| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EPHA1 | EPHA1_HUMAN | AF-P21709-K1A | P21709 | 616 | 890 | 976.0 | No_ligand | No_ligand | Active | DFGin | 6.0327 | 14.6832 | BLAminus | -138.4, -178.11 | 59.23, 67.7 | -84.1, 14.72 | 296.01, 92.0 | -60.59, -34.63 | in-in | in | 8.3875 | Saltbr-in | 2.7245 | HRD-in | -74.65, -44.09 | 68.7, -13.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9031 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.65, 144.12 | APE9-dihe-in | -120.74, 127.82 | APE8-dihe-in | -74.84, 77.33 | APE8-rot-na | 33.56 | APE67-dihe-in | -67.55, -20.32 | -45.2, -43.82 | APE12-dist-na | 11.3957 | APE11-dist-na | 8.9853 | APE10-dist-na | 9.7145 | APE9-dist-in | 6.3523 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 275.0 | 275.0 | 0 | 30 | 30 | 0 | [[624, 882]] | 1.0 | AF-P21709-K1 | TYR_EPHA1_HUMAN | TYR | 4.1e-101 | 343.6 | 3.0 | 260.0 | 258.0 | 766 | 767 | 768 | 770 | 772 | 656 | 673 | 677 | 746 | 748 | 747 | 749.0 | 808 | 796 | 791 | 790 | 789 | 788 | 787 | 786 | 785 | 703 | Ephrin type-A receptor 1 |
| TYR | EPHA1 | EPHA1_HUMAN | AF-P21709-K3A | P21709 | 616 | 890 | 976.0 | No_ligand | No_ligand | Active | DFGin | 5.8671 | 14.1273 | BLAminus | -139.82, -176.61 | 56.86, 65.42 | -78.07, 11.4 | 297.23, 94.02 | -60.31, -35.33 | in-in | in | 8.4837 | Saltbr-in | 2.812 | HRD-in | -75.32, -46.82 | 70.9, -7.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9093 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.88, 141.88 | APE9-dihe-in | -121.2, 130.06 | APE8-dihe-in | -76.18, 78.8 | APE8-rot-na | 35.3 | APE67-dihe-in | -62.82, -25.78 | -43.97, -44.95 | APE12-dist-na | 11.6361 | APE11-dist-na | 9.2606 | APE10-dist-na | 10.0232 | APE9-dist-in | 6.3952 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 275.0 | 275.0 | 0 | 30 | 30 | 0 | [[624, 882]] | 1.0 | AF-P21709-K3 | TYR_EPHA1_HUMAN | TYR | 4.1e-101 | 343.6 | 3.0 | 260.0 | 258.0 | 766 | 767 | 768 | 770 | 772 | 656 | 673 | 677 | 746 | 748 | 747 | 749.0 | 808 | 796 | 791 | 790 | 789 | 788 | 787 | 786 | 785 | 703 | Ephrin type-A receptor 1 |
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| TYR | EPHA1 | EPHA1_HUMAN | AF-P21709-K1A | P21709 | 616 | 890 | 976.0 | No_ligand | No_ligand | Active | DFGin | 6.0327 | 14.6832 | BLAminus | -138.4, -178.11 | 59.23, 67.7 | -84.1, 14.72 | 296.01, 92.0 | -60.59, -34.63 | in-in | in | 8.3875 | Saltbr-in | 2.7245 | HRD-in | -74.65, -44.09 | 68.7, -13.09 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9031 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.65, 144.12 | APE9-dihe-in | -120.74, 127.82 | APE8-dihe-in | -74.84, 77.33 | APE8-rot-na | 33.56 | APE67-dihe-in | -67.55, -20.32 | -45.2, -43.82 | APE12-dist-na | 11.3957 | APE11-dist-na | 8.9853 | APE10-dist-na | 9.7145 | APE9-dist-in | 6.3523 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 275.0 | 275.0 | 0 | 30 | 30 | 0 | [[624, 882]] | 1.0 | AF-P21709-K1 | Homo sapiens | TYR_EPHA1_HUMAN | TYR | 4.1e-101 | 343.6 | 3.0 | 260.0 | 258.0 | 766 | 767 | 768 | 770 | 772 | 656 | 673 | 677 | 746 | 748 | 747 | 749.0 | 808 | 796 | 791 | 790 | 789 | 788 | 787 | 786 | 785 | 703 | Ephrin type-A receptor 1 |
| TYR | EPHA1 | EPHA1_HUMAN | AF-P21709-K3A | P21709 | 616 | 890 | 976.0 | No_ligand | No_ligand | Active | DFGin | 5.8671 | 14.1273 | BLAminus | -139.82, -176.61 | 56.86, 65.42 | -78.07, 11.4 | 297.23, 94.02 | -60.31, -35.33 | in-in | in | 8.4837 | Saltbr-in | 2.812 | HRD-in | -75.32, -46.82 | 70.9, -7.99 | in-in-in | SNCiii | in-in | ActLoopNT-in | 2.9093 | ActLoopCT-in | TYR | APEdihe_iiiai | APEdist_aaai | APE10-dihe-in | -67.88, 141.88 | APE9-dihe-in | -121.2, 130.06 | APE8-dihe-in | -76.18, 78.8 | APE8-rot-na | 35.3 | APE67-dihe-in | -62.82, -25.78 | -43.97, -44.95 | APE12-dist-na | 11.6361 | APE11-dist-na | 9.2606 | APE10-dist-na | 10.0232 | APE9-dist-in | 6.3952 | None | None | None | AF2 | -1.0 | 1.0 | 1.0 | A | 275.0 | 275.0 | 0 | 30 | 30 | 0 | [[624, 882]] | 1.0 | AF-P21709-K3 | Homo sapiens | TYR_EPHA1_HUMAN | TYR | 4.1e-101 | 343.6 | 3.0 | 260.0 | 258.0 | 766 | 767 | 768 | 770 | 772 | 656 | 673 | 677 | 746 | 748 | 747 | 749.0 | 808 | 796 | 791 | 790 | 789 | 788 | 787 | 786 | 785 | 703 | Ephrin type-A receptor 1 |
| Spatial label | Dihedral label | Number of Chains | Percent | Representative |
|---|
| Group | Gene | SwissprotID | PDB | UniprotID | First_obs_res | Last_obs_res | Length_Unp | Ligand | Ligand_type | Activity_label | Spatial_label | Phe_Glu4_dis | Phe_Lys_dis | Dihedral_label | XDFG φ,ψ |
DFG-Asp φ,ψ |
DFG-Phe φ,ψ |
DFG-Phe χ1,χ2 |
DFG-Gly φ,ψ |
ChelixSaltbr_label | Chelix_label | Lys_Glu_dis | Saltbr_label | LysNZ_GluOE_dis | HRD_label | His φ,ψ | Arg φ,ψ | SNC_label | SNCpymol_label | ActLoop_label | ActLoopNT_label | DFG6_XHRD_dis | ActLoopCT_label | APEtype | APEdihe_label | APEdist_label | APE10_dihe_label | APE10 φ,ψ | APE9_dihe_label | APE9 φ,ψ | APE8_dihe_label | APE8 φ,ψ | APE8_rotamer_label | APE8 χ1 | APE67_label | APE6 φ,ψ | APE7 φ,ψ | APE12_dist_label | APE12_DFG4_dis | APE11_dist_label | APE11_DFG4_dis | APE10_dist_label | APE10_DFG4_dis | APE9_dist_label | APE9_Arg_dis | Chain_mut | Chain_phos | Modified_aa | Method | Resolution | Rvalue | FreeRvalue | Chain_id | ChainLen | Ordered_residues | DomainBreak | ActLoopLength | ActLoopResolvedResidues | ActLoopDisorderedResidues | Kinase_domains_Unp | N_Kinase_domains_Unp | pdb | Species | Kincore_name | hmm | Evalue | Score | hmmbeg | hmmend | hmmlen | XDFGnum | DFGnum | PHEnum | DFG4num | DFG6num | LYSnum | GLUnum | GLU4num | XHRDnum | ARGnum | HRDnum | HRDaspnum | aFaspnum | APEnum | APE6num | APE7num | APE8num | APE9num | APE10num | APE11num | APE12num | Hinge1num | Protein_name |
|---|