
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C4E |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3C4EC
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C4E |
Type1 |
34 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3C4ED
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C4E |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4K1BA
|
2.082 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1OC |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6NO8A
|
2.377 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
KUY |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6NO9A
|
1.712 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
KUV |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4K0YA
|
1.954 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1OA |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5TELA
|
2.214 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7AJ |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5TEXA
|
2.149 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7AU |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6VRUA
|
2.07 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ROY |
Type1 |
34 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6VRVA
|
1.74 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
WFY |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4DTKA
|
1.86 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7LI |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5KGDA
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6SL |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5KGEA
|
2.23 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6SN |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5KGGA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6SO |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5KGIA
|
2.13 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6SF |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5KGKA
|
2.66 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6SD |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6BSKA
|
2.573 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MVG |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4K18A
|
2.051 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1OB |
Type1 |
32 - 308 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5IISA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6CB |
Type1 |
32 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4TY1A
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
38W |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4WRSA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3U1 |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4WSYA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3U5 |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4WT6A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3U6 |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5EOLA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5QO |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5IPJA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6CD |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5KZIA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6YN |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6MT0A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
JYG |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4MTAA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2D2 |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5C1QB
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4YK |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6L11A
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E2C |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6L12A
|
1.87 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E2R |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6L13A
|
2.24 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E2F |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6L14A
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E2L |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6L15A
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E2O |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6L16A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E2U |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6L17A
|
1.75 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E2X |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
7XSVA
|
2.66 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
I4M |
Type1 |
32 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5KCXA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6S3 |
Type1 |
34 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4MBIA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
26K |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4MBLA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
26L |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YXVA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LI6 |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1YXXA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LI7 |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2O3PA
|
2.24 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
QUE |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2O63A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MYC |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2O64A
|
2.44 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MYU |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2O65A
|
2.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MYF |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3JXWA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LXG |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3JY0A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LYG |
Type1 |
33 - 307 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3JYAA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LWG |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5O11A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3NG |
Type1 |
34 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5O12A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1RO |
Type1 |
34 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5O13A
|
2.44 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9G5 |
Type1 |
34 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5DGZA
|
2.502 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
L20 |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5DHJA
|
2.457 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5E5 |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5DIAA
|
1.964 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5E6 |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5V80A
|
2.252 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
971 |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5V82A
|
1.888 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
96Y |
Type1 |
34 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3UIXA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Q17 |
Type1 |
37 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3UMWA
|
2.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
596 |
Type1 |
37 - 304 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3UMXA
|
2.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Q18 |
Type1 |
37 - 304 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4ENXA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Z20 |
Type1 |
37 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4ENYA
|
2.801 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
J19 |
Type1 |
37 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4LL5A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SK8 |
Type1 |
34 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4LM5A
|
2.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
Q17 |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4LMUA
|
2.38 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
QUE |
Type1 |
36 - 304 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5VUAB
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8GX |
Type1 |
36 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5VUBB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8GU |
Type1 |
36 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5VUCB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8GR |
Type1 |
36 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3R00A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UNJ |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3R01A
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UNE |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3R02A
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UNM |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3R04A
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UNQ |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3VBQA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0F5 |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3VBTA
|
2.23 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0F9 |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3VBVA
|
2.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0FK |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3VBWA
|
2.48 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0FN |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3VBXA
|
2.03 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0FO |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3VBYA
|
2.27 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0FR |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3VC4A
|
2.23 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0FS |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3F2AA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
985 |
Type1 |
32 - 308 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2XIXA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XIX |
Type1 |
33 - 306 |
0 |
SEP261,SEP276 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2XIYA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XIY |
Type1 |
33 - 306 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2XIZA
|
2.21 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XIZ |
Type1 |
33 - 306 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2XJ0A
|
3.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XJ0 |
Type1 |
33 - 307 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2XJ1A
|
2.13 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XJ1 |
Type1 |
33 - 306 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2XJ2A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
985 |
Type1 |
33 - 306 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4A7CA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
E46 |
Type1 |
32 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
1XWSA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI1 |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4BZNA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UGX |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4BZOA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
676 |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
7ZUNA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
JYO |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4XHKB
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3YR |
Type1 |
32 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4JX7A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1N6 |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4ALVA
|
2.59 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R9P |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4ALWA
|
1.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HY7 |
Type1 |
34 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3DCVA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
55E |
Type1 |
32 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4N6YA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2HV |
Type1 |
32 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4N6ZA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2HW |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4N70A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2HX |
Type1 |
32 - 306 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5DWRA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5H7 |
Type1 |
33 - 306 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6YKDA
|
1.86 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
OWB |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2OBJA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VRV |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3BGPA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VX1 |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3BGQA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VX2 |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3BGZA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VX3 |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3WE8A
|
1.954 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RUI |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4AS0A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RPS |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5TURA
|
2.948 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7LK |
Type1 |
34 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2J2IB
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LY4 |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
7QB2A
|
2.53 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A7X |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
7QFMA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AY3 |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3JPVA
|
2.35 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1DR |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3MA3A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
01I |
Type1 |
37 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3QF9A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NM8 |
Type1 |
32 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4GW8A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3RA |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6PCWA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
O97 |
Type1 |
32 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6PDIA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
OCJ |
Type1 |
32 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6PDNA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
OD4 |
Type1 |
32 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6PDOA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
OD1 |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6PDPA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
OBY |
Type1 |
36 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6QXKB
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
JKW |
Type1 |
35 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R0HA
|
1.88 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8UB |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R0QA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XGB |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R0WA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XGF |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R0YA
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XH3 |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R10A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XGQ |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R18A
|
1.89 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XGK |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R1KA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XHI |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R1NA
|
2.21 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XIT |
Type1 |
34 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R1PA
|
2.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XIP |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R1TA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XIJ |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R1WA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XIW |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R25A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XJL |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8R27A
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
XJW |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2BIKB
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI1 |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2BILB
|
2.55 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
BI1 |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2BZHB
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HB1 |
Type1 |
32 - 306 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2BZIB
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DW2 |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2BZJA
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ME3 |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2C3IB
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IYZ |
Type1 |
37 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
2OI4X
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
JM1 |
Type1 |
32 - 306 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3BWFA
|
2.35 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DWC |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5MZLA
|
1.955 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8ET |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N4NA
|
2.09 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8M8 |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N4OA
|
2.22 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8MB |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N4RA
|
2.13 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8MQ |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N4UA
|
2.202 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8MZ |
Type1 |
34 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N4VA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8MW |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N4XA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8MT |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N4YA
|
2.56 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8N5 |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N4ZA
|
2.257 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8MK |
Type1 |
34 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N50A
|
1.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8MN |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N51A
|
2.118 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8N8 |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N52A
|
2.252 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8N2 |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N5LA
|
1.97 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8NZ |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5N5MA
|
2.21 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8O8 |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
5NDTA
|
1.985 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
8UB |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
7Z6UA
|
2.28 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IJB |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3CXWA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7CP |
Type1 |
33 - 306 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3CY2A
|
2.01 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MB9 |
Type1 |
33 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3CY3A
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
JN5 |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4RPVA
|
3.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3UR |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
8AFRA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
M0F |
Type1 |
33 - 305 |
0 |
SEP261 |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4ALUA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
79O |
Type1 |
33 - 306 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
3T9IA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3T9 |
Type1.5_Back |
33 - 306 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6AYDA
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C2J |
Type1.5_Back |
34 - 305 |
0 |
None |
R250G |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
6KZIA
|
2.8 |
Inactive |
DFGin‑BLBminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RTX |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4IAAA
|
2.85 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RTZ |
Type1 |
33 - 305 |
0 |
SEP261 |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM1
|
PIM1_HUMAN
|
4XH6A
|
2.04 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HUL |
Type1 |
33 - 305 |
0 |
None |
None |
Serine/threonine-protein kinase pim-1 |
|
CAMK
|
PIM2
|
PIM2_HUMAN
|
AF-Q9P1W9-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
24 - 294 |
0 |
None |
None |
Serine/threonine-protein kinase pim-2 |
|
CAMK
|
PIM2
|
PIM2_HUMAN
|
AF-Q9P1W9-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
24 - 294 |
0 |
None |
None |
Serine/threonine-protein kinase pim-2 |
|
CAMK
|
PIM2
|
PIM2_HUMAN
|
2IWIA
|
2.8 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HB1 |
Type1 |
32 - 288 |
0 |
None |
None |
Serine/threonine-protein kinase pim-2 |
|
CAMK
|
PIM2
|
PIM2_HUMAN
|
2IWIB
|
2.8 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HB1 |
Type1 |
22 - 287 |
0 |
None |
None |
Serine/threonine-protein kinase pim-2 |
|
CAMK
|
PIM2
|
PIM2_HUMAN
|
4X7QA
|
2.33 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
3YR |
Type1 |
32 - 287 |
0 |
None |
None |
Serine/threonine-protein kinase pim-2 |
|
CAMK
|
PIM2
|
PIM2_HUMAN
|
4X7QB
|
2.33 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
3YR |
Type1 |
27 - 287 |
0 |
None |
None |
Serine/threonine-protein kinase pim-2 |
|
CAMK
|
PIM3
|
PIM3_HUMAN
|
AF-Q86V86-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
32 - 301 |
0 |
None |
None |
Serine/threonine-protein kinase pim-3 |
|
CAMK
|
PIM3
|
PIM3_HUMAN
|
AF-Q86V86-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
32 - 301 |
0 |
None |
None |
Serine/threonine-protein kinase pim-3 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
8X72A
|
2.2 |
Inactive |
DFGin‑BLAminus |
out-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
ANP |
ATPlike |
37 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2OU7A
|
2.4 |
Inactive |
DFGin‑BLAminus |
out-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
ANP |
ATPlike |
37 - 328 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
AF-P53350-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
45 - 313 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
AF-P53350-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
45 - 313 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2V5QA
|
2.3 |
Inactive |
DFGin‑BLAminus |
out-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
No_ligand |
No_ligand |
39 - 323 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2V5QB
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
No_ligand |
No_ligand |
39 - 323 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2YACA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_ioio |
937 |
Type1 |
39 - 329 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
3KB7A
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iooo |
071 |
Type1 |
39 - 328 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
4A4LA
|
2.35 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_ioio |
939 |
Type1 |
39 - 329 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
4A4OA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
664 |
Type1 |
39 - 329 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R8BA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
A1JCP |
Type1 |
37 - 326 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R8BB
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iiio |
A1JCP |
Type1 |
37 - 323 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R8CA
|
2.243 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
R78 |
Type1 |
38 - 326 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R8CB
|
2.243 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
R78 |
Type1 |
38 - 323 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
4J52A
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
1J3 |
Type1 |
38 - 330 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
4J53A
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
1J4 |
Type1 |
38 - 330 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2RKUA
|
1.95 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
R78 |
Type1 |
37 - 330 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
8BJTA
|
2.188 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iooo |
8X7 |
Type1 |
39 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
3THBA
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_ioio |
3TA |
Type1 |
42 - 328 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
2OWBA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
626 |
Type1 |
37 - 330 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
3FC2A
|
2.45 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
IBI |
Type1 |
37 - 329 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9D0PA
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
8X7 |
Type1 |
37 - 330 |
0 |
None |
T210V |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1WAAA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
A1JCP |
Type1 |
38 - 334 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1WBBB
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
A1JCP |
Type1 |
38 - 325 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1XA
|
2.84 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
R78 |
Type1 |
39 - 334 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1XB
|
2.84 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
R78 |
Type1 |
39 - 326 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1YAAA
|
2.602 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
A1JCQ |
Type1 |
38 - 334 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
9R1YBBB
|
2.602 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_ioio |
A1JCQ |
Type1 |
38 - 325 |
0 |
None |
K225D,K226A |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
5TA6A
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_ioio |
79D |
Type1 |
37 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK1
|
PLK1_HUMAN
|
5TA8A
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_ioio |
79C |
Type1 |
37 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase PLK1 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
AF-Q9NYY3-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
74 - 342 |
0 |
None |
None |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
AF-Q9NYY3-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
74 - 342 |
0 |
None |
None |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
4I5MA
|
1.801 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
R78 |
Type1 |
71 - 354 |
0 |
None |
C83S,V87T,A119S,A216S,C259A,C291S,L335T |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
4I5PA
|
1.738 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
1D1 |
Type1 |
71 - 354 |
0 |
None |
C83S,V87T,A119S,A216S,C259A,C291S,L335T |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
4I6BA
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
11G |
Type1 |
71 - 355 |
0 |
None |
C83S,V87T,A119S,A216S,C259A,C291S,L335T |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
4I6FA
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
1C7 |
Type1 |
71 - 355 |
0 |
None |
C83S,V87T,A119S,A216S,C259A,C291S,L335T |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK2
|
PLK2_HUMAN
|
4I6HA
|
1.91 |
Inactive |
DFGin‑BLBminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
1C8 |
Type1 |
71 - 355 |
0 |
None |
C83S,V87T,A119S,A216S,C259A,C291S,L335T |
Serine/threonine-protein kinase PLK2 |
|
CAMK
|
PLK3
|
PLK3_HUMAN
|
AF-Q9H4B4-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
54 - 322 |
0 |
None |
None |
Serine/threonine-protein kinase PLK3 |
|
CAMK
|
PLK3
|
PLK3_HUMAN
|
AF-Q9H4B4-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
54 - 322 |
0 |
None |
None |
Serine/threonine-protein kinase PLK3 |
|
CAMK
|
PLK3
|
PLK3_HUMAN
|
4B6LA
|
1.9 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9ZP |
Type1 |
52 - 332 |
0 |
None |
None |
Serine/threonine-protein kinase PLK3 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
9O63A
|
2.26 |
Inactive |
DFGin‑ABAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
A1CAD |
Type1 |
2 - 266 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
3COKA
|
2.25 |
Inactive |
DFGin‑BLAminus |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ANP |
ATPlike |
2 - 266 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
3COKB
|
2.25 |
Inactive |
DFGin‑BLAminus |
in-out |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ANP |
ATPlike |
2 - 266 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
AF-O00444-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
AF-O00444-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 273 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
4JXFA
|
2.4 |
Inactive |
DFGin‑None |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
631 |
Type1 |
4 - 267 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PLK4
|
PLK4_HUMAN
|
4YURA
|
2.65 |
Inactive |
DFGin‑None |
out-out |
none-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
4J7 |
Type1 |
5 - 266 |
0 |
None |
None |
Serine/threonine-protein kinase PLK4 |
|
CAMK
|
PNCK
|
KCC1B_HUMAN
|
AF-Q6P2M8-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 278 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1B |
|
CAMK
|
PNCK
|
KCC1B_HUMAN
|
AF-Q6P2M8-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
7 - 278 |
0 |
None |
None |
Calcium/calmodulin-dependent protein kinase type 1B |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
6C9FA
|
2.924 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
R34,
STU
|
Allosteric,
Type1
|
22 - 558 |
0 |
TPO183 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
7JIJA
|
5.5 |
Inactive |
DFGin‑ABAminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
22 - 559 |
0 |
TPO183 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
6C9GA
|
2.7 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
R93,
STU
|
Allosteric,
Type1
|
22 - 558 |
0 |
TPO183 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
6C9HA
|
2.65 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
R34,
STU
|
Allosteric,
Type1
|
22 - 558 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
6C9JA
|
3.05 |
Active |
DFGin‑BLAminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R34,
STU
|
Allosteric,
Type1
|
22 - 559 |
0 |
TPO183 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
AF-Q13131-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 287 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
AF-Q13131-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 287 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
7JHHA
|
3.92 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooo |
No_ligand |
No_ligand |
22 - 559 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
7JHGA
|
3.47 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
TAK |
Type1 |
22 - 559 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
7M74A
|
3.93 |
Inactive |
DFGin‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
TAK |
Type1 |
22 - 559 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
4RERA
|
4.047 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU |
Type1 |
20 - 559 |
0 |
TPO183 |
E480G,E483A,K485A |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
4REWA
|
4.58 |
Inactive |
DFGin‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
STU |
Type1 |
20 - 559 |
0 |
None |
E480G,E483A,K485A |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
4REDA
|
2.95 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoo |
APEdist_nnnn |
No_ligand |
No_ligand |
22 - 360 |
0 |
None |
K52A |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA1
|
AAPK1_HUMAN
|
4REDB
|
2.95 |
Inactive |
DFGinter‑None |
out-out |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
22 - 360 |
0 |
None |
K52A |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
5ISOA
|
2.63 |
Inactive |
DFGin‑ABAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
992
|
Type1,
Allosteric
|
9 - 551 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
5ISOC
|
2.63 |
Inactive |
DFGin‑ABAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
992
|
Type1,
Allosteric
|
9 - 550 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
6B1UC
|
2.77 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
CG7
|
Type1,
Allosteric
|
9 - 552 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
AF-P54646-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
8 - 276 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
AF-P54646-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
8 - 276 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4ZHXA
|
2.99 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
4O7 |
Type1 |
9 - 550 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4CFFA
|
3.924 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiii |
STU |
Type1 |
8 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
8BIKA
|
2.5 |
Inactive |
DFGin‑BLAminus |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
QTN
|
Type1,
Allosteric
|
8 - 551 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
8BIKD
|
2.5 |
Inactive |
DFGin‑BLAminus |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
QTN
|
Type1,
Allosteric
|
9 - 551 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
6B2EA
|
3.8 |
Inactive |
DFGin‑BLAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiio |
STU,
CG7
|
Type1,
Allosteric
|
9 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4CFEA
|
3.023 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiii |
STU,
992
|
Type1,
Allosteric
|
8 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4CFEC
|
3.023 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiii |
STU,
992
|
Type1,
Allosteric
|
10 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
7MYJA
|
2.95 |
Inactive |
DFGin‑BLBminus |
out-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4O7,
ZQV
|
Type1,
Allosteric
|
7 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
7MYJC
|
2.95 |
Inactive |
DFGin‑None |
out-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
4O7 |
Type1 |
8 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
5EZVA
|
2.99 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
STU,
C1V
|
Type1,
Allosteric
|
8 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
5EZVC
|
2.99 |
Inactive |
DFGin‑None |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
C1V
|
Type1,
Allosteric
|
9 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4ZHXC
|
2.99 |
Inactive |
DFGin‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_iiio |
4O7,
C1V
|
Type1,
Allosteric
|
9 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
6B1UA
|
2.77 |
Inactive |
DFGin‑None |
out-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
STU,
CG7
|
Type1,
Allosteric
|
8 - 550 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
4CFFC
|
3.924 |
Inactive |
DFGin‑None |
out-out |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_iiii |
STU,
C1V
|
Type1,
Allosteric
|
10 - 551 |
0 |
TPO172 |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
2H6DA
|
1.85 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
10 - 278 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
2YZAA
|
3.02 |
Inactive |
DFGout‑BBAminus |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
10 - 278 |
0 |
None |
T172D |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
9IC2A
|
2.5 |
Inactive |
None‑None |
out-out |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nooo |
A1I1Y |
Type1 |
8 - 279 |
0 |
None |
None |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
3AQVA
|
2.08 |
Inactive |
None‑None |
out-out |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
TAK |
Type1 |
7 - 279 |
0 |
None |
T172D |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKAA2
|
AAPK2_HUMAN
|
6BX6A
|
2.9 |
Inactive |
None‑None |
out-none |
out-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
EDJ |
Type1 |
13 - 277 |
0 |
None |
T172D |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
|
CAMK
|
PRKD1
|
KPCD1_HUMAN
|
AF-Q15139-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
575 - 847 |
0 |
None |
None |
Serine/threonine-protein kinase D1 |
|
CAMK
|
PRKD1
|
KPCD1_HUMAN
|
AF-Q15139-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
575 - 847 |
0 |
None |
None |
Serine/threonine-protein kinase D1 |
|
CAMK
|
PRKD2
|
KPCD2_HUMAN
|
AF-Q9BZL6-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
543 - 815 |
0 |
None |
None |
Serine/threonine-protein kinase D2 |
|
CAMK
|
PRKD2
|
KPCD2_HUMAN
|
AF-Q9BZL6-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
543 - 815 |
0 |
None |
None |
Serine/threonine-protein kinase D2 |
|
CAMK
|
PRKD3
|
KPCD3_HUMAN
|
AF-O94806-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
568 - 840 |
0 |
None |
None |
Serine/threonine-protein kinase D3 |
|
CAMK
|
PRKD3
|
KPCD3_HUMAN
|
AF-O94806-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
568 - 840 |
0 |
None |
None |
Serine/threonine-protein kinase D3 |
|
CAMK
|
PSKH1
|
KPSH1_HUMAN
|
AF-P11801-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
90 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase H1 |
|
CAMK
|
PSKH1
|
KPSH1_HUMAN
|
AF-P11801-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
90 - 363 |
0 |
None |
None |
Serine/threonine-protein kinase H1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
2WNTA
|
2.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanin |
APEdist_oooo |
No_ligand |
No_ligand |
416 - 708 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
2WNTB
|
2.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oooo |
No_ligand |
No_ligand |
415 - 709 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
3RNYA
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oooo |
No_ligand |
No_ligand |
418 - 707 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
3RNYB
|
2.7 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oooo |
No_ligand |
No_ligand |
419 - 708 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
AF-Q15418-K2A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
410 - 683 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
AF-Q15418-K4A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
410 - 683 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
8WF4A
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanin |
APEdist_oooo |
No_ligand |
No_ligand |
416 - 708 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
8WF4B
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiin |
APEdist_oooo |
No_ligand |
No_ligand |
415 - 708 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
4NIFA
|
2.15 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_oooo |
No_ligand |
No_ligand |
413 - 728 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA1-2
|
KS6A1_HUMAN
|
4NIFD
|
2.15 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aannn |
APEdist_ooon |
No_ligand |
No_ligand |
413 - 728 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-1 |
|
CAMK
|
RPS6KA2-2
|
KS6A2_HUMAN
|
AF-Q15349-K2A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
407 - 680 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-2 |
|
CAMK
|
RPS6KA2-2
|
KS6A2_HUMAN
|
AF-Q15349-K4A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
407 - 680 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-2 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
4D9TA
|
2.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oooo |
0JG |
Type1 |
415 - 713 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
4D9UA
|
2.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oooo |
0JH |
Type1 |
408 - 714 |
0 |
None |
K591E |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
AF-P51812-K2A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
414 - 687 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
AF-P51812-K4A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
414 - 687 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
8XEYA
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oooo |
No_ligand |
No_ligand |
403 - 714 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
4JG8A
|
3.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_oooo |
1LE |
Type1 |
415 - 714 |
0 |
None |
T493M |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
4JG6A
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oooo |
1LB |
Type1 |
406 - 712 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA3-2
|
KS6A3_HUMAN
|
4JG7A
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oooo |
1LC |
Type1 |
405 - 713 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-3 |
|
CAMK
|
RPS6KA4-2
|
KS6A4_HUMAN
|
AF-O75676-K2A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
400 - 682 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-4 |
|
CAMK
|
RPS6KA4-2
|
KS6A4_HUMAN
|
AF-O75676-K4A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
400 - 682 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-4 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
3KN5A
|
2.4 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ANP |
ATPlike |
415 - 729 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
3KN5B
|
2.4 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
ANP |
ATPlike |
415 - 729 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
AF-O75582-K2A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
415 - 695 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
AF-O75582-K4A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
415 - 695 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
3KN6A
|
2.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
415 - 729 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
3KN6B
|
2.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
No_ligand |
No_ligand |
415 - 729 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
7UP4A
|
3.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
O1K |
Type1 |
415 - 723 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
7UP4B
|
3.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
O1K |
Type1 |
415 - 728 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
7UP5A
|
2.8 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
O1R |
Type1 |
415 - 723 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
7UP5B
|
2.8 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
O1R |
Type1 |
415 - 728 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
7UP7A
|
2.8 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
1LE |
Type1 |
415 - 725 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
7UP7B
|
2.8 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
1LE |
Type1 |
416 - 728 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
7UP8A
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
O10 |
Type1 |
415 - 723 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
7UP8B
|
2.9 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
O10 |
Type1 |
415 - 727 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA5-2
|
KS6A5_HUMAN
|
7UP6A
|
2.6 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aannn |
APEdist_nnnn |
SUU,
OXM,
OXM
|
Type1,
Allosteric,
Allosteric
|
416 - 707 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-5 |
|
CAMK
|
RPS6KA6-2
|
KS6A6_HUMAN
|
AF-Q9UK32-K2A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
418 - 691 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
|
CAMK
|
RPS6KA6-2
|
KS6A6_HUMAN
|
AF-Q9UK32-K4A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
418 - 691 |
0 |
None |
None |
Ribosomal protein S6 kinase alpha-6 |
|
CAMK
|
SIK1
|
SIK1_HUMAN
|
AF-P57059-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 286 |
0 |
None |
None |
Serine/threonine-protein kinase SIK1 |
|
CAMK
|
SIK1
|
SIK1_HUMAN
|
AF-P57059-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 286 |
0 |
None |
None |
Serine/threonine-protein kinase SIK1 |
|
CAMK
|
SIK2
|
SIK2_HUMAN
|
AF-Q9H0K1-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 279 |
0 |
None |
None |
Serine/threonine-protein kinase SIK2 |
|
CAMK
|
SIK2
|
SIK2_HUMAN
|
AF-Q9H0K1-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 279 |
0 |
None |
None |
Serine/threonine-protein kinase SIK2 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4VB
|
1.9 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XWA |
Type1 |
61 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4VC
|
1.9 |
Inactive |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XWA |
Type1 |
61 - 385 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
AF-Q9Y2K2-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
58 - 325 |
0 |
None |
None |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
AF-Q9Y2K2-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
58 - 325 |
0 |
None |
None |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OA
|
2.725 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OC
|
2.725 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OE
|
2.725 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OG
|
2.725 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OI
|
2.725 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4OK
|
2.725 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XVI |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QA
|
2.838 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QC
|
2.838 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QE
|
2.838 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QG
|
2.838 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QI
|
2.838 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4QK
|
2.838 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DB8 |
Type1 |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4VA
|
1.9 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XWA |
Type1 |
62 - 385 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8OKUA
|
3.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VRU |
Type1 |
60 - 392 |
0 |
None |
T221D |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8OKUB
|
3.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
VRU |
Type1 |
60 - 390 |
0 |
None |
T221D |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4UA
|
2.416 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XW3 |
Type1.5_Front |
61 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4UC
|
2.416 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XW3 |
Type1.5_Front |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4UE
|
2.416 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XW3 |
Type1.5_Front |
61 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SIK3
|
SIK3_HUMAN
|
8R4UG
|
2.416 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
XW3 |
Type1.5_Front |
62 - 384 |
0 |
TPO221 |
C121S,C181S,C333S |
Serine/threonine-protein kinase SIK3 |
|
CAMK
|
SNRK
|
SNRK_HUMAN
|
AF-Q9NRH2-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
8 - 277 |
0 |
None |
None |
SNF-related serine/threonine-protein kinase |
|
CAMK
|
SNRK
|
SNRK_HUMAN
|
AF-Q9NRH2-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
8 - 277 |
0 |
None |
None |
SNF-related serine/threonine-protein kinase |
|
CAMK
|
SNRK
|
SNRK_HUMAN
|
5YKSA
|
2.9 |
Inactive |
DFGin‑BLBminus |
out-out |
none-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
1 - 344 |
0 |
None |
None |
SNF-related serine/threonine-protein kinase |
|
CAMK
|
SNRK
|
SNRK_HUMAN
|
5YKSB
|
2.9 |
Inactive |
DFGin‑BLBminus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 344 |
0 |
None |
None |
SNF-related serine/threonine-protein kinase |
|
CAMK
|
SPEG-1
|
SPEG_HUMAN
|
AF-Q15772-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1593 - 1862 |
0 |
None |
None |
Striated muscle preferentially expressed protein kinase |
|
CAMK
|
SPEG-1
|
SPEG_HUMAN
|
AF-Q15772-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1593 - 1862 |
0 |
None |
None |
Striated muscle preferentially expressed protein kinase |
|
CAMK
|
SPEG-2
|
SPEG_HUMAN
|
AF-Q15772-K2A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2958 - 3226 |
0 |
None |
None |
Striated muscle preferentially expressed protein kinase |
|
CAMK
|
SPEG-2
|
SPEG_HUMAN
|
AF-Q15772-K4A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2958 - 3226 |
0 |
None |
None |
Striated muscle preferentially expressed protein kinase |
|
CAMK
|
STK11
|
STK11_HUMAN
|
2WTKC
|
2.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
47 - 342 |
0 |
None |
D194A |
Serine/threonine-protein kinase STK11 |
|
CAMK
|
STK11
|
STK11_HUMAN
|
2WTKF
|
2.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ANP |
ATPlike |
45 - 340 |
0 |
None |
D194A |
Serine/threonine-protein kinase STK11 |
|
CAMK
|
STK11
|
STK11_HUMAN
|
AF-Q15831-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 317 |
0 |
None |
None |
Serine/threonine-protein kinase STK11 |
|
CAMK
|
STK11
|
STK11_HUMAN
|
AF-Q15831-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 317 |
0 |
None |
None |
Serine/threonine-protein kinase STK11 |
|
CAMK
|
STK11
|
STK11_HUMAN
|
8VSUC
|
2.86 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
41 - 347 |
0 |
None |
None |
Serine/threonine-protein kinase STK11 |
|
CAMK
|
STK17A
|
ST17A_HUMAN
|
7QUEB
|
2.4 |
Inactive |
DFGin‑ABAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_oooo |
F7I |
Type1 |
59 - 322 |
0 |
None |
None |
Serine/threonine-protein kinase 17A |
|
CAMK
|
STK17A
|
ST17A_HUMAN
|
7QUFA
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
F8I |
Type1 |
50 - 322 |
0 |
None |
None |
Serine/threonine-protein kinase 17A |
|
CAMK
|
STK17A
|
ST17A_HUMAN
|
7QUFB
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
F8I |
Type1 |
55 - 322 |
0 |
None |
None |
Serine/threonine-protein kinase 17A |
|
CAMK
|
STK17A
|
ST17A_HUMAN
|
AF-Q9UEE5-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
51 - 329 |
0 |
None |
None |
Serine/threonine-protein kinase 17A |
|
CAMK
|
STK17A
|
ST17A_HUMAN
|
AF-Q9UEE5-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
51 - 329 |
0 |
None |
None |
Serine/threonine-protein kinase 17A |
|
CAMK
|
STK17A
|
ST17A_HUMAN
|
7QUEA
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
F7I |
Type1 |
50 - 322 |
0 |
None |
None |
Serine/threonine-protein kinase 17A |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
6QF4A
|
2.495 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nioo |
ADP |
ATPlike |
18 - 308 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
7Q7CA
|
2.85 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
ADP |
ATPlike |
25 - 297 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
7Q7DA
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
ATP |
ATPlike |
25 - 297 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
7Q7EA
|
2.85 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
ATP |
ATPlike |
25 - 297 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
AF-O94768-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
24 - 301 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
AF-O94768-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
24 - 301 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
3LM0A
|
2.35 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
EBD |
Type1 |
25 - 304 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
6Y6FA
|
1.98 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
OD2 |
Type1 |
25 - 309 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
6Y6HA
|
1.95 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
OBW |
Type1 |
25 - 309 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
6ZJFA
|
1.75 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
QM2 |
Type1 |
25 - 309 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
7AKGA
|
2.08 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioo |
38O |
Type1 |
25 - 309 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK17B
|
ST17B_HUMAN
|
3LM5A
|
2.29 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
QUE |
Type1.5_Back |
25 - 301 |
0 |
None |
None |
Serine/threonine-protein kinase 17B |
|
CAMK
|
STK33
|
STK33_HUMAN
|
AF-Q9BYT3-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
108 - 389 |
0 |
None |
None |
Serine/threonine-protein kinase 33 |
|
CAMK
|
STK33
|
STK33_HUMAN
|
AF-Q9BYT3-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
108 - 389 |
0 |
None |
None |
Serine/threonine-protein kinase 33 |
|
CAMK
|
STK33
|
STK33_HUMAN
|
8VF6A
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-out |
in-none |
nonTYR |
APEdihe_aanii |
APEdist_nnnn |
A1AAY |
Type1 |
100 - 382 |
0 |
None |
None |
Serine/threonine-protein kinase 33 |
|
CAMK
|
STK33
|
STK33_HUMAN
|
8VF6B
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
A1AAY |
Type1 |
99 - 383 |
0 |
None |
None |
Serine/threonine-protein kinase 33 |
|
CAMK
|
STK40
|
STK40_HUMAN
|
5L2QA
|
2.53 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
26 - 336 |
0 |
None |
None |
Serine/threonine-protein kinase 40 |
|
CAMK
|
STK40
|
STK40_HUMAN
|
5L2QB
|
2.53 |
Pseudo |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
30 - 336 |
0 |
None |
None |
Serine/threonine-protein kinase 40 |
|
CAMK
|
STK40
|
STK40_HUMAN
|
5L2QC
|
2.53 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
37 - 335 |
0 |
None |
None |
Serine/threonine-protein kinase 40 |
|
CAMK
|
STK40
|
STK40_HUMAN
|
5L2QD
|
2.53 |
Pseudo |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
30 - 336 |
0 |
None |
None |
Serine/threonine-protein kinase 40 |
|
CAMK
|
TRIB1
|
TRIB1_HUMAN
|
6DC0A
|
2.8 |
Pseudo |
DFGin‑ABAminus |
in-na |
in-out |
nonTYR |
APEdihe_aaiai |
APEdist_iioi |
No_ligand |
No_ligand |
90 - 67 |
0 |
None |
None |
Tribbles homolog 1 |
|
CAMK
|
TRIB1
|
TRIB1_HUMAN
|
6DC0B
|
2.8 |
Pseudo |
DFGin‑ABAminus |
in-na |
in-out |
nonTYR |
APEdihe_aaiai |
APEdist_iioi |
No_ligand |
No_ligand |
90 - 74 |
0 |
None |
None |
Tribbles homolog 1 |
|
CAMK
|
TRIB1
|
TRIB1_HUMAN
|
5CEKA
|
2.8 |
Pseudo |
DFGinter‑None |
out-na |
none-out |
nonTYR |
APEdihe_aanao |
APEdist_nnnn |
No_ligand |
No_ligand |
88 - 342 |
0 |
None |
None |
Tribbles homolog 1 |
|
CAMK
|
TRIB1
|
TRIB1_HUMAN
|
5CEMA
|
2.1 |
Pseudo |
DFGinter‑None |
out-na |
none-out |
nonTYR |
APEdihe_aaiao |
APEdist_oooo |
No_ligand |
No_ligand |
88 - 364 |
0 |
None |
None |
Tribbles homolog 1 |
|
CAMK
|
TRIB2
|
TRIB2_HUMAN
|
7UPMA
|
2.7 |
Pseudo |
DFGin‑ABAminus |
in-na |
in-out |
nonTYR |
APEdihe_aaiai |
APEdist_iooi |
No_ligand |
No_ligand |
55 - 312 |
0 |
None |
None |
Tribbles homolog 2 |
|
CAMK
|
TRIO
|
TRIO_HUMAN
|
AF-O75962-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiai |
APEdist_iiii |
No_ligand |
No_ligand |
2788 - 3058 |
0 |
None |
None |
Triple functional domain protein |
|
CAMK
|
TRIO
|
TRIO_HUMAN
|
AF-O75962-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiai |
APEdist_iiii |
No_ligand |
No_ligand |
2788 - 3058 |
0 |
None |
None |
Triple functional domain protein |
|
CAMK
|
TSSK1B
|
TSSK1_HUMAN
|
AF-Q9BXA7-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 280 |
0 |
None |
None |
Testis-specific serine/threonine-protein kinase 1 |
|
CAMK
|
TSSK1B
|
TSSK1_HUMAN
|
AF-Q9BXA7-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 280 |
0 |
None |
None |
Testis-specific serine/threonine-protein kinase 1 |
|
CAMK
|
TSSK2
|
TSSK2_HUMAN
|
AF-Q96PF2-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 280 |
0 |
None |
None |
Testis-specific serine/threonine-protein kinase 2 |
|
CAMK
|
TSSK2
|
TSSK2_HUMAN
|
AF-Q96PF2-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 280 |
0 |
None |
None |
Testis-specific serine/threonine-protein kinase 2 |
|
CAMK
|
TSSK3
|
TSSK3_HUMAN
|
AF-Q96PN8-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 268 |
0 |
None |
None |
Testis-specific serine/threonine-protein kinase 3 |
|
CAMK
|
TSSK3
|
TSSK3_HUMAN
|
AF-Q96PN8-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 268 |
0 |
None |
None |
Testis-specific serine/threonine-protein kinase 3 |
|
CAMK
|
TSSK4
|
TSSK4_HUMAN
|
AF-Q6SA08-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
17 - 301 |
0 |
None |
None |
Testis-specific serine/threonine-protein kinase 4 |
|
CAMK
|
TSSK4
|
TSSK4_HUMAN
|
AF-Q6SA08-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
17 - 301 |
0 |
None |
None |
Testis-specific serine/threonine-protein kinase 4 |
|
CAMK
|
TSSK6
|
TSSK6_HUMAN
|
AF-Q9BXA6-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 273 |
0 |
None |
None |
Testis-specific serine/threonine-protein kinase 6 |
|
CAMK
|
TSSK6
|
TSSK6_HUMAN
|
AF-Q9BXA6-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 273 |
0 |
None |
None |
Testis-specific serine/threonine-protein kinase 6 |
|
CAMK
|
TTN
|
TITIN_HUMAN
|
1TKIA
|
2.0 |
Pseudo |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_iioo |
No_ligand |
No_ligand |
32172 - 32492 |
0 |
None |
None |
Titin |
|
CAMK
|
TTN
|
TITIN_HUMAN
|
1TKIB
|
2.0 |
Pseudo |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_iioo |
No_ligand |
No_ligand |
32172 - 32492 |
0 |
None |
None |
Titin |
|
CAMK
|
TTN
|
TITIN_HUMAN
|
4JNWA
|
2.06 |
Pseudo |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_iioo |
No_ligand |
No_ligand |
32172 - 32491 |
0 |
None |
None |
Titin |
|
CAMK
|
TTN
|
TITIN_HUMAN
|
4JNWB
|
2.06 |
Pseudo |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_iooo |
No_ligand |
No_ligand |
32172 - 32492 |
0 |
None |
None |
Titin |
|
CAMK
|
TTN
|
TITIN_HUMAN
|
6YGNA
|
2.4 |
Pseudo |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_iioo |
No_ligand |
No_ligand |
32046 - 32594 |
0 |
None |
None |
Titin |
|
CAMK
|
TTN
|
TITIN_HUMAN
|
6YGNB
|
2.4 |
Pseudo |
DFGin‑ABAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaini |
APEdist_iioo |
No_ligand |
No_ligand |
32046 - 32594 |
0 |
None |
None |
Titin |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
AF-P48729-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
9 - 291 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
AF-P48729-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
9 - 291 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
9OTYC
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
No_ligand |
No_ligand |
10 - 299 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
7WTTA
|
3.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
9 - 305 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
5FQDC
|
2.45 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 303 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
5FQDF
|
2.45 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 303 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
8G66C
|
3.45 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iini |
No_ligand |
No_ligand |
10 - 303 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
8G66F
|
3.45 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaini |
APEdist_iiii |
No_ligand |
No_ligand |
10 - 303 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1
|
KC1A_HUMAN
|
6GZDA
|
2.28 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LCI |
Type1 |
9 - 305 |
0 |
None |
None |
Casein kinase I isoform alpha |
|
CK1
|
CSNK1A1L
|
KC1AL_HUMAN
|
AF-Q8N752-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
9 - 291 |
0 |
None |
None |
Casein kinase I isoform alpha-like |
|
CK1
|
CSNK1A1L
|
KC1AL_HUMAN
|
AF-Q8N752-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
9 - 291 |
0 |
None |
None |
Casein kinase I isoform alpha-like |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RU6A
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ACP |
ATPlike |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RU6B
|
2.05 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
ACP |
ATPlike |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7P7FA
|
1.96 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
3 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7P7FB
|
1.96 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
3 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7P7GA
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
AMP |
ATPlike |
8 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7P7GB
|
1.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
AMP |
ATPlike |
7 - 293 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7P7HA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7P7HB
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AMP |
ATPlike |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
AF-P48730-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 283 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
AF-P48730-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 283 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5IH4A
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6PXOA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 292 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6PXOB
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 292 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RCHB
|
1.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
3UYSA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
3UYSB
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
3UYSC
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
3UYSD
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7MA
|
2.25 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7MB
|
2.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7NA
|
1.66 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7NB
|
1.66 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7OA
|
1.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7OB
|
1.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7PA
|
2.25 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8D7PB
|
2.25 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 290 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4TN6B
|
2.41 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 292 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
9B3SA
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 415 |
0 |
SEP411 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
9B3SB
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 414 |
0 |
SEP411 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6PXPA
|
2.35 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 293 |
0 |
None |
K171E |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6PXPB
|
2.35 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 294 |
0 |
None |
K171E |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6PXNA
|
1.551 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
2 - 291 |
0 |
None |
R178C |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6PXNB
|
1.551 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 294 |
0 |
None |
R178C |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8IZCA
|
1.45 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
S93 |
Type1 |
5 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8IZCB
|
1.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
S93 |
Type1 |
5 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5IH5A
|
2.25 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AUE |
Type1 |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5IH6A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
AUG |
Type1 |
2 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RCGA
|
1.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
K0E |
Type1 |
1 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7P7FC
|
1.96 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADN |
Type1 |
4 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7P7FD
|
1.96 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADN |
Type1 |
4 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QR9A
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZQ |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QR9B
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZQ |
Type1 |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QR9C
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZQ |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QR9D
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EZQ |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QRAA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EYI |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QRAB
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EYI |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QRAC
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EYI |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QRAD
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EYI |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QRBA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX9 |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QRBB
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX9 |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QRBC
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX9 |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7QRBD
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
EX9 |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
3UYTA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0CK |
Type1 |
5 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
3UYTB
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0CK |
Type1 |
5 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
3UYTC
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0CK |
Type1 |
4 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
3UYTD
|
2.0 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
0CK |
Type1 |
4 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
3UZPA
|
1.94 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0CK |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
3UZPB
|
1.94 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
0CK |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4HGTA
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
15G |
Type1 |
9 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4HGTB
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
15G |
Type1 |
2 - 292 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4HNFA
|
2.07 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
16W |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4HNFB
|
2.07 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
16W |
Type1 |
5 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8VXDA
|
2.47 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1AD7 |
Type1 |
1 - 292 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8VXDB
|
2.47 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnii |
A1AD7 |
Type1 |
2 - 298 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8VXFA
|
2.28 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AD8 |
Type1 |
4 - 298 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
8VXFB
|
2.28 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AD8 |
Type1 |
1 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5MQVA
|
2.154 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
D5Q |
Type1 |
8 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5MQVB
|
2.154 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D5Q |
Type1 |
8 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5MQVC
|
2.154 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
D5Q |
Type1 |
6 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5MQVD
|
2.154 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D5Q |
Type1 |
8 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5MQVE
|
2.154 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D5Q |
Type1 |
8 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5MQVF
|
2.154 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
D5Q |
Type1 |
7 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5OKTA
|
2.13 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9XK |
Type1 |
4 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5OKTB
|
2.13 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
9XK |
Type1 |
4 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5OKTC
|
2.13 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9XK |
Type1 |
4 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5OKTD
|
2.13 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9XK |
Type1 |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6F1WA
|
1.864 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CG5 |
Type1 |
3 - 292 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6F1WB
|
1.864 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CG5 |
Type1 |
1 - 291 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6F26A
|
1.83 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C9Z |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6F26B
|
1.83 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C9Z |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6HMPA
|
2.039 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GEW |
Type1 |
8 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6HMPB
|
2.039 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GEW |
Type1 |
1 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6HMRA
|
1.782 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GE5 |
Type1 |
7 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6HMRB
|
1.782 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
GE5 |
Type1 |
1 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7NZYA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UX2 |
Type1 |
4 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7NZYB
|
1.85 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_niii |
UX2 |
Type1 |
2 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7NZYC
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UX2 |
Type1 |
3 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
7NZYD
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UX2 |
Type1 |
3 - 294 |
0 |
TPO220 |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBCA
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QJ |
Type1 |
2 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBCB
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QJ |
Type1 |
1 - 291 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4TN6A
|
2.41 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PFO |
Type1 |
2 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4TW9A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
386 |
Type1 |
2 - 295 |
0 |
None |
R13N |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4TW9B
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
386 |
Type1 |
1 - 295 |
0 |
None |
R13N |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4TWCA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
37J |
Type1 |
2 - 295 |
0 |
None |
R13N |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4TWCB
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
37J |
Type1 |
1 - 295 |
0 |
None |
R13N |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6GZMA
|
1.59 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
LCI |
Type1 |
5 - 295 |
0 |
None |
R13N |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6GZMB
|
1.59 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
LCI |
Type1 |
1 - 295 |
0 |
None |
R13N |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KB8A
|
1.95 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
1QN |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KB8B
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QO |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KB8C
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QN |
Type1 |
7 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KB8D
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QO |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBAA
|
1.98 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
1QM |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBAB
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QM |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBAC
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QM |
Type1 |
7 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBAD
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QM |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBKA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QG |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBKB
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QG |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBKC
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QG |
Type1 |
4 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
4KBKD
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1QG |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5W4WA
|
1.99 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9WG |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5W4WB
|
1.99 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9WG |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5W4WC
|
1.99 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9WG |
Type1 |
4 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
5W4WD
|
1.99 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9WG |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RCHA
|
1.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
K0B |
Type1.5_Back |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RU7A
|
2.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
Type1.5_Back |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RU7B
|
2.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
Type1.5_Back |
3 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RU8A
|
1.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
Type1.5_Back |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RU8B
|
1.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
Type1.5_Back |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RU8C
|
1.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
Type1.5_Back |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1D
|
KC1D_HUMAN
|
6RU8D
|
1.92 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
Type1.5_Back |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform delta |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
AF-P49674-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 283 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
AF-P49674-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 283 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKA
|
2.77 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKC
|
2.77 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKE
|
2.77 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKG
|
2.77 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKI
|
2.77 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKK
|
2.77 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKM
|
2.77 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKO
|
2.77 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKQ
|
2.77 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKS
|
2.77 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
4 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKU
|
2.77 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 293 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HOKW
|
2.77 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 294 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HNIA
|
2.74 |
Inactive |
DFGout‑BBAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
16W |
Type1 |
3 - 293 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1E
|
KC1E_HUMAN
|
4HNIB
|
2.74 |
Inactive |
DFGout‑BBAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
16W |
Type1 |
1 - 293 |
0 |
None |
None |
Casein kinase I isoform epsilon |
|
CK1
|
CSNK1G1
|
KC1G1_HUMAN
|
AF-Q9HCP0-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 321 |
0 |
None |
None |
Casein kinase I isoform gamma-1 |
|
CK1
|
CSNK1G1
|
KC1G1_HUMAN
|
AF-Q9HCP0-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
36 - 321 |
0 |
None |
None |
Casein kinase I isoform gamma-1 |
|
CK1
|
CSNK1G1
|
KC1G1_HUMAN
|
2CMWA
|
1.75 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_iini |
OLP,
OLP,
OLP
|
Type1,
Allosteric,
Allosteric
|
44 - 339 |
0 |
None |
None |
Casein kinase I isoform gamma-1 |
|
CK1
|
CSNK1G2
|
KC1G2_HUMAN
|
AF-P78368-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
38 - 322 |
0 |
None |
None |
Casein kinase I isoform gamma-2 |
|
CK1
|
CSNK1G2
|
KC1G2_HUMAN
|
AF-P78368-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
38 - 322 |
0 |
None |
None |
Casein kinase I isoform gamma-2 |
|
CK1
|
CSNK1G2
|
KC1G2_HUMAN
|
2C47A
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5ID |
Type1 |
44 - 338 |
0 |
None |
None |
Casein kinase I isoform gamma-2 |
|
CK1
|
CSNK1G2
|
KC1G2_HUMAN
|
2C47B
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5ID |
Type1 |
44 - 338 |
0 |
None |
None |
Casein kinase I isoform gamma-2 |
|
CK1
|
CSNK1G2
|
KC1G2_HUMAN
|
2C47C
|
2.4 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5ID |
Type1 |
46 - 337 |
0 |
None |
None |
Casein kinase I isoform gamma-2 |
|
CK1
|
CSNK1G2
|
KC1G2_HUMAN
|
2C47D
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5ID |
Type1 |
43 - 338 |
0 |
None |
None |
Casein kinase I isoform gamma-2 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
AF-Q9Y6M4-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
35 - 318 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
AF-Q9Y6M4-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
35 - 318 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
4G16A
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
0VM |
Type1 |
34 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
4G17A
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
0VN |
Type1 |
34 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
4HGLA
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
0YO |
Type1 |
34 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
2IZRA
|
1.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
BRK |
Type1 |
36 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
2IZSA
|
1.95 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
BRQ |
Type1 |
36 - 333 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
2IZTA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
23D |
Type1 |
37 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
2IZUA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
P01 |
Type1 |
36 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
6GROA
|
1.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F92 |
Type1 |
37 - 329 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
2CHLA
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DKI |
Type1 |
36 - 333 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
CSNK1G3
|
KC1G3_HUMAN
|
4HGSA
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
15G |
Type1.5_Back |
34 - 334 |
0 |
None |
None |
Casein kinase I isoform gamma-3 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
8XPZA
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
20 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7QHWAAA
|
2.8 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CGI |
Type1 |
21 - 313 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7QHWCCC
|
2.8 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CGI |
Type1 |
21 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7Q8VA
|
2.13 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IV |
Type1 |
21 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7Q8WA
|
2.02 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IO |
Type1 |
21 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
4BTMA
|
2.54 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F8E |
Type1 |
21 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
4BTMB
|
2.54 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F8E |
Type1 |
21 - 313 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
4BTJA
|
2.16 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
21 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
4BTJB
|
2.16 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
21 - 313 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
AF-Q5TCY1-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
26 - 303 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
AF-Q5TCY1-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
26 - 303 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
4NFMA
|
2.12 |
None |
DFGin‑BLAminus |
in-none |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
22 - 314 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
9HHWA
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1IU7 |
Type1 |
21 - 313 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
4NFNA
|
1.42 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2KC |
Type1 |
22 - 314 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7ZHNA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VP7 |
Type1.5_Back |
21 - 313 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7ZHOA
|
2.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQR |
Type1.5_Back |
21 - 317 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7ZHPA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IQY |
Type1.5_Back |
21 - 313 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7ZHQA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IRD |
Type1.5_Back |
21 - 313 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7JXXA
|
1.56 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VP7 |
Type1.5_Back |
22 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7JXYA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VSY |
Type1.5_Back |
23 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
7JXYB
|
2.15 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_iini |
VSY |
Type1.5_Back |
20 - 312 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK1
|
TTBK1_HUMAN
|
4BTKA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
DTQ |
Type1.5_Back |
22 - 311 |
0 |
None |
None |
Tau-tubulin kinase 1 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q8YA
|
1.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IV |
Type1 |
6 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q8YB
|
1.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IV |
Type1 |
7 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q8ZA
|
1.57 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IK |
Type1 |
6 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q8ZB
|
1.57 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IK |
Type1 |
7 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q90A
|
1.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IS |
Type1 |
6 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
7Q90B
|
1.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
9IS |
Type1 |
7 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
6VRFA
|
1.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
9 - 298 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
6VRFB
|
1.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
9 - 298 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
AF-Q6IQ55-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 290 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
AF-Q6IQ55-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 290 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
6U0KA
|
1.744 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DTQ |
Type1 |
8 - 298 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
TTBK2
|
TTBK2_HUMAN
|
6U0KB
|
1.744 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DTQ |
Type1 |
8 - 299 |
0 |
None |
None |
Tau-tubulin kinase 2 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6AC9A
|
2.07 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
21 - 342 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6AC9B
|
2.07 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ANP |
ATPlike |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6AC9C
|
2.07 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ANP |
ATPlike |
24 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6AC9D
|
2.07 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
ANP |
ATPlike |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
AF-Q99986-K1A
|
-1.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
No_ligand |
No_ligand |
29 - 334 |
0 |
None |
None |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
AF-Q99986-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 334 |
0 |
None |
None |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
2LAVA
|
999.0 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iiio |
No_ligand |
No_ligand |
1 - 361 |
0 |
None |
None |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BP0A
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BP0C
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BRUA
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BRUC
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BTWC
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BU6C
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CFMC
|
2.45 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CMMA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CMMC
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CQHC
|
2.15 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CSWA
|
2.25 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CSWC
|
2.25 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6DD4A
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6DD4C
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VZHA
|
2.55 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VZHC
|
2.55 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
8V42A
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
8V42C
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
2RSVA
|
999.0 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
1 - 396 |
0 |
None |
None |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UKFA
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
8E1 |
Type1 |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UKFB
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8E1 |
Type1 |
51 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UKFC
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
8E1 |
Type1 |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UKFD
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
8E1 |
Type1 |
39 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
3OP5A
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
REB |
Type1 |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
3OP5B
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
REB |
Type1 |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
3OP5C
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
REB |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
3OP5D
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooi |
REB |
Type1 |
25 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UVFA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
7DZ |
Type1 |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UVFB
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
7DZ |
Type1 |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BP0B
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
E1D |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BTWB
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
E8D |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BU6B
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooi |
E8V |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BU6D
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
E8V |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CMMB
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F7D |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CMMD
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F7D |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CNXA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
F87 |
Type1 |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CQHA
|
2.15 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
F8Y |
Type1 |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CQHB
|
2.15 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F8Y |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CQHD
|
2.15 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F8Y |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CSWB
|
2.25 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
FBY |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CSWD
|
2.25 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
FBY |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6DD4B
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
G6J |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6DD4D
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
G6J |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VXUA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
RTJ |
Type1 |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VXUB
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RTJ |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VXUD
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RTJ |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
8V42B
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
YD9 |
Type1 |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
8V42D
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
YD9 |
Type1 |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UVFC
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
7DZ |
Type1.5_Back |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
5UVFD
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
7DZ |
Type1.5_Back |
25 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BP0D
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
E1D |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BRUB
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooi |
E5M |
Type1.5_Back |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BRUD
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
E5M |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BTWA
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
E8D |
Type1.5_Back |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BTWD
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
E8D |
Type1.5_Back |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6BU6A
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
E8V |
Type1.5_Back |
20 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CFMA
|
2.45 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
EA7 |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CFMB
|
2.45 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EA7 |
Type1.5_Back |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CFMD
|
2.45 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
EA7 |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CNXB
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F87 |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CNXC
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooi |
FCS |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6CNXD
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
F87 |
Type1.5_Back |
24 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6NPNA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KWJ |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6NPNB
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
KWJ |
Type1.5_Back |
24 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6NPNC
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KWJ |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6NPND
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
KWJ |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VXUC
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoi |
VBD |
Type1.5_Back |
21 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VZHB
|
2.55 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
RYA |
Type1.5_Back |
23 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
6VZHD
|
2.55 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RYA |
Type1.5_Back |
22 - 341 |
0 |
None |
K34A,K35A,E36A,E212A,K214A,E215A,E292A,K293A,K295A,K359A,K360A |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
2KTYA
|
999.0 |
Inactive |
DFGin‑None |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
1 - 360 |
0 |
None |
None |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK1
|
VRK1_HUMAN
|
2KULA
|
999.0 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
No_ligand |
No_ligand |
1 - 360 |
0 |
None |
None |
Serine/threonine-protein kinase VRK1 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
5UU1A
|
2.0 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
7DZ |
Type1.5_Back |
14 - 328 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
AF-Q86Y07-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
21 - 323 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
AF-Q86Y07-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
21 - 323 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
2V62A
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
2V62B
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
15 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
8Q1ZA
|
1.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IKD |
Type1 |
15 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
6NCGA
|
2.45 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
KJD |
Type1.5_Back |
14 - 326 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
6NCGB
|
2.45 |
Inactive |
DFGin‑BLAminus |
in-out |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
KJD |
Type1.5_Back |
16 - 326 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CK1
|
VRK2
|
VRK2_HUMAN
|
9FETA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
REB |
Type1.5_Back |
15 - 330 |
0 |
None |
None |
Serine/threonine-protein kinase VRK2 |
|
CK1
|
VRK3
|
VRK3_HUMAN
|
2JIIA
|
2.0 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiai |
APEdist_iiii |
No_ligand |
No_ligand |
141 - 472 |
0 |
None |
None |
Serine/threonine-protein kinase VRK3 |
|
CK1
|
VRK3
|
VRK3_HUMAN
|
2JIIB
|
2.0 |
Pseudo |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiai |
APEdist_iiii |
No_ligand |
No_ligand |
138 - 472 |
0 |
None |
None |
Serine/threonine-protein kinase VRK3 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
9SKQA
|
3.4 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iiii |
ANP |
ATPlike |
3 - 288 |
0 |
TPO161 |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
AF-P06493-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 295 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
AF-P06493-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 295 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4YC3A
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
7NJ0B
|
3.6 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 290 |
0 |
TPO161 |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4Y72A
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
LZ9 |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
5HQ0A
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
LZ9 |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
5LQFA
|
2.06 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
4SP |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
5LQFD
|
2.06 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
4SP |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU2A
|
2.0 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnno |
F9Z |
Type1 |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU3A
|
2.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
FB8 |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU4A
|
2.73 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
FC8 |
Type1 |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4YC6A
|
2.6 |
Inactive |
DFGin‑BLBplus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4YC6C
|
2.6 |
Inactive |
DFGin‑BLBplus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4YC6E
|
2.6 |
Inactive |
DFGin‑BLBplus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
4YC6G
|
2.6 |
Inactive |
DFGin‑BLBplus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 289 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU7C
|
2.75 |
Inactive |
DFGin‑BLBplus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
No_ligand |
No_ligand |
1 - 291 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU7E
|
2.75 |
Inactive |
DFGin‑BLBplus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
No_ligand |
No_ligand |
1 - 292 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU7G
|
2.75 |
Inactive |
DFGin‑BLBplus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
No_ligand |
No_ligand |
1 - 291 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU6A
|
2.33 |
Inactive |
DFGin‑BLBplus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_oooo |
1QK |
Type1 |
1 - 291 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK1
|
CDK1_HUMAN
|
6GU7A
|
2.75 |
Inactive |
DFGin‑BLBplus |
out-out |
out-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
FB8 |
Type1 |
1 - 293 |
0 |
None |
None |
Cyclin-dependent kinase 1 |
|
CMGC
|
CDK10
|
CDK10_HUMAN
|
AF-Q15131-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
31 - 331 |
0 |
None |
None |
Cyclin-dependent kinase 10 |
|
CMGC
|
CDK10
|
CDK10_HUMAN
|
AF-Q15131-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
31 - 331 |
0 |
None |
None |
Cyclin-dependent kinase 10 |
|
CMGC
|
CDK11A
|
CD11A_HUMAN
|
AF-Q9UQ88-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
418 - 719 |
0 |
None |
None |
Cyclin-dependent kinase 11A |
|
CMGC
|
CDK11A
|
CD11A_HUMAN
|
AF-Q9UQ88-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
418 - 719 |
0 |
None |
None |
Cyclin-dependent kinase 11A |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZA
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
436 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZB
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
436 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZC
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
436 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZD
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
437 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZE
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
435 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
7UKZF
|
2.6 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NK3 |
Type1 |
436 - 736 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
9I9IK
|
3.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
440 - 740 |
0 |
TPO595 |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
AF-P21127-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
430 - 731 |
0 |
None |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK11B
|
CD11B_HUMAN
|
AF-P21127-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
430 - 731 |
0 |
None |
None |
Cyclin-dependent kinase 11B |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU2H
|
3.13 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RVQ |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU4B
|
3.09 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU4H
|
3.09 |
Inactive |
DFGin‑ABAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU5B
|
3.134 |
Inactive |
DFGin‑ABAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RMF |
Type1 |
713 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU5H
|
3.134 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RMF |
Type1 |
713 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU9H
|
3.51 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RRC |
Type1 |
715 - 1038 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUAB
|
3.193 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RVH |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUAE
|
3.193 |
Inactive |
DFGin‑ABAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RVH |
Type1 |
715 - 1033 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUAH
|
3.193 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RVH |
Type1 |
715 - 1034 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUCB
|
3.85 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RKO |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUDB
|
3.2 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RP9 |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUDH
|
3.2 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RP9 |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUEH
|
3.25 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RVU |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUIB
|
3.5 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RV6 |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUIH
|
3.5 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RV6 |
Type1 |
715 - 1038 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BULH
|
3.4 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RSU |
Type1 |
715 - 1034 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUNB
|
3.08 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RNF |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUNH
|
3.08 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RNF |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUOB
|
3.58 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RLC |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BURE
|
3.64 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQU |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUSH
|
3.26 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RMX |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUTB
|
3.25 |
Inactive |
DFGin‑ABAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQ5 |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUTH
|
3.25 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RQ5 |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
7NXKA
|
3.0 |
Inactive |
DFGin‑ABAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
UUB |
Type1 |
715 - 1040 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
9FMRE
|
3.9 |
Inactive |
DFGin‑ABAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RMF |
Type1 |
714 - 1042 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
9FMRH
|
3.9 |
Inactive |
DFGin‑ABAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RMF |
Type1 |
714 - 1044 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4CXAA
|
3.15 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ANP |
ATPlike |
718 - 1050 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4NSTA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
716 - 1046 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4NSTC
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
717 - 1045 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
AF-Q9NYV4-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
719 - 1028 |
0 |
None |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
AF-Q9NYV4-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
719 - 1028 |
0 |
None |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4UN0C
|
3.15 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iiii |
No_ligand |
No_ligand |
719 - 1036 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4UN0D
|
3.15 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iiii |
No_ligand |
No_ligand |
723 - 1024 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
4CXAC
|
3.15 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
718 - 1048 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU2E
|
3.13 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU7B
|
3.245 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU7H
|
3.245 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUDE
|
3.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUGE
|
3.53 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6B3EA
|
3.06 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CJM |
Type1 |
717 - 1036 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6B3EC
|
3.06 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
CJM |
Type1 |
719 - 1036 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
5ACBC
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5I1 |
Type1 |
716 - 1040 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
5ACBD
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5I1 |
Type1 |
718 - 1044 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
9JK1A
|
2.72 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1EB3 |
Type1 |
717 - 1039 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
9JK1B
|
2.72 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
A1EB3 |
Type1 |
715 - 1039 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6TD3B
|
3.46 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RC8 |
Type1 |
715 - 1047 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6TD3E
|
3.46 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RC8 |
Type1 |
715 - 1047 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6TD3H
|
3.46 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iiii |
RC8 |
Type1 |
715 - 1047 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU1E
|
2.98 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU3E
|
3.42 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RSI |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU4E
|
3.09 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU6E
|
3.45 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQE |
Type1 |
715 - 1038 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU7E
|
3.245 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RS5 |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU9E
|
3.51 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RRC |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUBB
|
3.42 |
Inactive |
DFGin‑BLAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iioo |
RNU |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUBE
|
3.42 |
Inactive |
DFGin‑BLAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iooo |
RNU |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUCE
|
3.85 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RKO |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUEE
|
3.25 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RVU |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUFE
|
3.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RW6 |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUHE
|
3.79 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RR9 |
Type1 |
715 - 1034 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUIE
|
3.5 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
RV6 |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUJE
|
3.62 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RUW |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUKE
|
3.41 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RWE |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BULE
|
3.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RSU |
Type1 |
715 - 1038 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUME
|
3.36 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T6X |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUNE
|
3.08 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RNF |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUOE
|
3.58 |
Inactive |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RLC |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUPB
|
3.41 |
Inactive |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RWN |
Type1 |
715 - 1027 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUPE
|
3.41 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiio |
RWN |
Type1 |
715 - 1027 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUPH
|
3.41 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RWN |
Type1 |
715 - 1028 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUQB
|
3.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQ9 |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUQE
|
3.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQ9 |
Type1 |
715 - 1027 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BURB
|
3.64 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQU |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUSB
|
3.26 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RMX |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUTE
|
3.25 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQ5 |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6CKXA
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8M1 |
Type1 |
722 - 1024 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
6CKXC
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
8M1 |
Type1 |
722 - 1024 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
7NXKC
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
UUB |
Type1 |
717 - 1040 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8P81A
|
2.68 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RMF |
Type1 |
716 - 1035 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUGH
|
3.53 |
Inactive |
DFGin‑None |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU1B
|
2.98 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU1H
|
2.98 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQL |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU2B
|
3.13 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RVQ |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU3B
|
3.42 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RSI |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU3H
|
3.42 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RSI |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU5E
|
3.134 |
Inactive |
DFGin‑None |
in-out |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
RMF |
Type1 |
713 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU6B
|
3.45 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQE |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU6H
|
3.45 |
Inactive |
DFGin‑None |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQE |
Type1 |
715 - 1038 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BU9B
|
3.51 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RRC |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUBH
|
3.42 |
Inactive |
DFGin‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaooo |
APEdist_iiii |
RNU |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUCH
|
3.85 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RKO |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUEB
|
3.25 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RVU |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUFB
|
3.3 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RW6 |
Type1 |
715 - 1033 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUFH
|
3.3 |
Inactive |
DFGin‑None |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RW6 |
Type1 |
715 - 1032 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUGB
|
3.53 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RPW |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUHB
|
3.79 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RR9 |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUHH
|
3.79 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RR9 |
Type1 |
715 - 1033 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUJB
|
3.62 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RUW |
Type1 |
715 - 1041 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUJH
|
3.62 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RUW |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUKB
|
3.41 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RWE |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUKH
|
3.41 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RWE |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BULB
|
3.4 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RSU |
Type1 |
715 - 1039 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUMB
|
3.36 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T6X |
Type1 |
715 - 1040 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUMH
|
3.36 |
Inactive |
DFGin‑None |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T6X |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUOH
|
3.58 |
Inactive |
DFGin‑None |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RLC |
Type1 |
715 - 1044 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUQH
|
3.2 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQ9 |
Type1 |
715 - 1035 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BURH
|
3.64 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RQU |
Type1 |
715 - 1039 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
8BUSE
|
3.26 |
Inactive |
DFGin‑None |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RMX |
Type1 |
715 - 1043 |
0 |
TPO893 |
K965R |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK12
|
CDK12_HUMAN
|
9FMRB
|
3.9 |
Inactive |
DFGin‑None |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RMF |
Type1 |
714 - 1047 |
0 |
TPO893 |
None |
Cyclin-dependent kinase 12 |
|
CMGC
|
CDK13
|
CDK13_HUMAN
|
5EFQA
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
695 - 1025 |
0 |
TPO871 |
None |
Cyclin-dependent kinase 13 |
|
CMGC
|
CDK13
|
CDK13_HUMAN
|
5EFQC
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ADP |
ATPlike |
697 - 1031 |
0 |
TPO871 |
None |
Cyclin-dependent kinase 13 |
|
CMGC
|
CDK13
|
CDK13_HUMAN
|
AF-Q14004-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
697 - 1006 |
0 |
None |
None |
Cyclin-dependent kinase 13 |
|
CMGC
|
CDK13
|
CDK13_HUMAN
|
AF-Q14004-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
697 - 1006 |
0 |
None |
None |
Cyclin-dependent kinase 13 |
|
CMGC
|
CDK13
|
CDK13_HUMAN
|
7NXJA
|
2.36 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
5I1 |
Type1 |
695 - 1023 |
0 |
TPO871 |
None |
Cyclin-dependent kinase 13 |
|
CMGC
|
CDK13
|
CDK13_HUMAN
|
7NXJC
|
2.36 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
5I1 |
Type1 |
695 - 1017 |
0 |
TPO871 |
None |
Cyclin-dependent kinase 13 |
|
CMGC
|
CDK14
|
CDK14_HUMAN
|
AF-O94921-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
127 - 427 |
0 |
None |
None |
Cyclin-dependent kinase 14 |
|
CMGC
|
CDK14
|
CDK14_HUMAN
|
AF-O94921-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
127 - 427 |
0 |
None |
None |
Cyclin-dependent kinase 14 |
|
CMGC
|
CDK15
|
CDK15_HUMAN
|
AF-Q96Q40-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
95 - 395 |
0 |
None |
None |
Cyclin-dependent kinase 15 |
|
CMGC
|
CDK15
|
CDK15_HUMAN
|
AF-Q96Q40-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
95 - 395 |
0 |
None |
None |
Cyclin-dependent kinase 15 |
|
CMGC
|
CDK16
|
CDK16_HUMAN
|
AF-Q00536-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
157 - 454 |
0 |
None |
None |
Cyclin-dependent kinase 16 |
|
CMGC
|
CDK16
|
CDK16_HUMAN
|
AF-Q00536-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
157 - 454 |
0 |
None |
None |
Cyclin-dependent kinase 16 |
|
CMGC
|
CDK16
|
CDK16_HUMAN
|
5G6VA
|
2.2 |
Inactive |
DFGout‑BBAminus |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_iooo |
919 |
Type2 |
163 - 474 |
0 |
None |
S319D |
Cyclin-dependent kinase 16 |
|
CMGC
|
CDK16
|
CDK16_HUMAN
|
3MTLA
|
2.4 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
FEF |
Type1 |
163 - 473 |
0 |
None |
S319D |
Cyclin-dependent kinase 16 |
|
CMGC
|
CDK16
|
CDK16_HUMAN
|
5G6VB
|
2.2 |
Inactive |
DFGout‑None |
in-in |
out-out |
nonTYR |
APEdihe_aaoii |
APEdist_nnno |
919 |
Type2 |
163 - 475 |
0 |
None |
S319D |
Cyclin-dependent kinase 16 |
|
CMGC
|
CDK17
|
CDK17_HUMAN
|
AF-Q00537-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
184 - 481 |
0 |
None |
None |
Cyclin-dependent kinase 17 |
|
CMGC
|
CDK17
|
CDK17_HUMAN
|
AF-Q00537-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
184 - 481 |
0 |
None |
None |
Cyclin-dependent kinase 17 |
|
CMGC
|
CDK18
|
CDK18_HUMAN
|
AF-Q07002-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
136 - 433 |
0 |
None |
None |
Cyclin-dependent kinase 18 |
|
CMGC
|
CDK18
|
CDK18_HUMAN
|
AF-Q07002-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
136 - 433 |
0 |
None |
None |
Cyclin-dependent kinase 18 |
|
CMGC
|
CDK19
|
CDK19_HUMAN
|
AF-Q9BWU1-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 343 |
0 |
None |
None |
Cyclin-dependent kinase 19 |
|
CMGC
|
CDK19
|
CDK19_HUMAN
|
AF-Q9BWU1-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
12 - 343 |
0 |
None |
None |
Cyclin-dependent kinase 19 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8BZOA
|
3.5 |
Inactive |
DFGin‑ABAminus |
out-none |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
14 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5NEVA
|
2.97 |
Inactive |
DFGin‑ABAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
72L |
Type1 |
1 - 295 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5NEVC
|
2.97 |
Inactive |
DFGin‑ABAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
72L |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOOA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 297 |
0 |
TPO160 |
Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOOC
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOMA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 297 |
0 |
TPO160 |
H84S,Q85M,Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOMC
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
H84S,Q85M,Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4I3ZA
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4I3ZC
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QHRA
|
2.17 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QHRC
|
2.17 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QHWA
|
1.91 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QHWC
|
1.91 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1FINA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
ATP |
ATPlike |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1FINC
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
ATP |
ATPlike |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1FQ1B
|
3.0 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_oioo |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1JSTA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1JSTC
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2CJMA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 292 |
0 |
PTR15,TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2CJMC
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 297 |
0 |
PTR15,TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4II5A
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4II5C
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ADP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1GY3A
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1GY3C
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1QMZA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1QMZC
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2CCHA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2CCHC
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2CCIA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2CCIC
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9I9JK
|
3.1 |
Inactive |
DFGin‑BLAminus |
in-out |
none-out |
nonTYR |
APEdihe_aaooi |
APEdist_nnno |
ADP |
ATPlike |
6 - 284 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9I9KK
|
2.4 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioo |
ADP |
ATPlike |
2 - 292 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9QCVK
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
ANP |
ATPlike |
1 - 292 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOQA
|
2.15 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOQC
|
2.15 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOJA
|
1.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 298 |
0 |
TPO160 |
H84S,Q85M,K89D |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOJC
|
1.65 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
ATP |
ATPlike |
1 - 296 |
0 |
TPO160 |
H84S,Q85M,K89D |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8VQ3A
|
1.84 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
A1AC4 |
Allosteric |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8VQ4A
|
1.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnni |
A1AC5 |
Allosteric |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESOA
|
2.396 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W3A |
Allosteric |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESYA
|
2.394 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HH8,
HH8
|
Allosteric,
Type1
|
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ET1A
|
2.394 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IJL,
IJL
|
Allosteric,
Type1
|
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ET2A
|
2.37 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IJX,
IJX
|
Allosteric,
Type1
|
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESOC
|
2.396 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
W3A,
W3A,
W3A
|
Allosteric,
Type1,
Allosteric
|
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESQC
|
2.38 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IT4,
IT4,
IT4
|
Allosteric,
Type1,
Allosteric
|
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ET8A
|
2.31 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IIS,
IIS,
IIS
|
Allosteric,
Type1,
Allosteric
|
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESSA
|
2.44 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UUG,
UUG,
UUG,
UUG
|
Allosteric,
Type1,
Allosteric,
Allosteric
|
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESWA
|
2.38 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IJF,
IJF,
IJF,
IJF
|
Allosteric,
Type1,
Allosteric,
Allosteric
|
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESWC
|
2.38 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IJF,
IJF,
IJF,
IJF
|
Allosteric,
Type1,
Allosteric,
Allosteric
|
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ETBA
|
2.76 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
PYZ,
PYZ,
PYZ,
PYZ
|
Allosteric,
Type1,
Allosteric,
Allosteric
|
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ET3A
|
2.34 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1P8,
1P8,
1P8,
1P8,
1P8
|
Allosteric,
Type1,
Allosteric,
Allosteric,
Allosteric
|
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ET9A
|
2.494 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HEW,
HEW,
HEW,
HEW,
HEW
|
Allosteric,
Type1,
Allosteric,
Allosteric,
Allosteric
|
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ET6A
|
2.553 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HHQ,
HHQ,
HHQ,
HHQ,
HHQ
|
Allosteric,
Type1,
Type1,
Allosteric,
Allosteric
|
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESRA
|
2.388 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UU1,
UU1,
UU1,
UU1,
UU1
|
Allosteric,
Type1,
Type1.5_Back,
Allosteric,
Allosteric
|
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2JGZA
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 288 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
AF-P24941-K1A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
AF-P24941-K3A
|
-1.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9HIUB
|
3.2 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9HIWB
|
3.1 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9HJ1B
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aanoi |
APEdist_nnnn |
No_ligand |
No_ligand |
1 - 294 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1W98A
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1F5QA
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
No_ligand |
No_ligand |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1F5QC
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooo |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1JSUA
|
2.3 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
13 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OKVA
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OKVC
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OKWA
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OKWC
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OL1A
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OL1C
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OL2A
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OL2C
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1URCA
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioo |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1URCC
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiio |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2V22A
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2V22C
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WFYA
|
2.53 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WFYC
|
2.53 |
Inactive |
DFGin‑BLAminus |
in-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WHBA
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WHBC
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioi |
No_ligand |
No_ligand |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3EIDC
|
3.15 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_inni |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5IF1A
|
2.61 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5IF1C
|
2.61 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_iioo |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6P3WA
|
2.54 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6P3WC
|
2.54 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7B5LL
|
3.8 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
No_ligand |
No_ligand |
13 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7B5RL
|
3.8 |
Inactive |
DFGin‑BLAminus |
out-out |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
No_ligand |
No_ligand |
13 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8ROZA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 298 |
0 |
PTR15,TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9D0WC
|
2.95 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9D0XC
|
2.84 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7E34A
|
3.19 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6ATHA
|
1.82 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
17 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5UQ1A
|
3.201 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
3 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5UQ2A
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5UQ3A
|
3.6 |
Inactive |
DFGin‑BLAminus |
out-in |
in-out |
nonTYR |
APEdihe_aaiio |
APEdist_iiii |
No_ligand |
No_ligand |
19 - 292 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9QCXK
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
No_ligand |
No_ligand |
1 - 292 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6SG4A
|
2.43 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
28 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6SG4C
|
2.43 |
Inactive |
DFGin‑BLAminus |
out-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
29 - 295 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H24A
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 293 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H24C
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 293 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H25A
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 293 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H25C
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 293 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H26A
|
2.24 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H26C
|
2.24 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H27A
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H27C
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H28A
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H28C
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WMAA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WMAC
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WMBA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WMBC
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
No_ligand |
No_ligand |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOPA
|
1.99 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 297 |
0 |
TPO160 |
Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOPC
|
1.99 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 296 |
0 |
TPO160 |
Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EONA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1RO |
Type1 |
1 - 298 |
0 |
TPO160 |
H84S,Q85M,Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EONC
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1RO |
Type1 |
1 - 297 |
0 |
TPO160 |
H84S,Q85M,Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOIA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1RO |
Type1 |
1 - 298 |
0 |
TPO160 |
K89D,Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOIC
|
2.0 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 296 |
0 |
TPO160 |
K89D,Q131E |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2IW6A
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
QQ2 |
Type1 |
1 - 295 |
0 |
TPO160 |
K89T |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2IW6C
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
QQ2 |
Type1 |
1 - 295 |
0 |
TPO160 |
K89T |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2IW9A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4SP |
Type1 |
1 - 297 |
0 |
TPO160 |
K89T |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2IW9C
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4SP |
Type1 |
1 - 296 |
0 |
TPO160 |
K89T |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1E9HA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
INR |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1E9HC
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
INR |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PKDA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UCN |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1PKDC
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UCN |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5LMKC
|
2.4 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
6ZK |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9GLAA
|
2.18 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
YNK |
Type1 |
2 - 294 |
0 |
TPO160 |
E8D,K9F,I10L,T14Q,Y15F,V64I,L83M,H84E,Q85T,K88E,K89V,Q131N |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EORA
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4SP |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EORC
|
2.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
4SP |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1FVVA
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
107 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1FVVC
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oiii |
107 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5NA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
CK8 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5NC
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
CK8 |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5OA
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
CK2 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5OC
|
2.1 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
CK2 |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5VA
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
CK4 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5VC
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
CK4 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5XA
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_oioi |
MTW |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C5XC
|
2.9 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
MTW |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C6TA
|
2.61 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DT5 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2C6TC
|
2.61 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
DT5 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2I40A
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnii |
BLZ |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2I40C
|
2.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oioi |
BLZ |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UUEA
|
2.06 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
MTZ |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UUEC
|
2.06 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoii |
APEdist_oioi |
MTZ |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZBA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaoio |
APEdist_iioi |
C75 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZBC
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
C75 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZDA
|
2.72 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C85 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZDC
|
2.72 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C85 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZEA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C95 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZEC
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C95 |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZLA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C94 |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2UZLC
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
C94 |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WEVA
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
CK7 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2WEVC
|
2.3 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioo |
CK7 |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2X1NA
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooi |
APEdist_oioi |
X1N |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2X1NC
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaooo |
APEdist_iioi |
X1N |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3EIDA
|
3.15 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnii |
PO5 |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3EJ1A
|
3.22 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iioi |
5BP |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3EJ1C
|
3.22 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_oioi |
5BP |
Type1 |
1 - 297 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3EOCA
|
3.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T2A |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3EOCC
|
3.2 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_oiii |
T2A |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3TIYA
|
1.84 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_oooo |
TIY |
Type1 |
2 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FX3A
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iooi |
60K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4FX3C
|
2.75 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iooi |
60K |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7KJSA
|
2.187 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
WG1 |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8CURA
|
2.2 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaioi |
APEdist_nnoo |
OW6 |
Type1 |
1 - 296 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9D0VA
|
2.54 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1A1H |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9GOPA
|
2.158 |
None |
DFGin‑BLAminus |
in-in |
in-none |
nonTYR |
APEdihe_aaiii |
APEdist_nnni |
A1IOI |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9GP3A
|
2.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1IOP |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8H6PA
|
2.44 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
WZU |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8H6TA
|
3.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
WZZ |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1P5EA
|
2.22 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TBS |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1P5EC
|
2.22 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TBS |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2G9XA
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NU5 |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
2G9XC
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
NU5 |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3DDPA
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RC8 |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3DDPC
|
2.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RC8 |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3DDQA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RRC |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3DDQC
|
1.8 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
RRC |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3DOGA
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaiii |
APEdist_iioi |
NNN |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3DOGC
|
2.7 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
NNN |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5L2WA
|
2.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
1QK |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5LMKA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6ZK |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6GVAA
|
2.15 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
FCQ |
Type1 |
1 - 290 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6JGMA
|
2.3 |
Inactive |
DFGin‑BLAminus |
out-out |
none-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnno |
AQG |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6RIJA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
K4W |
Type1 |
1 - 290 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6RIJC
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
K4W |
Type1 |
1 - 290 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7ACKA
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R7B |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7ACKC
|
1.8 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
R7B |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7B7SA
|
2.54 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T1T |
Type1 |
1 - 293 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7B7SC
|
2.54 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T1T |
Type1 |
1 - 293 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7QHLA
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D5P |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7QHLC
|
1.7 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
D5P |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8B54A
|
2.6 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
P2V |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
8B54C
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
P2V |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9BJCA
|
2.22 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1AQZ |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4NJ3A
|
1.848 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nooo |
2KD |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3BHTA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MFR |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3BHTC
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MFR |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3BHUA
|
2.3 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
MHR |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3BHVA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VAR |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3BHVC
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
VAR |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3MY5A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RFZ |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3MY5C
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
RFZ |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3TNWA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F18 |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3TNWC
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F18 |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCKA
|
2.052 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T3E |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCKC
|
2.052 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T3E |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCNA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T9N |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCNC
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T9N |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCOA
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T6Q |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCOC
|
2.05 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T6Q |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCPA
|
2.26 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T3C |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCPC
|
2.26 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T3C |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOSA
|
2.57 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4EOSC
|
2.57 |
Inactive |
DFGin‑BLAminus |
in-in |
in-out |
nonTYR |
APEdihe_aaioi |
APEdist_iiii |
1RO |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9OB2A
|
2.12 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1CAE |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9OB3A
|
1.98 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1CAH |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9OB4A
|
1.95 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1CAF |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9OB5A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1CAG |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9OB6A
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1CAI |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCMA
|
2.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T7Z |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCMC
|
2.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
T7Z |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCQA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TJF |
Type1 |
1 - 295 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4BCQC
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
TJF |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OGUA
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ST8 |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OGUC
|
2.6 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ST8 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OI9A
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
N20 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OI9C
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
N20 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OIUA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
N76 |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OIUC
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
N76 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OIYA
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
N41 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1OIYC
|
2.4 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
N41 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFNA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
JYM |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFNC
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
JYM |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6GUBA
|
2.52 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F9Z |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6GUBC
|
2.52 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
F9Z |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6GUCA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SU9 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6GUCC
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SU9 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6GUEC
|
1.99 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
FB8 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6GUFA
|
2.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
23D |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
6GUFC
|
2.65 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
23D |
Type1 |
1 - 297 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESNA
|
2.393 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UUS |
Type1 |
1 - 294 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESPA
|
2.381 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UUV |
Type1 |
1 - 289 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESPC
|
2.381 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
UUV |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESUA
|
2.396 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IJU |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESUC
|
2.396 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IJU |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESXC
|
2.37 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
A1H6Y |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESYC
|
2.394 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HH8 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESZA
|
2.42 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HGW |
Type1 |
1 - 292 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ESZC
|
2.42 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HGW |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ET0A
|
2.239 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HHN |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ET0C
|
2.239 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HHN |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ET1C
|
2.394 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IJL |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ET2C
|
2.37 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
IJX |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ET7C
|
2.312 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
HGQ |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ETAA
|
2.512 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7ZX |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
9ETAC
|
2.512 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
7ZX |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H1PA
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CMG |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H1PC
|
2.1 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
CMG |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H1QA
|
2.5 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2A6 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H1QC
|
2.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2A6 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H1RA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6CP |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H1RC
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
6CP |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H1SA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4SP |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
1H1SC
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4SP |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFMA
|
2.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4QE |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFMC
|
2.85 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
4QE |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFWA
|
2.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SQ9 |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFWC
|
2.45 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
SQ9 |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFXA
|
3.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G6T |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFXC
|
3.5 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
G6T |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5CYIA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
55S |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
5CYIC
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
55S |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7MKXA
|
3.08 |
Inactive |
DFGin‑BLAminus |
in-out |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZGY |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
7MKXC
|
3.08 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
ZGY |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFUA
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2WC |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFUC
|
2.2 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
2WC |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFVA
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
75X |
Type1 |
1 - 298 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
4CFVC
|
2.0 |
Active |
DFGin‑BLAminus |
in-in |
in-in |
nonTYR |
APEdihe_aaiii |
APEdist_iiii |
75X |
Type1 |
1 - 296 |
0 |
TPO160 |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QTWA
|
1.85 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X3A |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3QU0A
|
1.95 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X40 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R9DA
|
1.95 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_oooo |
X6B |
Type1 |
1 - 298 |
0 |
None |
None |
Cyclin-dependent kinase 2 |
|
CMGC
|
CDK2
|
CDK2_HUMAN
|
3R9OA
|
1.9 |
Inactive |
DFGin‑BLAminus |
out-out |
out-out |
nonTYR |
APEdihe_aaiii |
APEdist_nnoo |
Z71 |
Type1 |
1 - 298 |
0 |
None |
None |
Cyc |