| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FLT3 | FLT3_HUMAN | AF-P36888-K1A | P36888 | 602 | 953 | 993.0 | No_ligand | No_ligand | Active | DFGin | 6.9519 | 14.1313 | BLAminus | -143.23, 178.77 | 67.08, 55.14 | -77.02, 14.59 | 286.19, 76.14 | -61.49, -31.53 | in-in | in | 7.4793 | Saltbr-in | 2.6983 | HRD-in | -78.74, -43.23 | 66.6, -14.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9188 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.73, 89.83 | APE9-dihe-in | -111.39, 151.17 | APE8-dihe-in | -77.59, 83.68 | APE8-rot-na | 35.47 | APE67-dihe-in | -70.07, -16.26 | -43.63, -37.27 | APE12-dist-na | 14.2956 | APE11-dist-na | 8.2372 | APE10-dist-na | 9.8964 | APE9-dist-in | 6.0185 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 352.0 | 352.0 | 0 | 30 | 30 | 0 | [[610, 945]] | 1.0 | AF-P36888-K1 | TYR_FLT3_HUMAN | TYR | 4.1e-102 | 346.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| TYR | FLT3 | FLT3_HUMAN | AF-P36888-K3A | P36888 | 602 | 953 | 993.0 | No_ligand | No_ligand | Active | DFGin | 7.2842 | 13.5426 | BLAminus | -131.51, -179.63 | 57.0, 62.49 | -72.98, 8.43 | 287.44, 96.64 | -61.83, -29.79 | in-in | in | 7.8544 | Saltbr-in | 2.7853 | HRD-in | -79.97, -43.81 | 68.78, -8.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8992 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.33, 109.47 | APE9-dihe-in | -88.85, 151.32 | APE8-dihe-in | -79.53, 61.94 | APE8-rot-na | 36.79 | APE67-dihe-in | -68.95, -18.44 | -45.43, -42.99 | APE12-dist-na | 14.4475 | APE11-dist-na | 8.7996 | APE10-dist-na | 12.3215 | APE9-dist-in | 7.3936 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 352.0 | 352.0 | 0 | 30 | 30 | 0 | [[610, 945]] | 1.0 | AF-P36888-K3 | TYR_FLT3_HUMAN | TYR | 4.1e-102 | 346.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FLT3 | FLT3_HUMAN | AF-P36888-K1A | P36888 | 602 | 953 | 993.0 | No_ligand | No_ligand | Active | DFGin | 6.9519 | 14.1313 | BLAminus | -143.23, 178.77 | 67.08, 55.14 | -77.02, 14.59 | 286.19, 76.14 | -61.49, -31.53 | in-in | in | 7.4793 | Saltbr-in | 2.6983 | HRD-in | -78.74, -43.23 | 66.6, -14.38 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9188 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -78.73, 89.83 | APE9-dihe-in | -111.39, 151.17 | APE8-dihe-in | -77.59, 83.68 | APE8-rot-na | 35.47 | APE67-dihe-in | -70.07, -16.26 | -43.63, -37.27 | APE12-dist-na | 14.2956 | APE11-dist-na | 8.2372 | APE10-dist-na | 9.8964 | APE9-dist-in | 6.0185 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 352.0 | 352.0 | 0 | 30 | 30 | 0 | [[610, 945]] | 1.0 | AF-P36888-K1 | Homo sapiens | TYR_FLT3_HUMAN | TYR | 4.1e-102 | 346.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| TYR | FLT3 | FLT3_HUMAN | AF-P36888-K3A | P36888 | 602 | 953 | 993.0 | No_ligand | No_ligand | Active | DFGin | 7.2842 | 13.5426 | BLAminus | -131.51, -179.63 | 57.0, 62.49 | -72.98, 8.43 | 287.44, 96.64 | -61.83, -29.79 | in-in | in | 7.8544 | Saltbr-in | 2.7853 | HRD-in | -79.97, -43.81 | 68.78, -8.23 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8992 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -70.33, 109.47 | APE9-dihe-in | -88.85, 151.32 | APE8-dihe-in | -79.53, 61.94 | APE8-rot-na | 36.79 | APE67-dihe-in | -68.95, -18.44 | -45.43, -42.99 | APE12-dist-na | 14.4475 | APE11-dist-na | 8.7996 | APE10-dist-na | 12.3215 | APE9-dist-in | 7.3936 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 352.0 | 352.0 | 0 | 30 | 30 | 0 | [[610, 945]] | 1.0 | AF-P36888-K3 | Homo sapiens | TYR_FLT3_HUMAN | TYR | 4.1e-102 | 346.9 | 1.0 | 259.0 | 259.0 | 828 | 829 | 830 | 832 | 834 | 644 | 661 | 665 | 808 | 810 | 809 | 811.0 | 870 | 858 | 853 | 852 | 851 | 850 | 849 | 848 | 847 | 692 | Receptor-type tyrosine-protein kinase FLT3 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|