| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR3 | FGFR3_HUMAN | AF-P22607-K1A | P22607 | 464 | 758 | 806.0 | No_ligand | No_ligand | Active | DFGin | 6.5621 | 13.7198 | BLAminus | -135.6, -172.84 | 54.36, 70.3 | -87.69, 11.11 | 291.08, 95.72 | -59.35, -30.65 | in-in | in | 7.4386 | Saltbr-in | 2.6502 | HRD-in | -71.1, -43.09 | 66.59, -18.9 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8909 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -62.08, 128.6 | APE9-dihe-in | -136.51, 151.31 | APE8-dihe-in | -81.26, 77.84 | APE8-rot-na | 37.52 | APE67-dihe-in | -66.67, -14.17 | -46.27, -41.56 | APE12-dist-na | 14.3905 | APE11-dist-na | 9.9039 | APE10-dist-na | 9.996 | APE9-dist-in | 6.5212 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 295.0 | 295.0 | 0 | 30 | 30 | 0 | [[472, 750]] | 1.0 | AF-P22607-K1 | TYR_FGFR3_HUMAN | TYR | 1.6e-104 | 354.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR3 | FGFR3_HUMAN | AF-P22607-K3A | P22607 | 464 | 758 | 806.0 | No_ligand | No_ligand | Active | DFGin | 6.3619 | 13.7626 | BLAminus | -140.11, -178.74 | 60.69, 64.92 | -81.11, 10.08 | 291.09, 95.14 | -60.2, -27.32 | in-in | in | 7.6939 | Saltbr-in | 2.724 | HRD-in | -81.64, -44.23 | 60.23, -5.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9077 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.46, 141.09 | APE9-dihe-in | -143.98, 144.08 | APE8-dihe-in | -81.78, 61.47 | APE8-rot-na | 36.97 | APE67-dihe-in | -68.61, -8.42 | -45.34, -43.48 | APE12-dist-na | 14.4543 | APE11-dist-na | 10.9342 | APE10-dist-na | 10.3642 | APE9-dist-in | 6.9461 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 295.0 | 295.0 | 0 | 30 | 30 | 0 | [[472, 750]] | 1.0 | AF-P22607-K3 | TYR_FGFR3_HUMAN | TYR | 1.6e-104 | 354.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | FGFR3 | FGFR3_HUMAN | AF-P22607-K1A | P22607 | 464 | 758 | 806.0 | No_ligand | No_ligand | Active | DFGin | 6.5621 | 13.7198 | BLAminus | -135.6, -172.84 | 54.36, 70.3 | -87.69, 11.11 | 291.08, 95.72 | -59.35, -30.65 | in-in | in | 7.4386 | Saltbr-in | 2.6502 | HRD-in | -71.1, -43.09 | 66.59, -18.9 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.8909 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -62.08, 128.6 | APE9-dihe-in | -136.51, 151.31 | APE8-dihe-in | -81.26, 77.84 | APE8-rot-na | 37.52 | APE67-dihe-in | -66.67, -14.17 | -46.27, -41.56 | APE12-dist-na | 14.3905 | APE11-dist-na | 9.9039 | APE10-dist-na | 9.996 | APE9-dist-in | 6.5212 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 295.0 | 295.0 | 0 | 30 | 30 | 0 | [[472, 750]] | 1.0 | AF-P22607-K1 | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 1.6e-104 | 354.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| TYR | FGFR3 | FGFR3_HUMAN | AF-P22607-K3A | P22607 | 464 | 758 | 806.0 | No_ligand | No_ligand | Active | DFGin | 6.3619 | 13.7626 | BLAminus | -140.11, -178.74 | 60.69, 64.92 | -81.11, 10.08 | 291.09, 95.14 | -60.2, -27.32 | in-in | in | 7.6939 | Saltbr-in | 2.724 | HRD-in | -81.64, -44.23 | 60.23, -5.49 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9077 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -64.46, 141.09 | APE9-dihe-in | -143.98, 144.08 | APE8-dihe-in | -81.78, 61.47 | APE8-rot-na | 36.97 | APE67-dihe-in | -68.61, -8.42 | -45.34, -43.48 | APE12-dist-na | 14.4543 | APE11-dist-na | 10.9342 | APE10-dist-na | 10.3642 | APE9-dist-in | 6.9461 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 295.0 | 295.0 | 0 | 30 | 30 | 0 | [[472, 750]] | 1.0 | AF-P22607-K3 | Homo sapiens | TYR_FGFR3_HUMAN | TYR | 1.6e-104 | 354.7 | 1.0 | 260.0 | 260.0 | 634 | 635 | 636 | 638 | 640 | 508 | 525 | 529 | 614 | 616 | 615 | 617.0 | 676 | 664 | 659 | 658 | 657 | 656 | 655 | 654 | 653 | 556 | Fibroblast growth factor receptor 3 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|